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7WF9
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BU of 7wf9 by Molmil
Crystal structure of mouse SNX25 RGS domain in space group P41212
分子名称: Sorting nexin-25
著者Zhang, Y, Xu, J, Liu, J.
登録日2021-12-26
公開日2022-10-26
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.55 Å)
主引用文献Structural Studies Reveal Unique Non-canonical Regulators of G Protein Signaling Homology (RH) Domains in Sorting Nexins.
J.Mol.Biol., 434, 2022
7WF6
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BU of 7wf6 by Molmil
Crystal structure of SNX13 RGS domain
分子名称: CHLORIDE ION, Sorting nexin-13
著者Xu, J, Zhu, J, Liu, J.
登録日2021-12-26
公開日2022-10-26
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (3.25 Å)
主引用文献Structural Studies Reveal Unique Non-canonical Regulators of G Protein Signaling Homology (RH) Domains in Sorting Nexins.
J.Mol.Biol., 434, 2022
1AI3
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BU of 1ai3 by Molmil
ORBITAL STEERING IN THE CATALYTIC POWER OF ENZYMES: SMALL STRUCTURAL CHANGES WITH LARGE CATALYTIC CONSEQUENCES
分子名称: ISOCITRATE DEHYDROGENASE, ISOCITRIC ACID, MAGNESIUM ION, ...
著者Stoddard, B.L, Mesecar, A, Koshland Junior, D.E.
登録日1997-04-30
公開日1997-11-12
最終更新日2023-08-02
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Orbital steering in the catalytic power of enzymes: small structural changes with large catalytic consequences.
Science, 277, 1997
1AI2
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BU of 1ai2 by Molmil
ISOCITRATE DEHYDROGENASE COMPLEXED WITH ISOCITRATE, NADP+, AND CALCIUM (FLASH-COOLED)
分子名称: ISOCITRATE CALCIUM COMPLEX, ISOCITRATE DEHYDROGENASE, NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE
著者Stoddard, B.L, Mesecar, A, Koshland Junior, D.E.
登録日1997-04-30
公開日1997-10-15
最終更新日2023-08-02
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Orbital steering in the catalytic power of enzymes: small structural changes with large catalytic consequences.
Science, 277, 1997
5Z02
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BU of 5z02 by Molmil
Crystal structure of HIS6-tagged Mdm2 with nutlin-3a
分子名称: 4-({(4S,5R)-4,5-bis(4-chlorophenyl)-2-[4-methoxy-2-(propan-2-yloxy)phenyl]-4,5-dihydro-1H-imidazol-1-yl}carbonyl)piperazin-2-one, E3 ubiquitin-protein ligase Mdm2
著者Su, Z.D, Cheng, X.Y, Chen, R, Pi, N.
登録日2017-12-18
公開日2018-01-03
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (1.35 Å)
主引用文献Crystal structure of HIS6-tagged Mdm2 with nutlin-3a
to be published
5ZXF
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BU of 5zxf by Molmil
The 1.25A Crystal structure of His6-tagged Mdm2 in complex with nutlin-3a
分子名称: 4-({(4S,5R)-4,5-bis(4-chlorophenyl)-2-[4-methoxy-2-(propan-2-yloxy)phenyl]-4,5-dihydro-1H-imidazol-1-yl}carbonyl)piperazin-2-one, E3 ubiquitin-protein ligase Mdm2
著者Cheng, X.Y, Su, Z.D, Pi, N, Cao, C.Z, Zhao, Z.T, Zhou, J.J, Chen, R, Kuang, Z.K, Huang, Y.Q.
登録日2018-05-19
公開日2018-08-22
最終更新日2024-03-27
実験手法X-RAY DIFFRACTION (1.25 Å)
主引用文献The 1.25A Crystal structure of His6-tagged Mdm2 in complex with nutlin-3a
To Be Published
3NDM
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BU of 3ndm by Molmil
Crystal structure of Rho-Associated Protein Kinase (ROCK1) with a potent isoquinolone derivative
分子名称: (3S,4R)-N-(7-chloro-1-oxo-1,4-dihydroisoquinolin-6-yl)-4-(4-chlorophenyl)pyrrolidine-3-carboxamide, Rho-Associated Protein Kinase (ROCK1)
著者Li, X.
登録日2010-06-07
公開日2010-12-08
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (3.3 Å)
主引用文献Substituted 2H-isoquinolin-1-ones as potent Rho-kinase inhibitors: part 3, aryl substituted pyrrolidines.
Bioorg.Med.Chem.Lett., 20, 2010

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件を2024-06-12に公開中

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