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1AUL
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BU of 1aul by Molmil
SOLUTION STRUCTURE OF A HIGHLY STABLE DNA DUPLEX CONJUGATED TO A MINOR GROOVE BINDER, NMR, MINIMIZED AVERAGE STRUCTURE
分子名称: DNA (5'-D(*CP*AP*GP*AP*TP*AP*AP*TP*CP*A)-3'), DNA (5'-D(P*THXP*GP*AP*TP*TP*AP*TP*CP*TP*G)-3')
著者Kumar, S, Reed, M.W, Gamper Junior, H.B, Gorn, V.V, Lukhtanov, E.A, Foti, M, West, J, Meyer Junior, R.B, Schweitzer, B.I.
登録日1997-08-29
公開日1997-12-24
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献Solution structure of a highly stable DNA duplex conjugated to a minor groove binder.
Nucleic Acids Res., 26, 1998
1JBL
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BU of 1jbl by Molmil
Solution structure of SFTI-1, A cyclic trypsin inhibitor from sunflower seeds
分子名称: CYCLIC TRYPSIN INHIBITOR
著者Korsinczky, M.L.J, Schirra, H.J, Rosengren, K.J, West, J, Condie, B.A, Otvos, L, Anderson, M.A, Craik, D.J.
登録日2001-06-05
公開日2001-08-22
最終更新日2015-04-15
実験手法SOLUTION NMR
主引用文献Solution structures by 1H NMR of the novel cyclic trypsin inhibitor SFTI-1 from sunflower seeds and an acyclic permutant.
J.Mol.Biol., 311, 2001
1JBN
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BU of 1jbn by Molmil
Solution structure of an acyclic permutant of SFTI-1, A trypsin inhibitor from sunflower seeds
分子名称: CYCLIC TRYPSIN INHIBITOR
著者Korsinczky, M.L.J, Schirra, H.J, Rosengren, K.J, West, J, Condie, B.A, Otvos, L, Anderson, M.A, Craik, D.J.
登録日2001-06-06
公開日2001-08-22
最終更新日2016-12-28
実験手法SOLUTION NMR
主引用文献Solution structures by 1H NMR of the novel cyclic trypsin inhibitor SFTI-1 from sunflower seeds and an acyclic permutant.
J.Mol.Biol., 311, 2001
1MI2
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BU of 1mi2 by Molmil
SOLUTION STRUCTURE OF MURINE MACROPHAGE INFLAMMATORY PROTEIN-2, NMR, 20 STRUCTURES
分子名称: MACROPHAGE INFLAMMATORY PROTEIN-2
著者Shao, W, Jerva, L.F, West, J, Lolis, E, Schweitzer, B.I.
登録日1997-10-24
公開日1998-04-29
最終更新日2022-02-23
実験手法SOLUTION NMR
主引用文献Solution structure of murine macrophage inflammatory protein-2.
Biochemistry, 37, 1998
2X4Z
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BU of 2x4z by Molmil
Crystal Structure of the Human p21-Activated Kinase 4 in Complex with PF-03758309
分子名称: GLYCEROL, PF-3758309, SERINE/THREONINE-PROTEIN KINASE PAK 4
著者Knighton, D.R, Deng, Y, Murray, B, Guo, C, Piraino, J, Westwick, J, Zhang, C, Lamerdin, J, Dagostino, E, Loi, C.-M, Zager, M, Kraynov, E, Christensen, J, Martinez, R, Kephart, S, Marakovits, J, Karlicek, S, Bergqvist, S, Smeal, T.
登録日2010-02-03
公開日2010-05-19
最終更新日2019-01-23
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Small-Molecule P21-Activated Kinase Inhibitor Pf- 3758309 is a Potent Inhibitor of Oncogenic Signaling and Tumor Growth.
Proc.Natl.Acad.Sci.USA, 107, 2010
1KCM
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BU of 1kcm by Molmil
Crystal Structure of Mouse PITP Alpha Void of Bound Phospholipid at 2.0 Angstroms Resolution
分子名称: Phosphatidylinositol Transfer Protein alpha
著者Schouten, A, Agianian, B, Westerman, J, Kroon, J, Wirtz, K.W.A, Gros, P.
登録日2001-11-09
公開日2002-05-08
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structure of apo-phosphatidylinositol transfer protein alpha provides insight into membrane association.
EMBO J., 21, 2002
3S2U
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BU of 3s2u by Molmil
Crystal structure of the Pseudomonas aeruginosa MurG:UDP-GlcNAc substrate complex
分子名称: UDP-N-acetylglucosamine--N-acetylmuramyl-(pentapeptide) pyrophosphoryl-undecaprenol N-acetylglucosamine transferase, URIDINE-DIPHOSPHATE-N-ACETYLGLUCOSAMINE
著者Brown, K, Vial, S.C.M, Dedi, N, Westcott, J, Scally, S, Bugg, T.D.H, Charlton, P.A, Cheetham, G.M.T.
登録日2011-05-17
公開日2012-09-26
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.23 Å)
主引用文献Crystal Structure of the Pseudomonas aeruginosa MurG: UDP-GlcNAc Substrate Complex.
