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3FDM
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alpha/beta foldamer in complex with Bcl-xL
分子名称: 1,2-ETHANEDIOL, Apoptosis regulator Bcl-X, alpha/beta-peptide foldamer
著者Fairlie, W.D, Lee, E.F, Smith, B.J, Czabotar, P.E, Colman, P.M, Sadowsky, J.D, Peterson-Kaufman, K.J, Gellman, S.H.
登録日2008-11-26
公開日2009-03-10
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.26 Å)
主引用文献High-Resolution Structural Characterization of a Helical alpha/beta-Peptide Foldamer Bound to the Anti-Apoptotic Protein Bcl-x(L)
Angew.Chem.Int.Ed.Engl., 48, 2009
2JM6
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BU of 2jm6 by Molmil
Solution structure of MCL-1 complexed with NOXAB
分子名称: Myeloid cell leukemia-1 protein Mcl-1 homolog, Noxa
著者Czabotar, P.E, Lee, E.F, van Delft, M.F, Day, C.L, Smith, B.J, Huang, D.C.S, Fairlie, W.D, Hinds, M.G, Colman, P.M.
登録日2006-10-17
公開日2007-03-20
最終更新日2023-12-20
実験手法SOLUTION NMR
主引用文献Structural insights into the degradation of Mcl-1 induced by BH3 domains
Proc.Natl.Acad.Sci.Usa, 104, 2007
2WLO
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BU of 2wlo by Molmil
POTASSIUM CHANNEL FROM MAGNETOSPIRILLUM MAGNETOTACTICUM
分子名称: POTASSIUM CHANNEL, POTASSIUM ION
著者Clarke, O.B, Caputo, A.T, Smith, B.J, Gulbis, J.M.
登録日2009-06-24
公開日2010-06-23
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (4.036 Å)
主引用文献Domain Reorientation and Rotation of an Intracellular Assembly Regulate Conduction in Kir Potassium Channels.
Cell(Cambridge,Mass.), 141, 2010
2X6A
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BU of 2x6a by Molmil
Potassium Channel from Magnetospirillum Magnetotacticum
分子名称: ATP-SENSITIVE INWARD RECTIFIER POTASSIUM CHANNEL 10, PHOSPHOCHOLINE, POTASSIUM ION
著者Clarke, O.B, Caputo, A.T, Hill, A.P, Vandenberg, J.I, Smith, B.J, Gulbis, J.M.
登録日2010-02-15
公開日2010-06-23
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献Domain Reorientation and Rotation of an Intracellular Assembly Regulate Conduction in Kir Potassium Channels.
Cell(Cambridge,Mass.), 141, 2010
2X6B
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BU of 2x6b by Molmil
Potassium Channel from Magnetospirillum Magnetotacticum
分子名称: ATP-SENSITIVE INWARD RECTIFIER POTASSIUM CHANNEL 10, BARIUM ION, PHOSPHOCHOLINE, ...
著者Clarke, O.B, Caputo, A.T, Hill, A.P, Vandenberg, J.I, Smith, B.J, Gulbis, J.M.
登録日2010-02-15
公開日2010-06-23
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (3.3 Å)
主引用文献Domain Reorientation and Rotation of an Intracellular Assembly Regulate Conduction in Kir Potassium Channels.
Cell(Cambridge,Mass.), 141, 2010
2WLN
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BU of 2wln by Molmil
POTASSIUM CHANNEL FROM MAGNETOSPIRILLUM MAGNETOTACTICUM
分子名称: POTASSIUM CHANNEL, POTASSIUM ION
著者Clarke, O.B, Caputo, A.T, Smith, B.J, Gulbis, J.M.
登録日2009-06-24
公開日2010-06-09
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (3.44 Å)
主引用文献Domain Reorientation and Rotation of an Intracellular Assembly Regulate Conduction in Kir Potassium Channels.
Cell(Cambridge,Mass.), 141, 2010
2WLI
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BU of 2wli by Molmil
POTASSIUM CHANNEL FROM MAGNETOSPIRILLUM MAGNETOTACTICUM
分子名称: KIRBAC3.1 POTASSIUM CHANNEL, POTASSIUM CHANNEL, POTASSIUM ION
著者Clarke, O.B, Caputo, A.T, Smith, B.J, Gulbis, J.M.
登録日2009-06-24
公開日2010-06-09
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (3.09 Å)
主引用文献Domain Reorientation and Rotation of an Intracellular Assembly Regulate Conduction in Kir Potassium Channels.
Cell(Cambridge,Mass.), 141, 2010
2WLH
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BU of 2wlh by Molmil
POTASSIUM CHANNEL FROM MAGNETOSPIRILLUM MAGNETOTACTICUM
分子名称: CHLORIDE ION, POTASSIUM CHANNEL, POTASSIUM ION
著者Clarke, O.B, Caputo, A.T, Smith, B.J, Gulbis, J.M.
登録日2009-06-24
公開日2010-06-09
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (3.28 Å)
主引用文献Domain Reorientation and Rotation of an Intracellular Assembly Regulate Conduction in Kir Potassium Channels.
