Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help
Search by PDB author
5AMH
DownloadVisualize
BU of 5amh by Molmil
Cereblon isoform 4 from Magnetospirillum gryphiswaldense in complex with Thalidomide, trigonal crystal form
Descriptor: CALCIUM ION, CEREBLON ISOFORM 4, CHLORIDE ION, ...
Authors:Hartmann, M.D, Lupas, A.N, Hernandez Alvarez, B.
Deposit date:2015-03-10
Release date:2015-07-01
Last modified:2024-01-10
Method:X-RAY DIFFRACTION (1.2 Å)
Cite:Structural Dynamics of the Cereblon Ligand Binding Domain.
Plos One, 10, 2015
5APS
DownloadVisualize
BU of 5aps by Molmil
Sequence IENKKAD inserted between GCN4 adaptors - Structure A7
Descriptor: GENERAL CONTROL PROTEIN GCN4
Authors:Hartmann, M.D, Mendler, C.T, Lupas, A.N, Hernandez Alvarez, B.
Deposit date:2015-09-17
Release date:2016-01-27
Last modified:2024-01-10
Method:X-RAY DIFFRACTION (1.37 Å)
Cite:alpha / beta coiled coils.
Elife, 5, 2016
5APQ
DownloadVisualize
BU of 5apq by Molmil
Sequence IENKAD inserted between GCN4 adaptors - Structure A6
Descriptor: GENERAL CONTROL PROTEIN GCN4
Authors:Hartmann, M.D, Mendler, C.T, Lupas, A.N, Hernandez Alvarez, B.
Deposit date:2015-09-17
Release date:2016-01-27
Last modified:2024-01-10
Method:X-RAY DIFFRACTION (2.1 Å)
Cite:alpha / beta coiled coils.
Elife, 5, 2016
5APX
DownloadVisualize
BU of 5apx by Molmil
Sequence MATKDDIAN inserted between GCN4 adaptors - Structure T9(6)
Descriptor: GENERAL CONTROL PROTEIN GCN4, PHOSPHATE ION
Authors:Hartmann, M.D, Mendler, C.T, Lupas, A.N, Hernandez Alvarez, B.
Deposit date:2015-09-17
Release date:2016-01-27
Last modified:2024-01-10
Method:X-RAY DIFFRACTION (1.8 Å)
Cite:alpha / beta coiled coils.
Elife, 5, 2016
2WPQ
DownloadVisualize
BU of 2wpq by Molmil
Salmonella enterica SadA 479-519 fused to GCN4 adaptors (SadAK3, in- register fusion)
Descriptor: CHLORIDE ION, NITRATE ION, TRIMERIC AUTOTRANSPORTER ADHESIN FRAGMENT
Authors:Hartmann, M.D, Hernandez Alvarez, B, Albrecht, R, Zeth, K, Lupas, A.N.
Deposit date:2009-08-09
Release date:2009-11-03
Last modified:2023-12-20
Method:X-RAY DIFFRACTION (1.85 Å)
Cite:A Coiled-Coil Motif that Sequesters Ions to the Hydrophobic Core.
Proc.Natl.Acad.Sci.USA, 106, 2009
5OH8
DownloadVisualize
BU of 5oh8 by Molmil
Cereblon isoform 4 from Magnetospirillum gryphiswaldense in complex with Rolipram
Descriptor: Cereblon isoform 4, ROLIPRAM, ZINC ION
Authors:Boichenko, I, Albrecht, R, Lupas, A.N, Hernandez Alvarez, B, Hartmann, M.D.
Deposit date:2017-07-14
Release date:2018-10-10
Last modified:2024-01-17
Method:X-RAY DIFFRACTION (1.95 Å)
Cite:Chemical Ligand Space of Cereblon.
Acs Omega, 3, 2018
5OH4
DownloadVisualize
BU of 5oh4 by Molmil
Cereblon isoform 4 from Magnetospirillum gryphiswaldense in complex with Piperidine-2,6-dione (Glutarimide)
Descriptor: Cereblon isoform 4, ZINC ION, piperidine-2,6-dione
Authors:Boichenko, I, Albrecht, R, Lupas, A.N, Hernandez Alvarez, B, Hartmann, M.D.
