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8AEY
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BU of 8aey by Molmil
3 A CRYO-EM STRUCTURE OF MYCOBACTERIUM TUBERCULOSIS FERRITIN FROM TIMEPIX3 detector
分子名称: Ferritin BfrB
著者Zhang, Y, van Schayck, J.P, Knoops, K, Peters, P.J, Ravelli, R.B.G.
登録日2022-07-14
公開日2023-01-18
最終更新日2023-03-01
実験手法ELECTRON MICROSCOPY (3.05 Å)
主引用文献Integration of an Event-driven Timepix3 Hybrid Pixel Detector into a Cryo-EM Workflow
Microsc Microanal, 2023
7P0Z
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BU of 7p0z by Molmil
2.43 A Mycobacterium marinum EspB.
分子名称: ESX-1 secretion-associated protein EspB
著者Gijsbers, A, Zhang, Y, Vinciauskaite, V, Siroy, A, Ye, G, Tria, G, Mathew, A, Sanchez-Puig, N, Lopez-Iglesias, C, Peters, P.J, Ravelli, R.B.G.
登録日2021-07-01
公開日2021-08-18
最終更新日2021-10-13
実験手法ELECTRON MICROSCOPY (2.43 Å)
主引用文献Priming mycobacterial ESX-secreted protein B to form a channel-like structure.
Curr Res Struct Biol, 3, 2021
7P13
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2.29 A Mycobacterium tuberculosis EspB.
分子名称: ESX-1 secretion-associated protein EspB
著者Gijsbers, A, Zhang, Y, Vinciauskaite, V, Siroy, A, Gao, Y, Tria, G, Mathew, A, Sanchez-Puig, N, Lopez-Iglesias, C, Peters, P.J, Ravelli, R.B.G.
登録日2021-07-01
公開日2021-08-18
最終更新日2021-10-13
実験手法ELECTRON MICROSCOPY (2.29 Å)
主引用文献Priming mycobacterial ESX-secreted protein B to form a channel-like structure.
Curr Res Struct Biol, 3, 2021
8QQK
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BU of 8qqk by Molmil
Cryo-EM structure of E. coli cytochrome bo3 quinol oxidase assembled in peptidiscs
分子名称: (2S)-3-(hexadecanoyloxy)-2-[(9Z)-octadec-9-enoyloxy]propyl 2-(trimethylammonio)ethyl phosphate, 1,2-Distearoyl-sn-glycerophosphoethanolamine, COPPER (II) ION, ...
著者Gao, Y, Zhang, Y, Hakke, S, Peters, P.J, Ravelli, R.B.G.
登録日2023-10-05
公開日2024-04-24
最終更新日2024-05-01
実験手法ELECTRON MICROSCOPY (2.8 Å)
主引用文献Cryo-EM structure of cytochrome bo 3 quinol oxidase assembled in peptidiscs reveals an "open" conformation for potential ubiquinone-8 release.
Biochim Biophys Acta Bioenerg, 1865, 2024
7O6E
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BU of 7o6e by Molmil
2.12 A cryo-EM structure of Mycobacterium tuberculosis Ferritin
分子名称: Ferritin BfrB
著者Gijsbers, A, Zhang, Y, Gao, Y, Peters, P.J, Ravelli, R.B.G.
登録日2021-04-10
公開日2021-05-19
最終更新日2024-07-10
実験手法ELECTRON MICROSCOPY (2.1 Å)
主引用文献Mycobacterium tuberculosis ferritin: a suitable workhorse protein for cryo-EM development.
Acta Crystallogr D Struct Biol, 77, 2021
1S1J
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BU of 1s1j by Molmil
Crystal Structure of ZipA in complex with indoloquinolizin inhibitor 1
分子名称: (12bS)-1,2,3,4,12,12b-hexahydroindolo[2,3-a]quinolizin-7(6H)-one, Cell division protein zipA
著者Jenning, L.D, Foreman, K.W, Rush III, T.S, Tsao, D.H, Mosyak, L, Li, Y, Sukhdeo, M.N, Ding, W, Dushin, E.G, Kenney, C.H, Moghazeh, S.L, Peterson, P.J, Ruzin, A.V, Tuckman, M, Sutherland, A.G.
登録日2004-01-06
公開日2004-05-04
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.18 Å)
主引用文献Design and synthesis of indolo[2,3-a]quinolizin-7-one inhibitors of the ZipA-FtsZ interaction
Bioorg.Med.Chem.Lett., 14, 2004
1S1S
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BU of 1s1s by Molmil
Crystal Structure of ZipA in complex with indoloquinolizin 10b
分子名称: Cell division protein zipA, N-{3-[(12bS)-7-oxo-1,3,4,6,7,12b-hexahydroindolo[2,3-a]quinolizin-12(2H)-yl]propyl}propane-2-sulfonamide
著者Jennings, L.D, Foreman, K.W, Rush III, T.S, Tsao, D.H, Mosyak, L, Li, Y, Sukhdeo, M.N, Ding, W, Dushin, E.G, Kenny, C.H, Moghazeh, S.L, Petersen, P.J, Ruzin, A.V, Tuckman, M, Sutherland, A.G.
