3ITN
| Crystal structure of Pseudo-activated Procaspase-3 | 分子名称: | ACETYL-ASP-GLU-VAL-ASP-CHLOROMETHYL KETONE inhibitor, Caspase-3 | 著者 | Walters, J, Pop, C, Scott, F.L, Drag, M, Swartz, P.D, Mattos, C, Salvesen, G.S, Clark, A.C. | 登録日 | 2009-08-28 | 公開日 | 2010-03-02 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.63 Å) | 主引用文献 | A constitutively active and uninhibitable caspase-3 zymogen efficiently induces apoptosis. Biochem.J., 424, 2009
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3PCX
| Caspase-3 E246A, K242A Double Mutant | 分子名称: | Caspase-3, Inhibitor Ac-DEVD-CMK | 著者 | Walters, J, Swartz, P, Mattos, C, Clark, A.C. | 登録日 | 2010-10-22 | 公開日 | 2011-02-23 | 最終更新日 | 2012-12-12 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Thermodynamic, enzymatic and structural effects of removing a salt bridge at the base of loop 4 in (pro)caspase-3. Arch.Biochem.Biophys., 508, 2011
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3PD1
| Caspase-3 K242A | 分子名称: | Caspase-3, Inhibitor Ac-DEVD-CMK | 著者 | Walters, J, Swartz, P, Mattos, C, Clark, A.C. | 登録日 | 2010-10-22 | 公開日 | 2011-02-23 | 最終更新日 | 2013-02-27 | 実験手法 | X-RAY DIFFRACTION (1.62 Å) | 主引用文献 | Thermodynamic, enzymatic and structural effects of removing a salt bridge at the base of loop 4 in (pro)caspase-3. Arch.Biochem.Biophys., 508, 2011
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3PD0
| Caspase-3 E246A | 分子名称: | CHLORIDE ION, Caspase-3, INHIBITOR AC-DEVD-CMK | 著者 | Walters, J, Swartz, P, Mattos, C, Clark, A.C. | 登録日 | 2010-10-22 | 公開日 | 2011-02-16 | 最終更新日 | 2012-12-12 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Thermodynamic, enzymatic and structural effects of removing a salt bridge at the base of loop 4 in (pro)caspase-3. Arch.Biochem.Biophys., 508, 2011
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4EHA
| Allosteric Modulation of Caspase-3 through Mutagenesis | 分子名称: | ACE-ASP-GLU-VAL-ASP-CHLOROMETHYLKETONE INHIBITOR, Caspase-3 | 著者 | Walters, J, Schipper, J.L, Swartz, P.D, Mattos, C, Clark, A.C. | 登録日 | 2012-04-02 | 公開日 | 2012-06-06 | 最終更新日 | 2017-11-15 | 実験手法 | X-RAY DIFFRACTION (1.696 Å) | 主引用文献 | Allosteric modulation of caspase 3 through mutagenesis. Biosci.Rep., 32, 2012
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4EHH
| Allosteric Modulation of Caspase-3 through Mutagenesis | 分子名称: | ACE-ASP-GLU-VAL-ASP-CHLOROMETHYLKETONE INHIBITOR, Caspase-3 | 著者 | Walters, J, Schipper, J.L, Swartz, P.D, Mattos, C, Clark, A.C. | 登録日 | 2012-04-02 | 公開日 | 2012-06-06 | 最終更新日 | 2017-11-15 | 実験手法 | X-RAY DIFFRACTION (1.78 Å) | 主引用文献 | Allosteric modulation of caspase 3 through mutagenesis. Biosci.Rep., 32, 2012
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4EHL
| Allosteric Modulation of Caspase-3 through Mutagenesis | 分子名称: | ACE-ASP-GLU-VAL-ASP-CHLOROMETHYLKETONE INHIBITOR, Caspase-3 | 著者 | Walters, J, Schipper, J.L, Swartz, P.D, Mattos, C, Clark, A.C. | 登録日 | 2012-04-02 | 公開日 | 2012-06-06 | 最終更新日 | 2017-11-15 | 実験手法 | X-RAY DIFFRACTION (1.799 Å) | 主引用文献 | Allosteric modulation of caspase 3 through mutagenesis. Biosci.Rep., 32, 2012
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4EHD
