6FHK
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8R9U
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![BU of 8r9u by Molmil](/molmil-images/mine/8r9u) | A soakable crystal form of human CDK7 in complex with AMP-PNP | 分子名称: | 7-dimethylphosphoryl-3-[2-[[(3~{S})-6,6-dimethylpiperidin-3-yl]amino]-5-(trifluoromethyl)pyrimidin-4-yl]-1~{H}-indole-6-carbonitrile, Cyclin-dependent kinase 7 | 著者 | Mukherjee, M, Cleasby, A. | 登録日 | 2023-11-30 | 公開日 | 2024-05-29 | 最終更新日 | 2024-06-26 | 実験手法 | X-RAY DIFFRACTION (1.937 Å) | 主引用文献 | Protein engineering enables a soakable crystal form of human CDK7 primed for high-throughput crystallography and structure-based drug design. Structure, 2024
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8R9S
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![BU of 8r9s by Molmil](/molmil-images/mine/8r9s) | A soakable crystal form of human CDK7 in complex with AMP-PNP | 分子名称: | 3,6,9,12,15,18,21,24,27,30,33,36,39-TRIDECAOXAHENTETRACONTANE-1,41-DIOL, Cyclin-dependent kinase 7, DI(HYDROXYETHYL)ETHER, ... | 著者 | Mukherjee, M, Cleasby, A. | 登録日 | 2023-11-30 | 公開日 | 2024-05-29 | 最終更新日 | 2024-06-26 | 実験手法 | X-RAY DIFFRACTION (2.78 Å) | 主引用文献 | Protein engineering enables a soakable crystal form of human CDK7 primed for high-throughput crystallography and structure-based drug design. Structure, 2024
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8R9A
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![BU of 8r9a by Molmil](/molmil-images/mine/8r9a) | A soakable crystal form of human CDK7 in complex with AMP-PNP | 分子名称: | (3R,4R)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-ol, Cyclin-dependent kinase 7, DI(HYDROXYETHYL)ETHER | 著者 | Mukherjee, M, Cleasby, A. | 登録日 | 2023-11-30 | 公開日 | 2024-05-29 | 最終更新日 | 2024-06-26 | 実験手法 | X-RAY DIFFRACTION (1.71 Å) | 主引用文献 | Protein engineering enables a soakable crystal form of human CDK7 primed for high-throughput crystallography and structure-based drug design. Structure, 2024
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8R9O
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![BU of 8r9o by Molmil](/molmil-images/mine/8r9o) | A soakable crystal form of human CDK7 in complex with AMP-PNP | 分子名称: | Cyclin-dependent kinase 7, ~{N}-[(1~{S})-2-(dimethylamino)-1-phenyl-ethyl]-6,6-dimethyl-3-[[4-(propanoylamino)phenyl]carbonylamino]-1,4-dihydropyrrolo[3,4-c]pyrazole-5-carboxamide | 著者 | Mukherjee, M, Cleasby, A. | 登録日 | 2023-11-30 | 公開日 | 2024-05-29 | 最終更新日 | 2024-06-26 | 実験手法 | X-RAY DIFFRACTION (2.22 Å) | 主引用文献 | Protein engineering enables a soakable crystal form of human CDK7 primed for high-throughput crystallography and structure-based drug design. Structure, 2024
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8R9B
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8R99
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8RU8
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![BU of 8ru8 by Molmil](/molmil-images/mine/8ru8) | A crystal form of a human CDK2-CDK7 chimera | 分子名称: | (3R,4R)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-ol, Cyclin-dependent kinase 2 | 著者 | Mukherjee, M, Cleasby, A. | 登録日 | 2024-01-30 | 公開日 | 2024-06-26 | 実験手法 | X-RAY DIFFRACTION (1.51 Å) | 主引用文献 | Protein engineering enables a soakable crystal form of human CDK7 primed for high-throughput crystallography and structure-based drug design. Structure, 2024
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1Z66
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![BU of 1z66 by Molmil](/molmil-images/mine/1z66) | NMR solution structure of domain III of E-protein of tick-borne Langat flavivirus (no RDC restraints) | 分子名称: | Major envelope protein E | 著者 | Mukherjee, M, Dutta, K, White, M.A, Cowburn, D, Fox, R.O. | 登録日 | 2005-03-21 | 公開日 | 2006-03-28 | 最終更新日 | 2022-03-02 | 実験手法 | SOLUTION NMR | 主引用文献 | NMR solution structure and backbone dynamics of domain III of the E protein of tick-borne Langat flavivirus suggests a potential site for molecular recognition. Protein Sci., 15, 2006
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2GG1
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![BU of 2gg1 by Molmil](/molmil-images/mine/2gg1) | NMR solution structure of domain III of the E-protein of tick-borne Langat flavivirus (includes RDC restraints) | 分子名称: | Genome polyprotein | 著者 | Mukherjee, M, Dutta, K, White, M.A, Cowburn, D, Fox, R.O. | 登録日 | 2006-03-23 | 公開日 | 2006-04-25 | 最終更新日 | 2023-11-29 | 実験手法 | SOLUTION NMR | 主引用文献 | NMR solution structure and backbone dynamics of domain III of the E protein of tick-borne Langat flavivirus suggests a potential site for molecular recognition. Protein Sci., 15, 2006
