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2VHH
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Crystal structure of a pyrimidine degrading enzyme from Drosophila melanogaster
分子名称: CG3027-PA
著者Lundgren, S, Lohkamp, B, Andersen, B, Piskur, J, Dobritzsch, D.
登録日2007-11-21
公開日2008-03-25
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献The Crystal Structure of Beta-Alanine Synthase from Drosophila Melanogaster Reveals a Homooctameric Helical Turn-Like Assembly.
J.Mol.Biol., 377, 2008
2VP5
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Structural Studies of Nucleoside Analog and Feedback Inhibitor Binding to Drosophila Melanogaster Multisubstrate Deoxyribonucleoside Kinase
分子名称: 2'-DEOXYCYTIDINE, DEOXYNUCLEOSIDE KINASE, SULFATE ION
著者Mikkelsen, N.E, Munch-Petersen, B, Eklund, H.
登録日2008-02-26
公開日2008-04-18
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Structural Studies of Nucleoside Analog and Feedback Inhibitor Binding to Drosophila Melanogaster Multisubstrate Deoxyribonucleoside Kinase.
FEBS J., 275, 2008
2VP2
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Structural Studies of Nucleoside Analog and Feedback Inhibitor Binding to Drosophila Melanogaster Multisubstrate Deoxyribonucleoside Kinase
分子名称: 2'-DEOXYGUANOSINE-5'-TRIPHOSPHATE, DEOXYNUCLEOSIDE KINASE
著者Mikkelsen, N.E, Munch-Petersen, B, Eklund, H.
登録日2008-02-26
公開日2008-04-29
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Structural Studies of Nucleoside Analog and Feedback Inhibitor Binding to Drosophila Melanogaster Multisubstrate Deoxyribonucleoside Kinase.
FEBS J., 275, 2008
2VHI
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Crystal structure of a pyrimidine degrading enzyme from Drosophila melanogaster
分子名称: CG3027-PA
著者Lundgren, S, Lohkamp, B, Andersen, B, Piskur, J, Dobritzsch, D.
登録日2007-11-21
公開日2008-03-25
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (3.3 Å)
主引用文献The Crystal Structure of Beta-Alanine Synthase from Drosophila Melanogaster Reveals a Homooctameric Helical Turn-Like Assembly.
J.Mol.Biol., 377, 2008
2UZ3
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Crystal Structure of Thymidine Kinase with dTTP from U. urealyticum
分子名称: MAGNESIUM ION, THYMIDINE KINASE, THYMIDINE-5'-TRIPHOSPHATE, ...
著者Welin, M, Kosinska, U, Mikkelsen, N.E, Carnrot, C, Zhu, C, Wang, L, Eriksson, S, Munch-Petersen, B, Eklund, H.
登録日2007-04-24
公開日2007-05-29
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Structures of Thymidine Kinase 1 of Human and Mycoplasmic Origin
Proc.Natl.Acad.Sci.USA, 101, 2004
1J90
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Crystal Structure of Drosophila Deoxyribonucleoside Kinase
分子名称: 2'-DEOXYCYTIDINE, Deoxyribonucleoside kinase, SULFATE ION
著者Johansson, K, Ramaswamy, S, Ljungkrantz, C, Knecht, W, Piskur, J, Munch-Petersen, B, Eriksson, S, Eklund, H.
登録日2001-05-23
公開日2001-11-28
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.56 Å)
主引用文献Structural basis for substrate specificities of cellular deoxyribonucleoside kinases.
Nat.Struct.Biol., 8, 2001
1S5O
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Structural and Mutational Characterization of L-carnitine Binding to Human carnitine Acetyltransferase
分子名称: CARNITINE, carnitine acetyltransferase isoform 2
著者Govindasamy, L, Kukar, T, Lian, W, Pedersen, B, Gu, Y, Agbandje-Mckenna, M, Jin, S, Mckenna, R, Wu, D.