Protein Pept.Lett., 20, 2013
8S2X
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BU of 8s2x by Molmil
SSX structure of Arabidopsis thaliana Pdx1.3 grown in microfluidic droplets
分子名称: CITRIC ACID, PHOSPHATE ION, Pyridoxal 5'-phosphate synthase subunit PDX1.3
著者Stubbs, J, Tews, I, Maly, M.
登録日2024-02-19
公開日2024-02-28
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Droplet microfluidics for time-resolved serial crystallography.
Iucrj, 11, 2024
8S2V
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BU of 8s2v by Molmil
SSX structure of Lysozyme grown in microfluidic droplets
分子名称: CHLORIDE ION, Lysozyme C
著者Stubbs, J, Tews, I, Maly, M.
登録日2024-02-19
公開日2024-02-28
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Droplet microfluidics for time-resolved serial crystallography.
Iucrj, 11, 2024
8S2W
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BU of 8s2w by Molmil
SSX structure of Arabidopsis thaliana Pdx1.3 grown in seeded batch conditions
分子名称: PHOSPHATE ION, Pyridoxal 5'-phosphate synthase subunit PDX1.3
著者Stubbs, J, Tews, I, Maly, M.
登録日2024-02-19
公開日2024-02-28
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Droplet microfluidics for time-resolved serial crystallography.
Iucrj, 11, 2024
8S2U
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BU of 8s2u by Molmil
SSX structure of Lysozyme grown in batch conditions
分子名称: CHLORIDE ION, Lysozyme C
著者Stubbs, J, Tews, I, Maly, M.
登録日2024-02-19
公開日2024-02-28
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Droplet microfluidics for time-resolved serial crystallography.
Iucrj, 11, 2024
6EUS
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BU of 6eus by Molmil
Crystal structure of the outer membrane channel DcaP of Acinetobacter baumannii
分子名称: DcaP-like protein
著者Zahn, M, van den Berg, B.
登録日2017-10-31
公開日2018-11-14
最終更新日2019-06-19
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献A Multidisciplinary Approach toward Identification of Antibiotic Scaffolds for Acinetobacter baumannii.
Structure, 27, 2019
5OW6
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BU of 5ow6 by Molmil
CryoEM structure of recombinant CMV particles with Tetanus-epitope
分子名称: Capsid protein, VP2, VP3, ...
著者Kotecha, A, Stuart, D.I, Backmann, M.
登録日2017-08-30
公開日2017-09-13
最終更新日2024-05-15
実験手法ELECTRON MICROSCOPY (4.2 Å)
主引用文献Incorporation of tetanus-epitope into virus-like particles achieves vaccine responses even in older recipients in models of psoriasis, Alzheimer's and cat allergy.
NPJ Vaccines, 2, 2017
5SZD
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BU of 5szd by Molmil
Crystal structure of Aquifex aeolicus Hfq at 1.5A
分子名称: (4R)-2-METHYLPENTANE-2,4-DIOL, (4S)-2-METHYL-2,4-PENTANEDIOL, CHLORIDE ION, ...
著者Stanek, K, Patterson, J, Randolph, P.S, Mura, C.
登録日2016-08-13
公開日2017-04-19
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (1.494 Å)
主引用文献Crystal structure and RNA-binding properties of an Hfq homolog from the deep-branching Aquificae: conservation of the lateral RNA-binding mode.
Acta Crystallogr D Struct Biol, 73, 2017
5SZE
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BU of 5sze by Molmil
Crystal structure of Aquifex aeolicus Hfq-RNA complex at 1.5A
分子名称: (4R)-2-METHYLPENTANE-2,4-DIOL, DI(HYDROXYETHYL)ETHER, RNA (5'-R(P*UP*UP*U)-3'), ...
著者Stanek, K, Patterson, J, Randolph, P.S, Mura, C.
登録日2016-08-13
公開日2017-04-12
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Crystal structure and RNA-binding properties of an Hfq homolog from the deep-branching Aquificae: conservation of the lateral RNA-binding mode.
Acta Crystallogr D Struct Biol, 73, 2017
1HHV
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BU of 1hhv by Molmil
SOLUTION STRUCTURE OF VIRUS CHEMOKINE VMIP-II
分子名称: VIRUS CHEMOKINE VMIP-II
著者Shao, W, Fernandez, E, Navenot, J.M, Wilken, J, Thompson, D.A, Pepiper, S, Schweitzer, B.I, Lolis, E.
登録日1998-12-06
公開日2003-09-16
最終更新日2023-12-27
実験手法SOLUTION NMR
主引用文献CCR2 and CCR5 receptor-binding properties of herpesvirus-8 vMIP-II based on sequence analysis and its solution structure
Eur.J.Biochem., 268, 2001
5LBM
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BU of 5lbm by Molmil
The asymmetric tetrameric structure of the formaldehyde sensing transcriptional repressor FrmR from Escherichia coli
分子名称: FORMYL GROUP, Transcriptional repressor FrmR
著者Bisson, C, Baker, P.J, Green, J, Chivers, P.T.
