1JNP
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![BU of 1jnp by Molmil](/molmil-images/mine/1jnp) | Crystal Structure of Murine Tcl1 at 2.5 Resolution | 分子名称: | T-CELL LEUKEMIA/LYMPHOMA PROTEIN 1A | 著者 | Petock, J.M, Torshin, I.Y, Wang, Y.F, DuBois, G.C, Croce, C.M, Harrison, R.W, Weber, I.T. | 登録日 | 2001-07-24 | 公開日 | 2001-11-07 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Structure of murine Tcl1 at 2.5 A resolution and implications for the TCL oncogene family. Acta Crystallogr.,Sect.D, 57, 2001
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1K1T
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![BU of 1k1t by Molmil](/molmil-images/mine/1k1t) | Combining Mutations in HIV-1 Protease to Understand Mechanisms of Resistance | 分子名称: | N-[(2R)-2-({N~5~-[amino(iminio)methyl]-L-ornithyl-L-valyl}amino)-4-methylpentyl]-L-phenylalanyl-L-alpha-glutamyl-L-alanyl-L-norleucinamide, PROTEASE RETROPEPSIN, SULFATE ION | 著者 | Mahalingam, B, Boross, P, Wang, Y.-F, Louis, J.M, Fischer, C, Tozser, J, Harrison, R.W, Weber, I.T. | 登録日 | 2001-09-25 | 公開日 | 2002-07-10 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (1.2 Å) | 主引用文献 | Combining mutations in HIV-1 protease to understand mechanisms of resistance. Proteins, 48, 2002
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1K2C
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![BU of 1k2c by Molmil](/molmil-images/mine/1k2c) | Combining Mutations in HIV-1 Protease to Understand Mechanisms of Resistance | 分子名称: | N-[(2R)-2-({N~5~-[amino(iminio)methyl]-L-ornithyl-L-valyl}amino)-4-methylpentyl]-L-phenylalanyl-L-alpha-glutamyl-L-alanyl-L-norleucinamide, PROTEASE RETROPEPSIN | 著者 | Mahalingam, B, Boross, P, Wang, Y.-F, Louis, J.M, Fischer, C, Tozser, J, W Harrison, R, Weber, I.T. | 登録日 | 2001-09-26 | 公開日 | 2002-07-10 | 最終更新日 | 2023-08-16 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Combining mutations in HIV-1 protease to understand mechanisms of resistance. Proteins, 48, 2002
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1K1U
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![BU of 1k1u by Molmil](/molmil-images/mine/1k1u) | Combining Mutations in HIV-1 Protease to Understand Mechanisms of Resistance | 分子名称: | N-[(2R)-2-({N~5~-[amino(iminio)methyl]-L-ornithyl-L-valyl}amino)-4-methylpentyl]-L-phenylalanyl-L-alpha-glutamyl-L-alanyl-L-norleucinamide, PROTEASE RETROPEPSIN | 著者 | Mahalingam, B, Boross, P, Wang, Y.-F, Louis, J.M, Fischer, C, Tozser, J, W Harrison, R, Weber, I.T. | 登録日 | 2001-09-25 | 公開日 | 2002-07-10 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | Combining mutations in HIV-1 protease to understand mechanisms of resistance. Proteins, 48, 2002
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1K2B
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![BU of 1k2b by Molmil](/molmil-images/mine/1k2b) | Combining Mutations in HIV-1 Protease to Understand Mechanisms of Resistance | 分子名称: | N-[(2R)-2-({N~5~-[amino(iminio)methyl]-L-ornithyl-L-valyl}amino)-4-methylpentyl]-L-phenylalanyl-L-alpha-glutamyl-L-alanyl-L-norleucinamide, PROTEASE RETROPEPSIN | 著者 | Mahalingam, B, Boross, P, Wang, Y.-F, Louis, J.M, Fischer, C, Tozser, J, W Harrison, R, Weber, I.T. | 登録日 | 2001-09-26 | 公開日 | 2002-07-10 | 最終更新日 | 2023-08-16 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Combining mutations in HIV-1 protease to understand mechanisms of resistance. Proteins, 48, 2002
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3LJP
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![BU of 3ljp by Molmil](/molmil-images/mine/3ljp) | Crystal structure of choline oxidase V464A mutant | 分子名称: | Choline oxidase, DIHYDROFLAVINE-ADENINE DINUCLEOTIDE | 著者 | Finnegan, S, Agniswamy, J, Weber, I.T, Giovanni, G. | 登録日 | 2010-01-26 | 公開日 | 2010-03-16 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Role of valine 464 in the flavin oxidation reaction catalyzed by choline oxidase. Biochemistry, 49, 2010
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3NYC
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![BU of 3nyc by Molmil](/molmil-images/mine/3nyc) | |
3NU6
