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2H65
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BU of 2h65 by Molmil
Crystal strusture of caspase-3 with inhibitor Ac-VDVAD-Cho
分子名称: Ac-VDVAD-Cho, caspase-3, p12 subunit, ...
著者Fang, B, Boross, P.I, Tozser, J, Weber, I.T.
登録日2006-05-30
公開日2006-09-19
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Structural and kinetic analysis of caspase-3 reveals role for s5 binding site in substrate recognition
J.Mol.Biol., 360, 2006
2H5J
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BU of 2h5j by Molmil
Crystal strusture of caspase-3 with inhibitor Ac-DMQD-Cho
分子名称: Ac-DMQD-Cho, caspase-3, p12 subunit, ...
著者Fang, B, Boross, P.I, Tozser, J, Weber, I.T.
登録日2006-05-26
公開日2006-09-19
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structural and kinetic analysis of caspase-3 reveals role for s5 binding site in substrate recognition
J.Mol.Biol., 360, 2006
2H5I
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BU of 2h5i by Molmil
Crystal structure of caspase-3 with inhibitor Ac-DEVD-Cho
分子名称: Ac-DEV(ASJ), caspase-3, p12 subunit, ...
著者Fang, B, Boross, P.I, Tozser, J, Weber, I.T.
登録日2006-05-26
公開日2006-09-19
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.69 Å)
主引用文献Structural and kinetic analysis of caspase-3 reveals role for s5 binding site in substrate recognition
J.Mol.Biol., 360, 2006
3GJS
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BU of 3gjs by Molmil
Caspase-3 Binds Diverse P4 Residues in Peptides
分子名称: Ac-YVAD-Cho inhibitor, Caspase-3 subunit p12, Caspase-3 subunit p17
著者Fang, B, Fu, G, Agniswamy, J, Harrison, R.W, Weber, I.T.
登録日2009-03-09
公開日2009-03-24
最終更新日2011-08-17
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Caspase-3 binds diverse P4 residues in peptides as revealed by crystallography and structural modeling.
Apoptosis, 14, 2009
3GJR
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BU of 3gjr by Molmil
Caspase-3 Binds Diverse P4 Residues in Peptides
分子名称: Caspase-3 subunit p12, Caspase-3 subunit p17, GLYCEROL, ...
著者Fang, B, Fu, G, Agniswamy, J, Harrison, R.W, Weber, I.T.
登録日2009-03-09
公開日2009-03-24
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Caspase-3 binds diverse P4 residues in peptides as revealed by crystallography and structural modeling.
Apoptosis, 14, 2009
3GJT
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BU of 3gjt by Molmil
Caspase-3 Binds Diverse P4 Residues in Peptides
分子名称: Caspase-3 subunit p12, Caspase-3 subunit p17, peptide inhibitor
著者Fang, B, Fu, G, Agniswamy, J, Harrison, R.W, Weber, I.T.
登録日2009-03-09
公開日2009-03-24
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Caspase-3 binds diverse P4 residues in peptides as revealed by crystallography and structural modeling.
Apoptosis, 14, 2009
3GJQ
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BU of 3gjq by Molmil
Caspase-3 Binds Diverse P4 Residues in Peptides
分子名称: Caspase-3 subunit p12, Caspase-3 subunit p17, peptide inhibitor
著者Fang, B, Fu, G, Agniswamy, J, Harrison, R.W, Weber, I.T.
登録日2009-03-09
公開日2009-03-24
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Caspase-3 binds diverse P4 residues in peptides as revealed by crystallography and structural modeling.
Apoptosis, 14, 2009
8KFO
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BU of 8kfo by Molmil
Crystal structure of BSA in complex with B3
分子名称: 6-[(~{E})-2-[1-[2-[2-(2-methoxyethoxy)ethoxy]ethyl]pyridin-1-ium-4-yl]ethenyl]-~{N},~{N}-dimethyl-naphthalen-2-amine, Albumin
著者Chen, X, Ge, Y.H, Yang, H, Fang, B, Li, L.
登録日2023-08-16
公開日2024-08-21
実験手法X-RAY DIFFRACTION (3.6 Å)
主引用文献Bioinspired two-stage assembled photosensitive protein engineering for tumor-specific mitochondrial targeted phototherapy
To Be Published
2QLJ
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BU of 2qlj by Molmil
Crystal Structure of Caspase-7 with Inhibitor AC-WEHD-CHO
分子名称: CITRIC ACID, Caspase-7, Inhibitor AC-WEHD-CHO, ...
