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2I89
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BU of 2i89 by Molmil
Structure of septuple mutant of Rat Outer Mitochondrial Membrane Cytochrome B5
分子名称: Cytochrome b5 type B, MAGNESIUM ION, PROTOPORPHYRIN IX CONTAINING FE
著者Terzyan, S, Zhang, X.C, Benson, D.R, Wang, L, Sun, N.
登録日2006-09-01
公開日2006-10-31
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献A histidine/tryptophan pi-stacking interaction stabilizes the heme-independent folding core of microsomal apocytochrome b5 relative to that of mitochondrial apocytochrome b5.
Biochemistry, 45, 2006
6MHE
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BU of 6mhe by Molmil
Galphai3 co-crystallized with KB752
分子名称: GLYCEROL, GUANOSINE-5'-DIPHOSPHATE, Guanine nucleotide-binding protein G(k) subunit alpha, ...
著者Rees, S.D, Kalogriopoulos, N.A, Ngo, T, Kopcho, N, Ilatovskiy, A, Sun, N, Komives, E, Chang, G, Ghosh, P, Kufareva, I.
登録日2018-09-17
公開日2019-07-31
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Structural basis for GPCR-independent activation of heterotrimeric Gi proteins.
Proc.Natl.Acad.Sci.USA, 116, 2019
6MHF
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BU of 6mhf by Molmil
Galphai3 co-crystallized with GIV/Girdin
分子名称: GLYCEROL, GUANOSINE-5'-DIPHOSPHATE, Girdin, ...
著者Rees, S.D, Kalogriopoulos, N.A, Ngo, T, Kopcho, N, Ilatovskiy, A, Sun, N, Komives, E, Chang, G, Ghosh, P, Kufareva, I.
登録日2018-09-17
公開日2019-07-31
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structural basis for GPCR-independent activation of heterotrimeric Gi proteins.
Proc.Natl.Acad.Sci.USA, 116, 2019
4HIL
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BU of 4hil by Molmil
1.25A Resolution Structure of Rat Type B Cytochrome b5
分子名称: Cytochrome b5 type B, PROTOPORPHYRIN IX CONTAINING FE, SODIUM ION
著者Lovell, S, Battaile, K.P, Parthasarathy, S, Sun, N, Terzyan, S, Zhang, X, Rivera, M, Kuczera, K, Benson, D.R.
登録日2012-10-11
公開日2013-10-16
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.25 Å)
主引用文献1.25A Resolution Structure of Rat Type B Cytochrome b5
To be Published
4HIN
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BU of 4hin by Molmil
2.4A Resolution Structure of Bovine Cytochrome b5 (S71L)
分子名称: COPPER (II) ION, Cytochrome b5, PROTOPORPHYRIN IX CONTAINING FE
著者Lovell, S, Battaile, K.P, Parthasarathy, S, Sun, N, Terzyan, S, Zhang, X, Rivera, M, Kuczera, K, Benson, D.R.
登録日2012-10-11
公開日2013-10-16
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献2.4A Resolution Structure of Bovine Cytochrome b5 (S71L)
To be Published
7XUQ
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BU of 7xuq by Molmil
Crystal structure of Tpe3.0 complexed with N-Boc-3-alkenylindole
分子名称: Transcriptional regulator, PadR-like family, dimethyl 2-[[2-methyl-1-[(2-methylpropan-2-yl)oxycarbonyl]indol-3-yl]methyl]-2-prop-2-enyl-propanedioate
著者Chen, X, Qian, J.Y, Sun, N.N, Zhong, F.R, Wu, Y.Z.
登録日2022-05-19
公開日2022-09-28
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Enantioselective [2+2]-cycloadditions with triplet photoenzymes.
Nature, 611, 2022
7XUP
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BU of 7xup by Molmil
Crystal structure of TPe3.0
分子名称: Transcriptional regulator, PadR-like family
著者Chen, X, Qian, J.Y, Sun, N.N, Zhong, F.R, Wu, Y.Z.
登録日2022-05-19
公開日2022-09-28
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.602 Å)
主引用文献Enantioselective [2+2]-cycloadditions with triplet photoenzymes.
Nature, 611, 2022
7CLF
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BU of 7clf by Molmil
PigF with SAH
分子名称: ACETATE ION, Methyltransferase domain-containing protein, S-ADENOSYL-L-HOMOCYSTEINE
