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5PTP
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BU of 5ptp by Molmil
STRUCTURE OF HYDROLASE (SERINE PROTEINASE)
分子名称: BETA TRYPSIN, CALCIUM ION
著者Stroud, R.M, Finer-Moore, J.
登録日1997-03-31
公開日1997-07-07
最終更新日2017-11-29
実験手法X-RAY DIFFRACTION (1.34 Å)
主引用文献Solvent structure in crystals of trypsin determined by X-ray and neutron diffraction.
Proteins, 12, 1992
7SP5
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BU of 7sp5 by Molmil
Crystal Structure of a Eukaryotic Phosphate Transporter
分子名称: PHOSPHATE ION, Phosphate transporter, nonyl beta-D-glucopyranoside
著者Stroud, R.M, Pedersen, B.P, Kumar, H, Waight, A.B, Risenmay, A.J, Roe-Zurz, Z, Chau, B.H, Schlessinger, A, Bonomi, M, Harries, W, Sali, A, Johri, A.K, Finer-Moore, J.
登録日2021-11-02
公開日2021-11-17
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Crystal structure of a eukaryotic phosphate transporter.
Nature, 496, 2013
6NNR
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BU of 6nnr by Molmil
high-resolution structure of wild-type E. coli thymidylate synthase
分子名称: 10-PROPARGYL-5,8-DIDEAZAFOLIC ACID, 2'-deoxy-5'-uridylic acid, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, ...
著者Stroud, R.M, Finer-Moore, J.
登録日2019-01-15
公開日2019-01-30
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (1.05 Å)
主引用文献Mg2+ binds to the surface of thymidylate synthase and affects hydride transfer at the interior active site.
J. Am. Chem. Soc., 135, 2013
3E2J
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BU of 3e2j by Molmil
Crystal structure of bovine coupling factor B
分子名称: ATP synthase subunit s, mitochondrial, MAGNESIUM ION
著者Stroud, R.M, Lee, J.K, Belogrudov, G.I.
登録日2008-08-05
公開日2008-08-19
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Crystal structure of bovine mitochondrial factor B at 0.96-A resolution.
Proc.Natl.Acad.Sci.Usa, 105, 2008
3E3Z
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BU of 3e3z by Molmil
Crystal structure of bovine coupling Factor B bound with phenylarsine oxide
分子名称: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, ATP synthase subunit s, mitochondrial, ...
著者Stroud, R.M, Lee, J.K, Belogrudov, G.I.
登録日2008-08-08
公開日2008-08-26
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Crystal structure of bovine mitochondrial factor B at 0.96-A resolution.
Proc.Natl.Acad.Sci.Usa, 105, 2008
3E4G
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BU of 3e4g by Molmil
Crystal structure of bovine coupling Factor B, G28E mutant
分子名称: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, ATP synthase subunit s, mitochondrial, ...
著者Stroud, R.M, Lee, J.K, Belogrudov, G.I.
登録日2008-08-11
公開日2008-08-26
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (0.96 Å)
主引用文献Crystal structure of bovine mitochondrial factor B at 0.96-A resolution.
Proc.Natl.Acad.Sci.Usa, 105, 2008
1BTW
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BU of 1btw by Molmil
Episelection: novel KI ~nanomolar inhibitors of serine proteases selected by binding or chemistry on an enzyme surface
分子名称: BETA-TRYPSIN, CALCIUM ION, N-(tert-butoxycarbonyl)-L-alanyl-N-{(1S)-5-ammonio-1-[hydroxy(3-hydroxypropoxy)boranyl]pentyl}-L-valinamide
著者Stroud, R.M, Katz, B.A, Finer-Moore, J.
登録日1995-05-17
公開日1995-10-15
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Episelection: novel Ki approximately nanomolar inhibitors of serine proteases selected by binding or chemistry on an enzyme surface.
Biochemistry, 34, 1995
1BTY
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BU of 1bty by Molmil
Crystal structure of beta-trypsin in complex with benzamidine
分子名称: BENZAMIDINE, BETA-TRYPSIN, CALCIUM ION
著者Stroud, R.M, Katz, B.A, Finer-Moore, J.
登録日1995-05-17
公開日1995-10-15
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Episelection: novel Ki approximately nanomolar inhibitors of serine proteases selected by binding or chemistry on an enzyme surface.
Biochemistry, 34, 1995
1BTZ
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BU of 1btz by Molmil
Episelection: novel KI ~nanomolar inhibitors of serine proteases selected by binding or chemistry on an enzyme surface
分子名称: BETA-TRYPSIN, CALCIUM ION, N-(tert-butoxycarbonyl)-L-alanyl-N-{(1R)-5-ammonio-1-[hydroxy(methoxy)boranyl]pentyl}-L-valinamide
著者Stroud, R.M, Katz, B.A, Finer-Moore, J.
