3KUZ
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![BU of 3kuz by Molmil](/molmil-images/mine/3kuz) | Crystal structure of the ubiquitin like domain of PLXNC1 | 分子名称: | Plexin-C1, UNKNOWN ATOM OR ION | 著者 | Wang, H, Li, B, Tempel, W, Tong, Y, Guan, X, Zhong, N, Crombet, L, MacKenzie, F, Buck, M, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Weigelt, J, Bochkarev, A, Park, H, Structural Genomics Consortium (SGC) | 登録日 | 2009-11-28 | 公開日 | 2009-12-08 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Crystal structure of the ubiquitin like domain of PLXNC1 to be published
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2PQE
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![BU of 2pqe by Molmil](/molmil-images/mine/2pqe) | Solution structure of proline-free mutant of staphylococcal nuclease | 分子名称: | Thermonuclease | 著者 | Shan, L, Tong, Y, Xie, T, Wang, M, Wang, J. | 登録日 | 2007-05-01 | 公開日 | 2007-06-19 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | Restricted backbone conformational and motional flexibilities of loops containing peptidyl-proline bonds dominate the enzyme activity of staphylococcal nuclease. Biochemistry, 46, 2007
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3LWE
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![BU of 3lwe by Molmil](/molmil-images/mine/3lwe) | The crystal structure of MPP8 | 分子名称: | M-phase phosphoprotein 8 | 著者 | Li, Z, Li, Z, Ruan, J, Xu, C, Tong, Y, Pan, P.W, Tempel, W, Crombet, L, Min, J, Zang, J, Structural Genomics Consortium (SGC) | 登録日 | 2010-02-23 | 公開日 | 2010-03-02 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.05 Å) | 主引用文献 | Structural basis for specific binding of human MPP8 chromodomain to histone H3 methylated at lysine 9. Plos One, 6, 2011
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3LLU
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![BU of 3llu by Molmil](/molmil-images/mine/3llu) | Crystal structure of the nucleotide-binding domain of Ras-related GTP-binding protein C | 分子名称: | MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-GUANYLATE ESTER, Ras-related GTP-binding protein C, ... | 著者 | Nedyalkova, L, Tempel, W, Tong, Y, Crombet, L, Zhong, N, Guan, X, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Weigelt, J, Bochkarev, A, Park, H, Structural Genomics Consortium (SGC) | 登録日 | 2010-01-29 | 公開日 | 2010-02-09 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.4 Å) | 主引用文献 | Crystal structure of the nucleotide-binding domain of Ras-related GTP-binding protein C to be published
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3O47
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![BU of 3o47 by Molmil](/molmil-images/mine/3o47) | Crystal structure of ARFGAP1-ARF1 fusion protein | 分子名称: | ADP-ribosylation factor GTPase-activating protein 1, ADP-ribosylation factor 1, GUANOSINE-5'-DIPHOSPHATE, ... | 著者 | Wang, H, Tong, Y, Nedyalkova, L, Tempel, W, Guan, X, Crombet, L, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Weigelt, J, Bochkarev, A, Park, H, Structural Genomics Consortium (SGC) | 登録日 | 2010-07-26 | 公開日 | 2010-08-11 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Crystal structure of ARFGAP1-ARF1 fusion protein to be published
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3O46
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![BU of 3o46 by Molmil](/molmil-images/mine/3o46) | Crystal structure of the PDZ domain of MPP7 | 分子名称: | MAGUK p55 subfamily member 7, UNKNOWN ATOM OR ION | 著者 | Nedyalkova, L, Tong, Y, Tempel, W, Zhong, N, Guan, X, Landry, R, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Weigelt, J, Bochkarev, A, Park, H, Structural Genomics Consortium (SGC) | 登録日 | 2010-07-26 | 公開日 | 2010-08-04 | 最終更新日 | 2017-11-08 | 実験手法 | X-RAY DIFFRACTION (1.3 Å) | 主引用文献 | Crystal structure of the PDZ domain of MPP7 TO BE PUBLISHED
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3MDB
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![BU of 3mdb by Molmil](/molmil-images/mine/3mdb) | Crystal structure of the ternary complex of full length centaurin alpha-1, KIF13B FHA domain, and IP4 | 分子名称: | (2R)-3-{[(R)-{[(1S,2S,3R,4S,5S,6S)-2,6-dihydroxy-3,4,5-tris(phosphonooxy)cyclohexyl]oxy}(hydroxy)phosphoryl]oxy}propane -1,2-diyl dioctanoate, Arf-GAP with dual PH domain-containing protein 1, Kinesin-like protein KIF13B, ... | 著者 | Shen, L, Tong, Y, Tempel, W, MacKenzie, F, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Weigelt, J, Bochkarev, A, Park, H, Structural Genomics Consortium (SGC) | 登録日 | 2010-03-30 | 公開日 | 2010-08-04 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.952 Å) | 主引用文献 | Crystal structure of the ternary complex of full length centaurin alpha-1, KIF13B FHA domain, and IP4 to be published
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3P1J