| Allosteric Modulation of Caspase-3 through Mutagenesis | 分子名称: | ACE-ASP-GLU-VAL-ASP-CHLOROMETHYLKETONE INHIBITOR, Caspase-3 | 著者 | Walters, J, Schipper, J.L, Swartz, P, Mattos, C, Clark, A.C. | 登録日 | 2012-04-02 | 公開日 | 2012-06-06 | 最終更新日 | 2017-11-15 | 実験手法 | X-RAY DIFFRACTION (1.581 Å) | 主引用文献 | Allosteric modulation of caspase 3 through mutagenesis. Biosci.Rep., 32, 2012
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4EHN
| Allosteric Modulation of Caspase-3 through Mutagenesis | 分子名称: | ACE-ASP-GLU-VAL-ASP-CHLOROMETHYLKETONE INHIBITOR, Caspase-3 | 著者 | Walters, J, Schipper, J.L, Swartz, P.D, Mattos, C, Clark, A.C. | 登録日 | 2012-04-02 | 公開日 | 2012-06-06 | 最終更新日 | 2017-11-15 | 実験手法 | X-RAY DIFFRACTION (1.69 Å) | 主引用文献 | Allosteric modulation of caspase 3 through mutagenesis. Biosci.Rep., 32, 2012
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4EHF
| Allosteric Modulation of Caspase-3 through Mutagenesis | 分子名称: | ACE-ASP-GLU-VAL-ASP-CHLOROMETHYLKETONE INHIBITOR, Caspase-3 | 著者 | Walters, J, Schipper, J.L, Swartz, P.D, Mattos, C, Clark, A.C. | 登録日 | 2012-04-02 | 公開日 | 2012-06-06 | 最終更新日 | 2017-11-15 | 実験手法 | X-RAY DIFFRACTION (1.655 Å) | 主引用文献 | Allosteric modulation of caspase 3 through mutagenesis. Biosci.Rep., 32, 2012
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4EHK
| Allosteric Modulation of Caspase-3 through Mutagenesis | 分子名称: | ACE-ASP-GLU-VAL-ASP-CHLOROMETHYLKETONE INHIBITOR, Caspase-3 | 著者 | Walters, J, Schipper, J.L, Swartz, P.D, Mattos, C, Clark, A.C. | 登録日 | 2012-04-02 | 公開日 | 2012-06-06 | 最終更新日 | 2017-11-15 | 実験手法 | X-RAY DIFFRACTION (1.668 Å) | 主引用文献 | Allosteric modulation of caspase 3 through mutagenesis. Biosci.Rep., 32, 2012
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3PTN
| ON THE DISORDERED ACTIVATION DOMAIN IN TRYPSINOGEN. CHEMICAL LABELLING AND LOW-TEMPERATURE CRYSTALLOGRAPHY | 分子名称: | CALCIUM ION, TRYPSIN | 著者 | Walter, J, Steigemann, W, Singh, T.P, Bartunik, H, Bode, W, Huber, R. | 登録日 | 1981-10-26 | 公開日 | 1982-03-04 | 最終更新日 | 2024-06-05 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | On the Disordered Activation Domain in Trypsinogen. Chemical Labelling and Low-Temperature Crystallography Acta Crystallogr.,Sect.B, 38, 1982
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2TGT
| ON THE DISORDERED ACTIVATION DOMAIN IN TRYPSINOGEN. CHEMICAL LABELLING AND LOW-TEMPERATURE CRYSTALLOGRAPHY | 分子名称: | CALCIUM ION, METHANOL, TRYPSINOGEN | 著者 | Walter, J, Steigemann, W, Singh, T.P, Bartunik, H, Bode, W, Huber, R. | 登録日 | 1981-10-26 | 公開日 | 1982-03-04 | 最終更新日 | 2024-06-05 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | On the Disordered Activation Domain in Trypsinogen. Chemical Labelling and Low-Temperature Crystallography Acta Crystallogr.,Sect.B, 38, 1982
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2TGA
| ON THE DISORDERED ACTIVATION DOMAIN IN TRYPSINOGEN. CHEMICAL LABELLING AND LOW-TEMPERATURE CRYSTALLOGRAPHY | 分子名称: | CALCIUM ION, TRYPSINOGEN | 著者 | Walter, J, Steigemann, W, Singh, T.P, Bartunik, H, Bode, W, Huber, R. | 登録日 | 1981-10-26 | 公開日 | 1982-03-04 | 最終更新日 | 2024-06-05 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | On the Disordered Activation Domain in Trypsinogen. Chemical Labelling and Low-Temperature Crystallography Acta Crystallogr.,Sect.B, 38, 1982
