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THE THREE-DIMENSIONAL STRUCTURE OF ASN102 MUTANT OF TRYPSIN. ROLE OF ASP102 IN SERINE PROTEASE CATALYSIS
Descriptor:	BENZAMIDINE, CALCIUM ION, TRYPSIN
Authors:	Sprang, S, Standing, T, Fletterick, R.J.
Deposit date:	1987-10-21
Release date:	1988-07-16
Last modified:	2017-11-29
Method:	X-RAY DIFFRACTION (2.3 Å)
Cite:	The three-dimensional structure of Asn102 mutant of trypsin: role of Asp102 in serine protease catalysis. Science, 237, 1987

1C1O

RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES
Descriptor:	CALCIUM ION, MAGNESIUM ION, SULFATE ION, ...
Authors:	Katz, B.A, Luong, C.
Deposit date:	1999-07-21
Release date:	2000-07-26
Last modified:	2023-12-27
Method:	X-RAY DIFFRACTION (1.4 Å)
Cite:	Design of potent selective zinc-mediated serine protease inhibitors. Nature, 391, 1998

1C1V

RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES
Descriptor:	BIS(5-AMIDINO-BENZIMIDAZOLYL)METHANE, Hirudin-2, SODIUM ION, ...
Authors:	Katz, B.A, Luong, C.
Deposit date:	1999-07-21
Release date:	2000-07-26
Last modified:	2023-11-15
Method:	X-RAY DIFFRACTION (1.98 Å)
Cite:	Design of potent selective zinc-mediated serine protease inhibitors. Nature, 391, 1998

1C2I

RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES
Descriptor:	BIS(5-AMIDINO-2-BENZIMIDAZOLYL)METHANE KETONE, CALCIUM ION, CHLORIDE ION, ...
Authors:	Katz, B.A, Luong, C.
Deposit date:	1999-07-21
Release date:	2000-07-26
Last modified:	2023-12-27
Method:	X-RAY DIFFRACTION (1.47 Å)
Cite:	Design of potent selective zinc-mediated serine protease inhibitors. Nature, 391, 1998

1C2D

RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES
Descriptor:	BIS(5-AMIDINO-2-BENZIMIDAZOLYL)METHANE KETONE, CALCIUM ION, MAGNESIUM ION, ...
Authors:	Katz, B.A, Luong, C.
Deposit date:	1999-07-21
Release date:	2000-07-26
Last modified:	2023-12-27
Method:	X-RAY DIFFRACTION (1.65 Å)
Cite:	Design of potent selective zinc-mediated serine protease inhibitors. Nature, 391, 1998

1C1P

RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES
Descriptor:	(5-AMIDINO-2-BENZIMIDAZOLYL)(2-BENZIMIDAZOLYL)METHANE, CALCIUM ION, DIMETHYL SULFOXIDE, ...
Authors:	Katz, B.A, Luong, C.
Deposit date:	1999-07-21
Release date:	2000-07-26
Last modified:	2023-12-27
Method:	X-RAY DIFFRACTION (1.37 Å)
Cite:	Design of potent selective zinc-mediated serine protease inhibitors. Nature, 391, 1998

1C1U

RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES
Descriptor:	(5-AMIDINO-2-BENZIMIDAZOLYL)(2-BENZIMIDAZOLYL)METHANE, ACETYL HIRUDIN, ALPHA THROMBIN, ...
Authors:	Katz, B.A, Luong, C.
Deposit date:	1999-07-21
Release date:	2000-07-26
Last modified:	2023-11-15
Method:	X-RAY DIFFRACTION (1.75 Å)
Cite:	Design of potent selective zinc-mediated serine protease inhibitors. Nature, 391, 1998

1C2F

RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES
Descriptor:	BIS(5-AMIDINO-2-BENZIMIDAZOLYL)METHANE KETONE HYDRATE, CALCIUM ION, DIMETHYL SULFOXIDE, ...
Authors:	Katz, B.A, Luong, C.
Deposit date:	1999-07-21
Release date:	2000-07-26
Last modified:	2023-12-27
Method:	X-RAY DIFFRACTION (1.7 Å)
Cite:	Design of potent selective zinc-mediated serine protease inhibitors. Nature, 391, 1998

1C1R

RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES
Descriptor:	(5-AMIDINO-2-BENZIMIDAZOLYL)(2-BENZIMIDAZOLYL)METHANE, CALCIUM ION, DIMETHYL SULFOXIDE, ...
Authors:	Katz, B.A, Luong, C.
Deposit date:	1999-07-21
Release date:	2000-07-26
Last modified:	2023-12-27
Method:	X-RAY DIFFRACTION (1.37 Å)
Cite:	Design of potent selective zinc-mediated serine protease inhibitors. Nature, 391, 1998