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![BU of 3p1j by Molmil](/molmil-images/mine/3p1j) | Crystal structure of human GTPase IMAP family member 2 in the nucleotide-free state | 分子名称: | GTPase IMAP family member 2, UNKNOWN ATOM OR ION | 著者 | Shen, L, Tempel, W, Tong, Y, Guan, X, Nedyalkova, L, Wernimont, A.K, Mackenzie, F, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Weigelt, J, Bochkarev, A, Andrews, D.W, Park, H, Structural Genomics Consortium (SGC) | 登録日 | 2010-09-30 | 公開日 | 2010-10-13 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.58 Å) | 主引用文献 | Crystal structure of human GTPase IMAP family member 2 in the nucleotide-free state to be published
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3OES
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![BU of 3oes by Molmil](/molmil-images/mine/3oes) | Crystal structure of the small GTPase RhebL1 | 分子名称: | GTPase RhebL1, MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-GUANYLATE ESTER | 著者 | Nedyalkova, L, Zhong, N, Tempel, W, Tong, Y, Shen, L, Loppnau, P, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Weigelt, J, Bochkarev, A, Park, H, Structural Genomics Consortium (SGC) | 登録日 | 2010-08-13 | 公開日 | 2010-08-25 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.301 Å) | 主引用文献 | Crystal structure of the small GTPase RhebL1 to be published
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3EO2
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![BU of 3eo2 by Molmil](/molmil-images/mine/3eo2) | Crystal structure of the RhoGEF domain of human neuroepithelial cell-transforming gene 1 protein | 分子名称: | Neuroepithelial cell-transforming gene 1 protein, UNKNOWN ATOM OR ION | 著者 | Nedyalkova, L, Tong, Y, Tempel, W, MacKenzie, F, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Weigelt, J, Bochkarev, A, Park, H, Structural Genomics Consortium (SGC) | 登録日 | 2008-09-26 | 公開日 | 2008-10-07 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Crystal structure of the RhoGEF domain of human neuroepithelial cell-transforming gene 1 protein To be Published
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3FK2
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![BU of 3fk2 by Molmil](/molmil-images/mine/3fk2) | Crystal structure of the RhoGAP domain of human glucocorticoid receptor DNA-binding factor 1 | 分子名称: | Glucocorticoid receptor DNA-binding factor 1, UNKNOWN ATOM OR ION | 著者 | Nedyalkova, L, Tong, Y, Tempel, W, Loppnau, P, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Weigelt, J, Bochkarev, A, Park, H, Structural Genomics Consortium (SGC) | 登録日 | 2008-12-15 | 公開日 | 2008-12-23 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Crystal structure of the RhoGAP domain of human glucocorticoid receptor DNA-binding factor 1 To be Published
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3CON
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![BU of 3con by Molmil](/molmil-images/mine/3con) | Crystal structure of the human NRAS GTPase bound with GDP | 分子名称: | GTPase NRas, GUANOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, ... | 著者 | Nedyalkova, L, Tong, Y, Tempel, W, Shen, L, Loppnau, P, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Weigelt, J, Bochkarev, A, Park, H, Structural Genomics Consortium (SGC) | 登録日 | 2008-03-28 | 公開日 | 2008-04-08 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (1.649 Å) | 主引用文献 | Crystal structure of the human NRAS GTPase bound with GDP. To be Published
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3CXL
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![BU of 3cxl by Molmil](/molmil-images/mine/3cxl) | Crystal structure of human chimerin 1 (CHN1) | 分子名称: | N-chimerin, UNKNOWN ATOM OR ION, ZINC ION | 著者 | Shen, L, Buck, M, Tong, Y, Tempel, W, MacKenzie, F, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Wilkstrom, M, Bochkarev, A, Park, H, Structural Genomics Consortium (SGC) | 登録日 | 2008-04-24 | 公開日 | 2008-08-05 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Crystal structure of human chimerin 1 (CHN1). To be Published
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3DWD
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![BU of 3dwd by Molmil](/molmil-images/mine/3dwd) | Crystal structure of the ArfGAP domain of human ARFGAP1 | 分子名称: | ADP-ribosylation factor GTPase-activating protein 1, UNKNOWN ATOM OR ION, ZINC ION | 著者 | Nedyalkova, L, Tong, Y, Tempel, W, Landry, R, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Wilkstrom, M, Bochkarev, A, Park, H, Structural Genomics Consortium (SGC) | 登録日 | 2008-07-22 | 公開日 | 2008-08-05 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Crystal structure of the ArfGAP domain of human ARFGAP1 To be Published
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3GRO
