1RZU
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![BU of 1rzu by Molmil](/molmil-images/mine/1rzu) | Crystal structure of the glycogen synthase from A. tumefaciens in complex with ADP | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, Glycogen synthase 1 | 著者 | Buschiazzo, A, Guerin, M.E, Ugalde, J.E, Ugalde, R.A, Shepard, W, Alzari, P.M. | 登録日 | 2003-12-29 | 公開日 | 2004-08-31 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Crystal structure of glycogen synthase: homologous enzymes catalyze glycogen synthesis and degradation. Embo J., 23, 2004
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6V54
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![BU of 6v54 by Molmil](/molmil-images/mine/6v54) | Crystal Structure of Metallo Beta Lactamase from Hirschia baltica | 分子名称: | 1,2-ETHANEDIOL, Beta-lactamase, CHLORIDE ION, ... | 著者 | Maltseva, N, Kim, Y, Clancy, S, Endres, M, Mulligan, R, Joachimiak, A, Center for Structural Genomics of Infectious Diseases (CSGID) | 登録日 | 2019-12-03 | 公開日 | 2019-12-25 | 実験手法 | X-RAY DIFFRACTION (1.45 Å) | 主引用文献 | Crystal Structure of Metallo Beta Lactamase from Hirschia baltica. To Be Published
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6V6N
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![BU of 6v6n by Molmil](/molmil-images/mine/6v6n) | The crystal structure of a class D beta-lactamase from Agrobacterium tumefaciens | 分子名称: | Beta-lactamase, FORMIC ACID, GLYCEROL, ... | 著者 | Tan, K, Wu, R, Endres, M, Joachimiak, A, Center for Structural Genomics of Infectious Diseases (CSGID) | 登録日 | 2019-12-05 | 公開日 | 2019-12-18 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | The crystal structure of a class D beta-lactamase from Agrobacterium tumefaciens To Be Published
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6V80
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7SWI
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![BU of 7swi by Molmil](/molmil-images/mine/7swi) | cTnC-TnI chimera complexed with A2 | 分子名称: | 4-(3-cyano-3-methylazetidine-1-carbonyl)-N-[(3R,4S)-7-fluoro-4-hydroxy-6-methyl-3,4-dihydro-2H-1-benzopyran-3-yl]-5-methyl-1H-pyrrole-2-sulfonamide, Troponin C, slow skeletal and cardiac muscles,Troponin I, ... | 著者 | Poppe, L, Hartman, J.J, Romero, A, Reagan, J.D. | 登録日 | 2021-11-19 | 公開日 | 2022-04-06 | 最終更新日 | 2024-05-15 | 実験手法 | SOLUTION NMR | 主引用文献 | Structural and Thermodynamic Model for the Activation of Cardiac Troponin. Biochemistry, 61, 2022
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6V7J
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![BU of 6v7j by Molmil](/molmil-images/mine/6v7j) | The C2221 crystal form of canavalin at 173 K | 分子名称: | BENZOIC ACID, CALCIUM ION, Canavalin, ... | 著者 | McPherson, A. | 登録日 | 2019-12-08 | 公開日 | 2020-02-19 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Binding of benzoic acid and anions within the cupin domains of the vicilin protein canavalin from jack bean (Canavalia ensiformis): Crystal structures. Biochem.Biophys.Res.Commun., 524, 2020
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7TFP
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![BU of 7tfp by Molmil](/molmil-images/mine/7tfp) | Human Ornithine Aminotransferase cocrystallized with its inhibitor, (1S,3S)-3-amino-4-(difluoromethylene)cyclopentane-1-carboxylic acid. | 分子名称: | (1S,3S,4S)-3-amino-4-(fluoromethyl)cyclopentane-1-carboxylic acid, Ornithine aminotransferase, mitochondrial, ... | 著者 | Butrin, A, Zhu, W, Silverman, R, Liu, D. | 登録日 | 2022-01-06 | 公開日 | 2022-04-06 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.71 Å) | 主引用文献 | Rational Design, Synthesis, and Mechanism of (3 S ,4 R )-3-Amino-4-(difluoromethyl)cyclopent-1-ene-1-carboxylic Acid: Employing a Second-Deprotonation Strategy for Selectivity of Human Ornithine Aminotransferase over GABA Aminotransferase. J.Am.Chem.Soc., 144, 2022
