6I1R
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![BU of 6i1r by Molmil](/molmil-images/mine/6i1r) | Crystal structure of CMP bound CST in an outward facing conformation | Descriptor: | CMP-sialic acid transporter 1, CYTIDINE-5'-MONOPHOSPHATE | Authors: | Nji, E, Gulati, A, Qureshi, A.A, Drew, D. | Deposit date: | 2018-10-30 | Release date: | 2019-06-05 | Last modified: | 2024-01-24 | Method: | X-RAY DIFFRACTION (2.8 Å) | Cite: | Structural basis for the delivery of activated sialic acid into Golgi for sialyation. Nat.Struct.Mol.Biol., 26, 2019
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6I1Z
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6SSR
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![BU of 6ssr by Molmil](/molmil-images/mine/6ssr) | |
6SSS
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![BU of 6sss by Molmil](/molmil-images/mine/6sss) | Crystal structure of Human Microsomal Glutathione S-Transferase 2 | Descriptor: | 1-(8Z-hexadecenoyl)-sn-glycerol, GLYCEROL, Microsomal glutathione S-transferase 2, ... | Authors: | Thulasingam, M, Nji, E, Haeggstrom, J.Z. | Deposit date: | 2019-09-09 | Release date: | 2021-02-03 | Last modified: | 2024-01-24 | Method: | X-RAY DIFFRACTION (2.498 Å) | Cite: | Crystal structures of human MGST2 reveal synchronized conformational changes regulating catalysis. Nat Commun, 12, 2021
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7OIX
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6SSW
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6SSU
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![BU of 6ssu by Molmil](/molmil-images/mine/6ssu) | |
5BZ2
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5BZ3
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![BU of 5bz3 by Molmil](/molmil-images/mine/5bz3) | CRYSTAL STRUCTURE OF SODIUM PROTON ANTIPORTER NAPA IN OUTWARD-FACING CONFORMATION. | Descriptor: | (2R)-2,3-DIHYDROXYPROPYL (7Z)-TETRADEC-7-ENOATE, Na(+)/H(+) antiporter | Authors: | Coincon, M, Uzdavinys, P, Emmanuel, N, Cameron, A, Drew, D. | Deposit date: | 2015-06-11 | Release date: | 2016-01-20 | Last modified: | 2024-05-08 | Method: | X-RAY DIFFRACTION (2.3 Å) | Cite: | Crystal structures reveal the molecular basis of ion translocation in sodium/proton antiporters. Nat.Struct.Mol.Biol., 23, 2016
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6RW3
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![BU of 6rw3 by Molmil](/molmil-images/mine/6rw3) | The molecular basis for sugar import in malaria parasites. | Descriptor: | Hexose transporter 1, alpha-D-glucopyranose, beta-D-glucopyranose | Authors: | Qureshi, A, Matsuoka, R, Brock, J, Drew, D. | Deposit date: | 2019-06-03 | Release date: | 2020-01-29 | Last modified: | 2024-01-24 | Method: | X-RAY DIFFRACTION (3.65 Å) | Cite: | The molecular basis for sugar import in malaria parasites. Nature, 578, 2020
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7WXX
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![BU of 7wxx by Molmil](/molmil-images/mine/7wxx) | Crystal structure of human MMP-7 in complex with inhibitor | Descriptor: | CALCIUM ION, Matrilysin, Peptide Inhibitor, ... | Authors: | Kamitani, M, Oka, Y, Tabuse, H. | Deposit date: | 2022-02-15 | Release date: | 2022-10-05 | Last modified: | 2023-11-29 | Method: | X-RAY DIFFRACTION (1.5 Å) | Cite: | Discovery of Highly Potent and Selective Matrix Metalloproteinase-7 Inhibitors by Hybridizing the S1' Subsite Binder with Short Peptides. J.Med.Chem., 65, 2022
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8JUD
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![BU of 8jud by Molmil](/molmil-images/mine/8jud) | Crystal structure of human MMP-7 in complex with inhibitor | Descriptor: | CALCIUM ION, Matrilysin, Peptide Inhibitor, ... | Authors: | Kamitani, M, Abe-Sato, K, Oka, Y. | Deposit date: | 2023-06-26 | Release date: | 2023-11-01 | Last modified: | 2023-11-22 | Method: | X-RAY DIFFRACTION (1.5 Å) | Cite: | Structure-Based Optimization and Biological Evaluation of Potent and Selective MMP-7 Inhibitors for Kidney Fibrosis. J.Med.Chem., 66, 2023
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8JUF
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![BU of 8juf by Molmil](/molmil-images/mine/8juf) | Crystal structure of human MMP-7 in complex with inhibitor | Descriptor: | CALCIUM ION, Matrilysin, Peptide Inhibitor, ... | Authors: | Kamitani, M, Abe-Sato, K, Oka, Y. | Deposit date: | 2023-06-26 | Release date: | 2023-11-01 | Last modified: | 2023-11-22 | Method: | X-RAY DIFFRACTION (1.39 Å) | Cite: | Structure-Based Optimization and Biological Evaluation of Potent and Selective MMP-7 Inhibitors for Kidney Fibrosis. J.Med.Chem., 66, 2023
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8JUG
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![BU of 8jug by Molmil](/molmil-images/mine/8jug) | Crystal structure of human MMP-7 in complex with inhibitor | Descriptor: | CALCIUM ION, Matrilysin, Peptide Inhibitor, ... | Authors: | Kamitani, M, Abe-Sato, K, Oka, Y. | Deposit date: | 2023-06-26 | Release date: | 2023-11-01 | Last modified: | 2023-11-22 | Method: | X-RAY DIFFRACTION (1.3 Å) | Cite: | Structure-Based Optimization and Biological Evaluation of Potent and Selective MMP-7 Inhibitors for Kidney Fibrosis. J.Med.Chem., 66, 2023
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8K4Z
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