7W3O
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![BU of 7w3o by Molmil](/molmil-images/mine/7w3o) | Crystal structure of human CYB5R3 | 分子名称: | FLAVIN-ADENINE DINUCLEOTIDE, NADH-cytochrome b5 reductase 3 soluble form | 著者 | Noda, N.N. | 登録日 | 2021-11-25 | 公開日 | 2022-12-07 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.46 Å) | 主引用文献 | The UFM1 system regulates ER-phagy through the ufmylation of CYB5R3. Nat Commun, 13, 2022
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7W3N
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5BRO
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![BU of 5bro by Molmil](/molmil-images/mine/5bro) | Crystal structure of modified HexB (modB) | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Beta-hexosaminidase subunit beta, FORMIC ACID, ... | 著者 | Kitakaze, K, Maita, N, Itoh, K. | 登録日 | 2015-06-01 | 公開日 | 2016-05-04 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Protease-resistant modified human beta-hexosaminidase B ameliorates symptoms in GM2 gangliosidosis model. J.Clin.Invest., 126, 2016
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3W0A
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![BU of 3w0a by Molmil](/molmil-images/mine/3w0a) | Crystal Structure Analysis of Vitamin D receptor | 分子名称: | (4S)-4-hydroxy-5-[2-methyl-4-(3-{3-methyl-4-[4,4,4-trifluoro-3-hydroxy-3-(trifluoromethyl)but-1-yn-1-yl]phenyl}pentan-3-yl)phenoxy]pentanoic acid, Vitamin D3 receptor | 著者 | Itoh, S, Iijima, S. | 登録日 | 2012-10-25 | 公開日 | 2013-11-13 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | structure analysis of vitamin D3 receptor To be Published
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3W0C
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![BU of 3w0c by Molmil](/molmil-images/mine/3w0c) | Crystal Structure Analysis of Vitamin D receptor | 分子名称: | (4S)-4-hydroxy-5-[2-methyl-4-(3-{3-methyl-4-[(1E)-4,4,4-trifluoro-3-hydroxy-3-(trifluoromethyl)but-1-en-1-yl]phenyl}pentan-3-yl)phenoxy]pentanoic acid, Vitamin D3 receptor | 著者 | Itoh, S, Iijima, S. | 登録日 | 2012-10-29 | 公開日 | 2013-11-13 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | structure analysis of vitamin D receptor To be Published
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3W0Y
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![BU of 3w0y by Molmil](/molmil-images/mine/3w0y) | Crystal Structure Analysis of Vitamin D receptor | 分子名称: | Vitamin D3 receptor, [3-fluoro-2'-methyl-4'-(3-{3-methyl-4-[(1E)-4,4,4-trifluoro-3-hydroxy-3-(trifluoromethyl)but-1-en-1-yl]phenyl}pentan-3-yl)biphenyl-4-yl]acetic acid | 著者 | Itoh, S, Iijima, S. | 登録日 | 2012-11-05 | 公開日 | 2013-11-13 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (1.98 Å) | 主引用文献 | Crystal Structure Analysis of Vitamin D receptor TO BE PUBLISHED
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3AZ1
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![BU of 3az1 by Molmil](/molmil-images/mine/3az1) | Crystal Structure Analysis of Vitamin D receptor | 分子名称: | Vitamin D3 receptor, {4-[3-(4-{[(2R)-2-hydroxy-3,3-dimethylbutyl]oxy}-3-methylphenyl)pentan-3-yl]-2-methylphenoxy}acetic acid | 著者 | Itoh, S, Iijima, S. | 登録日 | 2011-05-20 | 公開日 | 2011-11-02 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Novel nonsecosteroidal vitamin D(3) carboxylic acid analogs for osteoporosis, and SAR analysis. Bioorg.Med.Chem., 19, 2011
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3AZ2
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![BU of 3az2 by Molmil](/molmil-images/mine/3az2) | Crystal Structure Analysis of Vitamin D receptor | 分子名称: | 5-{4-[3-(4-{[(2R)-2-hydroxy-3,3-dimethylbutyl]oxy}-3-methylphenyl)pentan-3-yl]-2-methylphenoxy}pentanoic acid, Vitamin D3 receptor | 著者 | Itoh, S, Iijima, S. | 登録日 | 2011-05-20 | 公開日 | 2011-11-02 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (1.69 Å) | 主引用文献 | Novel nonsecosteroidal vitamin D(3) carboxylic acid analogs for osteoporosis, and SAR analysis. Bioorg.Med.Chem., 19, 2011
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3AZ3