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![BU of 3nu6 by Molmil](/molmil-images/mine/3nu6) | |
3NU5
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![BU of 3nu5 by Molmil](/molmil-images/mine/3nu5) | Crystal Structure of HIV-1 Protease Mutant I50V with Antiviral Drug Amprenavir | 分子名称: | ACETATE ION, CHLORIDE ION, SODIUM ION, ... | 著者 | Wang, Y.-F, Shen, C.H, Weber, I.T. | 登録日 | 2010-07-06 | 公開日 | 2010-08-25 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.29 Å) | 主引用文献 | Amprenavir complexes with HIV-1 protease and its drug-resistant mutants altering hydrophobic clusters. Febs J., 277, 2010
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3NYF
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![BU of 3nyf by Molmil](/molmil-images/mine/3nyf) | |
3NUJ
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![BU of 3nuj by Molmil](/molmil-images/mine/3nuj) | |
3NYE
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![BU of 3nye by Molmil](/molmil-images/mine/3nye) | |
3NU4
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![BU of 3nu4 by Molmil](/molmil-images/mine/3nu4) | Crystal Structure of HIV-1 Protease Mutant V32I with Antiviral Drug Amprenavir | 分子名称: | CHLORIDE ION, SODIUM ION, protease, ... | 著者 | Wang, Y.-F, Kovalevsky, A.Y, Weber, I.T. | 登録日 | 2010-07-06 | 公開日 | 2010-08-25 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.2 Å) | 主引用文献 | Amprenavir complexes with HIV-1 protease and its drug-resistant mutants altering hydrophobic clusters. Febs J., 277, 2010
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3NUO
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![BU of 3nuo by Molmil](/molmil-images/mine/3nuo) | |
3NU9
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![BU of 3nu9 by Molmil](/molmil-images/mine/3nu9) | |
3NU3
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![BU of 3nu3 by Molmil](/molmil-images/mine/3nu3) | Wild Type HIV-1 Protease with Antiviral Drug Amprenavir | 分子名称: | CHLORIDE ION, GLYCEROL, Protease, ... | 著者 | Wang, Y.-F, Kovalevsky, A.Y, Weber, I.T. | 登録日 | 2010-07-06 | 公開日 | 2010-08-25 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.02 Å) | 主引用文献 | Amprenavir complexes with HIV-1 protease and its drug-resistant mutants altering hydrophobic clusters. Febs J., 277, 2010
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3NNE
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![BU of 3nne by Molmil](/molmil-images/mine/3nne) | Crystal structure of choline oxidase S101A mutant | 分子名称: | ACETATE ION, Choline oxidase, FLAVIN-ADENINE DINUCLEOTIDE | 著者 | Wang, Y.-F, Finnegan, S, Yuan, H, Orville, A.M, Weber, I.T, Gadda, G. | 登録日 | 2010-06-23 | 公開日 | 2010-07-28 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.47 Å) | 主引用文献 | Structural and kinetic studies on the Ser101Ala variant of choline oxidase: Catalysis by compromise. Arch.Biochem.Biophys., 501, 2010
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3MWS
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![BU of 3mws by Molmil](/molmil-images/mine/3mws) | Crystal Structure of Group N HIV-1 Protease | 分子名称: | (3R,3AS,6AR)-HEXAHYDROFURO[2,3-B]FURAN-3-YL(1S,2R)-3-[[(4-AMINOPHENYL)SULFONYL](ISOBUTYL)AMINO]-1-BENZYL-2-HYDROXYPROPYLCARBAMATE, CHLORIDE ION, HIV-1 Protease | 著者 | Sayer, J.M, Agniswamy, J, Weber, I.T, Louis, J.M. | 登録日 | 2010-05-06 | 公開日 | 2011-03-23 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.09 Å) | 主引用文献 | Autocatalytic maturation, physical/chemical properties, and crystal structure of group N HIV-1 protease: relevance to drug resistance. Protein Sci., 19, 2010
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3OK9
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![BU of 3ok9 by Molmil](/molmil-images/mine/3ok9) | Crystal structure of wild-type HIV-1 protease with new oxatricyclic designed inhibitor GRL-0519A | 分子名称: | (3R,3aS,3bR,6aS,7aS)-octahydrodifuro[2,3-b:3',2'-d]furan-3-yl [(1S,2R)-1-benzyl-2-hydroxy-3-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}propyl]carbamate, CHLORIDE ION, GLYCEROL, ... | 著者 | Wang, Y.-F, Agniswamy, J, Weber, I.T. | 登録日 | 2010-08-24 | 公開日 | 2010-09-22 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.27 Å) | 主引用文献 | Probing Multidrug-Resistance and Protein-Ligand Interactions with Oxatricyclic Designed Ligands in HIV-1 Protease Inhibitors. Chemmedchem, 5, 2010