Deposit date:2017-07-14
Release date:2018-10-10
Last modified:2024-01-17
Method:X-RAY DIFFRACTION (2.3 Å)
Cite:Chemical Ligand Space of Cereblon.
Acs Omega, 3, 2018
5OH2
DownloadVisualize
BU of 5oh2 by Molmil
Cereblon isoform 4 from Magnetospirillum gryphiswaldense in complex with Pyrrolidin-2-one (Butyrolactam)
Descriptor: Cereblon isoform 4, ZINC ION, pyrrolidin-2-one
Authors:Boichenko, I, Albrecht, R, Lupas, A.N, Hernandez Alvarez, B, Hartmann, M.D.
Deposit date:2017-07-14
Release date:2018-10-10
Last modified:2024-01-17
Method:X-RAY DIFFRACTION (1.9 Å)
Cite:Chemical Ligand Space of Cereblon.
Acs Omega, 3, 2018
5OHB
DownloadVisualize
BU of 5ohb by Molmil
Cereblon isoform 4 from Magnetospirillum gryphiswaldense in complex with Piperidin-2-one (Valerolactam)
Descriptor: Cereblon isoform 4, ZINC ION, piperidin-2-one
Authors:Boichenko, I, Albrecht, R, Lupas, A.N, Hernandez Alvarez, B, Hartmann, M.D.
Deposit date:2017-07-14
Release date:2018-10-10
Last modified:2024-01-17
Method:X-RAY DIFFRACTION (1.7 Å)
Cite:Chemical Ligand Space of Cereblon.
Acs Omega, 3, 2018
5OH1
DownloadVisualize
BU of 5oh1 by Molmil
Cereblon isoform 4 from Magnetospirillum gryphiswaldense in complex with Aminoglutethimide
Descriptor: (3~{R})-3-(4-aminophenyl)-3-ethyl-piperidine-2,6-dione, Cereblon isoform 4, S-Thalidomide, ...
Authors:Boichenko, I, Albrecht, R, Lupas, A.N, Hernandez Alvarez, B, Hartmann, M.D.
Deposit date:2017-07-14
Release date:2018-10-10
Last modified:2024-01-17
Method:X-RAY DIFFRACTION (1.7 Å)
Cite:Chemical Ligand Space of Cereblon.
Acs Omega, 3, 2018
5OH9
DownloadVisualize
BU of 5oh9 by Molmil
Cereblon isoform 4 from Magnetospirillum gryphiswaldense in complex with Thiazolidine-2,4-dione
Descriptor: 1,3-thiazole-2,4-dione, Cereblon isoform 4, ZINC ION
Authors:Boichenko, I, Albrecht, R, Lupas, A.N, Hernandez Alvarez, B, Hartmann, M.D.
Deposit date:2017-07-14
Release date:2018-10-10
Last modified:2024-01-17
Method:X-RAY DIFFRACTION (1.65 Å)
Cite:Chemical Ligand Space of Cereblon.
Acs Omega, 3, 2018
5OH3
DownloadVisualize
BU of 5oh3 by Molmil
Cereblon isoform 4 from Magnetospirillum gryphiswaldense in complex with Ethosuximide
Descriptor: (3~{S})-3-ethyl-3-methyl-pyrrolidine-2,5-dione, Cereblon isoform 4, ZINC ION
Authors:Boichenko, I, Albrecht, R, Lupas, A.N, Hernandez Alvarez, B, Hartmann, M.D.
Deposit date:2017-07-14
Release date:2018-10-10
Last modified:2024-01-17
Method:X-RAY DIFFRACTION (2.1 Å)
Cite:Chemical Ligand Space of Cereblon.
Acs Omega, 3, 2018
5OHA
DownloadVisualize
BU of 5oha by Molmil
Cereblon isoform 4 from Magnetospirillum gryphiswaldense in complex with 2-Thiohydantoin
Descriptor: 2-sulfanylideneimidazol-4-one, Cereblon isoform 4, ZINC ION
Authors:Boichenko, I, Albrecht, R, Lupas, A.N, Hernandez Alvarez, B, Hartmann, M.D.
