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1MUO
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BU of 1muo by Molmil
CRYSTAL STRUCTURE OF AURORA-2, AN ONCOGENIC SERINE-THREONINE KINASE
分子名称: ADENOSINE, Aurora-related kinase 1
著者Cheetham, G.M.T, Knegtel, R.M.A, Coll, J.T, Renwick, S.B, Swenson, L, Weber, P, Lippke, J.A, Austen, D.A.
登録日2002-09-24
公開日2003-04-15
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Crystal Structure of Aurora-2, an Oncogenic Serine/Threonine Kinase
J.Biol.Chem., 277, 2002
1QLN
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STRUCTURE OF A TRANSCRIBING T7 RNA POLYMERASE INITIATION COMPLEX
分子名称: BACTERIOPHAGE T7 RNA POLYMERASE, DNA (5- D (P*CP*TP*CP*CP*CP*TP*AP*TP*AP*GP*TP*GP*AP*GP*TP*CP*GP*TP* AP*TP*TP*A)-3), DNA (5-D(P*TP*AP*AP*TP*AP*CP*GP*AP*CP*TP*CP*AP*CP*TP*A)-3), ...
著者Cheetham, G.M.T, Steitz, T.A.
登録日1999-09-01
公開日2000-02-04
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Structure of a Transcribing T7 RNA Polymerase Initiation Complex
Science, 286, 1999
1BEY
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BU of 1bey by Molmil
ANTIBODY TO CAMPATH-1H HUMANIZED FAB
分子名称: CAMPATH-1H ANTIBODY
著者Cheetham, G.M.T, Hale, G, Waldmann, H, Bloomer, A.C.
登録日1998-05-18
公開日1999-01-27
最終更新日2023-08-02
実験手法X-RAY DIFFRACTION (3.25 Å)
主引用文献Crystal structures of a rat anti-CD52 (CAMPATH-1) therapeutic antibody Fab fragment and its humanized counterpart.
J.Mol.Biol., 284, 1998
1BFO
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BU of 1bfo by Molmil
CAMPATH-1G IGG2B RAT MONOCLONAL FAB
分子名称: CAMPATH-1G ANTIBODY
著者Cheetham, G.M.T, Hale, G, Waldmann, H, Bloomer, A.C.
登録日1998-05-20
公開日1999-03-16
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Crystal structures of a rat anti-CD52 (CAMPATH-1) therapeutic antibody Fab fragment and its humanized counterpart.
J.Mol.Biol., 284, 1998
1CEZ
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BU of 1cez by Molmil
CRYSTAL STRUCTURE OF A T7 RNA POLYMERASE-T7 PROMOTER COMPLEX
分子名称: DNA (5'-D(P*TP*AP*AP*TP*AP*CP*GP*AP*CP*TP*CP*AP*CP*TP*A)-3'), DNA (5'-D(P*TP*AP*TP*AP*GP*TP*GP*AP*GP*TP*CP*GP*TP*AP*TP*TP*A)-3'), PROTEIN (BACTERIOPHAGE T7 RNA POLYMERASE)
著者Cheetham, G.M.T, Jeruzalmi, D, Steitz, T.A.
登録日1999-03-11
公開日1999-05-21
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Structural basis for initiation of transcription from an RNA polymerase-promoter complex.
Nature, 399, 1999
3S2U
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BU of 3s2u by Molmil
Crystal structure of the Pseudomonas aeruginosa MurG:UDP-GlcNAc substrate complex
分子名称: UDP-N-acetylglucosamine--N-acetylmuramyl-(pentapeptide) pyrophosphoryl-undecaprenol N-acetylglucosamine transferase, URIDINE-DIPHOSPHATE-N-ACETYLGLUCOSAMINE
著者Brown, K, Vial, S.C.M, Dedi, N, Westcott, J, Scally, S, Bugg, T.D.H, Charlton, P.A, Cheetham, G.M.T.
登録日2011-05-17
公開日2012-09-26
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.23 Å)
主引用文献Crystal Structure of the Pseudomonas aeruginosa MurG: UDP-GlcNAc Substrate Complex.
Protein Pept.Lett., 20, 2013
1GNH
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BU of 1gnh by Molmil
HUMAN C-REACTIVE PROTEIN
分子名称: C-REACTIVE PROTEIN, CALCIUM ION
著者Shrive, A.K, Cheetham, G.M.T, Holden, D, Myles, D.A, Turnell, W.G, Volanakis, J.E, Pepys, M.B, Bloomer, A.C, Greenhough, T.J.