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6V8D
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![BU of 6v8d by Molmil](/molmil-images/mine/6v8d) | Design, Synthesis, and Mechanism of Fluorine-substituted Cyclohexene Analogues of GAMA-Aminobutyric Acid (GABA) as Selective Ornithine Aminotransferase Inactivators | 分子名称: | (3Z)-3-iminocyclohex-1-ene-1-carboxylic acid, Ornithine aminotransferase, mitochondrial, ... | 著者 | Zhu, W, Doubleday, P.T, Catlin, D.S, Weerawarna, P, Butrin, A, Shen, S, Kelleher, N.L, Liu, D, Silverman, R.B. | 登録日 | 2019-12-10 | 公開日 | 2020-12-16 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (2.25 Å) | 主引用文献 | Design, Synthesis, and Mechanism of Fluorine-substituted Cyclohexene Analogues of GAMA-Aminobutyric Acid (GABA) as Selective Ornithine Aminotransferase Inactivators To Be Published
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7TEV
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![BU of 7tev by Molmil](/molmil-images/mine/7tev) | Human Ornithine Aminotransferase cocrystallized with its inhibitor, (3S,4R)-3-amino-4-(difluoromethyl)cyclopent-1-ene-1-carboxylate | 分子名称: | (1S,3R,4S)-3-formyl-4-[({3-hydroxy-2-methyl-5-[(phosphonooxy)methyl]pyridin-4-yl}methyl)amino]cyclopentane-1-carboxylic acid, Ornithine aminotransferase, mitochondrial | 著者 | Butrin, A, Zhu, W, Silverman, R, Liu, D. | 登録日 | 2022-01-05 | 公開日 | 2022-04-06 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.91 Å) | 主引用文献 | Rational Design, Synthesis, and Mechanism of (3 S ,4 R )-3-Amino-4-(difluoromethyl)cyclopent-1-ene-1-carboxylic Acid: Employing a Second-Deprotonation Strategy for Selectivity of Human Ornithine Aminotransferase over GABA Aminotransferase. J.Am.Chem.Soc., 144, 2022
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7SUP
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![BU of 7sup by Molmil](/molmil-images/mine/7sup) | NMR structure of cTnC-TnI chimera bound to calcium and A1 | 分子名称: | 4-(3-cyano-3-methylazetidine-1-carbonyl)-N-[(3S)-7-fluoro-6-methyl-3,4-dihydro-2H-1-benzopyran-3-yl]-5-methyl-1H-pyrrole-2-sulfonamide, CALCIUM ION, Troponin C, ... | 著者 | Poppe, L, Hartman, J.J, Romero, A, Reagan, J.D. | 登録日 | 2021-11-17 | 公開日 | 2022-04-06 | 最終更新日 | 2024-05-15 | 実験手法 | SOLUTION NMR | 主引用文献 | Structural and Thermodynamic Model for the Activation of Cardiac Troponin. Biochemistry, 61, 2022
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7SVC
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![BU of 7svc by Molmil](/molmil-images/mine/7svc) | NMR structure of cTnC-TnI chimera bound to calcium and A2 | 分子名称: | 4-(3-cyano-3-methylazetidine-1-carbonyl)-N-[(3R,4S)-7-fluoro-4-hydroxy-6-methyl-3,4-dihydro-2H-1-benzopyran-3-yl]-5-methyl-1H-pyrrole-2-sulfonamide, CALCIUM ION, Troponin C, ... | 著者 | Poppe, L, Hartman, J.J, Romero, A, Reagan, J.D. | 登録日 | 2021-11-18 | 公開日 | 2022-04-06 | 最終更新日 | 2024-05-15 | 実験手法 | SOLUTION NMR | 主引用文献 | Structural and Thermodynamic Model for the Activation of Cardiac Troponin. Biochemistry, 61, 2022
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7SOM
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![BU of 7som by Molmil](/molmil-images/mine/7som) | Ciliary C2 central pair apparatus isolated from Chlamydomonas reinhardtii | 分子名称: | Cilia- and flagella-associated protein 20, FAP147, FAP178, ... | 著者 | Gui, M, Wang, X, Dutcher, S.K, Brown, A, Zhang, R. | 登録日 | 2021-11-01 | 公開日 | 2022-04-13 | 最終更新日 | 2024-06-05 | 実験手法 | ELECTRON MICROSCOPY (3.7 Å) | 主引用文献 | Ciliary central apparatus structure reveals mechanisms of microtubule patterning. Nat.Struct.Mol.Biol., 29, 2022
