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7YP5
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BU of 7yp5 by Molmil
Crystal structure of elaiophylin glycosyltransferase in complex with TDP
分子名称: CHLORIDE ION, Glycosyltransferase, R-1,2-PROPANEDIOL, ...
著者Xu, T, Liu, Q, Gan, Q, Liu, J.
登録日2022-08-02
公開日2022-11-02
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.33 Å)
主引用文献Substrate-induced dimerization of elaiophylin glycosyltransferase reveals a novel self-activating form of glycosyltransferase for symmetric glycosylation.
Acta Crystallogr D Struct Biol, 78, 2022
7YP4
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BU of 7yp4 by Molmil
Crystal structure of elaiophylin glycosyltransferase in apo-form
分子名称: Glycosyltransferase, R-1,2-PROPANEDIOL
著者Xu, T, Liu, Q, Gan, Q, Liu, J.
登録日2022-08-02
公開日2022-11-02
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献Substrate-induced dimerization of elaiophylin glycosyltransferase reveals a novel self-activating form of glycosyltransferase for symmetric glycosylation.
Acta Crystallogr D Struct Biol, 78, 2022
3NDM
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BU of 3ndm by Molmil
Crystal structure of Rho-Associated Protein Kinase (ROCK1) with a potent isoquinolone derivative
分子名称: (3S,4R)-N-(7-chloro-1-oxo-1,4-dihydroisoquinolin-6-yl)-4-(4-chlorophenyl)pyrrolidine-3-carboxamide, Rho-Associated Protein Kinase (ROCK1)
著者Li, X.
登録日2010-06-07
公開日2010-12-08
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (3.3 Å)
主引用文献Substituted 2H-isoquinolin-1-ones as potent Rho-kinase inhibitors: part 3, aryl substituted pyrrolidines.
Bioorg.Med.Chem.Lett., 20, 2010
5Z02
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BU of 5z02 by Molmil
Crystal structure of HIS6-tagged Mdm2 with nutlin-3a
分子名称: 4-({(4S,5R)-4,5-bis(4-chlorophenyl)-2-[4-methoxy-2-(propan-2-yloxy)phenyl]-4,5-dihydro-1H-imidazol-1-yl}carbonyl)piperazin-2-one, E3 ubiquitin-protein ligase Mdm2
著者Su, Z.D, Cheng, X.Y, Chen, R, Pi, N.
登録日2017-12-18
公開日2018-01-03
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (1.35 Å)
主引用文献Crystal structure of HIS6-tagged Mdm2 with nutlin-3a
to be published
5ZXF
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BU of 5zxf by Molmil
The 1.25A Crystal structure of His6-tagged Mdm2 in complex with nutlin-3a
分子名称: 4-({(4S,5R)-4,5-bis(4-chlorophenyl)-2-[4-methoxy-2-(propan-2-yloxy)phenyl]-4,5-dihydro-1H-imidazol-1-yl}carbonyl)piperazin-2-one, E3 ubiquitin-protein ligase Mdm2
著者Cheng, X.Y, Su, Z.D, Pi, N, Cao, C.Z, Zhao, Z.T, Zhou, J.J, Chen, R, Kuang, Z.K, Huang, Y.Q.
登録日2018-05-19
公開日2018-08-22
最終更新日2024-03-27
実験手法X-RAY DIFFRACTION (1.25 Å)
主引用文献The 1.25A Crystal structure of His6-tagged Mdm2 in complex with nutlin-3a
To Be Published

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件を2024-05-15に公開中

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