登録日2016-06-16
公開日2016-12-21
最終更新日2017-08-30
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献The mechanism of a formaldehyde-sensing transcriptional regulator.
Sci Rep, 6, 2016
4ZFO
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BU of 4zfo by Molmil
J22.9-xi: chimeric mouse/human antibody against human BCMA (CD269)
分子名称: 2-[BIS-(2-HYDROXY-ETHYL)-AMINO]-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, COPPER (II) ION, J22.9-xi Fab, ...
著者Marino, S.F, Daumke, O, Olal, D.
登録日2015-04-21
公開日2015-05-20
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.895 Å)
主引用文献Potent anti-tumor response by targeting B cell maturation antigen (BCMA) in a mouse model of multiple myeloma.
Mol Oncol, 9, 2015
4ZPE
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BU of 4zpe by Molmil
BACE1 in complex with 4-(cyclohexylamino)-1-(3-fluorophenyl)-8-(3-isopropoxybenzyl)-1,3,8-triazaspiro[4.5]dec-3-en-2-one
分子名称: 4-(cyclohexylamino)-1-(3-fluorophenyl)-8-[3-(propan-2-yloxy)benzyl]-1,3,8-triazaspiro[4.5]dec-3-en-2-one, Beta-secretase 1
著者Orth, P.
登録日2015-05-07
公開日2015-08-05
最終更新日2015-10-28
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Methyl-substitution of an iminohydantoin spiropiperidine beta-secretase (BACE-1) inhibitor has a profound effect on its potency.
Bioorg.Med.Chem.Lett., 25, 2015
4ZPF
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BU of 4zpf by Molmil
BACE1 in complex with 8-(3-((1-aminopropan-2-yl)oxy)benzyl)-4-(cyclohexylamino)-1-(3-fluorophenyl)-1,3,8-triazaspiro[4.5]dec-3-en-2-one
分子名称: 8-(3-{[(2S)-1-aminopropan-2-yl]oxy}benzyl)-4-(cyclohexylamino)-1-(3-fluorophenyl)-1,3,8-triazaspiro[4.5]dec-3-en-2-one, Beta-secretase 1
著者Orth, P.
登録日2015-05-07
公開日2015-08-05
最終更新日2015-10-28
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Methyl-substitution of an iminohydantoin spiropiperidine beta-secretase (BACE-1) inhibitor has a profound effect on its potency.
Bioorg.Med.Chem.Lett., 25, 2015
4ZPG
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BU of 4zpg by Molmil
BACE1 in complex with 8-benzyl-4-(cyclohexylamino)-1-(3-fluorophenyl)-7-methyl-1,3,8-triazaspiro[4.5]dec-3-en-2-one
分子名称: (5R,7S)-8-benzyl-4-(cyclohexylamino)-1-(3-fluorophenyl)-7-methyl-1,3,8-triazaspiro[4.5]dec-3-en-2-one, Beta-secretase 1
著者Orth, P.
登録日2015-05-07
公開日2015-08-05
最終更新日2015-10-28
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Methyl-substitution of an iminohydantoin spiropiperidine beta-secretase (BACE-1) inhibitor has a profound effect on its potency.
Bioorg.Med.Chem.Lett., 25, 2015
7MKR
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BU of 7mkr by Molmil
Crystal structure of the GH12 domain from Acidothermus cellulolyticus GuxA
分子名称: 1,2-ETHANEDIOL, ACETATE ION, CHLORIDE ION, ...
著者Lunin, V.V.
登録日2021-04-26
公開日2022-05-04
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Characterization of the Biomass Degrading Enzyme GuxA from Acidothermus cellulolyticus.
Int J Mol Sci, 23, 2022
7MKS
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Crystal structure of the GH12 domain from Acidothermus cellulolyticus GuxA bound to cellobiose
分子名称: ACETATE ION, CHLORIDE ION, GLYCEROL, ...
著者Lunin, V.V.
登録日2021-04-26
公開日2022-05-04
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Characterization of the Biomass Degrading Enzyme GuxA from Acidothermus cellulolyticus.
Int J Mol Sci, 23, 2022
5UFL
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BU of 5ufl by Molmil
Crystal structure of a CIP2A core domain
分子名称: Protein CIP2A, ZINC ION
著者Wang, Z, Wang, J, Rao, Z, Xu, W.
登録日2017-01-04
公開日2017-02-15
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Oncoprotein CIP2A is stabilized via interaction with tumor suppressor PP2A/B56.
EMBO Rep., 18, 2017
6F0A
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BU of 6f0a by Molmil
Crystal structure of human indoleamine 2,3-dioxygenase bound to a triazole inhibitor and alanine molecule.
分子名称: ALANINE, Indoleamine 2,3-dioxygenase 1, PROTOPORPHYRIN IX CONTAINING FE, ...
著者Swan, M.K, Latchem, M.
登録日2017-11-17
公開日2017-12-27
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.26 Å)
主引用文献New 4-Amino-1,2,3-Triazole Inhibitors of Indoleamine 2,3-Dioxygenase Form a Long-Lived Complex with the Enzyme and Display Exquisite Cellular Potency.
Chembiochem, 19, 2018

 

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