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![BU of 3az3 by Molmil](/molmil-images/mine/3az3) | Crystal Structure Analysis of Vitamin D receptor | 分子名称: | (4S)-4-hydroxy-5-[4-(3-{4-[(3S)-3-hydroxy-4,4-dimethylpentyl]-3-methylphenyl}pentan-3-yl)-2-methylphenoxy]pentanoic acid, Vitamin D3 receptor | 著者 | Itoh, S, Iijima, S. | 登録日 | 2011-05-20 | 公開日 | 2011-11-02 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (1.36 Å) | 主引用文献 | Novel nonsecosteroidal vitamin D(3) carboxylic acid analogs for osteoporosis, and SAR analysis. Bioorg.Med.Chem., 19, 2011
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5EXA
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5EWZ
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7EA6
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![BU of 7ea6 by Molmil](/molmil-images/mine/7ea6) | Crystal structure of TCR-017 ectodomain | 分子名称: | T cell receptor 017 alpha chain, T cell receptor 017 beta chain | 著者 | Nagae, M, Yamasaki, S. | 登録日 | 2021-03-06 | 公開日 | 2021-10-13 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.18000245 Å) | 主引用文献 | Identification of conserved SARS-CoV-2 spike epitopes that expand public cTfh clonotypes in mild COVID-19 patients. J.Exp.Med., 218, 2021
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8X6R
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![BU of 8x6r by Molmil](/molmil-images/mine/8x6r) | KRasG12C in complex with inhibitor | 分子名称: | 1-[7-[6-ethenyl-8-ethoxy-7-(5-methyl-1~{H}-indazol-4-yl)-2-(1-methylpiperidin-4-yl)oxy-quinazolin-4-yl]-2,7-diazaspiro[3.5]nonan-2-yl]propan-1-one, GUANOSINE-5'-DIPHOSPHATE, Isoform 2B of GTPase KRas, ... | 著者 | Amano, Y, Tateishi, Y. | 登録日 | 2023-11-21 | 公開日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Discovery of ASP6918, a KRAS G12C inhibitor: Synthesis and structure-activity relationships of 1-{2,7-diazaspiro[3.5]non-2-yl}prop-2-en-1-one derivatives as covalent inhibitors with good potency and oral activity for the treatment of solid tumors. Bioorg.Med.Chem., 98, 2023
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4YB9
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![BU of 4yb9 by Molmil](/molmil-images/mine/4yb9) | Crystal structure of the Bovine Fructose transporter GLUT5 in an open inward-facing conformation | 分子名称: | Solute carrier family 2, facilitated glucose transporter member 5 | 著者 | Verdon, G, Kang, H.J, Iwata, S, Drew, D. | 登録日 | 2015-02-18 | 公開日 | 2015-10-14 | 最終更新日 | 2024-05-01 | 実験手法 | X-RAY DIFFRACTION (3.2 Å) | 主引用文献 | Structure and mechanism of the mammalian fructose transporter GLUT5. Nature, 526, 2015
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4YBQ
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![BU of 4ybq by Molmil](/molmil-images/mine/4ybq) | Rat GLUT5 with Fv in the outward-open form | 分子名称: | Solute carrier family 2, facilitated glucose transporter member 5, antibody Fv fragment heavy chain, ... | 著者 | Nomura, N, Shimamura, T, Iwata, S. | 登録日 | 2015-02-19 | 公開日 | 2015-10-07 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (3.27 Å) | 主引用文献 | Structure and mechanism of the mammalian fructose transporter GLUT5 Nature, 526, 2015
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8W85
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![BU of 8w85 by Molmil](/molmil-images/mine/8w85) | HLA-DQ2.5-gamma2 gliadin peptide in complex with DQN0385AE01 | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, DQN0385AE01 Fab heavy chain, DQN0385AE01 Fab light chain, ... | 著者 | Irie, M, Tsushima, T, Teranishi-Ikawa, Y, Takahashi, N, Ishii, S, Okura, Y, Fukami, T.A, Torizawa, T. | 登録日 | 2023-08-31 | 公開日 | 2023-11-08 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2.769 Å) | 主引用文献 | Characterizations of a neutralizing antibody broadly reactive to multiple gluten peptide:HLA-DQ2.5 complexes in the context of celiac disease. Nat Commun, 14, 2023
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8W86
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![BU of 8w86 by Molmil](/molmil-images/mine/8w86) | HLA-DQ2.5-B/C hordein peptide in complex with DQN0385AE02 | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, DQN0385AE02 Fab heavy chain, DQN0385AE02 Fab light chain, ... | 著者 | Irie, M, Tsushima, T, Teranishi-Ikawa, Y, Takahashi, N, Ishii, S, Okura, Y, Fukami, T.A, Torizawa, T. | 登録日 | 2023-08-31 | 公開日 | 2023-11-08 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2.236 Å) | 主引用文献 | Characterizations of a neutralizing antibody broadly reactive to multiple gluten peptide:HLA-DQ2.5 complexes in the context of celiac disease. Nat Commun, 14, 2023