登録日1995-05-17
公開日1995-10-15
最終更新日2012-12-12
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Episelection: novel Ki approximately nanomolar inhibitors of serine proteases selected by binding or chemistry on an enzyme surface.
Biochemistry, 34, 1995
1BTX
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BU of 1btx by Molmil
Episelection: Novel Ki ~Nanomolar Inhibitors of Serine Proteases Selected by Binding or Chemistry on an Enzyme Surface
分子名称: BETA-TRYPSIN, CALCIUM ION, N-(tert-butoxycarbonyl)-L-alanyl-N-[(1S)-5-amino-1-(diethoxyboranyl)pentyl]-L-valinamide
著者Stroud, R.M, Katz, B.A, Finer-Moore, J.
登録日1995-05-17
公開日1995-10-15
最終更新日2012-12-12
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Episelection: novel Ki approximately nanomolar inhibitors of serine proteases selected by binding or chemistry on an enzyme surface.
Biochemistry, 34, 1995
2TRM
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BU of 2trm by Molmil
THE THREE-DIMENSIONAL STRUCTURE OF ASN102 MUTANT OF TRYPSIN. ROLE OF ASP102 IN SERINE PROTEASE CATALYSIS
分子名称: BENZAMIDINE, CALCIUM ION, TRYPSIN
著者Stroud, R.M, Finer-Moore, J.
登録日1988-04-25
公開日1988-07-16
最終更新日2017-11-29
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献The three-dimensional structure of Asn102 mutant of trypsin: role of Asp102 in serine protease catalysis.
Science, 237, 1987
1CN4
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BU of 1cn4 by Molmil
ERYTHROPOIETIN COMPLEXED WITH EXTRACELLULAR DOMAINS OF ERYTHROPOIETIN RECEPTOR
分子名称: PROTEIN (ERYTHROPOIETIN RECEPTOR), PROTEIN (ERYTHROPOIETIN)
著者Stroud, R.M, Reid, S.W.
登録日1999-05-25
公開日1999-08-11
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Efficiency of signalling through cytokine receptors depends critically on receptor orientation.
Nature, 395, 1998
1DPO
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BU of 1dpo by Molmil
STRUCTURE OF RAT TRYPSIN
分子名称: BENZAMIDINE, CALCIUM ION, SULFATE ION, ...
著者Stroud, R.M.
登録日1997-03-31
公開日1997-07-07
最終更新日2021-11-03
実験手法X-RAY DIFFRACTION (1.59 Å)
主引用文献1.59 A structure of trypsin at 120 K: comparison of low temperature and room temperature structures.
Proteins, 10, 1991
9ICD
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BU of 9icd by Molmil
CATALYTIC MECHANISM OF NADP+-DEPENDENT ISOCITRATE DEHYDROGENASE: IMPLICATIONS FROM THE STRUCTURES OF MAGNESIUM-ISOCITRATE AND NADP+ COMPLEXES
分子名称: ISOCITRATE DEHYDROGENASE, NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE
著者Hurley, J.H, Dean, A.M, Koshland Jr, D.E, Stroud, R.M.
登録日1991-07-29
公開日1991-10-15
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Catalytic mechanism of NADP(+)-dependent isocitrate dehydrogenase: implications from the structures of magnesium-isocitrate and NADP+ complexes.
Biochemistry, 30, 1991
8ICD
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BU of 8icd by Molmil
REGULATION OF AN ENZYME BY PHOSPHORYLATION AT THE ACTIVE SITE
分子名称: ISOCITRATE DEHYDROGENASE, ISOCITRIC ACID, MAGNESIUM ION
著者Hurley, J.H, Dean, A.M, Sohl, J.L, Koshlandjunior, D.E, Stroud, R.M.
登録日1990-05-30
公開日1991-10-15
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Regulation of an enzyme by phosphorylation at the active site.
Science, 249, 1990
3TMS
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BU of 3tms by Molmil
PLASTIC ADAPTATION TOWARD MUTATIONS IN PROTEINS: STRUCTURAL COMPARISON OF THYMIDYLATE SYNTHASES
分子名称: PHOSPHATE ION, THYMIDYLATE SYNTHASE
著者Perry, K.M, Stroud, R.M.
登録日1991-09-19
公開日1991-10-15
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Plastic adaptation toward mutations in proteins: structural comparison of thymidylate synthases.
Proteins, 8, 1990
7UK4
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BU of 7uk4 by Molmil
KS-AT di-domain of mycobacterial Pks13 with endogenous KS ligand bound
分子名称: Polyketide synthase PKS13, UNKNOWN LIGAND
著者Kim, S.K, Dickinson, M.S, Finer-Moore, J.S, Rosenberg, O.S, Stroud, R.M.
