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3ZKT
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BU of 3zkt by Molmil
SOLUTION STRUCTURE OF THE SOMATOSTATIN SST3 RECEPTOR ANTAGONIST TAU- CONOTOXIN CnVA
分子名称: TAU-CNVA
著者Petrel, C, Hocking, H.G, Reynaud, M, Favreau, P, Paolini-Bertrand, M, Peigneur, S, Upert, G, Tytgat, J, Gilles, N, Hartley, O, Boelens, R, Stocklin, R, Servent, D.
登録日2013-01-24
公開日2013-04-24
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献Identification, Structural and Pharmacological Characterization of Tau-Cnva, a Conopeptide that Selectively Interacts with Somatostatin Sst3 Receptor.
Biochem.Pharmacol, 85, 2013
2XZ5
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BU of 2xz5 by Molmil
MMTS-modified Y53C mutant of Aplysia AChBP in complex with acetylcholine
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, 2-acetamido-2-deoxy-beta-D-glucopyranose, ACETYLCHOLINE, ...
著者Brams, M, Gay, E.A, Colon Saez, J, Guskov, A, van Elk, R, van der Schors, R.C, Peigneur, S, Tytgat, J, Strelkov, S.V, Smit, A.B, Yakel, J.L, Ulens, C.
登録日2010-11-23
公開日2010-12-08
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Crystal Structures of a Cysteine-Modified Mutant in Loop D of Acetylcholine Binding Protein
J.Biol.Chem., 286, 2011
2XZ6
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BU of 2xz6 by Molmil
MTSET-modified Y53C mutant of Aplysia AChBP
分子名称: 2-(TRIMETHYLAMMONIUM)ETHYL THIOL, SOLUBLE ACETYLCHOLINE RECEPTOR
著者Brams, M, Gay, E.A, Colon Saez, J, Guskov, A, Van Elk, R, Van Der Schors, R.C, Peigneur, S, Tytgat, J, Strelkov, S.V, Smit, A.B, Yakel, J.L, Ulens, C.
登録日2010-11-23
公開日2010-12-08
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (3.137 Å)
主引用文献Crystal Structures of a Cysteine-Modified Mutant in Loop D of Acetylcholine Binding Protein
J.Biol.Chem., 286, 2011
2LKB
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BU of 2lkb by Molmil
Evolutionary diversification of Mesobuthus alpha-scorpion toxins affecting sodium channels
分子名称: Neurotoxin MeuNaTx-5
著者Zhu, S, Peigneur, S, Gao, B, Lu, X, Cao, C, Tytgat, J.
登録日2011-10-09
公開日2011-11-02
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献Evolutionary diversification of Mesobuthus {alpha}-scorpion toxins affecting sodium channels
Mol.Cell Proteomics, 2011
2MD6
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BU of 2md6 by Molmil
NMR SOLUTION STRUCTURE OF ALPHA CONOTOXIN LO1A FROM Conus longurionis
分子名称: ALPHA CONOTOXIN LO1A
著者Maiti, M, Lescrinier, E, Herdewijn, P, Lebbe, E.K.M, Peigneur, S, D'Souza, L, Tytgat, J.
登録日2013-09-01
公開日2014-03-05
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献Structure-Function Elucidation of a New alpha-Conotoxin, Lo1a, from Conus longurionis.
J.Biol.Chem., 289, 2014
2LU6
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BU of 2lu6 by Molmil
NMR solution structure of Midi peptide designed based on m-conotoxins
分子名称: Midi peptide designed based on m-conotoxins
著者Dyubankova, N, Lescrinier, E, Stevens, M, Tytgat, J, Herdewijn, P, Peigneur, S.
登録日2012-06-08
公開日2012-06-27
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献Design of bioactive peptides from naturally occurring mu-conotoxin structures.
J.Biol.Chem., 287, 2012
2MSF
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BU of 2msf by Molmil
NMR SOLUTION STRUCTURE OF SCORPION VENOM TOXIN Ts11 (TsPep1) FROM Tityus serrulatus
分子名称: Peptide TsPep1
著者Maiti, M, Lescrinier, E, Herdewijn, P, Cremonez, C.M, Peigneur, S, Cassoli, J.S, Dutra, A.A.A, Waelkens, E, Pimenta, A.M.C, De Lima, M.H, Tytgat, J, Arantes, E.C.
