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6J90
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BU of 6j90 by Molmil
Crystal Structure of GyraseB N-Terminal Domain complex with ATP from Salmonella Typhi at 2.2A Resolution
分子名称: ADENOSINE-5'-TRIPHOSPHATE, CHLORIDE ION, DI(HYDROXYETHYL)ETHER, ...
著者Kaur, G, Sachdeva, E, Tiwari, P, Gupta, D, Ethayathulla, A.S, Kaur, P.
登録日2019-01-21
公開日2020-01-22
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Crystal Structure of GyraseB N-Terminal Domain complex with ATP from Salmonella Typhi at 2.2A Resolution
To Be Published
4MFR
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BU of 4mfr by Molmil
Crystal structure of Mycobacterium tuberculosis CarD
分子名称: GLYCEROL, IODIDE ION, RNA polymerase-binding transcription factor CarD, ...
著者Kaur, G, Thakur, K.G.
登録日2013-08-28
公開日2013-11-06
最終更新日2024-05-29
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Crystal structure of Mycobacterium tuberculosis CarD, an essential RNA polymerase binding protein, reveals a quasidomain-swapped dimeric structural architecture.
Proteins, 82, 2014
4ILU
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BU of 4ilu by Molmil
Crystal structure of Mycobacterium tuberculosis CarD
分子名称: RNA polymerase-binding transcription factor CarD, SULFATE ION
著者Thakur, K.G, Kaur, G.
登録日2013-01-01
公開日2013-10-30
最終更新日2024-05-29
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Crystal structure of Mycobacterium tuberculosis CarD, an essential RNA polymerase binding protein, reveals a quasidomain-swapped dimeric structural architecture.
Proteins, 82, 2014
5ZTJ
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BU of 5ztj by Molmil
Crystal Structure of GyraseA C-Terminal Domain from Salmonella typhi at 2.4A Resolution
分子名称: DNA gyrase subunit A
著者Sachdeva, E, Gupta, D, Tiwari, P, Kaur, G, Sharma, S, Singh, T.P, Ethayathulla, A.S, Kaur, P.
登録日2018-05-03
公開日2019-05-15
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献The pivot point arginines identified in the beta-pinwheel structure of C-terminal domain from Salmonella Typhi DNA Gyrase A subunit.
Sci Rep, 10, 2020
7L9A
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BU of 7l9a by Molmil
Crystal structure of BRDT bromodomain 2 in complex with CDD-1102
分子名称: BETA-MERCAPTOETHANOL, Bromodomain testis-specific protein, N~1~-(5-{[3-(4-amino-2-methylphenyl)-1-methyl-1H-indazole-5-carbonyl]amino}-2-methylphenyl)-N~4~-methylbenzene-1,4-dicarboxamide
著者Sharma, R, Kaur, G, Yu, Z, Ku, A.F, Anglin, J.L, Ucisik, M.N, Faver, J.C, Sankaran, B, Kim, C, Matzuk, M.M.
登録日2021-01-03
公開日2021-06-30
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.27 Å)
主引用文献Discovery and characterization of bromodomain 2-specific inhibitors of BRDT.
Proc.Natl.Acad.Sci.USA, 118, 2021
5VGD
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BU of 5vgd by Molmil
Crystal Structure of HLA-C*0501 in complex with SAE
分子名称: Beta-2-microglobulin, HLA class I histocompatibility antigen, Cw-5 alpha chain, ...
著者Gras, S, Rossjohn, J.
登録日2017-04-11
公開日2017-05-31
最終更新日2017-07-12
実験手法X-RAY DIFFRACTION (2.32 Å)
主引用文献Structural and regulatory diversity shape HLA-C protein expression levels.
Nat Commun, 8, 2017
5VGE
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BU of 5vge by Molmil
Crystal structure of HLA-C*07:02 in complex with RYR peptide
分子名称: ARG-TYR-ARG-PRO-GLY-THR-VAL-ALA-LEU, Beta-2-microglobulin, ZINC ION, ...
著者Mobbs, J.I, Vivian, J.P, Gras, S, Rossjohn, J.
登録日2017-04-11
公開日2017-06-07
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Structural and regulatory diversity shape HLA-C protein expression levels.
Nat Commun, 8, 2017
8RQU
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BU of 8rqu by Molmil
Structure of TEM1 beta-lactamase variant 70.a
分子名称: Beta-lactamase TEM-1, MAGNESIUM ION
著者Napier, E, Fram, B.F, Gauthier, N.P, Sander, C, Khan, A.R.
登録日2024-01-19
公開日2024-02-14
最終更新日2024-07-17
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Simultaneous enhancement of multiple functional properties using evolution-informed protein design.
Nat Commun, 15, 2024
7LV3
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BU of 7lv3 by Molmil
Crystal structure of human protein kinase G (PKG) R-C complex in inhibited state
分子名称: 1,2-ETHANEDIOL, Isoform Beta of cGMP-dependent protein kinase 1, MANGANESE (II) ION, ...
著者Sharma, R, Lying, Q, Casteel, D, Kim, C.
