8HPP
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![BU of 8hpp by Molmil](/molmil-images/mine/8hpp) | |
4ZMI
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![BU of 4zmi by Molmil](/molmil-images/mine/4zmi) | Crystal structure of the Helical domain of S. pombe Taz1 | 分子名称: | COBALT (II) ION, MAGNESIUM ION, Telomere length regulator taz1 | 著者 | Deng, W, Wu, J, Wang, F, Lei, M. | 登録日 | 2015-05-04 | 公開日 | 2015-09-23 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Fission yeast telomere-binding protein Taz1 is a functional but not a structural counterpart of human TRF1 and TRF2. Cell Res., 25, 2015
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4ZMK
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![BU of 4zmk by Molmil](/molmil-images/mine/4zmk) | |
5X7L
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![BU of 5x7l by Molmil](/molmil-images/mine/5x7l) | |
3BZO
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![BU of 3bzo by Molmil](/molmil-images/mine/3bzo) | Crystal structural of native EscU C-terminal domain | 分子名称: | EscU, SULFATE ION | 著者 | Zarivach, R, Deng, W, Vuckovic, M, Felise, H.B, Nguyen, H.V, Miller, S.I, Finlay, B.B, Strynadka, N.C.J. | 登録日 | 2008-01-18 | 公開日 | 2008-04-22 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Structural analysis of the essential self-cleaving type III secretion proteins EscU and SpaS. Nature, 453, 2008
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3BZV
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![BU of 3bzv by Molmil](/molmil-images/mine/3bzv) | Crystal structural of the mutated T264A EscU C-terminal domain | 分子名称: | EscU | 著者 | Zarivach, R, Deng, W, Vuckovic, M, Felise, H.B, Nguyen, H.V, Miller, S.I, Finlay, B.B, Strynadka, N.C.J. | 登録日 | 2008-01-18 | 公開日 | 2008-04-22 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (1.94 Å) | 主引用文献 | Structural analysis of the essential self-cleaving type III secretion proteins EscU and SpaS. Nature, 453, 2008
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3BZS
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![BU of 3bzs by Molmil](/molmil-images/mine/3bzs) | Crystal structure of EscU C-terminal domain with N262D mutation, Space group P 21 21 21 | 分子名称: | EscU | 著者 | Zarivach, R, Deng, W, Vuckovic, M, Felise, H.B, Nguyen, H.V, Miller, S.I, Finlay, B.B, Strynadka, N.C.J. | 登録日 | 2008-01-18 | 公開日 | 2008-04-22 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (1.48 Å) | 主引用文献 | Structural analysis of the essential self-cleaving type III secretion proteins EscU and SpaS. Nature, 453, 2008
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3BZR
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![BU of 3bzr by Molmil](/molmil-images/mine/3bzr) | Crystal structure of EscU C-terminal domain with N262D mutation, Space group P 41 21 2 | 分子名称: | EscU | 著者 | Zarivach, R, Deng, W, Vuckovic, M, Felise, H.B, Nguyen, H.V, Miller, S.I, Finlay, B.B, Strynadka, N.C.J. | 登録日 | 2008-01-18 | 公開日 | 2008-04-22 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (1.646 Å) | 主引用文献 | Structural analysis of the essential self-cleaving type III secretion proteins EscU and SpaS. Nature, 453, 2008
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3BZY
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![BU of 3bzy by Molmil](/molmil-images/mine/3bzy) | Crystal structure of the mutated Y316D EscU C-terminal domain | 分子名称: | EscU, SULFATE ION | 著者 | Zarivach, R, Deng, W, Vuckovic, M, Felise, H.B, Nguyen, H.V, Miller, S.I, Finlay, B.B, Strynadka, N.C.J. | 登録日 | 2008-01-18 | 公開日 | 2008-04-22 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (1.2 Å) | 主引用文献 | Structural analysis of the essential self-cleaving type III secretion proteins EscU and SpaS. Nature, 453, 2008
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3BZP
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![BU of 3bzp by Molmil](/molmil-images/mine/3bzp) | Crystal structural of the mutated N262A EscU C-terminal domain | 分子名称: | EscU | 著者 | Zarivach, R, Deng, W, Vuckovic, M, Felise, H.B, Nguyen, H.V, Miller, S.I, Finlay, B.B, Strynadka, N.C.J. | 登録日 | 2008-01-18 | 公開日 | 2008-04-22 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (1.499 Å) | 主引用文献 | Structural analysis of the essential self-cleaving type III secretion proteins EscU and SpaS. Nature, 453, 2008
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1ONJ
