1X96
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![BU of 1x96 by Molmil](/molmil-images/mine/1x96) | Crystal structure of Aldose Reductase with citrates bound in the active site | 分子名称: | CITRIC ACID, NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, aldose reductase | 著者 | El-Kabbani, O, Darmanin, C, Oka, M, Schulze-Briese, C, Tomizaki, T, Hazemann, I, Mitschler, A, Podjarny, A. | 登録日 | 2004-08-19 | 公開日 | 2004-09-07 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.4 Å) | 主引用文献 | High-Resolution Structures of Human Aldose Reductase Holoenzyme in Complex with Stereoisomers of the Potent Inhibitor Fidarestat: Stereospecific Interaction between the Enzyme and a Cyclic Imide Type Inhibitor J.Med.Chem., 47, 2004
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1X98
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![BU of 1x98 by Molmil](/molmil-images/mine/1x98) | Crystal structure of Aldose Reductase complexed with 2S4R (Stereoisomer of Fidarestat, 2S4S) | 分子名称: | (2S,4R)-2-AMINOFORMYL-6-FLUORO-SPIRO[CHROMAN-4,4'-IMIDAZOLIDINE]-2',5'-DIONE, Aldose Reductase, CITRIC ACID, ... | 著者 | El-Kabbani, O, Darmanin, C, Oka, M, Schulze-Briese, C, Tomizaki, T, Hazemann, I, Mitschler, A, Podjarny, A. | 登録日 | 2004-08-19 | 公開日 | 2004-09-07 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.3 Å) | 主引用文献 | High-Resolution Structures of Human Aldose Reductase Holoenzyme in Complex with Stereoisomers of the Potent Inhibitor Fidarestat: Stereospecific Interaction between the Enzyme and a Cyclic Imide Type Inhibitor J.Med.Chem., 47, 2004
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7F1I
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![BU of 7f1i by Molmil](/molmil-images/mine/7f1i) | Designed enzyme RA61 M48K/I72D mutant: form II | 分子名称: | Engineered Retroaldolase | 著者 | Fujioka, T, Oka, M, Numoto, N, Ito, N, Oda, M, Tanaka, F. | 登録日 | 2021-06-09 | 公開日 | 2021-11-24 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.4 Å) | 主引用文献 | Varying the Directionality of Protein Catalysts for Aldol and Retro-Aldol Reactions. Chembiochem, 23, 2022
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7F1H
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![BU of 7f1h by Molmil](/molmil-images/mine/7f1h) | Designed enzyme RA61 M48K/I72D mutant: form I | 分子名称: | Engineered Retroaldolase, FORMIC ACID, GLYCEROL | 著者 | Fujioka, T, Oka, M, Numoto, N, Ito, N, Oda, M, Tanaka, F. | 登録日 | 2021-06-09 | 公開日 | 2021-11-24 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.14 Å) | 主引用文献 | Varying the Directionality of Protein Catalysts for Aldol and Retro-Aldol Reactions. Chembiochem, 23, 2022
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7F1J
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![BU of 7f1j by Molmil](/molmil-images/mine/7f1j) | Designed enzyme RA61 M48K/I72D mutant: form III | 分子名称: | Engineered Retroaldolase | 著者 | Fujioka, T, Oka, M, Numoto, N, Ito, N, Oda, M, Tanaka, F. | 登録日 | 2021-06-09 | 公開日 | 2021-11-24 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Varying the Directionality of Protein Catalysts for Aldol and Retro-Aldol Reactions. Chembiochem, 23, 2022
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7F1K
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![BU of 7f1k by Molmil](/molmil-images/mine/7f1k) | Designed enzyme RA61 M48K/I72D mutant: form IV | 分子名称: | Engineered Retroaldolase | 著者 | Fujioka, T, Oka, M, Numoto, N, Ito, N, Oda, M, Tanaka, F. | 登録日 | 2021-06-09 | 公開日 | 2021-11-24 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.05 Å) | 主引用文献 | Varying the Directionality of Protein Catalysts for Aldol and Retro-Aldol Reactions. Chembiochem, 23, 2022
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7F1L
