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7YP5
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Crystal structure of elaiophylin glycosyltransferase in complex with TDP
分子名称: CHLORIDE ION, Glycosyltransferase, R-1,2-PROPANEDIOL, ...
著者Xu, T, Liu, Q, Gan, Q, Liu, J.
登録日2022-08-02
公開日2022-11-02
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.33 Å)
主引用文献Substrate-induced dimerization of elaiophylin glycosyltransferase reveals a novel self-activating form of glycosyltransferase for symmetric glycosylation.
Acta Crystallogr D Struct Biol, 78, 2022
7YP4
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Crystal structure of elaiophylin glycosyltransferase in apo-form
分子名称: Glycosyltransferase, R-1,2-PROPANEDIOL
著者Xu, T, Liu, Q, Gan, Q, Liu, J.
登録日2022-08-02
公開日2022-11-02
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献Substrate-induced dimerization of elaiophylin glycosyltransferase reveals a novel self-activating form of glycosyltransferase for symmetric glycosylation.
Acta Crystallogr D Struct Biol, 78, 2022
7WLK
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BU of 7wlk by Molmil
CryoEM structure of human low-voltage activated T-type calcium channel Cav3.3 in complex with Otilonium Bromide(OB)
分子名称: 1,2-Distearoyl-sn-glycerophosphoethanolamine, 2-[diethyl(methyl)-$l^{4}-azanyl]ethyl 4-[(2-octoxyphenyl)carbonylamino]benzoate, 2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者He, L, Yu, Z, Dong, Y, Chen, Q, Zhao, Y.
登録日2022-01-13
公開日2022-05-04
最終更新日2022-05-25
実験手法ELECTRON MICROSCOPY (3.6 Å)
主引用文献Structure, gating, and pharmacology of human Ca V 3.3 channel.
Nat Commun, 13, 2022
7WLI
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CryoEM structure of human low-voltage activated T-type calcium channel CaV3.3 (apo)
分子名称: 1,2-Distearoyl-sn-glycerophosphoethanolamine, 2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, ...
著者He, L, Yu, Z, Dong, Y, Chen, Q, Zhao, Y.
登録日2022-01-13
公開日2022-05-04
最終更新日2022-05-25
実験手法ELECTRON MICROSCOPY (3.3 Å)
主引用文献Structure, gating, and pharmacology of human Ca V 3.3 channel.
Nat Commun, 13, 2022
7WLL
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CryoEM structure of human low-voltage activated T-type calcium channel Cav3.3 in complex with pimozide(PMZ)
分子名称: 1,2-Distearoyl-sn-glycerophosphoethanolamine, 2-acetamido-2-deoxy-beta-D-glucopyranose, 3-[1-[4,4-bis(4-fluorophenyl)butyl]piperidin-4-yl]-1~{H}-benzimidazol-2-one, ...
著者He, L, Yu, Z, Dong, Y, Chen, Q, Zhao, Y.
登録日2022-01-13
公開日2022-05-04
最終更新日2022-05-25
実験手法ELECTRON MICROSCOPY (3.6 Å)
主引用文献Structure, gating, and pharmacology of human Ca V 3.3 channel.
Nat Commun, 13, 2022
7WLJ
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CryoEM structure of human low-voltage activated T-type calcium channel Cav3.3 in complex with mibefradil (MIB)
分子名称: (1S,2S)-2-(2-{[3-(1H-benzimidazol-2-yl)propyl](methyl)amino}ethyl)-6-fluoro-1-(propan-2-yl)-1,2,3,4-tetrahydronaphthalen-2-yl methoxyacetate, 1,2-Distearoyl-sn-glycerophosphoethanolamine, 2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者He, L, Yu, Z, Dong, Y, Chen, Q, Zhao, Y.
登録日2022-01-13
公開日2022-05-04
最終更新日2022-05-25
実験手法ELECTRON MICROSCOPY (3.9 Å)
主引用文献Structure, gating, and pharmacology of human Ca V 3.3 channel.
Nat Commun, 13, 2022
7JTN
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BU of 7jtn by Molmil
Human Complement Factor B Inhibited by a Slow Off-Rate Modified Aptamer of 29 Bases
分子名称: Complement factor B, DNA (30-MER)
著者Xu, X, Geisbrecht, B.V.
登録日2020-08-18
公開日2020-12-09
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献Inhibition of the Complement Alternative Pathway by Chemically Modified DNA Aptamers That Bind with Picomolar Affinity to Factor B.
J Immunol., 206, 2021
6IH0
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BU of 6ih0 by Molmil
Aquifex aeolicus LpxC complex with ACHN-975
分子名称: N-[(2S)-3-azanyl-3-methyl-1-(oxidanylamino)-1-oxidanylidene-butan-2-yl]-4-[4-[(1R,2R)-2-(hydroxymethyl)cyclopropyl]buta -1,3-diynyl]benzamide, UDP-3-O-acyl-N-acetylglucosamine deacetylase, ZINC ION, ...
著者Li, D.Y, Fan, S, Jin, Y.Y, Zhang, C, Lv, G.X, Wu, G.T, Yang, Z.Y.
登録日2018-09-27
公開日2019-01-30
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (1.21 Å)
主引用文献The Complex Structure of Protein AaLpxC from Aquifex aeolicus with ACHN-975 Molecule Suggests an Inhibitory Mechanism at Atomic-Level against Gram-Negative Bacteria
Molecules, 26, 2021
7EN0
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BU of 7en0 by Molmil
Structure and Activity of SLAC1 Channels for Stomatal Signaling in Leaves
分子名称: DIUNDECYL PHOSPHATIDYL CHOLINE, SLow Anion Channel 1, SPHINGOSINE
著者Deng, Y, Kashtoh, H, Wang, Q, Zhen, G, Li, Q, Tang, L, Gao, H, Zhang, C, Qin, L, Su, M, Li, F, Huang, X, Wang, Y, Xie, Q, Clarke, O.B, Hendrickson, W.A, Chen, Y.
登録日2021-04-15
公開日2021-05-19
最終更新日2024-06-05
実験手法ELECTRON MICROSCOPY (2.97 Å)
主引用文献Structure and activity of SLAC1 channels for stomatal signaling in leaves.
Proc.Natl.Acad.Sci.USA, 118, 2021
5CM4
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BU of 5cm4 by Molmil
Crystal structure of human Frizzled 4 Cysteine-Rich Domain (CRD)
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Frizzled-4
著者Ke, J, Parker, N, Gu, X, Zhang, C, Melcher, K, Xu, H.E.
登録日2015-07-16
公開日2015-08-12
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Structural basis of the Norrin-Frizzled 4 interaction.
Cell Res., 25, 2015
7BYI
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BU of 7byi by Molmil
Structure of SHMT2 in complex with CBX
分子名称: CARBENOXOLONE, DI(HYDROXYETHYL)ETHER, PHOSPHATE ION, ...
著者Li, L, Chen, Y, Lu, D, Zhang, C, Su, D.
登録日2020-04-23
公開日2021-09-15
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.76 Å)
主引用文献Structure of SHMT2 with CBX
To Be Published

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件を2024-07-24に公開中

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