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8W84
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![BU of 8w84 by Molmil](/molmil-images/mine/8w84) | HLA-DQ2.5-alpha2 gliadin peptide in complex with DQN0344AE02 | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, DQN0344AE02 Fab heavy chain, DQN0344AE02 Fab light chain, ... | 著者 | Irie, M, Tsushima, T, Teranishi-Ikawa, Y, Takahashi, N, Ishii, S, Okura, Y, Fukami, T.A, Torizawa, T. | 登録日 | 2023-08-31 | 公開日 | 2023-11-08 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2.105 Å) | 主引用文献 | Characterizations of a neutralizing antibody broadly reactive to multiple gluten peptide:HLA-DQ2.5 complexes in the context of celiac disease. Nat Commun, 14, 2023
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8W83
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![BU of 8w83 by Molmil](/molmil-images/mine/8w83) | HLA-DQ2.5-alpha1 gliadin peptide in complex with DQN0344AE02 | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, DQN0344AE02 Fab heavy chain, DQN0344AE02 Fab light chain, ... | 著者 | Irie, M, Tsushima, T, Teranishi-Ikawa, Y, Takahashi, N, Ishii, S, Okura, Y, Fukami, T.A, Torizawa, T. | 登録日 | 2023-08-31 | 公開日 | 2023-11-08 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2.818 Å) | 主引用文献 | Characterizations of a neutralizing antibody broadly reactive to multiple gluten peptide:HLA-DQ2.5 complexes in the context of celiac disease. Nat Commun, 14, 2023
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8SDH
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8JS5
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![BU of 8js5 by Molmil](/molmil-images/mine/8js5) | Dimeric PAS domains of oxygen sensor FixL with ferric unliganded heme | 分子名称: | GLYCEROL, PROTOPORPHYRIN IX CONTAINING FE, Sensor protein FixL | 著者 | Kamaya, M, Koteishi, H, Sawai, H, Sugimoto, H, Shiro, Y. | 登録日 | 2023-06-19 | 公開日 | 2024-06-26 | 実験手法 | X-RAY DIFFRACTION (2.95 Å) | 主引用文献 | Dimeric PAS domains of oxygen sensor FixL in complex with imidazole-bound heme. To be published
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8JS7
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![BU of 8js7 by Molmil](/molmil-images/mine/8js7) | Dimeric PAS domains of oxygen sensor FixL in complex with imidazole-bound heme | 分子名称: | GLYCEROL, IMIDAZOLE, PROTOPORPHYRIN IX CONTAINING FE, ... | 著者 | Kamaya, M, Koteishi, H, Sawai, H, Sugimoto, H, Shiro, Y. | 登録日 | 2023-06-19 | 公開日 | 2024-06-26 | 実験手法 | X-RAY DIFFRACTION (2.85 Å) | 主引用文献 | Dimeric PAS domains of oxygen sensor FixL in complex with imidazole-bound heme. To be published
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8JS6
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![BU of 8js6 by Molmil](/molmil-images/mine/8js6) | Dimeric PAS domains of oxygen sensor FixL in complex with cyanide-bound ferric heme | 分子名称: | CYANIDE ION, GLYCEROL, PROTOPORPHYRIN IX CONTAINING FE, ... | 著者 | Kamaya, M, Koteishi, H, Sawai, H, Sugimoto, H, Shiro, Y. | 登録日 | 2023-06-19 | 公開日 | 2024-06-26 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Dimeric PAS domains of oxygen sensor FixL in complex with imidazole-bound heme. To be published
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5H9W
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![BU of 5h9w by Molmil](/molmil-images/mine/5h9w) | Crystal structure of Regnase PIN domain, form II | 分子名称: | Ribonuclease ZC3H12A, SODIUM ION | 著者 | Yokogawa, M, Tsushima, T, Adachi, W, Noda, N.N, Inagaki, F. | 登録日 | 2015-12-29 | 公開日 | 2016-03-16 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Structural basis for the regulation of enzymatic activity of Regnase-1 by domain-domain interactions Sci Rep, 6, 2016
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5H9V
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![BU of 5h9v by Molmil](/molmil-images/mine/5h9v) | Crystal structure of Regnase PIN domain, form I | 分子名称: | Ribonuclease ZC3H12A, SODIUM ION | 著者 | Yokogawa, M, Tsushima, T, Adachi, W, Noda, N.N, Inagaki, F. | 登録日 | 2015-12-29 | 公開日 | 2016-03-16 | 最終更新日 | 2020-02-19 | 実験手法 | X-RAY DIFFRACTION (2.75 Å) | 主引用文献 | Structural basis for the regulation of enzymatic activity of Regnase-1 by domain-domain interactions Sci Rep, 6, 2016
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