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1TGC
| ON THE DISORDERED ACTIVATION DOMAIN IN TRYPSINOGEN. CHEMICAL LABELLING AND LOW-TEMPERATURE CRYSTALLOGRAPHY | 分子名称: | CALCIUM ION, TRYPSINOGEN | 著者 | Walter, J, Steigemann, W, Singh, T.P, Bartunik, H, Bode, W, Huber, R. | 登録日 | 1981-10-26 | 公開日 | 1982-03-04 | 最終更新日 | 2024-10-09 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | On the Disordered Activation Domain in Trypsinogen. Chemical Labelling and Low-Temperature Crystallography Acta Crystallogr.,Sect.B, 38, 1982
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1TGT
| ON THE DISORDERED ACTIVATION DOMAIN IN TRYPSINOGEN. CHEMICAL LABELLING AND LOW-TEMPERATURE CRYSTALLOGRAPHY | 分子名称: | CALCIUM ION, METHANOL, TRYPSINOGEN | 著者 | Walter, J, Steigemann, W, Singh, T.P, Bartunik, H, Bode, W, Huber, R. | 登録日 | 1981-10-26 | 公開日 | 1982-03-04 | 最終更新日 | 2024-06-05 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | On the Disordered Activation Domain in Trypsinogen. Chemical Labelling and Low-Temperature Crystallography Acta Crystallogr.,Sect.B, 38, 1982
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2TPI
| ON THE DISORDERED ACTIVATION DOMAIN IN TRYPSINOGEN. CHEMICAL LABELLING AND LOW-TEMPERATURE CRYSTALLOGRAPHY | 分子名称: | ISOLEUCINE, MERCURY (II) ION, TRYPSIN INHIBITOR, ... | 著者 | Walter, J, Steigemann, W, Singh, T.P, Bartunik, H, Bode, W, Huber, R. | 登録日 | 1981-10-26 | 公開日 | 1982-03-04 | 最終更新日 | 2024-06-05 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | On the Disordered Activation Domain in Trypsinogen. Chemical Labelling and Low-Temperature Crystallography Acta Crystallogr.,Sect.B, 38, 1982
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2PTN
| ON THE DISORDERED ACTIVATION DOMAIN IN TRYPSINOGEN. CHEMICAL LABELLING AND LOW-TEMPERATURE CRYSTALLOGRAPHY | 分子名称: | CALCIUM ION, TRYPSIN | 著者 | Walter, J, Steigemann, W, Singh, T.P, Bartunik, H, Bode, W, Huber, R. | 登録日 | 1981-10-26 | 公開日 | 1982-03-04 | 最終更新日 | 2024-10-09 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | On the Disordered Activation Domain in Trypsinogen. Chemical Labelling and Low-Temperature Crystallography Acta Crystallogr.,Sect.B, 38, 1982
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1TPP
| THE GEOMETRY OF THE REACTIVE SITE AND OF THE PEPTIDE GROUPS IN TRYPSIN, TRYPSINOGEN AND ITS COMPLEXES WITH INHIBITORS | 分子名称: | (2S)-3-(4-carbamimidoylphenyl)-2-hydroxypropanoic acid, BETA-TRYPSIN, CALCIUM ION, ... | 著者 | Walter, J, Bode, W, Huber, R. | 登録日 | 1982-09-27 | 公開日 | 1983-01-18 | 最終更新日 | 2024-06-05 | 実験手法 | X-RAY DIFFRACTION (1.4 Å) | 主引用文献 | The Geometry of the Reactive Site and of the Peptide Groups in Trypsin, Trypsinogen and its Complexes with Inhibitors Acta Crystallogr.,Sect.B, 39, 1983
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4TPI
