5JOG
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![BU of 5jog by Molmil](/molmil-images/mine/5jog) | CRYSTAL STRUCTURE OF CSN5(2-257) IN COMPLEX WITH CNS5i-3 | 分子名称: | 3-(difluoromethyl)-N-{6-[(5S,6S)-6-hydroxy-6,7,8,9-tetrahydro-5H-imidazo[1,5-a]azepin-5-yl][1,1'-biphenyl]-3-yl}-1-(propan-2-yl)-1H-pyrazole-5-carboxamide, COP9 signalosome complex subunit 5, ZINC ION | 著者 | Renatus, M, Wiesmann, C. | 登録日 | 2016-05-02 | 公開日 | 2016-11-02 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.46 Å) | 主引用文献 | Targeted inhibition of the COP9 signalosome for treatment of cancer. Nat Commun, 7, 2016
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4WAS
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![BU of 4was by Molmil](/molmil-images/mine/4was) | STRUCTURE OF THE ETR1P/NADP/CROTONYL-COA COMPLEX | 分子名称: | CROTONYL COENZYME A, Enoyl-[acyl-carrier-protein] reductase [NADPH, B-specific] 1, ... | 著者 | Quade, N, Voegeli, B, Rosenthal, R, Capitani, G, Erb, T.J. | 登録日 | 2014-08-31 | 公開日 | 2015-03-18 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | The use of ene adducts to study and engineer enoyl-thioester reductases. Nat.Chem.Biol., 11, 2015
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5C37
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![BU of 5c37 by Molmil](/molmil-images/mine/5c37) | Structure of the beta-ketoacyl reductase domain of human fatty acid synthase bound to a spiro-imidazolone inhibitor | 分子名称: | 6-{[(3R)-1-(cyclopropylcarbonyl)pyrrolidin-3-yl]methyl}-5-[4-(1-methyl-1H-indazol-5-yl)phenyl]-4,6-diazaspiro[2.4]hept-4-en-7-one, CHLORIDE ION, Fatty acid synthase, ... | 著者 | Schubert, C, Milligan, C.M, Vo, K, Grasberger, B. | 登録日 | 2015-06-17 | 公開日 | 2016-06-22 | 最終更新日 | 2024-06-19 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Design and synthesis of a series of bioavailable fatty acid synthase (FASN) KR domain inhibitors for cancer therapy. Bioorg.Med.Chem.Lett., 28, 2018
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3S2Q
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![BU of 3s2q by Molmil](/molmil-images/mine/3s2q) | The crystal structure of AT5g51720 (AT-NEET) | 分子名称: | AT5g51720/MIO24_14, FE2/S2 (INORGANIC) CLUSTER, ZINC ION | 著者 | Livnah, O, Eisenberg-Domovich, Y, Nechushtai, R. | 登録日 | 2011-05-17 | 公開日 | 2012-05-23 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | Arabidopsis thaliana ChloroNEET, a Member of the New NEET Family of Human Proteins, is Involved in Development, Senescence and Iron Metabolism. To be Published
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6GS0
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![BU of 6gs0 by Molmil](/molmil-images/mine/6gs0) | Native Glucuronoyl Esterase from Opitutus terrae | 分子名称: | 1,2-ETHANEDIOL, MAGNESIUM ION, Putative acetyl xylan esterase, ... | 著者 | Lo Leggio, L, Larsbrink, J, Meland Knudsen, R, Mazurkewich, S, Navarro Poulsen, J.C. | 登録日 | 2018-06-13 | 公開日 | 2018-08-22 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (1.34 Å) | 主引用文献 | Biochemical and structural features of diverse bacterial glucuronoyl esterases facilitating recalcitrant biomass conversion. Biotechnol Biofuels, 11, 2018
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6GRY
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![BU of 6gry by Molmil](/molmil-images/mine/6gry) | Glucuronoyl Esterase from Solibacter usitatus. | 分子名称: | 1,2-ETHANEDIOL, DI(HYDROXYETHYL)ETHER, Putative acetyl xylan esterase, ... | 著者 | Lo Leggio, L, Larsbrink, J, Meland Knudsen, R, Mazurkewich, S, Navarro Poulsen, J.C. | 登録日 | 2018-06-12 | 公開日 | 2018-08-15 | 最終更新日 | 2024-05-01 | 実験手法 | X-RAY DIFFRACTION (2.0003376 Å) | 主引用文献 | Biochemical and structural features of diverse bacterial glucuronoyl esterases facilitating recalcitrant biomass conversion. Biotechnol Biofuels, 11, 2018
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6GU8