登録日2004-01-21
公開日2004-02-03
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Structural and mutational characterization of l-carnitine binding to human carnitine acetyltransferase.
J.Struct.Biol., 146, 2004
2V8G
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Crystal structure of beta-alanine synthase from Saccharomyces kluyveri in complex with the product beta-alanine
分子名称: BETA-ALANINE, BETA-ALANINE SYNTHASE, BICINE, ...
著者Lundgren, S, Andersen, B, Piskur, J, Dobritzsch, D.
登録日2007-08-07
公開日2007-10-02
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Crystal Structures of Yeast -Alanine Synthase Complexes Reveal the Mode of Substrate Binding and Large Scale Domain Closure Movements.
J.Biol.Chem., 282, 2007
2V8V
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Crystal structure of mutant R322A of beta-alanine synthase from Saccharomyces kluyveri
分子名称: 2,3-DIHYDROXY-1,4-DITHIOBUTANE, BETA-ALANINE SYNTHASE, N-(AMINOCARBONYL)-BETA-ALANINE, ...
著者Lundgren, S, Andersen, B, Piskur, J, Dobritzsch, D.
登録日2007-08-15
公開日2007-10-02
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Crystal Structures of Yeast -Alanine Synthase Complexes Reveal the Mode of Substrate Binding and Large Scale Domain Closure Movements.
J.Biol.Chem., 282, 2007
2V8D
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Crystal structure of mutant E159A of beta-alanine synthase from Saccharomyces kluyveri
分子名称: BETA-ALANINE SYNTHASE, ZINC ION
著者Lundgren, S, Andersen, B, Piskur, J, Dobritzsch, D.
登録日2007-08-07
公開日2007-10-02
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Crystal Structures of Yeast -Alanine Synthase Complexes Reveal the Mode of Substrate Binding and Large Scale Domain Closure Movements.
J.Biol.Chem., 282, 2007
2V8H
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BU of 2v8h by Molmil
Crystal structure of mutant E159A of beta-alanine synthase from Saccharomyces kluyveri in complex with its substrate N-carbamyl-beta- alanine
分子名称: BETA-ALANINE SYNTHASE, BICINE, N-(AMINOCARBONYL)-BETA-ALANINE, ...
著者Lundgren, S, Andersen, B, Piskur, J, Dobritzsch, D.
登録日2007-08-08
公開日2007-10-02
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Crystal Structures of Yeast -Alanine Synthase Complexes Reveal the Mode of Substrate Binding and Large Scale Domain Closure Movements.
J.Biol.Chem., 282, 2007
2WVJ
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BU of 2wvj by Molmil
Mutation of Thr163 to Ser in Human Thymidine Kinase Shifts the Specificity from Thymidine towards the Nucleoside Analogue Azidothymidine
分子名称: MAGNESIUM ION, THYMIDINE KINASE, CYTOSOLIC, ...
著者Skovgaard, T, Uhlin, U, Munch-Petersen, B.
登録日2009-10-17
公開日2009-10-27
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Comparative Active-Site Mutation Study of Human and Caenorhabditis Elegans Thymidine Kinase 1.
FEBS J., 279, 2012
1T1U
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BU of 1t1u by Molmil
Structural Insights and Functional Implications of Choline Acetyltransferase
分子名称: Choline O-acetyltransferase
著者Govindasamy, L, Pedersen, B, Lian, W, Kukar, T, Gu, Y, Jin, S, Agbandje-McKenna, M, Wu, D.
登録日2004-04-18
公開日2005-04-12
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (1.55 Å)
主引用文献Structural insights and functional implications of choline acetyltransferase
J.Struct.Biol., 148, 2004
1ELA
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BU of 1ela by Molmil
Analogous inhibitors of elastase do not always bind analogously
分子名称: 6-ammonio-N-(trifluoroacetyl)-L-norleucyl-N-[4-(1-methylethyl)phenyl]-L-prolinamide, ACETIC ACID, CALCIUM ION, ...