著者Agniswamy, J, Fang, B, Weber, I.
登録日2007-07-12
公開日2007-08-28
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Plasticity of S2-S4 specificity pockets of executioner caspase-7 revealed by structural and kinetic analysis.
Febs J., 274, 2007
2QL5
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BU of 2ql5 by Molmil
Crystal Structure of caspase-7 with inhibitor AC-DMQD-CHO
分子名称: CITRIC ACID, Caspase-7, inhibitor, ...
著者Agniswamy, J, Fang, B, Weber, I.
登録日2007-07-12
公開日2007-08-28
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.34 Å)
主引用文献Plasticity of S2-S4 specificity pockets of executioner caspase-7 revealed by structural and kinetic analysis.
Febs J., 274, 2007
2QL9
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BU of 2ql9 by Molmil
Crystal Structure of Caspase-7 with inhibitor AC-DQMD-CHO
分子名称: CITRIC ACID, Caspase-7, Inhibitor AC-DQMD-CHO, ...
著者Agniswamy, J, Fang, B, Weber, I.
登録日2007-07-12
公開日2007-08-28
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.14 Å)
主引用文献Plasticity of S2-S4 specificity pockets of executioner caspase-7 revealed by structural and kinetic analysis.
Febs J., 274, 2007
2QLF
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BU of 2qlf by Molmil
Crystal Structure of Caspase-7 with inhibitor AC-DNLD-CHO
分子名称: Caspase-7, Inhibitor AC-DNLD-CHO, Peptide QGHGE
著者Agniswamy, J, Fang, B, Weber, I.
登録日2007-07-12
公開日2007-08-28
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Plasticity of S2-S4 specificity pockets of executioner caspase-7 revealed by structural and kinetic analysis.
Febs J., 274, 2007
2QLB
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BU of 2qlb by Molmil
Crystal Structure of caspase-7 with inhibitor AC-ESMD-CHO
分子名称: CITRIC ACID, Caspase-7, Inhibitor AC-ESMD-CHO, ...
著者Agniswamy, J, Fang, B, Weber, I.
登録日2007-07-12
公開日2007-08-28
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.25 Å)
主引用文献Plasticity of S2-S4 specificity pockets of executioner caspase-7 revealed by structural and kinetic analysis.
Febs J., 274, 2007
2QL7
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BU of 2ql7 by Molmil
Crystal Structure of Caspase-7 with inhibitor AC-IEPD-CHO
分子名称: CITRIC ACID, Caspase-7, Inhibitor AC-IEPD_CHO, ...
著者Agniswamy, J, Fang, B, Weber, I.
登録日2007-07-12
公開日2007-08-28
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Plasticity of S2-S4 specificity pockets of executioner caspase-7 revealed by structural and kinetic analysis.
Febs J., 274, 2007
6LKG
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BU of 6lkg by Molmil
two-component system protein mediate signal transduction
分子名称: 6-O-phosphono-alpha-D-glucopyranose, ABC transporter, solute-binding protein, ...
著者Wang, M, Tao, Y.
登録日2019-12-19
公開日2020-12-02
最終更新日2024-03-27
実験手法X-RAY DIFFRACTION (1.948 Å)
主引用文献Interface switch mediates signal transmission in a two-component system.
Proc.Natl.Acad.Sci.USA, 117, 2020
6LKK
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BU of 6lkk by Molmil
Two-component system protein mediate signal transduction
分子名称: 6-O-phosphono-alpha-D-glucopyranose, ABC transporter, solute-binding protein
著者Wang, M, Tao, Y.
登録日2019-12-19
公開日2020-12-02
最終更新日2024-03-27
実験手法X-RAY DIFFRACTION (1.502 Å)
主引用文献Interface switch mediates signal transmission in a two-component system.
Proc.Natl.Acad.Sci.USA, 117, 2020
6LKL
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BU of 6lkl by Molmil
Two-component system protein mediate signal transduction
分子名称: ABC transporter, solute-binding protein, MALONIC ACID
著者Wang, M, Tao, Y.
登録日2019-12-19
公開日2020-12-02
最終更新日2024-03-27
実験手法X-RAY DIFFRACTION (2.213 Å)
主引用文献Interface switch mediates signal transmission in a two-component system.
