5DYA
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![BU of 5dya by Molmil](/molmil-images/mine/5dya) | Crystal structure of the human BRPF1 bromodomain in complex with SEED5 | 分子名称: | (2R)-2-ethyl-3-oxo-1,2,3,4-tetrahydroquinoxaline-6-carboxylic acid, NITRATE ION, Peregrin | 著者 | Zhu, J, Caflisch, A. | 登録日 | 2015-09-24 | 公開日 | 2016-05-25 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.65 Å) | 主引用文献 | Twenty Crystal Structures of Bromodomain and PHD Finger Containing Protein 1 (BRPF1)/Ligand Complexes Reveal Conserved Binding Motifs and Rare Interactions. J.Med.Chem., 59, 2016
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7RK6
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![BU of 7rk6 by Molmil](/molmil-images/mine/7rk6) | Aplysia Slo1 with Barium | 分子名称: | (1R)-2-{[(S)-{[(2S)-2,3-dihydroxypropyl]oxy}(hydroxy)phosphoryl]oxy}-1-[(hexadecanoyloxy)methyl]ethyl (9Z)-octadec-9-enoate, BARIUM ION, BK channel, ... | 著者 | Zhu, J, Srivastava, S, Cachau, R, Holmgren, M. | 登録日 | 2021-07-22 | 公開日 | 2022-06-22 | 最終更新日 | 2023-04-05 | 実験手法 | ELECTRON MICROSCOPY (2.91 Å) | 主引用文献 | CryoEM structure of Aplysia Slo1 with 0 mM Ba2+ at 2.91 A To Be Published
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7RJT
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![BU of 7rjt by Molmil](/molmil-images/mine/7rjt) | Aplysia Slo1 with Barium | 分子名称: | (1R)-2-{[(S)-{[(2S)-2,3-dihydroxypropyl]oxy}(hydroxy)phosphoryl]oxy}-1-[(hexadecanoyloxy)methyl]ethyl (9Z)-octadec-9-enoate, BARIUM ION, BK channel, ... | 著者 | Zhu, J, Srivastava, S, Cachau, R, Holmgren, M. | 登録日 | 2021-07-21 | 公開日 | 2022-06-22 | 最終更新日 | 2024-06-05 | 実験手法 | ELECTRON MICROSCOPY (2.93 Å) | 主引用文献 | CryoEM structure of Aplysia Slo1 with 10 mM Ba2+ at 2.93 A To Be Published
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5DY7
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![BU of 5dy7 by Molmil](/molmil-images/mine/5dy7) | |
5EPR
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![BU of 5epr by Molmil](/molmil-images/mine/5epr) | |
5ETD
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![BU of 5etd by Molmil](/molmil-images/mine/5etd) | |
5EVA
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![BU of 5eva by Molmil](/molmil-images/mine/5eva) | |
5EV9
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![BU of 5ev9 by Molmil](/molmil-images/mine/5ev9) | |
5EWW
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![BU of 5eww by Molmil](/molmil-images/mine/5eww) | Crystal structure of the human BRPF1 bromodomain in complex with SEED21 | 分子名称: | NITRATE ION, Peregrin, ~{N}-[(2~{R})-butan-2-yl]-1-methyl-[1,2,4]triazolo[4,3-a]quinoxalin-4-amine | 著者 | Zhu, J, Wiedmer, L, Caflisch, A. | 登録日 | 2015-11-21 | 公開日 | 2016-11-02 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.73 Å) | 主引用文献 | Crystal structure of the human BRPF1 bromodomain in complex with SEED21 To Be Published
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5EWH
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![BU of 5ewh by Molmil](/molmil-images/mine/5ewh) | |
5EWC
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![BU of 5ewc by Molmil](/molmil-images/mine/5ewc) | Crystal structure of the human BRPF1 bromodomain in complex with SEED17 | 分子名称: | NITRATE ION, Peregrin, ethyl (2~{R})-2-methyl-3-oxidanylidene-2,4-dihydro-1~{H}-quinoxaline-6-carboxylate | 著者 | Zhu, J, Caflisch, A. | 登録日 | 2015-11-20 | 公開日 | 2016-05-25 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | Twenty Crystal Structures of Bromodomain and PHD Finger Containing Protein 1 (BRPF1)/Ligand Complexes Reveal Conserved Binding Motifs and Rare Interactions. J.Med.Chem., 59, 2016
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5EWV
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![BU of 5ewv by Molmil](/molmil-images/mine/5ewv) | Crystal structure of the human BRPF1 bromodomain in complex with SEED20 | 分子名称: | 1,5-dimethyl-[1,2,4]triazolo[4,3-a]quinoline, NITRATE ION, Peregrin | 著者 | Zhu, J, Wiedmer, L, Caflisch, A. | 登録日 | 2015-11-21 | 公開日 | 2016-11-02 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.67 Å) | 主引用文献 | Crystal structure of the human BRPF1 bromodomain in complex with SEED20 To Be Published
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5ETB
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![BU of 5etb by Molmil](/molmil-images/mine/5etb) | |
5E3D
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![BU of 5e3d by Molmil](/molmil-images/mine/5e3d) | Crystal structure of the human BRPF1 bromodomain in complex with SEED7 | 分子名称: | 2,8-dithioxo-1,2,3,7,8,9-hexahydro-6H-purin-6-one, NITRATE ION, Peregrin | 著者 | Zhu, J, Caflisch, A. | 登録日 | 2015-10-02 | 公開日 | 2016-05-25 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.71 Å) | 主引用文献 | Twenty Crystal Structures of Bromodomain and PHD Finger Containing Protein 1 (BRPF1)/Ligand Complexes Reveal Conserved Binding Motifs and Rare Interactions. J.Med.Chem., 59, 2016
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5DYC