| THE REFINED 2.2-ANGSTROMS (0.22-NM) X-RAY CRYSTAL STRUCTURE OF THE TERNARY COMPLEX FORMED BY BOVINE TRYPSINOGEN, VALINE-VALINE AND THE ARG15 ANALOGUE OF BOVINE PANCREATIC TRYPSIN INHIBITOR | 分子名称: | BOVINE PANCREATIC TRYPSIN INHIBITOR, CALCIUM ION, SULFATE ION, ... | 著者 | Bode, W, Walter, J. | 登録日 | 1985-06-11 | 公開日 | 1985-11-08 | 最終更新日 | 2024-06-05 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | The refined 2.2-A (0.22-nm) X-ray crystal structure of the ternary complex formed by bovine trypsinogen, valine-valine and the Arg15 analogue of bovine pancreatic trypsin inhibitor Eur.J.Biochem., 144, 1984
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3PTB
| THE GEOMETRY OF THE REACTIVE SITE AND OF THE PEPTIDE GROUPS IN TRYPSIN, TRYPSINOGEN AND ITS COMPLEXES WITH INHIBITORS | 分子名称: | BENZAMIDINE, BETA-TRYPSIN, CALCIUM ION | 著者 | Bode, W, Schwager, P, Walter, J. | 登録日 | 1982-09-27 | 公開日 | 1983-01-18 | 最終更新日 | 2024-06-05 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | The Geometry of the Reactive Site and of the Peptide Groups in Trypsin, Trypsinogen and its Complexes with Inhibitors Acta Crystallogr.,Sect.B, 39, 1983
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1TPO
| THE GEOMETRY OF THE REACTIVE SITE AND OF THE PEPTIDE GROUPS IN TRYPSIN, TRYPSINOGEN AND ITS COMPLEXES WITH INHIBITORS | 分子名称: | BETA-TRYPSIN, CALCIUM ION | 著者 | Bode, W, Walter, J, Huber, R. | 登録日 | 1982-09-27 | 公開日 | 1983-01-18 | 最終更新日 | 2024-06-05 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | The Geometry of the Reactive Site and of the Peptide Groups in Trypsin, Trypsinogen and its Complexes with Inhibitors Acta Crystallogr.,Sect.B, 39, 1983
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5WMG
| N-terminal bromodomain of BRD4 in complex with OTX-015 | 分子名称: | 1,2-ETHANEDIOL, 4-{6-(3,5-dimethyl-1,2-oxazol-4-yl)-1-[(1S)-1-(pyridin-2-yl)ethyl]-1H-pyrrolo[3,2-b]pyridin-3-yl}benzoic acid, Bromodomain-containing protein 4 | 著者 | Zhang, Y. | 登録日 | 2017-07-28 | 公開日 | 2018-08-01 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (1.19 Å) | 主引用文献 | BRD4 Profiling Identifies Critical Chronic Lymphocytic Leukemia Oncogenic Circuits and Reveals Sensitivity to PLX51107, a Novel Structurally Distinct BET Inhibitor. Cancer Discov, 8, 2018
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5WMD
| N-terminal bromodomain of BRD4 in complex with OTX-015 | 分子名称: | 2-[(6S)-4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl]-N-(4-hydroxyphenyl)acetamide, Bromodomain-containing protein 4 | 著者 | Zhang, Y. | 登録日 | 2017-07-28 | 公開日 | 2018-08-01 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (1.27 Å) | 主引用文献 | BRD4 Profiling Identifies Critical Chronic Lymphocytic Leukemia Oncogenic Circuits and Reveals Sensitivity to PLX51107, a Novel Structurally Distinct BET Inhibitor. Cancer Discov, 8, 2018
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5WMA
| N-terminal bromodomain of BRD4 in complex with PLX5981 | 分子名称: | 1,2-ETHANEDIOL, 5-(3,5-dimethyl-1,2-oxazol-4-yl)-1H-pyrrolo[2,3-b]pyridine, Bromodomain-containing protein 4 | 著者 | Zhang, Y. | 登録日 | 2017-07-28 | 公開日 | 2018-08-01 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (1.401 Å) | 主引用文献 | BRD4 Profiling Identifies Critical Chronic Lymphocytic Leukemia Oncogenic Circuits and Reveals Sensitivity to PLX51107, a Novel Structurally Distinct BET Inhibitor. Cancer Discov, 8, 2018
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