登録日2004-01-07
公開日2005-01-18
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Design and synthesis of indolo[2,3-a]quinolizin-7-one inhibitors of the ZipA-FtsZ interaction
BIOORG.MED.CHEM.LETT., 14, 2004
6KZM
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BU of 6kzm by Molmil
GluK3 receptor complex with kainate
分子名称: Glutamate receptor ionotropic, kainate 3
著者Kumar, J, Kumari, J, Burada, A.P.
登録日2019-09-24
公開日2020-03-04
実験手法ELECTRON MICROSCOPY (9.6 Å)
主引用文献Structural dynamics of the GluK3-kainate receptor neurotransmitter binding domains revealed by cryo-EM.
Int.J.Biol.Macromol., 149, 2020
8AKO
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BU of 8ako by Molmil
Structure of EspB-EspK complex: the non-identical twin of the PE-PPE-EspG secretion mechanism.
分子名称: ESX-1 secretion-associated protein EspB, ESX-1 secretion-associated protein EspK
著者Gijsbers, A, Eymery, M, Menart, I, Vinciauskaite, V, Gao, Y, Siliqi, D, Peters, P, Mccarthy, A, Ravelli, R.B.G.
登録日2022-07-30
公開日2022-12-14
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.293 Å)
主引用文献The crystal structure of the EspB-EspK virulence factor-chaperone complex suggests an additional type VII secretion mechanism in Mycobacterium tuberculosis.
J.Biol.Chem., 299, 2022
7P1T
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BU of 7p1t by Molmil
Cryo-EM structure of encapsulin from Mycobacterium tuberculosis
分子名称: 29 kDa antigen, Cfp29
著者Lewis, C.J, Berger, C, Ravelli, R.B.G.
登録日2021-07-02
公開日2022-07-13
実験手法ELECTRON MICROSCOPY (2.29 Å)
主引用文献Encapsulins in mycobacteria: from single particle to in situ
To Be Published
6L6F
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BU of 6l6f by Molmil
GluK3 receptor complex with UBP301
分子名称: Glutamate receptor ionotropic, kainate 3
著者Kumar, J, Kumari, J, Burada, A.P.
登録日2019-10-28
公開日2020-03-04
実験手法ELECTRON MICROSCOPY (10.6 Å)
主引用文献Structural dynamics of the GluK3-kainate receptor neurotransmitter binding domains revealed by cryo-EM.
Int.J.Biol.Macromol., 149, 2020
2Q85
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BU of 2q85 by Molmil
Crystal Structure of E. Coli Mur B bound to a Naphthyl Tetronic Acid inihibitor
分子名称: (5Z)-3-(4-CHLOROPHENYL)-4-HYDROXY-5-(1-NAPHTHYLMETHYLENE)FURAN-2(5H)-ONE, FLAVIN-ADENINE DINUCLEOTIDE, UDP-N-acetylenolpyruvoylglucosamine reductase
著者Chopra, R, Bard, J, Svenson, K, Mansour, T.
登録日2007-06-08
公開日2007-06-26
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.51 Å)
主引用文献Crystal Structure of E. Coli Mur B bound to a napthyl tetronic acid inhibitor
TO BE PUBLISHED
1Q2Q
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BU of 1q2q by Molmil
Enterobacter cloacae GC1 class C beta-lactamase complexed with penem WAY185229
分子名称: (6,7-DIHYDRO-5H-CYCLOPENTA[D]IMIDAZO[2,1-B]THIAZOL-2-YL]-4,7-DIHYDRO[1,4]THIAZEPINE-3,6-DICARBOXYLIC ACID, GLYCEROL, class C beta-lactamase
著者Nukaga, M, Venkatesan, A.M, Mansour, T.S, Hujer, A, Bonomo, R.A, Knox, J.R.
登録日2003-07-25
公開日2004-09-14
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献Structure-activity relationship of 6-methylidene penems bearing tricyclic heterocycles as broad-spectrum beta-lactamase inhibitors: crystallographic structures show unexpected binding of 1,4-thiazepine intermediates
J.Med.Chem., 47, 2004
1Q2P
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BU of 1q2p by Molmil
SHV-1 class A beta-lactamase complexed with penem WAY185229
分子名称: (6,7-DIHYDRO-5H-CYCLOPENTA[D]IMIDAZO[2,1-B]THIAZOL-2-YL]-4,7-DIHYDRO[1,4]THIAZEPINE-3,6-DICARBOXYLIC ACID, CYCLOHEXYL-HEXYL-BETA-D-MALTOSIDE, beta-lactamase SHV-1
著者Nukaga, M, Venkatesan, A.M, Mansour, T.S, Hujer, A, Bonomo, R.A, Knox, J.R.
登録日2003-07-25
公開日2004-09-14
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structure-activity relationship of 6-methylidene penems bearing tricyclic heterocycles as broad-spectrum beta-lactamase inhibitors: crystallographic structures show unexpected binding of 1,4-thiazepine intermediates
J.Med.Chem., 47, 2004

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件を2024-07-10に公開中

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