Cell(Cambridge,Mass.), 141, 2010
2WLL
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BU of 2wll by Molmil
POTASSIUM CHANNEL FROM BURKHOLDERIA PSEUDOMALLEI
分子名称: DIUNDECYL PHOSPHATIDYL CHOLINE, MAGNESIUM ION, POTASSIUM CHANNEL, ...
著者Clarke, O.B, Caputo, A.T, Hill, A.P, VandenBerg, J.I, Smith, B.J, Gulbis, J.M.
登録日2009-06-24
公開日2010-06-09
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (3.65 Å)
主引用文献Domain Reorientation and Rotation of an Intracellular Assembly Regulate Conduction in Kir Potassium Channels.
Cell(Cambridge,Mass.), 141, 2010
2WLM
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POTASSIUM CHANNEL FROM MAGNETOSPIRILLUM MAGNETOTACTICUM
分子名称: POTASSIUM CHANNEL, POTASSIUM ION
著者Clarke, O.B, Caputo, A.T, Smith, B.J, Gulbis, J.M.
登録日2009-06-24
公開日2010-06-09
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (3.61 Å)
主引用文献Domain Reorientation and Rotation of an Intracellular Assembly Regulate Conduction in Kir Potassium Channels.
Cell(Cambridge,Mass.), 141, 2010
2X6C
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BU of 2x6c by Molmil
Potassium Channel from Magnetospirillum Magnetotacticum
分子名称: ATP-SENSITIVE INWARD RECTIFIER POTASSIUM CHANNEL 10, CHLORIDE ION, PHOSPHOCHOLINE, ...
著者Clarke, O.B, Caputo, A.T, Hill, A.P, Vandenberg, J.I, Smith, B.J, Gulbis, J.M.
登録日2010-02-15
公開日2010-06-23
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Domain Reorientation and Rotation of an Intracellular Assembly Regulate Conduction in Kir Potassium Channels.
Cell(Cambridge,Mass.), 141, 2010
7KD6
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BU of 7kd6 by Molmil
Insulin Receptor L1-CR plus alphaCT fragment in co-complex with Fv 83-7 and single-chain insulin SCI-b
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Lawrence, M.C, Menting, J.G.
登録日2020-10-08
公開日2021-10-13
最終更新日2024-10-09
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Single-chain insulin analogs threaded by the insulin receptor alpha CT domain.
Biophys.J., 2022
4WAT
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BU of 4wat by Molmil
Crystal structure of PfRh5, an essential P. falciparum ligand for invasion of human erythrocytes
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, IMIDAZOLE, PfRh5
著者Chen, L.
登録日2014-09-01
公開日2014-10-22
最終更新日2024-10-16
実験手法X-RAY DIFFRACTION (2.18 Å)
主引用文献Crystal structure of PfRh5, an essential P. falciparum ligand for invasion of human erythrocytes.
Elife, 3, 2014
4BD7
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BU of 4bd7 by Molmil
Bax domain swapped dimer induced by octylmaltoside
分子名称: APOPTOSIS REGULATOR BAX, CHLORIDE ION, PRASEODYMIUM ION
著者Czabotar, P.E, Westphal, D, Adams, J.M, Colman, P.M.
登録日2012-10-05
公開日2013-02-13
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.801 Å)
主引用文献Bax Crystal Structures Reveal How Bh3 Domains Activate Bax and Nucleate its Oligomerization to Induce Apoptosis.
Cell(Cambridge,Mass.), 152, 2013
4BD2
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BU of 4bd2 by Molmil
Bax domain swapped dimer in complex with BidBH3
分子名称: APOPTOSIS REGULATOR BAX, BH3-INTERACTING DOMAIN DEATH AGONIST
著者Czabotar, P.E, Westphal, D, Adams, J.M, Colman, P.M.
登録日2012-10-04
公開日2013-02-13
最終更新日2024-05-01
実験手法X-RAY DIFFRACTION (2.206 Å)
主引用文献Bax Crystal Structures Reveal How Bh3 Domains Activate Bax and Nucleate its Oligomerization to Induce Apoptosis.
Cell(Cambridge,Mass.), 152, 2013
4BD6
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BU of 4bd6 by Molmil
Bax domain swapped dimer in complex with BaxBH3
分子名称: APOPTOSIS REGULATOR BAX
著者Czabotar, P.E, Westphal, D, Adams, J.M, Colman, P.M.
登録日2012-10-05
公開日2013-02-13
最終更新日2024-05-01
実験手法X-RAY DIFFRACTION (2.494 Å)
主引用文献Bax Crystal Structures Reveal How Bh3 Domains Activate Bax and Nucleate its Oligomerization to Induce Apoptosis.
Cell(Cambridge,Mass.), 152, 2013
5WBT
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BU of 5wbt by Molmil
Solution Structure and Dynamics of an Ultra-Stable Single-Chain Insulin Analog STUDIES OF AN ENGINEERED MONOMER AND IMPLICATIONS FOR RECEPTOR BINDING
分子名称: Insulin
著者Glidden, M.D, Yang, Y, Wickramasinghe, N.P, Weiss, M.A.