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7TGH
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![BU of 7tgh by Molmil](/molmil-images/mine/7tgh) | Cryo-EM structure of respiratory super-complex CI+III2 from Tetrahymena thermophila | 分子名称: | 1,2-DIACYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 1,2-Distearoyl-sn-glycerophosphoethanolamine, 2 iron, ... | 著者 | Zhou, L, Maldonado, M, Padavannil, A, Guo, F, Letts, J.A. | 登録日 | 2022-01-07 | 公開日 | 2022-04-06 | 最終更新日 | 2022-07-20 | 実験手法 | ELECTRON MICROSCOPY (2.6 Å) | 主引用文献 | Structures of Tetrahymena 's respiratory chain reveal the diversity of eukaryotic core metabolism. Science, 376, 2022
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7TED
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![BU of 7ted by Molmil](/molmil-images/mine/7ted) | Human Ornithine Aminotransferase cocrystallized with its inhibitor, (S,E)-3-amino-4-(fluoromethylene)cyclopent-1-ene-1-carboxylate | 分子名称: | (1S,3R,4S)-3-formyl-4-[({3-hydroxy-2-methyl-5-[(phosphonooxy)methyl]pyridin-4-yl}methyl)amino]cyclopentane-1-carboxylic acid, Ornithine aminotransferase, mitochondrial, ... | 著者 | Butrin, A, Zhu, W, Silverman, R, Liu, D. | 登録日 | 2022-01-04 | 公開日 | 2022-04-06 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.63 Å) | 主引用文献 | Rational Design, Synthesis, and Mechanism of (3 S ,4 R )-3-Amino-4-(difluoromethyl)cyclopent-1-ene-1-carboxylic Acid: Employing a Second-Deprotonation Strategy for Selectivity of Human Ornithine Aminotransferase over GABA Aminotransferase. J.Am.Chem.Soc., 144, 2022
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7SQC
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![BU of 7sqc by Molmil](/molmil-images/mine/7sqc) | Ciliary C1 central pair apparatus isolated from Chlamydomonas reinhardtii | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, CPC1, Calmodulin, ... | 著者 | Gui, M, Wang, X, Dutcher, S.K, Brown, A, Zhang, R. | 登録日 | 2021-11-05 | 公開日 | 2022-04-13 | 最終更新日 | 2024-06-05 | 実験手法 | ELECTRON MICROSCOPY (3.8 Å) | 主引用文献 | Ciliary central apparatus structure reveals mechanisms of microtubule patterning. Nat.Struct.Mol.Biol., 29, 2022
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2MK3
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![BU of 2mk3 by Molmil](/molmil-images/mine/2mk3) | Solution NMR structure of gp41 ectodomain monomer on a DPC micelle | 分子名称: | Transmembrane glycoprotein, chimeric construct | 著者 | Roche, J, Louis, J.M, Grishaev, A, Ying, J, Bax, A. | 登録日 | 2014-01-23 | 公開日 | 2014-02-19 | 最終更新日 | 2024-05-01 | 実験手法 | SOLUTION NMR | 主引用文献 | Dissociation of the trimeric gp41 ectodomain at the lipid-water interface suggests an active role in HIV-1 Env-mediated membrane fusion. Proc.Natl.Acad.Sci.USA, 111, 2014
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2MB0
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6VBU
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![BU of 6vbu by Molmil](/molmil-images/mine/6vbu) | Structure of the bovine BBSome complex | 分子名称: | BBS1 domain-containing protein, Bardet-Biedl syndrome 18 protein, Bardet-Biedl syndrome 2 protein homolog, ... | 著者 | Singh, S.K, Gui, M, Koh, F, Yip, M.C.J, Brown, A. | 登録日 | 2019-12-19 | 公開日 | 2020-01-29 | 最終更新日 | 2024-03-06 | 実験手法 | ELECTRON MICROSCOPY (3.1 Å) | 主引用文献 | Structure and activation mechanism of the BBSome membrane protein trafficking complex. Elife, 9, 2020
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7AHR
