6ZSZ
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6ZSY
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6H6W
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![BU of 6h6w by Molmil](/molmil-images/mine/6h6w) | Molybdenum storage protein- H156A | 分子名称: | ADENOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, MOLYBDATE ION, ... | 著者 | Ermler, U, Bruenle, S. | 登録日 | 2018-07-30 | 公開日 | 2018-12-05 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | The molybdenum storage protein - A bionanolab for creating experimentally alterable polyoxomolybdate clusters. J. Inorg. Biochem., 189, 2018
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3KZ7
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4BQR
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![BU of 4bqr by Molmil](/molmil-images/mine/4bqr) | Mtb InhA complex with Methyl-thiazole compound 11 | 分子名称: | (NZ)-2-[2,6-bis(fluoranyl)phenyl]-N-[5-[(1S)-1-(4-methyl-1,3-thiazol-2-yl)-1-oxidanyl-ethyl]-3H-1,3,4-thiadiazol-2-ylidene]ethanamide, ENOYL-[ACYL-CARRIER-PROTEIN] REDUCTASE [NADH], NICOTINAMIDE-ADENINE-DINUCLEOTIDE | 著者 | Read, J.A, Gingell, H, Madhavapeddi, P, Shirude, P.S. | 登録日 | 2013-05-31 | 公開日 | 2013-12-11 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2.05 Å) | 主引用文献 | Methyl-Thiazoles: A Novel Mode of Inhibition with the Potential to Develop Novel Inhibitors Targeting Inha in Mycobacterium Tuberculosis. J.Med.Chem., 56, 2013
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4BQP
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![BU of 4bqp by Molmil](/molmil-images/mine/4bqp) | Mtb InhA complex with Methyl-thiazole compound 7 | 分子名称: | (1S)-1-(5-{[1-(2,6-DIFLUOROBENZYL)-1H-PYRAZOL-3-YL]AMINO}-1,3,4-THIADIAZOL-2-YL)-1-(4-METHYL-1,3-THIAZOL-2-YL)ETHANOL, ENOYL-[ACYL-CARRIER-PROTEIN] REDUCTASE [NADH], NICOTINAMIDE-ADENINE-DINUCLEOTIDE, ... | 著者 | Read, J.A, Gingell, H, Madhavapeddi, P, Shirude, P.S. | 登録日 | 2013-05-31 | 公開日 | 2013-12-11 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (1.89 Å) | 主引用文献 | Methyl-Thiazoles: A Novel Mode of Inhibition with the Potential to Develop Novel Inhibitors Targeting Inha in Mycobacterium Tuberculosis. J.Med.Chem., 56, 2013
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1E5I
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![BU of 1e5i by Molmil](/molmil-images/mine/1e5i) | DELTA-R306 DEACETOXYCEPHALOSPORIN C SYNTHASE COMPLEXED WITH IRON AND 2-OXOGLUTARATE. | 分子名称: | 2-OXOGLUTARIC ACID, DEACETOXYCEPHALOSPORIN C SYNTHASE, FE (II) ION | 著者 | Lee, H.J, Lloyd, M.D, Harlos, K, Clifton, I.J, Baldwin, J.E, Schofield, C.J. | 登録日 | 2000-07-26 | 公開日 | 2001-07-26 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Kinetic and Crystallographic Studies on Deacetoxycephalosporin C Synthase (Daocs) J.Mol.Biol., 308, 2001
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1E5H
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![BU of 1e5h by Molmil](/molmil-images/mine/1e5h) | DELTA-R307A DEACETOXYCEPHALOSPORIN C SYNTHASE COMPLEXED WITH SUCCINATE AND CARBON DIOXIDE | 分子名称: | CARBON DIOXIDE, DEACETOXYCEPHALOSPORIN C SYNTHASE, FE (II) ION, ... | 著者 | Lee, H.J, Lloyd, M.D, Harlos, K, Clifton, I.J, Baldwin, J.E, Schofield, C.J. | 登録日 | 2000-07-26 | 公開日 | 2001-07-26 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (1.96 Å) | 主引用文献 | Kinetic and Crystallographic Studies on Deacetoxycephalosporin C Synthase (Daocs) J.Mol.Biol., 308, 2001
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4NKN
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3OQV