著者Qiu, S, Xu, D, Han, N, Sun, B, Ran, T, Wang, W.
登録日2020-07-20
公開日2021-07-28
最終更新日2022-03-16
実験手法X-RAY DIFFRACTION (1.982 Å)
主引用文献Crystal structures of PigF, an O-methyltransferase involved in the prodigiosin synthetic pathway, reveal an induced-fit substrate-recognition mechanism.
Iucrj, 9, 2022
7CLU
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BU of 7clu by Molmil
PigF with SAH
分子名称: ACETATE ION, GLYCEROL, Methyltransferase domain-containing protein
著者Qiu, S, Xu, D, Han, N, Sun, B, Ran, T, Wang, W.
登録日2020-07-22
公開日2021-07-28
最終更新日2022-03-16
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Crystal structures of PigF, an O-methyltransferase involved in the prodigiosin synthetic pathway, reveal an induced-fit substrate-recognition mechanism.
Iucrj, 9, 2022
3TWJ
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BU of 3twj by Molmil
Rho-associated protein kinase 1 (ROCK 1) IN COMPLEX WITH RKI1447
分子名称: 1,2-ETHANEDIOL, 1-[(3-hydroxyphenyl)methyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)urea, Rho-associated protein kinase 1
著者Martin, M.P, Zhu, J.-Y, Schonbrunn, E.
登録日2011-09-21
公開日2012-08-22
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献RKI-1447 Is a Potent Inhibitor of the Rho-Associated ROCK Kinases with Anti-Invasive and Antitumor Activities in Breast Cancer.
Cancer Res., 72, 2012
8WD2
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BU of 8wd2 by Molmil
The Crystal Structure of p53 from Biortus.
分子名称: 1,2-ETHANEDIOL, Cellular tumor antigen p53, PHOSPHATE ION, ...
著者Wang, F, Cheng, W, Yuan, Z, Qi, J, Lu, Y.
登録日2023-09-14
公開日2023-10-04
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献The Crystal Structure of p53 from Biortus.
To Be Published
6CCA
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BU of 6cca by Molmil
Crystal structure of DszA carbon methyltransferase
分子名称: DisA protein
著者Meinke, J.L, Keatinge-Clay, A.T.
登録日2018-02-06
公開日2018-12-05
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Structural and Functional Studies of a gem-Dimethylating Methyltransferase from a trans-Acyltransferase Assembly Line.
ACS Chem. Biol., 13, 2018
7EFT
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BU of 7eft by Molmil
Crystal structure of cell shape-determining protein MreC
分子名称: CHLORIDE ION, Cell shape protein MreC
著者Xu, Q, Xiao, Q.J, Sun, B.
登録日2021-03-23
公開日2021-10-20
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献The crystal structure of MreC provides insights into polymer formation.
Febs Open Bio, 12, 2022
3V8S
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BU of 3v8s by Molmil
Human RHO-ASSOCIATED PROTEIN KINASE 1 (ROCK 1) IN COMPLEX WITH INDAZOLE DERIVATIVE (COMPOUND 18)
分子名称: 1-(1H-indazol-5-yl)-3-(2-phenylethyl)urea, Rho-associated protein kinase 1
著者Martin, M.P, Zhu, J.-Yi, Schonbrunn, E.
登録日2011-12-23
公開日2012-02-08
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (2.286 Å)
主引用文献Fragment-based and structure-guided discovery and optimization of rho kinase inhibitors.
J.Med.Chem., 55, 2012
6NO7
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BU of 6no7 by Molmil
Crystal Structure of the full-length wild-type PKA RIa Holoenzyme
分子名称: ADENOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, cAMP-dependent protein kinase catalytic subunit alpha, ...
著者Lu, T, Wu, J, Taylor, S.S.
登録日2019-01-15
公開日2019-07-24
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (3.55 Å)
主引用文献Two PKA RI alpha holoenzyme states define ATP as an isoform-specific orthosteric inhibitor that competes with the allosteric activator, cAMP.
Proc.Natl.Acad.Sci.USA, 116, 2019

219869

件を2024-05-15に公開中

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