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![BU of 1onj by Molmil](/molmil-images/mine/1onj) | Crystal structure of Atratoxin-b from Chinese cobra venom of Naja atra | 分子名称: | Cobrotoxin b, SULFATE ION | 著者 | Lou, X, Tu, X, Pan, G, Xu, C, Fan, R, Lu, W, Deng, W, Rao, P, Teng, M, Niu, L. | 登録日 | 2003-02-28 | 公開日 | 2004-02-28 | 最終更新日 | 2017-10-11 | 実験手法 | X-RAY DIFFRACTION (1.555 Å) | 主引用文献 | Purification, N-terminal sequencing, crystallization and preliminary structural determination of atratoxin-b, a short-chain alpha-neurotoxin from Naja atra venom. Acta Crystallogr.,Sect.D, 59, 2003
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2OBL
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![BU of 2obl by Molmil](/molmil-images/mine/2obl) | Structural and biochemical analysis of a prototypical ATPase from the type III secretion system of pathogenic bacteria | 分子名称: | ACETATE ION, CALCIUM ION, EscN, ... | 著者 | Zarivach, R, Vuckovic, M, Deng, W, Finlay, B.B, Strynadka, N.C.J. | 登録日 | 2006-12-19 | 公開日 | 2007-01-30 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Structural analysis of a prototypical ATPase from the type III secretion system. Nat.Struct.Mol.Biol., 14, 2007
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2OBM
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![BU of 2obm by Molmil](/molmil-images/mine/2obm) | Structural and biochemical analysis of a prototypical ATPase from the type III secretion system of pathogenic bacteria | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, CALCIUM ION, EscN | 著者 | Zarivach, R, Vuckovic, M, Deng, W, Finlay, B.B, Strynadka, N.C.J. | 登録日 | 2006-12-19 | 公開日 | 2007-01-30 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (2.25 Å) | 主引用文献 | Structural analysis of a prototypical ATPase from the type III secretion system. Nat.Struct.Mol.Biol., 14, 2007
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3C00
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![BU of 3c00 by Molmil](/molmil-images/mine/3c00) | Crystal structural of the mutated G247T EscU/SpaS C-terminal domain | 分子名称: | EscU | 著者 | Zarivach, R, Deng, W, Vuckovic, M, Felise, H.B, Nguyen, H.V, Miller, S.I, Finlay, B.B, Strynadka, N.C.J. | 登録日 | 2008-01-18 | 公開日 | 2008-04-22 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (1.41 Å) | 主引用文献 | Structural analysis of the essential self-cleaving type III secretion proteins EscU and SpaS. Nature, 453, 2008
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3BZT
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![BU of 3bzt by Molmil](/molmil-images/mine/3bzt) | Crystal structural of the mutated P263A EscU C-terminal domain | 分子名称: | EscU | 著者 | Zarivach, R, Deng, W, Vuckovic, M, Felise, H.B, Nguyen, H.V, Miller, S.I, Finlay, B.B, Strynadka, N.C.J. | 登録日 | 2008-01-18 | 公開日 | 2008-04-22 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Structural analysis of the essential self-cleaving type III secretion proteins EscU and SpaS. Nature, 453, 2008
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3C03
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![BU of 3c03 by Molmil](/molmil-images/mine/3c03) | Crystal structure of the EscU C-terminal domain with P263A mutation,space group P 1 21 1 | 分子名称: | EscU, PROLINE | 著者 | Zarivach, R, Deng, W, Vuckovic, M, Felise, H.B, Nguyen, H.V, Miller, S.I, Finlay, B.B, Strynadka, N.C.J. | 登録日 | 2008-01-18 | 公開日 | 2008-04-22 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Structural analysis of the essential self-cleaving type III secretion proteins EscU and SpaS. Nature, 453, 2008
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3BZL
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![BU of 3bzl by Molmil](/molmil-images/mine/3bzl) | Crystal structural of native EscU C-terminal domain | 分子名称: | EscU, FORMIC ACID, SODIUM ION | 著者 | Zarivach, R, Deng, W, Vuckovic, M, Felise, H.B, Nguyen, H.V, Miller, S.I, Finlay, B.B, Strynadka, N.C.J. | 登録日 | 2008-01-18 | 公開日 | 2008-04-22 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (1.71 Å) | 主引用文献 | Structural analysis of the essential self-cleaving type III secretion proteins EscU and SpaS. Nature, 453, 2008
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3BZX