登録日2022-03-31
公開日2023-02-15
最終更新日2023-03-29
実験手法ELECTRON MICROSCOPY (1.94 Å)
主引用文献Structure and dynamics of the essential endogenous mycobacterial polyketide synthase Pks13.
Nat.Struct.Mol.Biol., 30, 2023
6ICD
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BU of 6icd by Molmil
REGULATION OF AN ENZYME BY PHOSPHORYLATION AT THE ACTIVE SITE
分子名称: ISOCITRATE DEHYDROGENASE
著者Hurley, J.H, Dean, A.M, Sohl, J.L, Koshlandjunior, D.E, Stroud, R.M.
登録日1990-05-30
公開日1991-10-15
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Regulation of an enzyme by phosphorylation at the active site.
Science, 249, 1990
8FVZ
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BU of 8fvz by Molmil
PiPT Y150A
分子名称: CITRATE ANION, PHOSPHATE ION, Phosphate transporter
著者Gupta, M, Finer-Moore, J, Stroud, R.M.
登録日2023-01-20
公開日2024-01-03
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献Roles of PiPT residues in phosphate binding and transport tested by mutagenesis
To be published
5ICD
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BU of 5icd by Molmil
REGULATION OF AN ENZYME BY PHOSPHORYLATION AT THE ACTIVE SITE
分子名称: ISOCITRATE DEHYDROGENASE, ISOCITRIC ACID, MAGNESIUM ION
著者Hurley, J.H, Dean, A.M, Sohl, J.L, Koshlandjunior, D.E, Stroud, R.M.
登録日1990-05-30
公開日1991-10-15
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Regulation of an enzyme by phosphorylation at the active site.
Science, 249, 1990
3KOU
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BU of 3kou by Molmil
Structural insights into the catalytic mechanism of CD38: Evidence for a conformationally flexible covalent enzyme-substrate complex.
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CD38 molecule, ...
著者Egea, P.F, Muller-Steffner, H, Stroud, R.M, Oppenheimer, N.J, Kellenberger, E, Schuber, F.
登録日2009-11-13
公開日2010-10-27
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.78 Å)
主引用文献Insights into the mechanism of bovine CD38/NAD+glycohydrolase from the X-ray structures of its Michaelis complex and covalently-trapped intermediates.
Plos One, 7, 2012
4FGT
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BU of 4fgt by Molmil
Allosteric peptidic inhibitor of human thymidylate synthase that stabilizes inactive conformation of the enzyme.
分子名称: CG peptide, SULFATE ION, Thymidylate synthase
著者Tochowicz, A, Finer-Moore, J, Stroud, R.M, Costi, M.P.
登録日2012-06-04
公開日2013-03-06
最終更新日2017-11-15
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Alanine mutants of the interface residues of human thymidylate synthase decode key features of the binding mode of allosteric anticancer peptides.
J.Med.Chem., 58, 2015
4N1A
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BU of 4n1a by Molmil
Thermomonospora curvata EccC (ATPases 2 and 3) in complex with a signal sequence peptide
分子名称: ADENOSINE-5'-TRIPHOSPHATE, Cell divisionFtsK/SpoIIIE, MAGNESIUM ION, ...
著者Dovala, D.L, Bendebury, A, Cox, J.S, Stroud, R.M, Rosenberg, O.S.
登録日2013-10-03
公開日2015-02-11
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (3.24 Å)
主引用文献Substrates Control Multimerization and Activation of the Multi-Domain ATPase Motor of Type VII Secretion.
Cell(Cambridge,Mass.), 161, 2015
7TDF
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BU of 7tdf by Molmil
AtTPC1 D454N with 1 mM EDTA state I
分子名称: Two pore calcium channel protein 1
著者Dickinson, M.S, Stroud, R.M.
登録日2021-12-31
公開日2022-02-02
最終更新日2022-03-09
実験手法ELECTRON MICROSCOPY (2.7 Å)
主引用文献Molecular basis of multistep voltage activation in plant two-pore channel 1.
Proc.Natl.Acad.Sci.USA, 119, 2022
3C02
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BU of 3c02 by Molmil
X-ray structure of the aquaglyceroporin from Plasmodium falciparum
分子名称: Aquaglyceroporin, GLYCEROL, octyl beta-D-glucopyranoside
著者Newby, Z.E, Stroud, R.M, Center for Structures of Membrane Proteins (CSMP)
登録日2008-01-18
公開日2008-05-27
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献Crystal structure of the aquaglyceroporin PfAQP from the malarial parasite Plasmodium falciparum.
Nat.Struct.Mol.Biol., 15, 2008

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