登録日1996-03-01
公開日1997-01-27
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Three dimensional structure of human C-reactive protein.
Nat.Struct.Biol., 3, 1996
1SNU
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BU of 1snu by Molmil
CRYSTAL STRUCTURE OF THE UNPHOSPHORYLATED INTERLEUKIN-2 TYROSINE KINASE CATALYTIC DOMAIN
分子名称: STAUROSPORINE, Tyrosine-protein kinase ITK/TSK
著者Brown, K, Long, J.M, Vial, S.C, Dedi, N, Dunster, N.J, Renwick, S.B, Tanner, A.J, Frantz, J.D, Fleming, M.A, Cheetham, G.M.T.
登録日2004-03-12
公開日2004-07-20
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Crystal structures of interleukin-2 tyrosine kinase and their implications for the design of selective inhibitors.
J.Biol.Chem., 279, 2004
1SM2
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BU of 1sm2 by Molmil
Crystal structure of the phosphorylated Interleukin-2 tyrosine kinase catalytic domain
分子名称: STAUROSPORINE, Tyrosine-protein kinase ITK/TSK
著者Brown, K, Long, J.M, Vial, S.C.M, Dedi, N, Dunster, N.J, Renwick, S.B, Tanner, A.J, Frantz, J.D, Fleming, M.A, Cheetham, G.M.T.
登録日2004-03-08
公開日2004-07-16
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Crystal structures of interleukin-2 tyrosine kinase and their implications for the design of selective inhibitors.
J.Biol.Chem., 279, 2004
1SNX
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CRYSTAL STRUCTURE OF APO INTERLEUKIN-2 TYROSINE KINASE CATALYTIC DOMAIN
分子名称: Tyrosine-protein kinase ITK/TSK
著者Brown, K, Long, J.M, Vial, S.C, Dedi, N, Dunster, N.J, Renwick, S.B, Tanner, A.J, Frantz, J.D, Fleming, M.A, Cheetham, G.M.T.
登録日2004-03-12
公開日2004-07-20
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Crystal structures of interleukin-2 tyrosine kinase and their implications for the design of selective inhibitors.
J.Biol.Chem., 279, 2004
3QGW
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BU of 3qgw by Molmil
Crystal Structure of ITK kinase bound to an inhibitor
分子名称: 3-[(8-phenylthieno[2,3-h]quinazolin-2-yl)amino]benzenesulfonamide, N-(6-oxo-1,6-dihydro-3,4'-bipyridin-5-yl)benzamide, Tyrosine-protein kinase ITK/TSK
著者Brown, K, Cheetham, G.M.T.
登録日2011-01-25
公開日2011-06-22
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Discovery and structure-activity relationship of 3-aminopyrid-2-ones as potent and selective interleukin-2 inducible T-cell kinase (Itk) inhibitors
J.Med.Chem., 54, 2011
3QGY
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Crystal structure of ITK inhibitor complex
分子名称: 3-[(8-phenylthieno[2,3-h]quinazolin-2-yl)amino]benzenesulfonamide, N-{5-[2-(methylamino)pyrimidin-4-yl]-2-oxo-1,2-dihydropyridin-3-yl}-4-(piperidin-1-yl)benzamide, Tyrosine-protein kinase ITK/TSK
著者Brown, K, Cheetham, G.M.T.
登録日2011-01-25
公開日2011-06-22
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Discovery and structure-activity relationship of 3-aminopyrid-2-ones as potent and selective interleukin-2 inducible T-cell kinase (Itk) inhibitors
J.Med.Chem., 54, 2011
1QTJ
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BU of 1qtj by Molmil
CRYSTAL STRUCTURE OF LIMULUS POLYPHEMUS SAP
分子名称: PROTEIN (SERUM AMYLOID P COMPONENT)
著者Shrive, A.K, Metcalfe, A.M, Cartwright, J.R, Greenhough, T.J.
登録日1999-06-28
公開日2000-06-28
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献C-reactive protein and SAP-like pentraxin are both present in Limulus polyphemus haemolymph: crystal structure of Limulus SAP.
J.Mol.Biol., 290, 1999

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