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![BU of 3bzx by Molmil](/molmil-images/mine/3bzx) | Crystal structure of the mutated H265A EscU C-terminal domain | 分子名称: | EscU, SULFATE ION | 著者 | Zarivach, R, Deng, W, Vuckovic, M, Felise, H.B, Nguyen, H.V, Miller, S.I, Finlay, B.B, Strynadka, N.C.J. | 登録日 | 2008-01-18 | 公開日 | 2008-04-22 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Structural analysis of the essential self-cleaving type III secretion proteins EscU and SpaS. Nature, 453, 2008
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3C01
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![BU of 3c01 by Molmil](/molmil-images/mine/3c01) | Crystal structural of native SpaS C-terminal domain | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, CYSTEINE, SULFATE ION, ... | 著者 | Zarivach, R, Deng, W, Vuckovic, M, Felise, H.B, Nguyen, H.V, Miller, S.I, Finlay, B.B, Strynadka, N.C.J. | 登録日 | 2008-01-18 | 公開日 | 2008-04-22 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Structural analysis of the essential self-cleaving type III secretion proteins EscU and SpaS. Nature, 453, 2008
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3BZZ
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![BU of 3bzz by Molmil](/molmil-images/mine/3bzz) | Crystal structural of the mutated R313T EscU/SpaS C-terminal domain | 分子名称: | EscU | 著者 | Zarivach, R, Deng, W, Vuckovic, M, Felise, H.B, Nguyen, H.V, Miller, S.I, Finlay, B.B, Strynadka, N.C.J. | 登録日 | 2008-01-18 | 公開日 | 2008-04-22 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (1.407 Å) | 主引用文献 | Structural analysis of the essential self-cleaving type III secretion proteins EscU and SpaS. Nature, 453, 2008
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5TO2
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![BU of 5to2 by Molmil](/molmil-images/mine/5to2) | |
7VKO
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![BU of 7vko by Molmil](/molmil-images/mine/7vko) | Crystal structure of TrkA kinase with repotrectinib | 分子名称: | Repotrectinib, SULFATE ION, Tyrosine-protein kinase receptor | 著者 | Murray, B.W, Rogers, E, Zhai, D, Deng, W, Chen, X, Sprengeler, P.A, Zhang, X, Graber, A, Reich, S.H, Stopatschinskaja, S, Solomon, B, Besse, B, Drilon, A. | 登録日 | 2021-09-30 | 公開日 | 2021-10-13 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | Molecular Characteristics of Repotrectinib That Enable Potent Inhibition of TRK Fusion Proteins and Resistant Mutations. Mol.Cancer Ther., 20, 2021
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7VKM
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![BU of 7vkm by Molmil](/molmil-images/mine/7vkm) | Crystal structure of TrkA (G595R) kinase domain | 分子名称: | Tyrosine-protein kinase receptor | 著者 | Murray, B.W, Rogers, E, Zhai, D, Deng, W, Chen, X, Sprengeler, P.A, Zhang, X, Graber, A, Reich, S.H, Stopatschinskaja, S, Solomon, B, Besse, B, Drilon, A. | 登録日 | 2021-09-30 | 公開日 | 2021-10-13 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.55 Å) | 主引用文献 | Molecular Characteristics of Repotrectinib That Enable Potent Inhibition of TRK Fusion Proteins and Resistant Mutations. Mol.Cancer Ther., 20, 2021
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7VKN
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![BU of 7vkn by Molmil](/molmil-images/mine/7vkn) | Crystal structure of TrkA (G595R) kinase with repotrectinib | 分子名称: | Repotrectinib, SULFATE ION, Tyrosine-protein kinase receptor | 著者 | Murray, B.W, Rogers, E, Zhai, D, Deng, W, Chen, X, Sprengeler, P.A, Zhang, X, Graber, A, Reich, S.H, Stopatschinskaja, S, Solomon, B, Besse, B, Drilon, A. | 登録日 | 2021-09-30 | 公開日 | 2021-10-13 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Molecular Characteristics of Repotrectinib That Enable Potent Inhibition of TRK Fusion Proteins and Resistant Mutations. Mol.Cancer Ther., 20, 2021
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7DTZ
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![BU of 7dtz by Molmil](/molmil-images/mine/7dtz) | FGFR4 complex with a covalent inhibitor | 分子名称: | Fibroblast growth factor receptor 4, N-[2-[[5-[[2,6-bis(chloranyl)-3,5-dimethoxy-phenyl]methoxy]pyrimidin-2-yl]amino]-3-methyl-phenyl]-2-fluoranyl-prop-2-enamide, SULFATE ION | 著者 | Chen, X.J, Dai, S.Y, Chen, Y.H. | 登録日 | 2021-01-07 | 公開日 | 2021-04-14 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.01 Å) | 主引用文献 | Investigation of Covalent Warheads in the Design of 2-Aminopyrimidine-based FGFR4 Inhibitors. Acs Med.Chem.Lett., 12, 2021
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