登録日2017-06-29
公開日2017-11-15
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献Solution structure of an ultra-stable single-chain insulin analog connects protein dynamics to a novel mechanism of receptor binding.
J. Biol. Chem., 293, 2018
4QVX
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BU of 4qvx by Molmil
Discovery of a Potent and Selective BCL-XL Inhibitor That Demonstrates Thrombocytopenia and Inhibits Tumor Growth in Vivo
分子名称: 2-[8-(1,3-benzothiazol-2-ylcarbamoyl)-3,4-dihydroisoquinolin-2(1H)-yl]-5-(3-{4-[3-(dimethylamino)prop-1-yn-1-yl]-2-fluorophenoxy}propyl)-1,3-thiazole-4-carboxylic acid, Bcl-2-like protein 1
著者Park, C.H.
登録日2014-07-16
公開日2015-07-22
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Discovery of a Potent and Selective BCL-XL Inhibitor with in Vivo Activity.
ACS MED.CHEM.LETT., 5, 2014
5JYQ
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BU of 5jyq by Molmil
Structure of Conus Geographus insulin G1
分子名称: Insulin 1, Insulin 1b, SULFATE ION
著者Lawrence, M.C, Menting, J, Norton, R.S, Safavi-Hemami, H.
登録日2016-05-15
公開日2016-09-07
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献A minimized human insulin-receptor-binding motif revealed in a Conus geographus venom insulin.
Nat.Struct.Mol.Biol., 23, 2016
5J3H
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BU of 5j3h by Molmil
Human insulin receptor domains L1-CR in complex with peptide S519C16 and 83-7 Fv
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-3)-[alpha-D-mannopyranose-(1-6)]beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Lawrence, M, Menting, J, Lawrence, C.
登録日2016-03-30
公開日2016-06-15
最終更新日2024-10-16
実験手法X-RAY DIFFRACTION (3.27 Å)
主引用文献Insulin Mimetic Peptide Disrupts the Primary Binding Site of the Insulin Receptor.
J.Biol.Chem., 291, 2016
2TMP
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BU of 2tmp by Molmil
N-TERMINAL DOMAIN OF TISSUE INHIBITOR OF METALLOPROTEINASE-2 (N-TIMP-2), NMR, 49 STRUCTURES
分子名称: TISSUE INHIBITOR OF METALLOPROTEINASES-2
著者Muskett, F.W, Frenkiel, T.A, Feeney, J, Freedman, R.B, Carr, M.D, Williamson, R.A.
登録日1998-05-26
公開日1998-12-09
最終更新日2022-03-16
実験手法SOLUTION NMR
主引用文献High resolution structure of the N-terminal domain of tissue inhibitor of metalloproteinases-2 and characterization of its interaction site with matrix metalloproteinase-3.
J.Biol.Chem., 273, 1998
6VEP
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BU of 6vep by Molmil
Human insulin in complex with the human insulin microreceptor in turn in complex with Fv 83-7
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Lawrence, M.C, Menting, J.G.T.
登録日2020-01-02
公開日2020-06-03
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献A structurally minimized yet fully active insulin based on cone-snail venom insulin principles.
Nat.Struct.Mol.Biol., 27, 2020
6UXQ
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BU of 6uxq by Molmil
Crystal structure of BAK core domain BH3-groove-dimer in complex with POPC and C8E4
分子名称: (HYDROXYETHYLOXY)TRI(ETHYLOXY)OCTANE, 1,2-ETHANEDIOL, 1-palmitoyl-2-oleoyl-sn-glycero-3-phosphocholine, ...
著者Cowan, A.D, Colman, P.M, Czabotar, P.E.
登録日2019-11-07
公開日2020-09-02
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (1.696 Å)
主引用文献BAK core dimers bind lipids and can be bridged by them.
Nat.Struct.Mol.Biol., 27, 2020
6UXN
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BU of 6uxn by Molmil
Crystal structure of BAK core domain BH3-groove-dimer in complex with phosphatidylserine
分子名称: Bcl-2 homologous antagonist/killer, GLYCEROL, O-[(R)-{[(2R)-2,3-bis(octanoyloxy)propyl]oxy}(hydroxy)phosphoryl]-L-serine, ...
著者Cowan, A.D, Colman, P.M, Czabotar, P.E.
登録日2019-11-07
公開日2020-09-02
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2.49 Å)
主引用文献BAK core dimers bind lipids and can be bridged by them.
Nat.Struct.Mol.Biol., 27, 2020
6VET
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BU of 6vet by Molmil
Human insulin analog: [GluB10,HisA8,ArgA9,TyrB20]-DOI
分子名称: Insulin A chain, Insulin B chain
著者Menting, J.G, Chou, D.H.-C, Lawrence, M.C, Xiong, X.
登録日2020-01-02
公開日2020-06-03
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (1.46 Å)
主引用文献A structurally minimized yet fully active insulin based on cone-snail venom insulin principles.
Nat.Struct.Mol.Biol., 27, 2020

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