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![BU of 3gro by Molmil](/molmil-images/mine/3gro) | Human palmitoyl-protein thioesterase 1 | 分子名称: | Palmitoyl-protein thioesterase 1, UNKNOWN ATOM OR ION | 著者 | Dobrovetsky, E, Seitova, A, Tong, Y, Tempel, W, Dong, A, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Weigelt, J, Bochkarev, A, Cossar, D, Park, H, Structural Genomics Consortium (SGC) | 登録日 | 2009-03-26 | 公開日 | 2009-04-07 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.53 Å) | 主引用文献 | Human palmitoyl-protein thioesterase 1 To be Published
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7Y47
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![BU of 7y47 by Molmil](/molmil-images/mine/7y47) | Crystal structure of bifunctional miltiradiene synthase from selaginella moellendorffii that complexed with GGPP | 分子名称: | Bifunctional diterpene synthase, chloroplastic, GERANYLGERANYL DIPHOSPHATE, ... | 著者 | Ma, X, Tao, Y, Jiang, T. | 登録日 | 2022-06-14 | 公開日 | 2022-10-26 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Structural and mechanistic insights into the precise product synthesis by a bifunctional miltiradiene synthase. Plant Biotechnol J, 21, 2023
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8P2A
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![BU of 8p2a by Molmil](/molmil-images/mine/8p2a) | Crystal structure of SaFMN3 domain 2 | 分子名称: | FLAVIN MONONUCLEOTIDE, FMN-binding domain-containing protein | 著者 | Rozeboom, H.J, Fraaije, M.W. | 登録日 | 2023-05-15 | 公開日 | 2023-07-19 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Characterization of two bacterial multi-flavinylated proteins harboring multiple covalent flavin cofactors. Bba Adv, 4, 2023
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8P2B
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![BU of 8p2b by Molmil](/molmil-images/mine/8p2b) | Crystal structure of CbFMN4 domain 1 | 分子名称: | Clostridiaceae bacterium FMN4 domain 1, FLAVIN MONONUCLEOTIDE | 著者 | Rozeboom, H.J, Fraaije, M.W. | 登録日 | 2023-05-15 | 公開日 | 2023-07-19 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Characterization of two bacterial multi-flavinylated proteins harboring multiple covalent flavin cofactors. Bba Adv, 4, 2023
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8Q5E
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![BU of 8q5e by Molmil](/molmil-images/mine/8q5e) | |
8Q5F
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8Q5G
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2E9N
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![BU of 2e9n by Molmil](/molmil-images/mine/2e9n) | Structure of h-CHK1 complexed with A767085 | 分子名称: | 3-(4'-HYDROXYBIPHENYL-4-YL)-N-(4-HYDROXYCYCLOHEXYL)-1,4-DIHYDROINDENO[1,2-C]PYRAZOLE-6-CARBOXAMIDE, Serine/threonine-protein kinase Chk1 | 著者 | Park, C. | 登録日 | 2007-01-26 | 公開日 | 2008-01-29 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Discovery of 1,4-dihydroindeno[1,2-c]pyrazoles as a novel class of potent and selective checkpoint kinase 1 inhibitors. Bioorg.Med.Chem., 15, 2007
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2E9O
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![BU of 2e9o by Molmil](/molmil-images/mine/2e9o) | Structure of h-CHK1 complexed with AA582939 | 分子名称: | 4-(6-{[(4-METHYLCYCLOHEXYL)AMINO]METHYL}-1,4-DIHYDROINDENO[1,2-C]PYRAZOL-3-YL)BENZOIC ACID, Serine/threonine-protein kinase Chk1 | 著者 | Park, C. | 登録日 | 2007-01-26 | 公開日 | 2008-01-29 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Discovery of 1,4-dihydroindeno[1,2-c]pyrazoles as a novel class of potent and selective checkpoint kinase 1 inhibitors. Bioorg.Med.Chem., 15, 2007
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2E9V
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![BU of 2e9v by Molmil](/molmil-images/mine/2e9v) | Structure of h-CHK1 complexed with A859017 | 分子名称: | 18-CHLORO-2-OXO-17-[(PYRIDIN-4-YLMETHYL)AMINO]-2,3,11,12,13,14-HEXAHYDRO-1H,10H-4,8-(AZENO)-9,15,1,3,6-BENZODIOXATRIAZACYCLOHEPTADECINE-7-CARBONITRILE, Serine/threonine-protein kinase Chk1 | 著者 | Park, C. | 登録日 | 2007-01-27 | 公開日 | 2008-01-29 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Structure-Based Design, Synthesis and Biological Evaluation of Potent Selective Macrocyclic Chk1 Inhibitors To be Published
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2E9P
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![BU of 2e9p by Molmil](/molmil-images/mine/2e9p) | Structure of h-CHK1 complexed with A771129 | 分子名称: | 1-(5-CHLORO-2-METHOXYPHENYL)-3-{6-[2-(DIMETHYLAMINO)-1-METHYLETHOXY]PYRAZIN-2-YL}UREA, Serine/threonine-protein kinase Chk1 | 著者 | Park, C. | 登録日 | 2007-01-26 | 公開日 | 2008-01-29 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Structure-Based Design, Synthesis and Biological Evaluation of Potent and Selective Macrocyclic Chk1 Inhibitors To be Published
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