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![BU of 7f1l by Molmil](/molmil-images/mine/7f1l) | Designed enzyme RA61 M48K/I72D mutant: form V | 分子名称: | CHLORIDE ION, Engineered Retroaldolase, IMIDAZOLE | 著者 | Fujioka, T, Oka, M, Numoto, N, Ito, N, Oda, M, Tanaka, F. | 登録日 | 2021-06-09 | 公開日 | 2021-11-24 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Varying the Directionality of Protein Catalysts for Aldol and Retro-Aldol Reactions. Chembiochem, 23, 2022
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3WQH
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![BU of 3wqh by Molmil](/molmil-images/mine/3wqh) | Crystal Structure of human DPP-IV in complex with Anagliptin | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, Dipeptidyl peptidase 4, N-[2-({2-[(2S)-2-cyanopyrrolidin-1-yl]-2-oxoethyl}amino)-2-methylpropyl]-2-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide | 著者 | Watanabe, Y.S, Okada, S, Motoyama, T, Takahashi, R, Adachi, H, Oka, M. | 登録日 | 2014-01-27 | 公開日 | 2015-07-15 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.85 Å) | 主引用文献 | Anagliptin, a potent dipeptidyl peptidase IV inhibitor: its single-crystal structure and enzyme interactions. J Enzyme Inhib Med Chem, 30, 2015
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5XB7
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![BU of 5xb7 by Molmil](/molmil-images/mine/5xb7) | GH42 alpha-L-arabinopyranosidase from Bifidobacterium animalis subsp. lactis Bl-04 | 分子名称: | Beta-galactosidase, GLYCEROL, SULFATE ION | 著者 | Viborg, A.H, Katayama, T, Arakawa, T, Abou Hachem, M, Lo Leggio, L, Kitaoka, M, Svensson, B, Fushinobu, S. | 登録日 | 2017-03-16 | 公開日 | 2017-11-01 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Discovery of alpha-l-arabinopyranosidases from human gut microbiome expands the diversity within glycoside hydrolase family 42. J. Biol. Chem., 292, 2017
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5X6V
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![BU of 5x6v by Molmil](/molmil-images/mine/5x6v) | Crystal structure of human heteroheptameric complex | 分子名称: | ACETATE ION, Ragulator complex protein LAMTOR1, Ragulator complex protein LAMTOR2, ... | 著者 | Yonehara, R, Nada, S, Nakai, T, Nakai, M, Kitamura, A, Ogawa, A, Nakatsumi, H, Nakayama, K.I, Li, S, Standley, D.M, Yamashita, E, Nakagawa, A, Okada, M. | 登録日 | 2017-02-23 | 公開日 | 2017-12-06 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.02 Å) | 主引用文献 | Structural basis for the assembly of the Ragulator-Rag GTPase complex. Nat Commun, 8, 2017
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4WH2
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![BU of 4wh2 by Molmil](/molmil-images/mine/4wh2) | N-acetylhexosamine 1-kinase in complex with ADP | 分子名称: | ACETIC ACID, ADENOSINE-5'-DIPHOSPHATE, GLYCEROL, ... | 著者 | Sato, M, Arakawa, T, Nam, Y.W, Nishimoto, M, Kitaoka, M, Fushinobu, S. | 登録日 | 2014-09-19 | 公開日 | 2015-02-18 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (1.847 Å) | 主引用文献 | Open-close structural change upon ligand binding and two magnesium ions required for the catalysis of N-acetylhexosamine 1-kinase Biochim.Biophys.Acta, 1854, 2015
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4WH1
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![BU of 4wh1 by Molmil](/molmil-images/mine/4wh1) | N-Acetylhexosamine 1-kinase (ligand free) | 分子名称: | ACETIC ACID, GLYCEROL, N-acetylhexosamine 1-kinase | 著者 | Sato, M, Arakawa, T, Nam, Y.W, Nishimoto, M, Kitaoka, M, Fushinobu, S. | 登録日 | 2014-09-19 | 公開日 | 2015-02-11 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (2.05 Å) | 主引用文献 | Open-close structural change upon ligand binding and two magnesium ions required for the catalysis of N-acetylhexosamine 1-kinase Biochim.Biophys.Acta, 1854, 2015
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4WH3
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![BU of 4wh3 by Molmil](/molmil-images/mine/4wh3) | N-acetylhexosamine 1-kinase in complex with ATP | 分子名称: | ACETIC ACID, ADENOSINE-5'-TRIPHOSPHATE, GLYCEROL, ... | 著者 | Sato, M, Arakawa, T, Nam, Y.W, Nishimoto, M, Kitaoka, M, Fushinobu, S. | 登録日 | 2014-09-19 | 公開日 | 2015-02-18 | 最終更新日 | 2020-02-05 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Open-close structural change upon ligand binding and two magnesium ions required for the catalysis of N-acetylhexosamine 1-kinase Biochim.Biophys.Acta, 1854, 2015