1C2K

RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES
Descriptor:	5-AMIDINO-BENZIMIDAZOLE, CALCIUM ION, CHLORIDE ION, ...
Authors:	Katz, B.A, Luong, C.
Deposit date:	1999-07-21
Release date:	2000-07-26
Last modified:	2023-12-27
Method:	X-RAY DIFFRACTION (1.65 Å)
Cite:	Design of potent selective zinc-mediated serine protease inhibitors. Nature, 391, 1998

1AJM

CRYSTAL STRUCTURE OF THYMIDYLATE SYNTHASE R126E MUTANT
Descriptor:	THYMIDYLATE SYNTHASE
Authors:	Strop, P, Montfort, W.R.
Deposit date:	1997-05-06
Release date:	1997-11-12
Last modified:	2021-11-03
Method:	X-RAY DIFFRACTION (2.4 Å)
Cite:	Crystal structures of a marginally active thymidylate synthase mutant, Arg 126-->Glu. Protein Sci., 6, 1997

1C2M

RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES
Descriptor:	CALCIUM ION, MAGNESIUM ION, SULFATE ION, ...
Authors:	Katz, B.A, Luong, C.
Deposit date:	1999-07-21
Release date:	2000-07-26
Last modified:	2023-12-27
Method:	X-RAY DIFFRACTION (1.4 Å)
Cite:	Design of potent selective zinc-mediated serine protease inhibitors. Nature, 391, 1998

1C2G

RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES
Descriptor:	BIS(5-AMIDINO-2-BENZIMIDAZOLYL)METHANE KETONE HYDRATE, CALCIUM ION, DIMETHYL SULFOXIDE, ...
Authors:	Katz, B.A, Luong, C.
Deposit date:	1999-07-21
Release date:	2000-07-26
Last modified:	2023-12-27
Method:	X-RAY DIFFRACTION (1.65 Å)
Cite:	Design of potent selective zinc-mediated serine protease inhibitors. Nature, 391, 1998

1C2E

RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES
Descriptor:	BIS(5-AMIDINO-2-BENZIMIDAZOLYL)METHANE KETONE, CALCIUM ION, MAGNESIUM ION, ...
Authors:	Katz, B.A, Luong, C.
Deposit date:	1999-07-22
Release date:	2000-07-26
Last modified:	2023-12-27
Method:	X-RAY DIFFRACTION (1.65 Å)
Cite:	Design of potent selective zinc-mediated serine protease inhibitors. Nature, 391, 1998

1C1N

RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES
Descriptor:	BENZAMIDINE, CALCIUM ION, SULFATE ION, ...
Authors:	Katz, B.A, Luong, C.
Deposit date:	1999-07-21
Release date:	2000-07-26
Last modified:	2023-12-27
Method:	X-RAY DIFFRACTION (1.4 Å)
Cite:	Design of potent selective zinc-mediated serine protease inhibitors. Nature, 391, 1998

1C1W

RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES
Descriptor:	BIS(5-AMIDINO-2-BENZIMIDAZOLYL)METHANE KETONE HYDRATE, Hirudin-2, SODIUM ION, ...
Authors:	Katz, B.A, Luong, C.
Deposit date:	1999-07-21
Release date:	2000-07-26
Last modified:	2023-11-15
Method:	X-RAY DIFFRACTION (1.9 Å)
Cite:	Design of potent selective zinc-mediated serine protease inhibitors. Nature, 391, 1998

1C2H

RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES
Descriptor:	BIS(5-AMIDINO-2-BENZIMIDAZOLYL)METHANE KETONE, CALCIUM ION, MAGNESIUM ION, ...
Authors:	Katz, B.A, Luong, C.
Deposit date:	1999-07-21
Release date:	2000-07-26
Last modified:	2023-12-27
Method:	X-RAY DIFFRACTION (1.4 Å)
Cite:	Design of potent selective zinc-mediated serine protease inhibitors. Nature, 391, 1998

1C2J

RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES
Descriptor:	BIS(5-AMIDINO-2-BENZIMIDAZOLYL)METHANE KETONE, CALCIUM ION, MAGNESIUM ION, ...
Authors:	Katz, B.A, Luong, C.
Deposit date:	1999-07-21
Release date:	2000-07-26
Last modified:	2023-12-27
Method:	X-RAY DIFFRACTION (1.4 Å)
Cite:	Design of potent selective zinc-mediated serine protease inhibitors. Nature, 391, 1998