登録日2014-08-01
公開日2015-08-26
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献Structural and Functional Elucidation of Peptide Ts11 Shows Evidence of a Novel Subfamily of Scorpion Venom Toxins.
Toxins (Basel), 8, 2016
2LER
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BU of 2ler by Molmil
Conotoxin pc16a
分子名称: Conotoxin pc16a
著者Dyubankova, N, Lescrinier, E, Van Der Haegen, A, Peigneur, S, Tytgat, J.
登録日2011-06-22
公開日2012-04-11
最終更新日2012-04-18
実験手法SOLUTION NMR
主引用文献Pc16a, the first characterized peptide from Conus pictus venom, shows a novel disulfide connectivity.
Peptides, 34, 2012
2RTY
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BU of 2rty by Molmil
Solution structure of navitoxin
分子名称: navitoxin
著者Umetsu, Y, Ohki, S.
登録日2013-10-16
公開日2014-04-23
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献Experimental conversion of a defensin into a neurotoxin: implications for origin of toxic function
MOL.BIOL.EVOL., 31, 2014
5WCV
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BU of 5wcv by Molmil
AsK132958: A minimal homologue of ShK identified in the transcriptome of Anemonia sulcata
分子名称: ShK homolog AsK132958
著者Krishnarjuna, B, MacRaild, C.A, Norton, R.S.
登録日2017-07-02
公開日2017-10-25
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献Structure, folding and stability of a minimal homologue from Anemonia sulcata of the sea anemone potassium channel blocker ShK.
Peptides, 99, 2018
7AY8
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BU of 7ay8 by Molmil
NMR solution structure of Tbo-IT2
分子名称: Tbo-IT2
著者Mineev, K.S, Kornilov, F.D, Lushpa, V.A, Korolkova, Y.A, Maleeva, E.E, Andreev, Y.A, Kozlov, S.A, Arseniev, A.S.
登録日2020-11-11
公開日2021-03-03
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献New Insectotoxin from Tibellus Oblongus Spider Venom Presents Novel Adaptation of ICK Fold.
Toxins, 13, 2021
7K1M
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BU of 7k1m by Molmil
Peptide from stony coral Heliofungia actiniformis: Hact-1
分子名称: GLY-CYS-HIS-TYR-THR-PRO-PHE-GLY-LEU-ILE-CYS-PHE peptide
著者Daly, N.L, Schmidt, C.A.
登録日2020-09-08
公開日2020-11-25
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献Identification and Characterization of a Peptide from the Stony Coral Heliofungia actiniformis .
J.Nat.Prod., 83, 2020
6OQP
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BU of 6oqp by Molmil
U-AITx-Ate1
分子名称: SER-LYS-TRP-ILE-CYS-ALA-ASN-ARG-SER-VAL-CYS-PRO-ILE
著者Elnahriry, K.A, Wai, D.C.C, Norton, R.S.
登録日2019-04-28
公開日2019-07-31
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献Structural and functional characterisation of a novel peptide from the Australian sea anemone Actinia tenebrosa.
Toxicon, 168, 2019
6WQR
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BU of 6wqr by Molmil
NMR solution structure of leech peptide HSTX-I
分子名称: HSTX-I
著者Schroeder, C.I, McMahon, K.L.
登録日2020-04-29
公開日2020-06-24
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献Pharmacological activity and NMR solution structure of the leech peptide HSTX-I.
Biochem Pharmacol, 181, 2020
6ENA
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BU of 6ena by Molmil
Nemertide alpha-1
分子名称: Nemertide alpha-1
著者Jacobsson, E, Rosengren, K.J, Goransson, U.
登録日2017-10-04
公開日2018-03-14
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献Lineus longissimus, the longest animal on earth, expresses peptide toxins targeting voltage gated sodium channels
Sci Rep, 2018
6SAB
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BU of 6sab by Molmil
M-BUTX-Ptr1a (Parabuthus transvaalicus)
分子名称: M-BUTX-Ptr1a
著者Meudal, H, Landon, C, Delmas, A.F.
登録日2019-07-16
公開日2020-07-22
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献A Venomics Approach Coupled to High-Throughput Toxin Production Strategies Identifies the First Venom-Derived Melanocortin Receptor Agonists.
J.Med.Chem., 63, 2020
6SAA
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BU of 6saa by Molmil
M-TRTX-Preg1a (Poecilotheria regalis)
分子名称: U1-theraphotoxin-Pf3
著者Meudal, H, Landon, C, Delmas, A.F.