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![BU of 5dyc by Molmil](/molmil-images/mine/5dyc) | |
5EM3
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![BU of 5em3 by Molmil](/molmil-images/mine/5em3) | |
5EPS
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![BU of 5eps by Molmil](/molmil-images/mine/5eps) | |
5EQ1
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![BU of 5eq1 by Molmil](/molmil-images/mine/5eq1) | Crystal structure of the human BRPF1 bromodomain in complex with SEED12 | 分子名称: | 5-METHYL-1,2,4-TRIAZOLO[3,4-B]BENZOTHIAZOLE, NITRATE ION, Peregrin | 著者 | Zhu, J, Caflisch, A. | 登録日 | 2015-11-12 | 公開日 | 2016-05-25 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | Twenty Crystal Structures of Bromodomain and PHD Finger Containing Protein 1 (BRPF1)/Ligand Complexes Reveal Conserved Binding Motifs and Rare Interactions. J.Med.Chem., 59, 2016
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6JMT
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![BU of 6jmt by Molmil](/molmil-images/mine/6jmt) | Crystal structure of GIT/PIX complex | 分子名称: | ARF GTPase-activating protein GIT2, ZINC ION, beta PIX | 著者 | Zhu, J, Lin, L, Xia, Y, Zhang, R, Zhang, M. | 登録日 | 2019-03-13 | 公開日 | 2020-05-20 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | GIT/PIX Condensates Are Modular and Ideal for Distinct Compartmentalized Cell Signaling. Mol.Cell, 79, 2020
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6JMU
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![BU of 6jmu by Molmil](/molmil-images/mine/6jmu) | Crystal structure of GIT1/Paxillin complex | 分子名称: | ARF GTPase-activating protein GIT1, Paxillin | 著者 | Zhu, J, Lin, L, Xia, Y, Zhang, R, Zhang, M. | 登録日 | 2019-03-13 | 公開日 | 2020-05-20 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | GIT/PIX Condensates Are Modular and Ideal for Distinct Compartmentalized Cell Signaling. Mol.Cell, 79, 2020
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2QVO
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![BU of 2qvo by Molmil](/molmil-images/mine/2qvo) | Crystal structure of AF1382 from Archaeoglobus fulgidus | 分子名称: | Uncharacterized protein AF_1382 | 著者 | Zhu, J, Zhao, M, Fu, Z.-Q, Yang, H, Chang, J, Hao, X, Chen, L, Liu, Z.J, Rose, J.P, Wang, B.C, Southeast Collaboratory for Structural Genomics (SECSG) | 登録日 | 2007-08-08 | 公開日 | 2007-09-04 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Crystal structure of AF1382 from Archaeoglobus fulgidus. To be Published
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3RO3
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![BU of 3ro3 by Molmil](/molmil-images/mine/3ro3) | crystal structure of LGN/mInscuteable complex | 分子名称: | CHLORIDE ION, ETHANOL, G-protein-signaling modulator 2, ... | 著者 | Zhu, J, Wen, W, Shang, Y, Wei, Z, Pan, Z, Wang, W, Zhang, M. | 登録日 | 2011-04-25 | 公開日 | 2012-03-07 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (1.1 Å) | 主引用文献 | LGN/mInsc and LGN/NuMA complex structures suggest distinct functions in asymmetric cell division for the Par3/mInsc/LGN and G[alpha]i/LGN/NuMA pathways Mol.Cell, 43, 2011
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4HTX
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![BU of 4htx by Molmil](/molmil-images/mine/4htx) | Crystal structure of PDE2 catalytic domain in complex with BAY60-7550 | 分子名称: | 2-(3,4-dimethoxybenzyl)-7-[(2R,3R)-2-hydroxy-6-phenylhexan-3-yl]-5-methylimidazo[5,1-f][1,2,4]triazin-4(3H)-one, MAGNESIUM ION, ZINC ION, ... | 著者 | Zhu, J, Huang, Q. | 登録日 | 2012-11-02 | 公開日 | 2013-08-28 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | X-ray Crystal Structure of Phosphodiesterase 2 in Complex with a Highly Selective, Nanomolar Inhibitor Reveals a Binding-Induced Pocket Important for Selectivity. J.Am.Chem.Soc., 135, 2013
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4HTZ
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![BU of 4htz by Molmil](/molmil-images/mine/4htz) | Crystal structure of PDE2 catalytic domain in space group P1 | 分子名称: | MAGNESIUM ION, ZINC ION, cGMP-dependent 3',5'-cyclic phosphodiesterase | 著者 | Zhu, J, Huang, Q. | 登録日 | 2012-11-02 | 公開日 | 2013-08-28 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | X-ray Crystal Structure of Phosphodiesterase 2 in Complex with a Highly Selective, Nanomolar Inhibitor Reveals a Binding-Induced Pocket Important for Selectivity. J.Am.Chem.Soc., 135, 2013
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5YPR
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![BU of 5ypr by Molmil](/molmil-images/mine/5ypr) | Crystal Structure of PSD-95 SH3-GK domain in complex with a synthesized inhibitor | 分子名称: | Disks large homolog 4, Synthesized GK inhibitor | 著者 | Zhu, J, Zhou, Q, Shang, Y, Weng, Z, Zhu, R, Zhang, M. | 登録日 | 2017-11-02 | 公開日 | 2018-03-14 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.349 Å) | 主引用文献 | Synaptic Targeting and Function of SAPAPs Mediated by Phosphorylation-Dependent Binding to PSD-95 MAGUKs. Cell Rep, 21, 2017
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