Proc.Natl.Acad.Sci.USA, 117, 2020
6LKI
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BU of 6lki by Molmil
Two-component system protein mediate signal transduction
分子名称: ABC transporter, solute-binding protein, MALONIC ACID, ...
著者Wang, M, Tao, Y.
登録日2019-12-19
公開日2020-12-02
最終更新日2024-03-27
実験手法X-RAY DIFFRACTION (1.781 Å)
主引用文献Interface switch mediates signal transmission in a two-component system.
Proc.Natl.Acad.Sci.USA, 117, 2020
6LKJ
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BU of 6lkj by Molmil
Two-component system protein mediate signal transduction
分子名称: 6-O-phosphono-beta-D-galactopyranose, ABC transporter, solute-binding protein
著者Wang, M, Tao, Y.
登録日2019-12-19
公開日2020-12-02
最終更新日2024-03-27
実験手法X-RAY DIFFRACTION (2.004 Å)
主引用文献Interface switch mediates signal transmission in a two-component system.
Proc.Natl.Acad.Sci.USA, 117, 2020
6LKH
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BU of 6lkh by Molmil
Two-component system protein mediate signal transduction
分子名称: 6-O-phosphono-alpha-D-glucopyranose, ABC transporter, solute-binding protein, ...
著者Wang, M, Tao, Y.
登録日2019-12-19
公開日2021-03-17
最終更新日2024-05-29
実験手法X-RAY DIFFRACTION (2.534 Å)
主引用文献Interface switch mediates signal transmission in a two-component system.
Proc.Natl.Acad.Sci.USA, 117, 2020
3IBF
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BU of 3ibf by Molmil
Crystal structure of unliganded caspase-7
分子名称: Caspase-7
著者Agniswamy, J.
登録日2009-07-15
公開日2009-09-01
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Conformational similarity in the activation of caspase-3 and -7 revealed by the unliganded and inhibited structures of caspase-7.
Apoptosis, 14, 2009
3EDR
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BU of 3edr by Molmil
The crystal structure of caspase-7 in complex with Acetyl-LDESD-CHO
分子名称: Caspase-7, Inhibitor Ac-ldesd-cho peptide
著者Agniswamy, J.
登録日2008-09-03
公開日2008-10-28
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.45 Å)
主引用文献Structural basis for executioner caspase recognition of P5 position in substrates.
Apoptosis, 13, 2008
3IBC
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BU of 3ibc by Molmil
Crystal Structure of Caspase-7 incomplex with Acetyl-YVAD-CHO
分子名称: Acetyl-YVAD-CHO, Caspase-7
著者Agniswamy, J.
登録日2009-07-15
公開日2009-09-01
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.75 Å)
主引用文献Conformational similarity in the activation of caspase-3 and -7 revealed by the unliganded and inhibited structures of caspase-7.
Apoptosis, 14, 2009
3EDQ
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BU of 3edq by Molmil
Crystal structure of Caspase-3 with inhibitor AC-LDESD-CHO
分子名称: AC-LDESD-CHO peptide, Caspase-3
著者Fu, G.
登録日2008-09-03
公開日2008-10-28
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.61 Å)
主引用文献Structural basis for executioner caspase recognition of P5 position in substrates.
Apoptosis, 13, 2008
8X73
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BU of 8x73 by Molmil
Crystal structure of Peroxiredoxin I in complex with compound 19-069
分子名称: Peroxiredoxin-1, methyl (2~{S})-2-[[(2~{R},4~{a}~{S},6~{a}~{R},6~{a}~{S},14~{a}~{S},14~{b}~{R})-2,4~{a},6~{a},6~{a},9,14~{a}-hexamethyl-10-oxidanyl-11-oxidanylidene-1,3,4,5,6,13,14,14~{b}-octahydropicen-2-yl]carbamoylamino]-3-oxidanyl-propanoate
著者Zhang, H, Luo, C.
登録日2023-11-22
公開日2024-06-19
実験手法X-RAY DIFFRACTION (1.61 Å)
主引用文献Discovery of a Novel Orally Bioavailable FLT3-PROTAC Degrader for Efficient Treatment of Acute Myeloid Leukemia and Overcoming Resistance of FLT3 Inhibitors.
J.Med.Chem., 67, 2024

 

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