著者Mattos, C, Rasmussen, B, Ding, X, Petsko, G.A, Ringe, D.
登録日1993-12-07
公開日1994-04-30
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Analogous inhibitors of elastase do not always bind analogously.
Nat.Struct.Biol., 1, 1994
1ELB
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BU of 1elb by Molmil
Analogous inhibitors of elastase do not always bind analogously
分子名称: 6-ammonio-N-(trifluoroacetyl)-L-norleucyl-N-[4-(1-methylethyl)phenyl]-L-leucinamide, CALCIUM ION, ELASTASE, ...
著者Mattos, C, Rasmussen, B, Ding, X, Petsko, G.A, Ringe, D.
登録日1993-12-07
公開日1994-06-22
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Analogous inhibitors of elastase do not always bind analogously.
Nat.Struct.Biol., 1, 1994
1KJ3
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BU of 1kj3 by Molmil
Mhc Class I H-2Kb molecule complexed with pKB1 peptide
分子名称: BETA-2 MICROGLOBULIN, H-2KB MHC CLASS I MOLECULE ALPHA CHAIN, NATURALLY PROCESSED OCTAPEPTIDE PKB1
著者Reiser, J.-B, Gregoire, C, Darnault, C, Mosser, T, Guimezanes, A, Schmitt-Verhulst, A.-M, Fontecilla-Camps, J.C, Mazza, G, Malissen, B, Housset, D.
登録日2001-12-04
公開日2002-03-27
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献A T cell receptor CDR3beta loop undergoes conformational changes of unprecedented magnitude upon binding to a peptide/MHC class I complex.
Immunity, 16, 2002
1DUX
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BU of 1dux by Molmil
ELK-1/DNA STRUCTURE REVEALS HOW RESIDUES DISTAL FROM DNA-BINDING SURFACE AFFECT DNA-RECOGNITION
分子名称: DNA (5'-D(*AP*CP*AP*CP*TP*TP*CP*CP*GP*GP*TP*CP*A)-3'), DNA (5'-D(*TP*GP*AP*CP*CP*GP*GP*AP*AP*GP*TP*GP*T)-3'), ETS-DOMAIN PROTEIN ELK-1
著者Mo, Y, Vaessen, B, Johnston, K, Marmorstein, R.
登録日2000-01-19
公開日2000-04-17
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Structure of the elk-1-DNA complex reveals how DNA-distal residues affect ETS domain recognition of DNA.
Nat.Struct.Biol., 7, 2000
1ELC
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BU of 1elc by Molmil
Analogous inhibitors of elastase do not always bind analogously
分子名称: 6-ammonio-N-(trifluoroacetyl)-L-norleucyl-N-[4-(1-methylethyl)phenyl]-L-phenylalaninamide, CALCIUM ION, ELASTASE
著者Mattos, C, Rasmussen, B, Ding, X, Petsko, G.A, Ringe, D.
登録日1993-12-07
公開日1994-04-30
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Analogous inhibitors of elastase do not always bind analogously.
Nat.Struct.Biol., 1, 1994
1FU5
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NMR STRUCTURE OF THE N-SH2 DOMAIN OF THE P85 SUBUNIT OF PI3-KINASE COMPLEXED TO A DOUBLY PHOSPHORYLATED PEPTIDE DERIVED FROM POLYOMAVIRUS MIDDLE T ANTIGEN
分子名称: DOUBLY PHOSPHORYLATED MIDDLE T ANTIGEN, PHOSPHATIDYLINOSITOL 3-KINASE REGULATORY ALPHA SUBUNIT
著者Weber, T, Schaffhausen, B, Liu, Y, Guenther, U.L.