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5B3A
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![BU of 5b3a by Molmil](/molmil-images/mine/5b3a) | Crystal Structure of O-Phoshoserine Sulfhydrylase from Aeropyrum pernix in Complexed with the alpha-Aminoacrylate Intermediate | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, 2-{[(E)-{3-hydroxy-2-methyl-5-[(phosphonooxy)methyl]pyridin-4-yl}methylidene]amino}prop-2-enoic acid, Protein CysO | 著者 | Nakamura, T, Takeda, E, Kawai, Y, Kataoka, M, Ishikawa, K. | 登録日 | 2016-02-12 | 公開日 | 2016-03-16 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.14 Å) | 主引用文献 | Role of F225 in O-phosphoserine sulfhydrylase from Aeropyrum pernix K1 Extremophiles, 20, 2016
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5AZZ
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![BU of 5azz by Molmil](/molmil-images/mine/5azz) | Crystal structure of seleno-insulin | 分子名称: | Insulin A chain, Insulin B chain | 著者 | Watanabe, S, Okumura, M, Arai, K, Takei, T, Asahina, Y, Hojo, H, Iwaoka, M, Inaba, K. | 登録日 | 2015-10-23 | 公開日 | 2017-05-03 | 最終更新日 | 2017-06-14 | 実験手法 | X-RAY DIFFRACTION (1.45 Å) | 主引用文献 | Preparation of Selenoinsulin as a Long-Lasting Insulin Analogue. Angew. Chem. Int. Ed. Engl., 56, 2017
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8OZ0
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![BU of 8oz0 by Molmil](/molmil-images/mine/8oz0) | Structure of a human 48S translation initiation complex with eIF4F and eIF4A | 分子名称: | 18S rRNA, 40S ribosomal protein S10, 40S ribosomal protein S11, ... | 著者 | Brito Querido, J, Sokabe, M, Diaz-Lopez, I, Gordiyenko, Y, Fraser, C.S, Ramakrishnan, V. | 登録日 | 2023-05-06 | 公開日 | 2024-02-07 | 最終更新日 | 2024-04-24 | 実験手法 | ELECTRON MICROSCOPY (3.5 Å) | 主引用文献 | The structure of a human translation initiation complex reveals two independent roles for the helicase eIF4A. Nat.Struct.Mol.Biol., 31, 2024
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1C1B
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![BU of 1c1b by Molmil](/molmil-images/mine/1c1b) | CRYSTAL STRUCTURE OF HIV-1 REVERSE TRANSCRIPTASE IN COMPLEX WITH GCA-186 | 分子名称: | 6-(3',5'-DIMETHYLBENZYL)-1-ETHOXYMETHYL-5-ISOPROPYLURACIL, HIV-1 REVERSE TRANSCRIPTASE (A-CHAIN), HIV-1 REVERSE TRANSCRIPTASE (B-CHAIN) | 著者 | Hopkins, A.L, Ren, J, Tanaka, H, Baba, B, Okamato, M, Stuart, D.I, Stammers, D.K. | 登録日 | 1999-07-21 | 公開日 | 2000-07-21 | 最終更新日 | 2014-11-12 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Design of MKC-442 (emivirine) analogues with improved activity against drug-resistant HIV mutants. J.Med.Chem., 42, 1999
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3ED1
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![BU of 3ed1 by Molmil](/molmil-images/mine/3ed1) | Crystal Structure of Rice GID1 complexed with GA3 | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, GIBBERELLIN A3, Gibberellin receptor GID1, ... | 著者 | Shimada, A, Nakatsu, T, Ueguchi-Tanaka, M, Kato, H, Matsuoka, M. | 登録日 | 2008-09-02 | 公開日 | 2008-11-25 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Structural basis for gibberellin recognition by its receptor GID1. Nature, 456, 2008
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3EBL
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![BU of 3ebl by Molmil](/molmil-images/mine/3ebl) | Crystal Structure of Rice GID1 complexed with GA4 | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, GIBBERELLIN A4, Gibberellin receptor GID1, ... | 著者 | Shimada, A, Nakatsu, T, Ueguchi-Tanaka, M, Kato, H, Matsuoka, M. | 登録日 | 2008-08-28 | 公開日 | 2008-11-25 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Structural basis for gibberellin recognition by its receptor GID1. Nature, 456, 2008