1EER

CRYSTAL STRUCTURE OF HUMAN ERYTHROPOIETIN COMPLEXED TO ITS RECEPTOR AT 1.9 ANGSTROMS
Descriptor:	ERYTHROPOIETIN, ERYTHROPOIETIN RECEPTOR
Authors:	Syed, R.S, Li, C.
Deposit date:	1998-07-24
Release date:	1999-10-01
Last modified:	2021-11-03
Method:	X-RAY DIFFRACTION (1.9 Å)
Cite:	Efficiency of signalling through cytokine receptors depends critically on receptor orientation. Nature, 395, 1998

1C1T

RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES
Descriptor:	BIS(5-AMIDINO-BENZIMIDAZOLYL)METHANE, CALCIUM ION, MAGNESIUM ION, ...
Authors:	Katz, B.A, Luong, C.
Deposit date:	1999-07-21
Release date:	2000-07-26
Last modified:	2023-12-27
Method:	X-RAY DIFFRACTION (1.37 Å)
Cite:	Design of potent selective zinc-mediated serine protease inhibitors. Nature, 391, 1998

1C2L

RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES
Descriptor:	CALCIUM ION, CHLORIDE ION, TRYPSIN, ...
Authors:	Katz, B.A, Luong, C.
Deposit date:	1999-07-21
Release date:	2000-07-26
Last modified:	2023-12-27
Method:	X-RAY DIFFRACTION (1.5 Å)
Cite:	Design of potent selective zinc-mediated serine protease inhibitors. Nature, 391, 1998

1C1Q

RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES
Descriptor:	(5-AMIDINO-2-BENZIMIDAZOLYL)(2-BENZIMIDAZOLYL)METHANE, CALCIUM ION, MAGNESIUM ION, ...
Authors:	Katz, B.A, Luong, C.
Deposit date:	1999-07-21
Release date:	2000-07-26
Last modified:	2023-12-27
Method:	X-RAY DIFFRACTION (1.37 Å)
Cite:	Design of potent selective zinc-mediated serine protease inhibitors. Nature, 391, 1998

5ESI

Saccharomyces cerevisiae CYP51 (Lanosterol 14-alpha demethylase) G73W mutant
Descriptor:	Lanosterol 14-alpha demethylase, PROTOPORPHYRIN IX CONTAINING FE
Authors:	Sagatova, A, Keniya, M.V, Wilson, R, Sabherwal, M, Tyndall, J.D.A, Monk, B.C.
Deposit date:	2015-11-16
Release date:	2016-11-23
Last modified:	2023-09-27
Method:	X-RAY DIFFRACTION (2.1 Å)
Cite:	Impact of Homologous Resistance Mutations from Pathogenic Yeast on Saccharomyces cerevisiae Lanosterol 14 alpha-Demethylase. Antimicrob.Agents Chemother., 62, 2018

5ESE

Saccharomyces cerevisiae CYP51 (Lanosterol 14-alpha demethylase) G73R mutant complexed with fluconazole
Descriptor:	2-(2,4-DIFLUOROPHENYL)-1,3-DI(1H-1,2,4-TRIAZOL-1-YL)PROPAN-2-OL, Lanosterol 14-alpha demethylase, PROTOPORPHYRIN IX CONTAINING FE
Authors:	Sagatova, A, Keniya, M.V, Wilson, R.K, Sabherwal, M, Tyndall, J.D.A, Monk, B.C.
Deposit date:	2015-11-16
Release date:	2016-11-23
Last modified:	2023-09-27
Method:	X-RAY DIFFRACTION (2.2 Å)
Cite:	Impact of Homologous Resistance Mutations from Pathogenic Yeast on Saccharomyces cerevisiae Lanosterol 14 alpha-Demethylase. Antimicrob.Agents Chemother., 62, 2018

5ESF

Saccharomyces cerevisiae CYP51 (Lanosterol 14-alpha demethylase) G73E mutant complexed with fluconazole
Descriptor:	2-(2,4-DIFLUOROPHENYL)-1,3-DI(1H-1,2,4-TRIAZOL-1-YL)PROPAN-2-OL, Lanosterol 14-alpha demethylase, PROTOPORPHYRIN IX CONTAINING FE
Authors:	Sagatova, A, Keniya, M.V, Wilson, R.K, Sabherwal, M, Tyndall, J.D.A, Monk, B.C.
Deposit date:	2015-11-16
Release date:	2016-11-23
Last modified:	2023-09-27
Method:	X-RAY DIFFRACTION (2.25 Å)
Cite:	Impact of Homologous Resistance Mutations from Pathogenic Yeast on Saccharomyces cerevisiae Lanosterol 14 alpha-Demethylase. Antimicrob.Agents Chemother., 62, 2018

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