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5ODS
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2MQ1
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3VK6
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![BU of 3vk6 by Molmil](/molmil-images/mine/3vk6) | |
2G6U
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![BU of 2g6u by Molmil](/molmil-images/mine/2g6u) | |
1R8T
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![BU of 1r8t by Molmil](/molmil-images/mine/1r8t) | Solution structures of high affinity miniprotein ligands to Streptavidin | 分子名称: | MP1 | 著者 | Luo, J, Mukherjee, M, Fan, X, Yang, H, Liu, D, Khan, R, White, M, Fox, R.O. | 登録日 | 2003-10-28 | 公開日 | 2005-02-15 | 最終更新日 | 2022-03-02 | 実験手法 | SOLUTION NMR | 主引用文献 | Structure-based design of high affinity miniprotein ligands To be Published
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5HPK
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![BU of 5hpk by Molmil](/molmil-images/mine/5hpk) | System-wide modulation of HECT E3 ligases with selective ubiquitin variant probes: NEDD4L and UbV NL.1 | 分子名称: | E3 ubiquitin-protein ligase NEDD4-like, Ubiquitin variant NL.1 | 著者 | Wu, K.-P, Mukherjee, M, Mercredi, P.Y, Schulman, B.A. | 登録日 | 2016-01-20 | 公開日 | 2016-03-16 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2.431 Å) | 主引用文献 | System-Wide Modulation of HECT E3 Ligases with Selective Ubiquitin Variant Probes. Mol.Cell, 62, 2016
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7ELJ
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5HPT
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5HPL
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5HPS
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5ODT
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![BU of 5odt by Molmil](/molmil-images/mine/5odt) | Aurora-A in complex with TACC3 | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, Aurora kinase A, GLYCEROL, ... | 著者 | Burgess, S.G, Bayliss, R. | 登録日 | 2017-07-06 | 公開日 | 2018-03-14 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (2.021 Å) | 主引用文献 | Mitotic spindle association of TACC3 requires Aurora-A-dependent stabilization of a cryptic alpha-helix. EMBO J., 37, 2018
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5C7J
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![BU of 5c7j by Molmil](/molmil-images/mine/5c7j) | CRYSTAL STRUCTURE OF NEDD4 WITH A UB VARIANT | 分子名称: | E3 ubiquitin-protein ligase NEDD4, Polyubiquitin-C | 著者 | Walker, J.R, Hu, J, Dong, A, Bountra, C, Edwards, A.M, Arrowsmith, C.H, Tong, Y, Structural Genomics Consortium (SGC) | 登録日 | 2015-06-24 | 公開日 | 2016-03-16 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | System-Wide Modulation of HECT E3 Ligases with Selective Ubiquitin Variant Probes. Mol.Cell, 62, 2016
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5C7M
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![BU of 5c7m by Molmil](/molmil-images/mine/5c7m) | CRYSTAL STRUCTURE OF E3 LIGASE ITCH WITH A UB VARIANT | 分子名称: | E3 ubiquitin-protein ligase Itchy homolog, Polyubiquitin-C | 著者 | Walker, J.R, Hu, J, Dong, A, Wernimont, A, Zhang, W, Sidhu, S, Bountra, C, Edwards, A.M, Arrowsmith, C.H, Tong, Y, Structural Genomics Consortium (SGC) | 登録日 | 2015-06-24 | 公開日 | 2016-03-16 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (3.03 Å) | 主引用文献 | System-Wide Modulation of HECT E3 Ligases with Selective Ubiquitin Variant Probes. Mol.Cell, 62, 2016
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4G1A
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5XCE
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![BU of 5xce by Molmil](/molmil-images/mine/5xce) | Crystal structure of Wild type Vps29 from Entamoeba histolytica | 分子名称: | Vacuolar protein sorting-associated protein 29 | 著者 | Srivastava, V.K, Yadav, R, Tomar, P, Gourinath, S, Datta, S. | 登録日 | 2017-03-22 | 公開日 | 2017-10-04 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.86 Å) | 主引用文献 | Structural and thermodynamic characterization of metal binding in Vps29 from Entamoeba histolytica: implication in retromer function. Mol. Microbiol., 106, 2017
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