5JLJ
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![BU of 5jlj by Molmil](/molmil-images/mine/5jlj) | Crystal Structure of KPT8602 in complex with CRM1-Ran-RanBP1 | Descriptor: | (2R)-3-{3-[3,5-bis(trifluoromethyl)phenyl]-1H-1,2,4-triazol-1-yl}-2-(pyrimidin-5-yl)propanamide, CHLORIDE ION, Exportin-1, ... | Authors: | Fung, H.Y, Chook, Y.M. | Deposit date: | 2016-04-27 | Release date: | 2016-06-29 | Last modified: | 2023-09-27 | Method: | X-RAY DIFFRACTION (2.5 Å) | Cite: | Next-generation XPO1 inhibitor shows improved efficacy and in vivo tolerability in hematological malignancies. Leukemia, 30, 2016
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7L5E
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![BU of 7l5e by Molmil](/molmil-images/mine/7l5e) | |
2M4M
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![BU of 2m4m by Molmil](/molmil-images/mine/2m4m) | Solution structure of the RRM domain of the hypothetical protein CAGL0M09691g from Candida glabrata | Descriptor: | hypothetical protein | Authors: | Harris, R, Hillerich, B, Ahmed, M, Bonanno, J.B, Chamala, S, Evans, B, Lafleur, J, Hammonds, J, Washington, E, Stead, M, Love, J, Attonito, J, Patel, H, Seidel, R.D, Chook, Y.M, Rout, M.P, Girvin, M.E, Almo, S.C, New York Structural Genomics Research Consortium (NYSGRC), Nucleocytoplasmic Transport: a Target for Cellular Control (NPCXstals) | Deposit date: | 2013-02-07 | Release date: | 2013-02-27 | Last modified: | 2024-05-15 | Method: | SOLUTION NMR | Cite: | Solution structure of the RRM domain of the hypothetical protein CAGL0M09691g from Candida glabrata To be Published
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2OT8
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![BU of 2ot8 by Molmil](/molmil-images/mine/2ot8) | |
2QMR
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![BU of 2qmr by Molmil](/molmil-images/mine/2qmr) | Karyopherin beta2/transportin | Descriptor: | Transportin-1 | Authors: | Cansizoglu, A.E, Chook, Y.M. | Deposit date: | 2007-07-16 | Release date: | 2007-10-30 | Last modified: | 2023-08-30 | Method: | X-RAY DIFFRACTION (3 Å) | Cite: | Conformational heterogeneity of karyopherin beta2 is segmental Structure, 15, 2007
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5YVG
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![BU of 5yvg by Molmil](/molmil-images/mine/5yvg) | |
5YVI
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![BU of 5yvi by Molmil](/molmil-images/mine/5yvi) | |
5YVH
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![BU of 5yvh by Molmil](/molmil-images/mine/5yvh) | |
5DHF
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![BU of 5dhf by Molmil](/molmil-images/mine/5dhf) | |
5DH9
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![BU of 5dh9 by Molmil](/molmil-images/mine/5dh9) | |
5DHA
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![BU of 5dha by Molmil](/molmil-images/mine/5dha) | |
5DIF
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![BU of 5dif by Molmil](/molmil-images/mine/5dif) | |
5DI9
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![BU of 5di9 by Molmil](/molmil-images/mine/5di9) | |
5UWJ
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![BU of 5uwj by Molmil](/molmil-images/mine/5uwj) | |
5UWQ
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![BU of 5uwq by Molmil](/molmil-images/mine/5uwq) | |
5UWI
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![BU of 5uwi by Molmil](/molmil-images/mine/5uwi) | |
5UWU
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![BU of 5uwu by Molmil](/molmil-images/mine/5uwu) | |
5UWR
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![BU of 5uwr by Molmil](/molmil-images/mine/5uwr) | |
5UWP
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![BU of 5uwp by Molmil](/molmil-images/mine/5uwp) | |
5UWO
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![BU of 5uwo by Molmil](/molmil-images/mine/5uwo) | |
5UWH
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![BU of 5uwh by Molmil](/molmil-images/mine/5uwh) | |
5UWT
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![BU of 5uwt by Molmil](/molmil-images/mine/5uwt) | |
5UWS
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![BU of 5uws by Molmil](/molmil-images/mine/5uws) | |
5UWW
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![BU of 5uww by Molmil](/molmil-images/mine/5uww) | |
6XJT
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![BU of 6xjt by Molmil](/molmil-images/mine/6xjt) | Crystal Structure of KPT-8602 bound to CRM1 (537-DLTVK-541 to GLCEQ) | Descriptor: | (2R)-3-{3-[3,5-bis(trifluoromethyl)phenyl]-1H-1,2,4-triazol-1-yl}-2-(pyrimidin-5-yl)propanamide, Exportin-1, GTP-binding nuclear protein Ran, ... | Authors: | Baumhardt, J.M, Chook, Y.M. | Deposit date: | 2020-06-24 | Release date: | 2021-01-27 | Last modified: | 2023-10-18 | Method: | X-RAY DIFFRACTION (2.406 Å) | Cite: | Recurrent XPO1 mutations alter pathogenesis of chronic lymphocytic leukemia. J Hematol Oncol, 14, 2021
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