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![BU of 3oqv by Molmil](/molmil-images/mine/3oqv) | AlbC, a cyclodipeptide synthase from Streptomyces noursei | 分子名称: | AlbC, DITHIANE DIOL, PHOSPHATE ION | 著者 | Sauguet, L, Ledu, M.H, Charbonnier, J.B, Gondry, M. | 登録日 | 2010-09-04 | 公開日 | 2011-02-16 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Cyclodipeptide synthases, a family of class-I aminoacyl-tRNA synthetase-like enzymes involved in non-ribosomal peptide synthesis. Nucleic Acids Res., 39, 2011
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4MOT
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4OE9
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4P2I
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![BU of 4p2i by Molmil](/molmil-images/mine/4p2i) | Crystal structure of the mouse SNX19 PX domain | 分子名称: | MKIAA0254 protein | 著者 | Collins, B.M. | 登録日 | 2014-03-04 | 公開日 | 2014-09-03 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Structural Basis for Different Phosphoinositide Specificities of the PX Domains of Sorting Nexins Regulating G-protein Signaling. J.Biol.Chem., 289, 2014
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4P2J
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6XS7
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![BU of 6xs7 by Molmil](/molmil-images/mine/6xs7) | Crystal structure of human Vps29 complexed with RaPID-derived cyclic peptide RT-D2 | 分子名称: | 48V-DTY-THR-THR-ILE-TYR-TRP-THR-PRO-LEU-GLY-THR-PHE-PRO-ARG-ILE-ARG, FORMIC ACID, GLYCEROL, ... | 著者 | Chen, K.-E, Guo, Q, Collins, B.M. | 登録日 | 2020-07-15 | 公開日 | 2021-07-14 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.58 Å) | 主引用文献 | De novo macrocyclic peptides for inhibiting, stabilizing, and probing the function of the retromer endosomal trafficking complex. Sci Adv, 7, 2021
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6XSA
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![BU of 6xsa by Molmil](/molmil-images/mine/6xsa) | Crystal structure of human Vps29 complexed with RaPID-derived cyclic peptide RT-L2 | 分子名称: | 48V-TYR-LEU-PRO-THR-ILE-THR-GLY-VAL-GLY-HIS-LEU-TRP-HIS-PRO-LEU, SULFATE ION, Vacuolar protein sorting-associated protein 29 | 著者 | Chen, K.-E, Guo, Q, Collins, B.M. | 登録日 | 2020-07-15 | 公開日 | 2021-07-14 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.83 Å) | 主引用文献 | De novo macrocyclic peptides for inhibiting, stabilizing, and probing the function of the retromer endosomal trafficking complex. Sci Adv, 7, 2021
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6XS5
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![BU of 6xs5 by Molmil](/molmil-images/mine/6xs5) | Crystal structure of human Vps29 complexed with RaPID-derived cyclic peptide RT-D1 | 分子名称: | 48V-DTY-ILE-ILE-ASP-THR-PRO-LEU-GLY-VAL-PHE-LEU-SER-SER-LEU-LYS-ARG, FORMIC ACID, GLYCEROL, ... | 著者 | Chen, K.-E, Guo, Q, Collins, B.M. | 登録日 | 2020-07-15 | 公開日 | 2021-07-14 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.01 Å) | 主引用文献 | De novo macrocyclic peptides for inhibiting, stabilizing, and probing the function of the retromer endosomal trafficking complex. Sci Adv, 7, 2021
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6XS8
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![BU of 6xs8 by Molmil](/molmil-images/mine/6xs8) | Crystal structure of Chaetomium thermophilum Vps29 complexed with RaPID-derived cyclic peptide RT-D3 | 分子名称: | 48V-DTY-GLY-TYR-ASP-PRO-LEU-GLY-LEU-LYS-TYR-PHE-ALA, Vacuolar protein sorting-associated protein 29 | 著者 | Chen, K.-E, Guo, Q, Collins, B.M. | 登録日 | 2020-07-15 | 公開日 | 2021-07-14 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.95009851 Å) | 主引用文献 | De novo macrocyclic peptides for inhibiting, stabilizing, and probing the function of the retromer endosomal trafficking complex. Sci Adv, 7, 2021