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3GJR
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![BU of 3gjr by Molmil](/molmil-images/mine/3gjr) | Caspase-3 Binds Diverse P4 Residues in Peptides | 分子名称: | Caspase-3 subunit p12, Caspase-3 subunit p17, GLYCEROL, ... | 著者 | Fang, B, Fu, G, Agniswamy, J, Harrison, R.W, Weber, I.T. | 登録日 | 2009-03-09 | 公開日 | 2009-03-24 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Caspase-3 binds diverse P4 residues in peptides as revealed by crystallography and structural modeling. Apoptosis, 14, 2009
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3GJT
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![BU of 3gjt by Molmil](/molmil-images/mine/3gjt) | Caspase-3 Binds Diverse P4 Residues in Peptides | 分子名称: | Caspase-3 subunit p12, Caspase-3 subunit p17, peptide inhibitor | 著者 | Fang, B, Fu, G, Agniswamy, J, Harrison, R.W, Weber, I.T. | 登録日 | 2009-03-09 | 公開日 | 2009-03-24 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Caspase-3 binds diverse P4 residues in peptides as revealed by crystallography and structural modeling. Apoptosis, 14, 2009
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3EC0
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![BU of 3ec0 by Molmil](/molmil-images/mine/3ec0) | High Resolution HIV-2 Protease Structure in Complex with Antiviral Inhibitor GRL-06579A | 分子名称: | (3AS,5R,6AR)-HEXAHYDRO-2H-CYCLOPENTA[B]FURAN-5-YL (2S,3S)-3-HYDROXY-4-(4-(HYDROXYMETHYL)-N-ISOBUTYLPHENYLSULFONAMIDO)-1-PHENYLBUTAN-2-YLCARBAMATE, CHLORIDE ION, IMIDAZOLE, ... | 著者 | Kovalevsky, A.Y, Weber, I.T. | 登録日 | 2008-08-28 | 公開日 | 2008-09-16 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.18 Å) | 主引用文献 | Structural evidence for effectiveness of darunavir and two related antiviral inhibitors against HIV-2 protease J.Mol.Biol., 384, 2008
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3GJS
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![BU of 3gjs by Molmil](/molmil-images/mine/3gjs) | Caspase-3 Binds Diverse P4 Residues in Peptides | 分子名称: | Ac-YVAD-Cho inhibitor, Caspase-3 subunit p12, Caspase-3 subunit p17 | 著者 | Fang, B, Fu, G, Agniswamy, J, Harrison, R.W, Weber, I.T. | 登録日 | 2009-03-09 | 公開日 | 2009-03-24 | 最終更新日 | 2011-08-17 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Caspase-3 binds diverse P4 residues in peptides as revealed by crystallography and structural modeling. Apoptosis, 14, 2009
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3EBZ
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![BU of 3ebz by Molmil](/molmil-images/mine/3ebz) | High Resolution HIV-2 Protease Structure in Complex with Clinical Drug Darunavir | 分子名称: | (3R,3AS,6AR)-HEXAHYDROFURO[2,3-B]FURAN-3-YL(1S,2R)-3-[[(4-AMINOPHENYL)SULFONYL](ISOBUTYL)AMINO]-1-BENZYL-2-HYDROXYPROPYLCARBAMATE, CHLORIDE ION, IMIDAZOLE, ... | 著者 | Kovalevsky, A.Y, Weber, I.T. | 登録日 | 2008-08-28 | 公開日 | 2008-09-16 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.2 Å) | 主引用文献 | Structural evidence for effectiveness of darunavir and two related antiviral inhibitors against HIV-2 protease J.Mol.Biol., 384, 2008
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3ECG
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![BU of 3ecg by Molmil](/molmil-images/mine/3ecg) | High Resolution HIV-2 Protease Structure in Complex with Antiviral Inhibitor GRL-98065 | 分子名称: | (3R,3AS,6AR)-HEXAHYDROFURO[2,3-B]FURAN-3-YL(2S,3R)-3-HYDROXY-4-(N-ISOBUTYLBENZO[D][1,3]DIOXOLE-5-SULFONAMIDO)-1-PHENYLBUTAN-2-YLCARBAMATE, CHLORIDE ION, IMIDAZOLE, ... | 著者 | Kovalevsky, A.Y, Weber, I.T. | 登録日 | 2008-08-29 | 公開日 | 2008-09-16 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.18 Å) | 主引用文献 | Structural evidence for effectiveness of darunavir and two related antiviral inhibitors against HIV-2 protease J.Mol.Biol., 384, 2008
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