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3LOO
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BU of 3loo by Molmil
Crystal structure of Anopheles gambiae adenosine kinase in complex with P1,P4-di(adenosine-5) tetraphosphate
分子名称: Anopheles gambiae adenosine kinase, BIS(ADENOSINE)-5'-TETRAPHOSPHATE, CHLORIDE ION, ...
著者Ho, M.-C, Cassera, M.B, Almo, S.C, Schramm, V.L.
登録日2010-02-04
公開日2011-02-02
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献A High-Affinity Adenosine Kinase from Anopheles gambiae.
Biochemistry, 50, 2011
3EWC
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BU of 3ewc by Molmil
Crystal Structure of adenosine deaminase from Plasmodial vivax in complex with MT-coformycin
分子名称: (8R)-3-(5-S-methyl-5-thio-beta-D-ribofuranosyl)-3,6,7,8-tetrahydroimidazo[4,5-d][1,3]diazepin-8-ol, Adenosine deaminase, ZINC ION
著者Schramm, V.L, Almo, S.C, Cassera, M.B, Ho, M.C.
登録日2008-10-14
公開日2009-09-22
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.11 Å)
主引用文献Structural and metabolic specificity of methylthiocoformycin for malarial adenosine deaminases.
Biochemistry, 48, 2009
3EWD
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BU of 3ewd by Molmil
Crystal structure of adenosine deaminase mutant (delta Asp172) from Plasmodium vivax in complex with MT-coformycin
分子名称: (8R)-3-(5-S-methyl-5-thio-beta-D-ribofuranosyl)-3,6,7,8-tetrahydroimidazo[4,5-d][1,3]diazepin-8-ol, Adenosine deaminase, ZINC ION
著者Schramm, V.L, Almo, S.C, Cassera, M.B, Ho, M.C.
登録日2008-10-14
公開日2009-09-22
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Structural and metabolic specificity of methylthiocoformycin for malarial adenosine deaminases.
Biochemistry, 48, 2009
3PHB
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BU of 3phb by Molmil
Crystal Structure of human purine nucleoside phosphorylase in complex with DADMe-ImmG
分子名称: 2-amino-7-{[(3R,4R)-3-hydroxy-4-(hydroxymethyl)pyrrolidin-1-yl]methyl}-3,5-dihydro-4H-pyrrolo[3,2-d]pyrimidin-4-one, PHOSPHATE ION, Purine nucleoside phosphorylase
著者Ho, M, Cassera, M.B, Murkin, A.S, Almo, S.C, Schramm, V.L.
登録日2010-11-03
公開日2011-11-09
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Crystal Structure of human purine nucleoside phosphorylase in complex with DADMe-ImmG
to be published
3MB8
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BU of 3mb8 by Molmil
Crystal structure of purine nucleoside phosphorylase from toxoplasma gondii in complex with immucillin-H
分子名称: 1,4-DIDEOXY-4-AZA-1-(S)-(9-DEAZAHYPOXANTHIN-9-YL)-D-RIBITOL, GLYCEROL, PHOSPHATE ION, ...
著者Ho, M, Almo, S.C, Schramm, V.L.
登録日2010-03-25
公開日2011-04-06
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Inhibition and Structure of Toxoplasma gondii Purine Nucleoside Phosphorylase.
Eukaryot Cell, 13, 2014
2P4S
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BU of 2p4s by Molmil
Structure of Purine Nucleoside Phosphorylase from Anopheles gambiae in complex with DADMe-ImmH
分子名称: 7-[[(3R,4R)-3-(hydroxymethyl)-4-oxidanyl-pyrrolidin-1-ium-1-yl]methyl]-3,5-dihydropyrrolo[3,2-d]pyrimidin-4-one, PHOSPHATE ION, Purine nucleoside phosphorylase
著者Rinaldo-Matthis, A, Almo, S.C, Schramm, V.L.
登録日2007-03-13
公開日2008-01-15
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Anopheles gambiae purine nucleoside phosphorylase: catalysis, structure, and inhibition.
Biochemistry, 46, 2007
3OZG
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BU of 3ozg by Molmil
Crystal Structure of Plasmodium falciparum Hypoxanthine-Guanine-Xanthine Phosphoribosyltransferase in complex with S-SerMe-ImmH phosphonate
分子名称: Hypoxanthine-guanine-xanthine phosphoribosyltransferase, MAGNESIUM ION, PYROPHOSPHATE 2-, ...
著者Ho, M, Hazleton, K.Z, Almo, S.C, Schramm, V.L.
登録日2010-09-24
公開日2011-09-28
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.993 Å)
主引用文献Acyclic Immucillin Phosphonates: Second-Generation Inhibitors of Plasmodium falciparum Hypoxanthine- Guanine-Xanthine Phosphoribosyltransferase.
Chem.Biol., 19, 2012
3OZF
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Crystal Structure of Plasmodium falciparum Hypoxanthine-Guanine-Xanthine Phosphoribosyltransferase in complex with hypoxanthine
分子名称: HYPOXANTHINE, Hypoxanthine-guanine-xanthine phosphoribosyltransferase, MAGNESIUM ION, ...
著者Ho, M, Hazleton, K.Z, Almo, S.C, Schramm, V.L.
登録日2010-09-24
公開日2011-09-28
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.944 Å)
主引用文献Acyclic Immucillin Phosphonates: Second-Generation Inhibitors of Plasmodium falciparum Hypoxanthine- Guanine-Xanthine Phosphoribosyltransferase.
Chem.Biol., 19, 2012

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件を2024-09-18に公開中

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