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6XS9
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![BU of 6xs9 by Molmil](/molmil-images/mine/6xs9) | Crystal structure of human Vps29 complexed with RaPID-derived cyclic peptide RT-L1 | 分子名称: | 1,4,7,10,13,16-HEXAOXACYCLOOCTADECANE, 48V-TYR-ILE-LYS-THR-PRO-LEU-GLY-THR-PHE-PRO-ASN-ARG-HIS-GLY, GLYCEROL, ... | 著者 | Chen, K.-E, Guo, Q, Collins, B.M. | 登録日 | 2020-07-15 | 公開日 | 2021-07-21 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.69 Å) | 主引用文献 | De novo macrocyclic peptides for inhibiting, stabilizing, and probing the function of the retromer endosomal trafficking complex. Sci Adv, 7, 2021
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7YAC
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![BU of 7yac by Molmil](/molmil-images/mine/7yac) | Paltusotine-bound SSTR2-Gi complex | 分子名称: | Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2, Guanine nucleotide-binding protein G(I)/G(S)/G(T) subunit beta-1, Guanine nucleotide-binding protein G(i) subunit alpha-1, ... | 著者 | Zhao, J, Shao, Z. | 登録日 | 2022-06-27 | 公開日 | 2023-04-19 | 最終更新日 | 2023-09-27 | 実験手法 | ELECTRON MICROSCOPY (3.24 Å) | 主引用文献 | Prospect of acromegaly therapy: molecular mechanism of clinical drugs octreotide and paltusotine. Nat Commun, 14, 2023
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7YAE
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![BU of 7yae by Molmil](/molmil-images/mine/7yae) | Octreotide-bound SSTR2-Gi complex | 分子名称: | CHOLESTEROL, DPN-CYS-PHE-DTR-LYS-THR-CYS-THO, Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2, ... | 著者 | Zhao, J, Shao, Z. | 登録日 | 2022-06-28 | 公開日 | 2023-04-19 | 実験手法 | ELECTRON MICROSCOPY (3.37 Å) | 主引用文献 | Prospect of acromegaly therapy: molecular mechanism of clinical drugs octreotide and paltusotine. Nat Commun, 14, 2023
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7X31
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7X4B
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![BU of 7x4b by Molmil](/molmil-images/mine/7x4b) | Crystal Structure of An Anti-CRISPR Protein | 分子名称: | Anti-CRISPR protein (AcrIIC1), SULFATE ION | 著者 | Hu, J, Zhang, S, Gao, J.Y, Liu, X, Liu, J. | 登録日 | 2022-03-02 | 公開日 | 2022-10-26 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.61 Å) | 主引用文献 | A redox switch regulates the assembly and anti-CRISPR activity of AcrIIC1. Nat Commun, 13, 2022
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2HGO
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![BU of 2hgo by Molmil](/molmil-images/mine/2hgo) | NMR structure of Cassiicolin | 分子名称: | 1,5-anhydro-3-O-methyl-D-mannitol, CASSIICOLIN | 著者 | Barthe, P, Pujade-Renault, V, Roumestand, C, de Lamotte, F. | 登録日 | 2006-06-27 | 公開日 | 2007-02-27 | 最終更新日 | 2020-07-29 | 実験手法 | SOLUTION NMR | 主引用文献 | Structural Analysis of Cassiicolin, a Host-selective Protein Toxin from Corynespora cassiicola J.Mol.Biol., 367, 2007
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1HJG
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![BU of 1hjg by Molmil](/molmil-images/mine/1hjg) | Alteration of the co-substrate selectivity of deacetoxycephalosporin C synthase: The role of arginine-258 | 分子名称: | 3-METHYL-2-OXOBUTANOIC ACID, DEACETOXYCEPHALOSPORIN C SYNTHASE, FE (II) ION | 著者 | Lee, H.J, Lloyd, M.D, Clifton, I.J, Harlos, K, Dubus, A, Baldwin, J.E, Frere, J.M, Schofield, C.J. | 登録日 | 2001-01-15 | 公開日 | 2001-06-01 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Alteration of the 2-Oxoacid Cosubstrate Selectivity in Deacetoxycephalosporin C Synthase: The Role of Arginine-258 J.Biol.Chem., 276, 2001
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