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![BU of 6gu8 by Molmil](/molmil-images/mine/6gu8) | Glucuronoyl Esterase from Solibacter usitatus | 分子名称: | 1,2-ETHANEDIOL, DI(HYDROXYETHYL)ETHER, Putative acetyl xylan esterase | 著者 | Lo Leggio, L, Larsbrink, J, Meland Knudsen, R, Mazurkewich, S, Navarro Poulsen, J.C. | 登録日 | 2018-06-19 | 公開日 | 2018-08-15 | 実験手法 | X-RAY DIFFRACTION (2.01807833 Å) | 主引用文献 | Biochemical and structural features of diverse bacterial glucuronoyl esterases facilitating recalcitrant biomass conversion. Biotechnol Biofuels, 11, 2018
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6GRW
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![BU of 6grw by Molmil](/molmil-images/mine/6grw) | Glucuronoyl Esterase from Opitutus terrae (Au derivative) | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, 1,2-ETHANEDIOL, CALCIUM ION, ... | 著者 | Lo Leggio, L, Larsbrink, J, Meland Knudsen, R, Mazurkewich, S, Navarro Poulsen, J.C. | 登録日 | 2018-06-12 | 公開日 | 2018-08-15 | 最終更新日 | 2024-05-01 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Biochemical and structural features of diverse bacterial glucuronoyl esterases facilitating recalcitrant biomass conversion. Biotechnol Biofuels, 11, 2018
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6WTU
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6WN1
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6WQO
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6WNO
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6WOZ
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6WTY
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6WTV
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5WHZ
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![BU of 5whz by Molmil](/molmil-images/mine/5whz) | PGDM1400-10E8v4 CODV Fab | 分子名称: | Anti-HIV CODV-Fab Heavy chain, Anti-HIV CODV-Fab Light chain | 著者 | Lord, D.M, Wei, R.R. | 登録日 | 2017-07-18 | 公開日 | 2017-10-11 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (3.549 Å) | 主引用文献 | Trispecific broadly neutralizing HIV antibodies mediate potent SHIV protection in macaques. Science, 358, 2017
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6WM9
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5Y27
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![BU of 5y27 by Molmil](/molmil-images/mine/5y27) | Crystal structure of Se-Met Dpb4-Dpb3 | 分子名称: | DNA polymerase epsilon subunit D, GLYCEROL, Putative transcription factor C16C4.22 | 著者 | Li, Y, Gao, F, Su, M, Zhang, F.B, Chen, Y.H. | 登録日 | 2017-07-24 | 公開日 | 2018-01-24 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Coordinated regulation of heterochromatin inheritance by Dpb3-Dpb4 complex. Proc. Natl. Acad. Sci. U.S.A., 114, 2017
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5Y26
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![BU of 5y26 by Molmil](/molmil-images/mine/5y26) | Crystal structure of native Dpb4-Dpb3 | 分子名称: | DNA polymerase epsilon subunit D, GLYCEROL, Putative transcription factor C16C4.22 | 著者 | Chen, Y.H, Li, Y, Gao, F. | 登録日 | 2017-07-24 | 公開日 | 2018-01-24 | 最終更新日 | 2024-03-27 | 実験手法 | X-RAY DIFFRACTION (2.003 Å) | 主引用文献 | Coordinated regulation of heterochromatin inheritance by Dpb3-Dpb4 complex. Proc. Natl. Acad. Sci. U.S.A., 114, 2017
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4HVH
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4HVI
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4HVG
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4HVD
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![BU of 4hvd by Molmil](/molmil-images/mine/4hvd) | JAK3 kinase domain in complex with 2-Cyclopropyl-5H-pyrrolo[2,3-b]pyrazine-7-carboxylic acid ((S)-1,2,2-trimethyl-propyl)-amide | 分子名称: | 1-phenylurea, 2-cyclopropyl-N-[(2S)-3,3-dimethylbutan-2-yl]-5H-pyrrolo[2,3-b]pyrazine-7-carboxamide, Tyrosine-protein kinase JAK3 | 著者 | Kuglstatter, A, Shao, A. | 登録日 | 2012-11-06 | 公開日 | 2013-01-16 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | 3-Amido Pyrrolopyrazine JAK Kinase Inhibitors: Development of a JAK3 vs JAK1 Selective Inhibitor and Evaluation in Cellular and in Vivo Models. J.Med.Chem., 56, 2013
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8TNS
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6UF2
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