登録日2019-07-16
公開日2020-07-22
最終更新日2020-08-26
実験手法SOLUTION NMR
主引用文献A Venomics Approach Coupled to High-Throughput Toxin Production Strategies Identifies the First Venom-Derived Melanocortin Receptor Agonists.
J.Med.Chem., 63, 2020
5OUG
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BU of 5oug by Molmil
Humanized alpha-AChBP (acetylcholine binding protein) in complex with lobeline and allosteric binder fragment 4.
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 4,5-dibromo-N-(3-hydroxypropyl)-1H-pyrrole-2-carboxamide, Alpha-Lobeline, ...
著者Delbart, F, Gruss, F, Ulens, C.
登録日2017-08-23
公開日2017-12-20
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2.57 Å)
主引用文献An allosteric binding site of the alpha 7 nicotinic acetylcholine receptor revealed in a humanized acetylcholine-binding protein.
J. Biol. Chem., 293, 2018
5OUI
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BU of 5oui by Molmil
Humanized alpha-AChBP (acetylcholine binding protein) in complex with allosteric binder fragment CU2017
分子名称: (3~{R})-~{N}-(5-bromanylpyridin-2-yl)piperidine-3-carboxamide, 1,2-ETHANEDIOL, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Delbart, F, Gruss, F, Ulens, C.
登録日2017-08-23
公開日2017-11-29
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献An allosteric binding site of the alpha 7 nicotinic acetylcholine receptor revealed in a humanized acetylcholine-binding protein.
J. Biol. Chem., 293, 2018
5OUH
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BU of 5ouh by Molmil
Humanized alpha-AChBP (acetylcholine binding protein) in complex with lobeline.
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Acetylcholine binding protein, Alpha-Lobeline, ...
著者Delbart, F, Gruss, F, Ulens, C.
登録日2017-08-23
公開日2017-11-29
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献An allosteric binding site of the alpha 7 nicotinic acetylcholine receptor revealed in a humanized acetylcholine-binding protein.
J. Biol. Chem., 293, 2018
7OXF
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BU of 7oxf by Molmil
Solution structure of bee apamin
分子名称: Apamin
著者Mineev, K, Kuzmenkov, A, Vassilevski, A.
登録日2021-06-22
公開日2022-07-13
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献Apamin structure and pharmacology revisited.
Front Pharmacol, 13, 2022
5M4V
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BU of 5m4v by Molmil
X-ray structure of the mambaquaretin-1, a selective antagonist of the vasopressin type 2 receptor
分子名称: CHLORIDE ION, Mambaquaretin-1, S-1,2-PROPANEDIOL
著者Stura, E.A, Vera, L, Ciolek, J, Mourier, G, Gilles, N.
登録日2016-10-19
公開日2017-05-03
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.06 Å)
主引用文献Green mamba peptide targets type-2 vasopressin receptor against polycystic kidney disease.
Proc. Natl. Acad. Sci. U.S.A., 114, 2017
7QXJ
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BU of 7qxj by Molmil
Solution structure of Tk-hefu-11
分子名称: Tk-hefu-11
著者Mineev, K.S, Lushpa, V.A, Vassilevski, A.A, Gigolaev, A.M.
登録日2022-01-26
公開日2022-09-21
最終更新日2022-11-16
実験手法SOLUTION NMR
主引用文献Artificial pore blocker acts specifically on voltage-gated potassium channel isoform K V 1.6.
J.Biol.Chem., 298, 2022
8CIQ
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BU of 8ciq by Molmil
JzTx-34 toxin peptide
分子名称: Mu-theraphotoxin-Cg1a
著者Landon, C, Meudal, H.
登録日2023-02-10
公開日2023-07-26
実験手法SOLUTION NMR
主引用文献Structure-function relationship of new peptides activating human Na v 1.1.
Biomed Pharmacother, 165, 2023
8CJP
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JzTx-34 toxin peptide H18A mutant
分子名称: Mu-theraphotoxin-Cg1a
著者Landon, C, Meudal, H.
登録日2023-02-13
公開日2023-07-26
実験手法SOLUTION NMR
主引用文献Structure-function relationship of new peptides activating human Na v 1.1.
Biomed Pharmacother, 165, 2023

 

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