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![BU of 7ahr by Molmil](/molmil-images/mine/7ahr) | Enzyme of biosynthetic pathway | 分子名称: | 3-[(1-Carboxyvinyl)oxy]benzoic acid, Chorismate dehydratase, GLYCEROL | 著者 | Archna, A, Breithaupt, C, Stubbs, M.T. | 登録日 | 2020-09-25 | 公開日 | 2021-10-06 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (2.21 Å) | 主引用文献 | Mechanism of chorismate dehydratase MqnA, the first enzyme of the futalosine pathway, proceeds via substrate-assisted catalysis J.Biol.Chem., 2022
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6USU
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![BU of 6usu by Molmil](/molmil-images/mine/6usu) | Crystal structure of GluN1/GluN2A ligand-binding domain in complex with L689,560 and glutamate | 分子名称: | (2R,4S)-5,7-dichloro-4-[(phenylcarbamoyl)amino]-1,2,3,4-tetrahydroquinoline-2-carboxylic acid, GLUTAMIC ACID, Glutamate receptor ionotropic, ... | 著者 | Romero-Hernandez, A, Tajima, N, Chou, T, Furukawa, H. | 登録日 | 2019-10-28 | 公開日 | 2020-07-15 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (2.092 Å) | 主引用文献 | Structural Basis of Functional Transitions in Mammalian NMDA Receptors. Cell, 182, 2020
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2MJX
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![BU of 2mjx by Molmil](/molmil-images/mine/2mjx) | Solution NMR structure of a mismatch DNA | 分子名称: | DNA (5'-D(*CP*GP*CP*GP*TP*AP*CP*GP*AP*TP*GP*CP*GP*C)-3'), DNA (5'-D(*GP*CP*GP*CP*AP*TP*GP*CP*TP*AP*CP*GP*CP*G)-3') | 著者 | Ghosh, A, Kumar, K.R, Bhunia, A, Chatterjee, S. | 登録日 | 2014-01-21 | 公開日 | 2014-03-05 | 最終更新日 | 2024-05-15 | 実験手法 | SOLUTION NMR | 主引用文献 | Double GC:GC mismatch in dsDNA enhances local dynamics retaining the DNA footprint: a high-resolution NMR study Chemmedchem, 9, 2014
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7T7N
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![BU of 7t7n by Molmil](/molmil-images/mine/7t7n) | Structure of SPCC1393.13 protein from fission yeast | 分子名称: | 1-METHOXY-2-[2-(2-METHOXY-ETHOXY]-ETHANE, Damage-control phosphatase SPCC1393.13, PHOSPHATE ION | 著者 | Jacewicz, A, Sanchez, A.M, Shuman, S. | 登録日 | 2021-12-15 | 公開日 | 2022-06-01 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Fission yeast Duf89 and Duf8901 are cobalt/nickel-dependent phosphatase-pyrophosphatases that act via a covalent aspartyl-phosphate intermediate. J.Biol.Chem., 298, 2022
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7T7O
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7T7K
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![BU of 7t7k by Molmil](/molmil-images/mine/7t7k) | Structure of SPAC806.04c protein from fission yeast bound to Co2+ | 分子名称: | CHLORIDE ION, COBALT (II) ION, Damage-control phosphatase SPAC806.04c, ... | 著者 | Jacewicz, A, Sanchez, A.M, Shuman, S. | 登録日 | 2021-12-15 | 公開日 | 2022-06-01 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Fission yeast Duf89 and Duf8901 are cobalt/nickel-dependent phosphatase-pyrophosphatases that act via a covalent aspartyl-phosphate intermediate. J.Biol.Chem., 298, 2022
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6VFM
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![BU of 6vfm by Molmil](/molmil-images/mine/6vfm) | Crystal structure of SpeG allosteric polyamine acetyltransferase from Bacillus thuringiensis | 分子名称: | Spermidine N1-acetyltransferase | 著者 | Tsimbalyuk, S, Shornikov, A, Le, V.T.B, Kuhn, M.L, Forwood, J.K. | 登録日 | 2020-01-05 | 公開日 | 2020-02-19 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (2.67 Å) | 主引用文献 | SpeG polyamine acetyltransferase enzyme from Bacillus thuringiensis forms a dodecameric structure and exhibits high catalytic efficiency. J.Struct.Biol., 210, 2020
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