Deposit date:2017-07-14
Release date:2018-10-10
Last modified:2024-01-17
Method:X-RAY DIFFRACTION (1.55 Å)
Cite:Chemical Ligand Space of Cereblon.
Acs Omega, 3, 2018
5OH7
DownloadVisualize
BU of 5oh7 by Molmil
Cereblon isoform 4 from Magnetospirillum gryphiswaldense in complex with Imidazolidine-2,4-dione (Hydantoin)
Descriptor: Cereblon isoform 4, ZINC ION, imidazolidine-2,4-dione
Authors:Boichenko, I, Albrecht, R, Lupas, A.N, Hernandez Alvarez, B, Hartmann, M.D.
Deposit date:2017-07-14
Release date:2018-10-10
Last modified:2024-01-17
Method:X-RAY DIFFRACTION (1.85 Å)
Cite:Chemical Ligand Space of Cereblon.
Acs Omega, 3, 2018
6Y06
DownloadVisualize
BU of 6y06 by Molmil
Moevan: a designed granulopoietic protein by topological rescaffolding
Descriptor: Moevan
Authors:ElGamacy, M, Coles, M.
Deposit date:2020-02-06
Release date:2020-03-18
Last modified:2023-06-14
Method:SOLUTION NMR
Cite:Design of novel granulopoietic proteins by topological rescaffolding.
Plos Biol., 18, 2020
6Y07
DownloadVisualize
BU of 6y07 by Molmil
Designing a Granulopoietic Protein by Topological Rescaffolding 1: Sohair
Descriptor: sohair
Authors:ElGamacy, M, Coles, M.
Deposit date:2020-02-06
Release date:2020-03-18
Last modified:2024-05-15
Method:SOLUTION NMR
Cite:Design of novel granulopoietic proteins by topological rescaffolding.
Plos Biol., 18, 2020
7NY0
DownloadVisualize
BU of 7ny0 by Molmil
Solution structure of Boskar4; a de novo designed G-CSF agonist
Descriptor: Boskar4
Authors:ElGamacy, M, Coles, M.
Deposit date:2021-03-19
Release date:2021-10-06
Last modified:2022-06-08
Method:SOLUTION NMR
Cite:A topological refactoring design strategy yields highly stable granulopoietic proteins.
Nat Commun, 13, 2022
6R18
DownloadVisualize
BU of 6r18 by Molmil
Cereblon isoform 4 from Magnetospirillum gryphiswaldense in complex with compound 11a
Descriptor: CHLORIDE ION, Cereblon isoform 4, PHOSPHATE ION, ...
Authors:Heim, C, Hartmann, M.D.
Deposit date:2019-03-14
Release date:2019-08-07
Last modified:2024-01-24
Method:X-RAY DIFFRACTION (1.35 Å)
Cite:De-Novo Design of Cereblon (CRBN) Effectors Guided by Natural Hydrolysis Products of Thalidomide Derivatives.
J.Med.Chem., 62, 2019
6R19
DownloadVisualize
BU of 6r19 by Molmil
Cereblon isoform 4 from Magnetospirillum gryphiswaldense in complex with compound 20a
Descriptor: Cereblon isoform 4, PHOSPHATE ION, S-Thalidomide, ...
Authors:Heim, C, Hartmann, M.D.
Deposit date:2019-03-14
Release date:2019-08-07
Last modified:2024-01-24
Method:X-RAY DIFFRACTION (1.45 Å)
Cite:De-Novo Design of Cereblon (CRBN) Effectors Guided by Natural Hydrolysis Products of Thalidomide Derivatives.
J.Med.Chem., 62, 2019
6R1A
DownloadVisualize
BU of 6r1a by Molmil
Cereblon isoform 4 from Magnetospirillum gryphiswaldense in complex with compound 20b
Descriptor: Cereblon isoform 4, PHOSPHATE ION, S-Thalidomide, ...
Authors:Heim, C, Hartmann, M.D.