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7DZY
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![BU of 7dzy by Molmil](/molmil-images/mine/7dzy) | Spike protein from SARS-CoV2 with Fab fragment of enhancing antibody 2490 | 分子名称: | Fab Heavy chain of enhancing antibody 2490, Fab light chain of enhancing antibody 2490, Spike glycoprotein | 著者 | Liu, Y, Soh, W.T, Li, S, Kishikawa, J, Hirose, M, Kato, T, Standley, D, Okada, M, Arase, H. | 登録日 | 2021-01-26 | 公開日 | 2021-06-02 | 最終更新日 | 2024-06-05 | 実験手法 | ELECTRON MICROSCOPY (3.6 Å) | 主引用文献 | An infectivity-enhancing site on the SARS-CoV-2 spike protein targeted by antibodies. Cell, 184, 2021
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7DZW
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![BU of 7dzw by Molmil](/molmil-images/mine/7dzw) | Apo spike protein from SARS-CoV2 | 分子名称: | Spike glycoprotein | 著者 | Liu, Y, Soh, W.T, Li, S, Kishikawa, J, Hirose, M, Kato, T, Standley, D, Okada, M, Arase, H. | 登録日 | 2021-01-26 | 公開日 | 2021-06-02 | 最終更新日 | 2024-03-27 | 実験手法 | ELECTRON MICROSCOPY (3.45 Å) | 主引用文献 | An infectivity-enhancing site on the SARS-CoV-2 spike protein targeted by antibodies. Cell, 184, 2021
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7DZX
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![BU of 7dzx by Molmil](/molmil-images/mine/7dzx) | Spike protein from SARS-CoV2 with Fab fragment of enhancing antibody 8D2 | 分子名称: | Fab Heavy chain of enhancing antibody, Fab light chain of enhancing antibody, Spike glycoprotein | 著者 | Liu, Y, Soh, W.T, Li, S, Kishikawa, J, Hirose, M, Kato, T, Standley, D, Okada, M, Arase, H. | 登録日 | 2021-01-26 | 公開日 | 2021-06-02 | 最終更新日 | 2024-03-27 | 実験手法 | ELECTRON MICROSCOPY (3.53 Å) | 主引用文献 | An infectivity-enhancing site on the SARS-CoV-2 spike protein targeted by antibodies. Cell, 184, 2021
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3EQN
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![BU of 3eqn by Molmil](/molmil-images/mine/3eqn) | Crystal structure of beta-1,3-glucanase from Phanerochaete chrysosporium (Lam55A) | 分子名称: | ACETATE ION, GLYCEROL, Glucan 1,3-beta-glucosidase, ... | 著者 | Ishida, T, Fushinobu, S, Kawai, R, Kitaoka, M, Igarashi, K, Samejima, M. | 登録日 | 2008-10-01 | 公開日 | 2009-02-03 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Crystal structure of glycoside hydrolase family 55 beta -1,3-glucanase from the basidiomycete Phanerochaete chrysosporium J.Biol.Chem., 284, 2009
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3EQO
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![BU of 3eqo by Molmil](/molmil-images/mine/3eqo) | Crystal structure of beta-1,3-glucanase from Phanerochaete chrysosporium (Lam55A) gluconolactone complex | 分子名称: | D-glucono-1,5-lactone, Glucan 1,3-beta-glucosidase, ZINC ION, ... | 著者 | Ishida, T, Fushinobu, S, Kawai, R, Kitaoka, M, Igarashi, K, Samejima, M. | 登録日 | 2008-10-01 | 公開日 | 2009-02-03 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (2.25 Å) | 主引用文献 | Crystal structure of glycoside hydrolase family 55 beta -1,3-glucanase from the basidiomycete Phanerochaete chrysosporium J.Biol.Chem., 284, 2009
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8R5J
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![BU of 8r5j by Molmil](/molmil-images/mine/8r5j) | Crystal structure of MERS-CoV main protease | 分子名称: | Non-structural protein 11 | 著者 | Balcomb, B.H, Fairhead, M, Koekemoer, L, Lithgo, R.M, Aschenbrenner, J.C, Chandran, A.V, Godoy, A.S, Lukacik, P, Marples, P.G, Mazzorana, M, Ni, X, Strain-Damerell, C, Thompson, W, Tomlinson, C.W.E, Wild, C, Winokan, M, Fearon, D, Walsh, M.A, von Delft, F. | 登録日 | 2023-11-16 | 公開日 | 2023-12-06 | 実験手法 | X-RAY DIFFRACTION (1.898 Å) | 主引用文献 | Crystal structure of MERS-CoV main protease To Be Published
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