4RSS
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![BU of 4rss by Molmil](/molmil-images/mine/4rss) | Crystal structure of tyrosine-protein kinase SYK with an inhibitor | 分子名称: | 1-[(3-methyl-1-{2-[(1,2,3-trimethyl-1H-indol-5-yl)amino]pyrimidin-4-yl}-1H-pyrazol-4-yl)methyl]azetidin-3-ol, Tyrosine-protein kinase SYK | 著者 | Lee, B.I, Lee, S.J, Choi, J.-S. | 登録日 | 2014-11-11 | 公開日 | 2015-10-21 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (1.83 Å) | 主引用文献 | Highly potent and selective pyrazolylpyrimidines as Syk kinase inhibitors. Bioorg.Med.Chem.Lett., 25, 2015
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7C90
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![BU of 7c90 by Molmil](/molmil-images/mine/7c90) | Crystal structure of Cytochrome CL from the marine methylotrophic bacterium Methylophaga aminisulfidivorans MPT (Ma-CytcL) | 分子名称: | 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, CALCIUM ION, Cytochrome c, ... | 著者 | Ghosh, S, Dhanasingh, I, Lee, S.H. | 登録日 | 2020-06-04 | 公開日 | 2020-07-22 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.13 Å) | 主引用文献 | Crystal Structure of CytochromecLfrom the Aquatic Methylotrophic BacteriumMethylophaga aminisulfidivoransMPT. J Microbiol Biotechnol., 30, 2020
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4HAC
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5YCN
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![BU of 5ycn by Molmil](/molmil-images/mine/5ycn) | Human PPARgamma ligand binding domain complexed with Lobeglitazone | 分子名称: | (5S)-5-[[4-[2-[[6-(4-methoxyphenoxy)pyrimidin-4-yl]-methyl-amino]ethoxy]phenyl]methyl]-1,3-thiazolidine-2,4-dione, Nuclear receptor coactivator 1, Peroxisome proliferator-activated receptor gamma | 著者 | Jang, J.Y, Han, B.W. | 登録日 | 2017-09-07 | 公開日 | 2018-09-12 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.15 Å) | 主引用文献 | Structural Basis for the Enhanced Anti-Diabetic Efficacy of Lobeglitazone on PPAR gamma. Sci Rep, 8, 2018
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5YCP
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3RUJ
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3RUI
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![BU of 3rui by Molmil](/molmil-images/mine/3rui) | Crystal structure of Atg7C-Atg8 complex | 分子名称: | Autophagy-related protein 8, Ubiquitin-like modifier-activating enzyme ATG7, ZINC ION | 著者 | Hong, S.B, Kim, B.W, Song, H.K. | 登録日 | 2011-05-05 | 公開日 | 2011-11-23 | 最終更新日 | 2013-07-03 | 実験手法 | X-RAY DIFFRACTION (1.906 Å) | 主引用文献 | Insights into noncanonical E1 enzyme activation from the structure of autophagic E1 Atg7 with Atg8. Nat.Struct.Mol.Biol., 18, 2011
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1CZV
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![BU of 1czv by Molmil](/molmil-images/mine/1czv) | CRYSTAL STRUCTURE OF THE C2 DOMAIN OF HUMAN COAGULATION FACTOR V: DIMERIC CRYSTAL FORM | 分子名称: | PROTEIN (COAGULATION FACTOR V) | 著者 | Macedo-Ribeiro, S, Bode, W, Huber, R, Kane, W.H, Fuentes-Prior, P. | 登録日 | 1999-09-07 | 公開日 | 1999-11-26 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Crystal structures of the membrane-binding C2 domain of human coagulation factor V. Nature, 402, 1999
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1CZT
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![BU of 1czt by Molmil](/molmil-images/mine/1czt) | CRYSTAL STRUCTURE OF THE C2 DOMAIN OF HUMAN COAGULATION FACTOR V | 分子名称: | PROTEIN (COAGULATION FACTOR V) | 著者 | Macedo-Ribeiro, S, Bode, W, Huber, R, Kane, W.H, Fuentes-Prior, P. | 登録日 | 1999-09-07 | 公開日 | 1999-11-26 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (1.87 Å) | 主引用文献 | Crystal structures of the membrane-binding C2 domain of human coagulation factor V. Nature, 402, 1999