登録日2000-09-14
公開日2001-02-21
最終更新日2022-02-23
実験手法SOLUTION NMR
主引用文献NMR structure of the N-SH2 of the p85 subunit of phosphoinositide 3-kinase complexed to a doubly phosphorylated peptide reveals a second phosphotyrosine binding site.
Biochemistry, 39, 2000
1FU6
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NMR STRUCTURE OF THE N-SH2 DOMAIN OF THE P85 SUBUNIT OF PI3-KINASE
分子名称: PHOSPHATIDYLINOSITOL 3-KINASE REGULATORY ALPHA SUBUNIT
著者Weber, T, Schaffhausen, B, Liu, Y, Guenther, U.L.
登録日2000-09-14
公開日2001-02-21
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献NMR structure of the N-SH2 of the p85 subunit of phosphoinositide 3-kinase complexed to a doubly phosphorylated peptide reveals a second phosphotyrosine binding site.
Biochemistry, 39, 2000
1HRV
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BU of 1hrv by Molmil
HRV14/SDZ 35-682 COMPLEX
分子名称: 1-[2-HYDROXY-3-(4-CYCLOHEXYL-PHENOXY)-PROPYL]-4-(2-PYRIDYL)-PIPERAZINE, HUMAN RHINOVIRUS 14 COAT PROTEIN (SUBUNIT VP1), HUMAN RHINOVIRUS 14 COAT PROTEIN (SUBUNIT VP2), ...
著者Oren, D.A, Zhang, A, Arnold, E.
登録日1995-03-02
公開日1995-06-03
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献SDZ 35-682, a new picornavirus capsid-binding agent with potent antiviral activity.
Antiviral Res., 26, 1995
6L2B
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BU of 6l2b by Molmil
Crystal structure of cyclophilin mutant I164M from Leishmania donovani at 2.65 angstrom resolution
分子名称: Peptidyl-prolyl cis-trans isomerase
著者Ghosh, S, Biswas, G, Datta, A.K, Banerjee, R.
登録日2019-10-03
公開日2019-10-23
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.65 Å)
主引用文献Crystal structure of cyclophilin mutant I164M from Leishmania donovani at 2.65 angstrom resolution.
To Be Published
2FVM
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Crystal structure of dihydropyrimidinase from Saccharomyces kluyveri in complex with the reaction product N-carbamyl-beta-alanine
分子名称: N-(AMINOCARBONYL)-BETA-ALANINE, ZINC ION, dihydropyrimidinase
著者Dobritzsch, D, Lohkamp, B.
登録日2006-01-31
公開日2006-03-14
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.45 Å)
主引用文献The Crystal Structures of Dihydropyrimidinases Reaffirm the Close Relationship between Cyclic Amidohydrolases and Explain Their Substrate Specificity.
J.Biol.Chem., 281, 2006
4O5Q
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Crystal Structure of the Alkylhydroperoxide Reductase AhpF from Escherichia coli
分子名称: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Alkyl hydroperoxide reductase subunit F, CADMIUM ION, ...
著者Dip, P.V, Kamariah, N, Manimekalai, M.S.S, Balakrishna, A.M, Gruber, G.
登録日2013-12-20
公開日2014-11-05
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structure, mechanism and ensemble formation of the alkylhydroperoxide reductase subunits AhpC and AhpF from Escherichia coli
Acta Crystallogr.,Sect.D, 70, 2014
1VRH
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HRV14/SDZ 880-061 COMPLEX
分子名称: 2-[4-(2H-1,4-BENZOTHIAZINE-3-YL)-PIPERAZINE-1-LY]-1,3-THIAZOLE-4-CARBOXYLIC ACID ETHYLESTER, RHINOVIRUS 14
著者Oren, D.A, Zhang, A, Arnold, E.
登録日1996-02-26
公開日1997-02-12
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Synthesis and activity of piperazine-containing antirhinoviral agents and crystal structure of SDZ 880-061 bound to human rhinovirus 14.
J.Mol.Biol., 259, 1996

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