登録日2021-02-23
公開日2022-08-24
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.41 Å)
主引用文献An auto-inhibited state of protein kinase G and implications for selective activation.
Elife, 11, 2022
7MBJ
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BU of 7mbj by Molmil
Crystal structure of cGMP dependent protein kinase I alpha (PKG I alpha)CNB-A domain with R177Q mutation
分子名称: cGMP-dependent protein kinase 1
著者Kim, J.J, Casteel, D.E, Kim, C.
登録日2021-03-31
公開日2022-05-11
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (1.26 Å)
主引用文献An auto-inhibited state of protein kinase G and implications for selective activation.
Elife, 11, 2022
5HEZ
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BU of 5hez by Molmil
JAK2 kinase (JH1 domain) mutant P1057A in complex with TG101209
分子名称: CHLORIDE ION, N-tert-butyl-3-[(5-methyl-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]benzenesulfonamide, Tyrosine-protein kinase JAK2, ...
著者Ultsch, M, Eigenbrot, C.
登録日2016-01-06
公開日2016-11-09
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.66 Å)
主引用文献Resolving TYK2 locus genotype-to-phenotype differences in autoimmunity.
Sci Transl Med, 8, 2016
8GII
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BU of 8gii by Molmil
TEM-1 Beta Lactamase Variant 80.a
分子名称: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, TEM-1 Variant 80.a
著者Fram, B.F, Gauthier, N.P, Khan, A.R, Sander, C.
登録日2023-03-14
公開日2024-04-17
最終更新日2024-07-17
実験手法X-RAY DIFFRACTION (1.83 Å)
主引用文献Simultaneous enhancement of multiple functional properties using evolution-informed protein design.
Nat Commun, 15, 2024
8GIJ
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BU of 8gij by Molmil
TEM-1 Beta Lactamase Variant 80.b
分子名称: TEM-1 Beta Lactmase Variant 80.b
著者Fram, B.F, Gauthier, N.P, Khan, A, Sander, C.
登録日2023-03-14
公開日2024-04-17
最終更新日2024-07-17
実験手法X-RAY DIFFRACTION (1.59 Å)
主引用文献Simultaneous enhancement of multiple functional properties using evolution-informed protein design.
Nat Commun, 15, 2024
7L99
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BU of 7l99 by Molmil
Crystal structure of BRDT bromodomain 2 in complex with CDD-1302
分子名称: Bromodomain testis-specific protein, N-[3-(acetylamino)-4-methylphenyl]-3-(4-amino-2-methylphenyl)-1-methyl-1H-indazole-5-carboxamide, O-(O-(2-AMINOPROPYL)-O'-(2-METHOXYETHYL)POLYPROPYLENE GLYCOL 500)
著者Sharma, R, Yu, Z, Ku, A.F, Anglin, J.L, Ucisik, M.N, Faver, J.C, Sankaran, B, Kim, C, Matzuk, M.M.
登録日2021-01-03
公開日2021-06-30
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Discovery and characterization of bromodomain 2-specific inhibitors of BRDT.
Proc.Natl.Acad.Sci.USA, 118, 2021
8S9M
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BU of 8s9m by Molmil
DNA cytosine-N4 methyltransferase (residues 79-324) from the Bdelloid rotifer Adineta vaga
分子名称: 1,2-ETHANEDIOL, DNA cytosine-N4 methyltransferase, SINEFUNGIN
著者Zhou, J, Horton, J.R, Cheng, X.
登録日2023-03-29
公開日2023-08-02
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (1.49 Å)
主引用文献Biochemical and structural characterization of the first-discovered metazoan DNA cytosine-N4 methyltransferase from the bdelloid rotifer Adineta vaga.
J.Biol.Chem., 299, 2023
8S9N
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BU of 8s9n by Molmil
DNA cytosine-N4 methyltransferase (residues 61-324) from the Bdelloid rotifer Adineta vaga - C2 crystal form
分子名称: 1,2-ETHANEDIOL, DNA cytosine-N4 methyltransferase, SINEFUNGIN
著者Zhou, J, Horton, J.R, Cheng, X.
登録日2023-03-29
公開日2023-08-02
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (1.89 Å)
主引用文献Biochemical and structural characterization of the first-discovered metazoan DNA cytosine-N4 methyltransferase from the bdelloid rotifer Adineta vaga.
J.Biol.Chem., 299, 2023
8S9O
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BU of 8s9o by Molmil
DNA cytosine-N4 methyltransferase (residues 61-324) from the Bdelloid rotifer Adineta vaga - P1 crystal form
分子名称: 1,2-ETHANEDIOL, DNA cytosine-N4 methyltransferase, SINEFUNGIN
著者Zhou, J, Horton, J.R, Cheng, X.
登録日2023-03-29
公開日2023-08-02
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (1.94 Å)
主引用文献Biochemical and structural characterization of the first-discovered metazoan DNA cytosine-N4 methyltransferase from the bdelloid rotifer Adineta vaga.
J.Biol.Chem., 299, 2023

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件を2024-07-24に公開中

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