Deposit date:2019-03-14
Release date:2019-08-07
Last modified:2024-01-24
Method:X-RAY DIFFRACTION (1.54 Å)
Cite:De-Novo Design of Cereblon (CRBN) Effectors Guided by Natural Hydrolysis Products of Thalidomide Derivatives.
J.Med.Chem., 62, 2019
6R1D
DownloadVisualize
BU of 6r1d by Molmil
Cereblon isoform 4 from Magnetospirillum gryphiswaldense in complex with compound 7d, co-crystallized
Descriptor: (phenylmethyl) ~{N}-[(3~{S})-2,5-bis(oxidanylidene)pyrrolidin-3-yl]carbamate, Cereblon isoform 4, ZINC ION
Authors:Heim, C, Hartmann, M.D.
Deposit date:2019-03-14
Release date:2019-08-07
Last modified:2024-01-24
Method:X-RAY DIFFRACTION (1.1 Å)
Cite:De-Novo Design of Cereblon (CRBN) Effectors Guided by Natural Hydrolysis Products of Thalidomide Derivatives.
J.Med.Chem., 62, 2019
6R1K
DownloadVisualize
BU of 6r1k by Molmil
Cereblon isoform 4 from Magnetospirillum gryphiswaldense in complex with compound 7c
Descriptor: Cereblon isoform 4, PHOSPHATE ION, ZINC ION, ...
Authors:Heim, C, Hartmann, M.D.
Deposit date:2019-03-14
Release date:2019-08-07
Last modified:2024-01-24
Method:X-RAY DIFFRACTION (1.94 Å)
Cite:De-Novo Design of Cereblon (CRBN) Effectors Guided by Natural Hydrolysis Products of Thalidomide Derivatives.
J.Med.Chem., 62, 2019
6R1W
DownloadVisualize
BU of 6r1w by Molmil
Cereblon isoform 4 from Magnetospirillum gryphiswaldense in complex with compound 16b
Descriptor: (4-azanylcyclohexyl)methyl ~{N}-[(3~{S})-2,6-bis(oxidanylidene)piperidin-3-yl]carbamate, Cereblon isoform 4, PHOSPHATE ION, ...
Authors:Heim, C, Hartmann, M.D.
Deposit date:2019-03-15
Release date:2019-08-07
Last modified:2024-01-24
Method:X-RAY DIFFRACTION (1.35 Å)
Cite:De-Novo Design of Cereblon (CRBN) Effectors Guided by Natural Hydrolysis Products of Thalidomide Derivatives.
J.Med.Chem., 62, 2019
6R1X
DownloadVisualize
BU of 6r1x by Molmil
Cereblon isoform 4 from Magnetospirillum gryphiswaldense in complex with compound 7a
Descriptor: Cereblon isoform 4, ZINC ION, ~{N}-[(3~{S})-2,5-bis(oxidanylidene)pyrrolidin-3-yl]-3-methyl-but-2-enamide
Authors:Heim, C, Hartmann, M.D.
Deposit date:2019-03-15
Release date:2019-08-07
Last modified:2024-05-15
Method:X-RAY DIFFRACTION (1.8 Å)
Cite:De-Novo Design of Cereblon (CRBN) Effectors Guided by Natural Hydrolysis Products of Thalidomide Derivatives.
J.Med.Chem., 62, 2019
6R1C
DownloadVisualize
BU of 6r1c by Molmil
Cereblon isoform 4 from Magnetospirillum gryphiswaldense in complex with compound 12a
Descriptor: 4-[[4-[[(3~{S})-2,5-bis(oxidanylidene)pyrrolidin-3-yl]carbamoyloxymethyl]phenyl]methylamino]-4-oxidanylidene-butanoic acid, ASPARTIC ACID, CHLORIDE ION, ...
Authors:Heim, C, Hartmann, M.D.
Deposit date:2019-03-14
Release date:2019-08-07
Last modified:2024-01-24
Method:X-RAY DIFFRACTION (1.5 Å)
Cite:De-Novo Design of Cereblon (CRBN) Effectors Guided by Natural Hydrolysis Products of Thalidomide Derivatives.
J.Med.Chem., 62, 2019

221051

數據於2024-06-12公開中

PDB statisticsPDBj update infoContact PDBjnumon