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1CZS
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![BU of 1czs by Molmil](/molmil-images/mine/1czs) | CRYSTAL STRUCTURE OF THE C2 DOMAIN OF HUMAN COAGULATION FACTOR V: COMPLEX WITH PHENYLMERCURY | 分子名称: | PHENYLMERCURY, PROTEIN (COAGULATION FACTOR V) | 著者 | Macedo-Ribeiro, S, Bode, W, Huber, R, Kane, W.H, Fuentes-Prior, P. | 登録日 | 1999-09-07 | 公開日 | 1999-11-26 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Crystal structures of the membrane-binding C2 domain of human coagulation factor V. Nature, 402, 1999
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2AEB
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![BU of 2aeb by Molmil](/molmil-images/mine/2aeb) | Crystal structure of human arginase I at 1.29 A resolution and exploration of inhibition in immune response. | 分子名称: | 2(S)-AMINO-6-BORONOHEXANOIC ACID, Arginase 1, MANGANESE (II) ION | 著者 | Di Costanzo, L, Sabio, G, Mora, A, Rodriguez, P.C, Ochoa, A.C, Centeno, F, Christianson, D.W. | 登録日 | 2005-07-21 | 公開日 | 2005-09-06 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (1.29 Å) | 主引用文献 | Crystal structure of human arginase I at 1.29 A resolution and exploration of inhibition in the immune response. Proc.Natl.Acad.Sci.Usa, 102, 2005
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1WVA
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![BU of 1wva by Molmil](/molmil-images/mine/1wva) | Crystal structure of human arginase I from twinned crystal | 分子名称: | Arginase 1, MANGANESE (II) ION, S-2-(BORONOETHYL)-L-CYSTEINE | 著者 | Di Costanzo, L, Sabio, G, Mora, A, Rodriguez, P.C, Ochoa, A.C, Centeno, F, Christianson, D.W. | 登録日 | 2004-12-14 | 公開日 | 2005-09-06 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.94 Å) | 主引用文献 | Crystal structure of human arginase I at 1.29 A resolution and exploration of inhibition in the immune response Proc.Natl.Acad.Sci.Usa, 102, 2005
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5XM3
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![BU of 5xm3 by Molmil](/molmil-images/mine/5xm3) | Crystal Structure of Methanol dehydrogenase from Methylophaga aminisulfidivorans | 分子名称: | Glucose dehydrogenase, MAGNESIUM ION, Methanol dehydrogenase [cytochrome c] subunit 2, ... | 著者 | Cao, T.P, Choi, J.M, Lee, S.H. | 登録日 | 2017-05-12 | 公開日 | 2018-03-21 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.701 Å) | 主引用文献 | The crystal structure of methanol dehydrogenase, a quinoprotein from the marine methylotrophic bacterium Methylophaga aminisulfidivorans MPT J. Microbiol., 56, 2018
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7UFV
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![BU of 7ufv by Molmil](/molmil-images/mine/7ufv) | Crystal structure of the WDR domain of human DCAF1 in complex with OICR-6766 | 分子名称: | (3P)-N-[(1S)-3-amino-1-(3-chlorophenyl)-3-oxopropyl]-3-(2-fluorophenyl)-1H-pyrazole-4-carboxamide, DDB1- and CUL4-associated factor 1, UNKNOWN ATOM OR ION | 著者 | Kimani, S, Li, A, Li, Y, Dong, A, Hutchinson, A, Seitova, A, Wilson, B, Al-Awar, R, Vedadi, M, Brown, P, Arrowsmith, C.H, Edwards, A.M, Halabelian, L, Structural Genomics Consortium (SGC) | 登録日 | 2022-03-23 | 公開日 | 2022-05-04 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Discovery of Nanomolar DCAF1 Small Molecule Ligands. J.Med.Chem., 66, 2023
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