5EU7
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![BU of 5eu7 by Molmil](/molmil-images/mine/5eu7) | Crystal structure of HIV-1 integrase catalytic core in complex with Fab | 分子名称: | FAB Heavy Chain, FAB light chain, Integrase | 著者 | Galilee, M, Griner, S.L, Stroud, R.M, Alian, A. | 登録日 | 2015-11-18 | 公開日 | 2016-09-28 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.64 Å) | 主引用文献 | The Preserved HTH-Docking Cleft of HIV-1 Integrase Is Functionally Critical. Structure, 24, 2016
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5OVN
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4B7O
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1MKA
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1MKB
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6EX9
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4PA1
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7JGV
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![BU of 7jgv by Molmil](/molmil-images/mine/7jgv) | CRYSTAL STRUCTURE OF BCL-XL IN COMPLEX WITH COMPOUND 1620116, CRYSTAL FORM 2 | 分子名称: | 6-[(8E)-8-{2-[4-(benzylcarbamoyl)-1,3-thiazol-2-yl]hydrazinylidene}-5,6,7,8-tetrahydronaphthalen-2-yl]-3-(2-phenylethoxy)pyridine-2-carboxylic acid, Bcl-2-like protein 1 | 著者 | Lee, M, Fairlie, W.D, Smith, B.J, Lee, E.F. | 登録日 | 2020-07-19 | 公開日 | 2021-02-24 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.05 Å) | 主引用文献 | Optimization of Benzothiazole and Thiazole Hydrazones as Inhibitors of Schistosome BCL-2. Acs Infect Dis., 7, 2021
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7JGW
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![BU of 7jgw by Molmil](/molmil-images/mine/7jgw) | Crystal structure of BCL-XL in complex with COMPOUND 1620116, CRYSTAL FORM 1 | 分子名称: | 6-[(8E)-8-{2-[4-(benzylcarbamoyl)-1,3-thiazol-2-yl]hydrazinylidene}-5,6,7,8-tetrahydronaphthalen-2-yl]-3-(2-phenylethoxy)pyridine-2-carboxylic acid, Bcl-2-like protein 1 | 著者 | Lee, M, Fairlie, W.D, Smith, B.J, Lee, E.F. | 登録日 | 2020-07-19 | 公開日 | 2021-02-24 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.3 Å) | 主引用文献 | Optimization of Benzothiazole and Thiazole Hydrazones as Inhibitors of Schistosome BCL-2. Acs Infect Dis., 7, 2021
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6XFM
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![BU of 6xfm by Molmil](/molmil-images/mine/6xfm) | Molecular structure of the core of amyloid-like fibrils formed by residues 111-214 of FUS | 分子名称: | RNA-binding protein FUS | 著者 | Tycko, R, Lee, M, Ghosh, U, Thurber, K, Kato, M. | 登録日 | 2020-06-15 | 公開日 | 2020-10-07 | 最終更新日 | 2024-03-06 | 実験手法 | ELECTRON MICROSCOPY (2.62 Å) | 主引用文献 | Molecular structure and interactions within amyloid-like fibrils formed by a low-complexity protein sequence from FUS. Nat Commun, 11, 2020
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7SP0
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6OWJ
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![BU of 6owj by Molmil](/molmil-images/mine/6owj) | Zn-mediated polymerization of human SFPQ | 分子名称: | Splicing factor, proline- and glutamine-rich, ZINC ION | 著者 | Lee, M. | 登録日 | 2019-05-10 | 公開日 | 2020-02-05 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (1.94 Å) | 主引用文献 | Structural basis of the zinc-induced cytoplasmic aggregation of the RNA-binding protein SFPQ. Nucleic Acids Res., 48, 2020
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6VVI
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6VVH
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5K3X
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![BU of 5k3x by Molmil](/molmil-images/mine/5k3x) | Crystal Structure of the sulfite dehydrogenase, SorT R78K mutant from Sinorhizobium meliloti | 分子名称: | (MOLYBDOPTERIN-S,S)-OXO-MOLYBDENUM, GLYCEROL, Putative sulfite oxidase | 著者 | Lee, M, McGrath, A, Maher, M. | 登録日 | 2016-05-20 | 公開日 | 2017-05-24 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | The central active site arginine in sulfite oxidizing enzymes alters kinetic properties by controlling electron transfer and redox interactions. Biochim. Biophys. Acta, 1859, 2017
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6NCQ
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8EZE
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5WPA
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![BU of 5wpa by Molmil](/molmil-images/mine/5wpa) | Structure of human SFPQ/PSPC1 heterodimer | 分子名称: | Paraspeckle component 1, Splicing factor, proline- and glutamine-rich | 著者 | Lee, M. | 登録日 | 2017-08-04 | 公開日 | 2018-03-21 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.29 Å) | 主引用文献 | Crystal structure of a SFPQ/PSPC1 heterodimer provides insights into preferential heterodimerization of human DBHS family proteins. J. Biol. Chem., 293, 2018
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8EZD
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4OCA
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![BU of 4oca by Molmil](/molmil-images/mine/4oca) | Cryatal structure of ArnB K188A complexted with PLP and UDP-Ara4N | 分子名称: | (2R,3R,4S,5S)-3,4-dihydroxy-5-[({3-hydroxy-2-methyl-5-[(phosphonooxy)methyl]pyridin-4-yl}methyl)amino]tetrahydro-2H-pyr an-2-yl [(2R,3S,4R,5R)-5-(2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)-3,4-dihydroxytetrahydrofuran-2-yl]methyl dihydrogen diphosphate, UDP-4-amino-4-deoxy-L-arabinose--oxoglutarate aminotransferase | 著者 | Sousa, M.C, Lee, M. | 登録日 | 2014-01-08 | 公開日 | 2014-03-12 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Structural Basis for Substrate Specificity in ArnB. A Key Enzyme in the Polymyxin Resistance Pathway of Gram-Negative Bacteria. Biochemistry, 53, 2014
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6YAR
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![BU of 6yar by Molmil](/molmil-images/mine/6yar) | Crystal structure of a Selenium-derivatized complex of the bacterial cellulose secretion regulators BcsR and BcsQ, crystallized in the presence of AppCp | 分子名称: | ADENOSINE-5'-TRIPHOSPHATE, Bacterial cellulose secretion regulator BcsQ, Bacterial cellulose secretion regulator BcsR, ... | 著者 | Caleechurn, M, Abidi, W, Zouhir, S, Roche, S, Krasteva, P.V. | 登録日 | 2020-03-12 | 公開日 | 2021-02-24 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Architecture and regulation of an enterobacterial cellulose secretion system. Sci Adv, 7, 2021
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6YB3
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![BU of 6yb3 by Molmil](/molmil-images/mine/6yb3) | Crystal structure of a native BcsRQ complex purified and crystallized in the absence of nucleotide | 分子名称: | ADENOSINE-5'-TRIPHOSPHATE, Bacterial cellulose secretion regulator BcsQ, Bacterial cellulose secretion regulator BcsR, ... | 著者 | Caleechurn, M, Abidi, W, Zouhir, S, Roche, S, Krasteva, P.V. | 登録日 | 2020-03-15 | 公開日 | 2021-02-24 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.59 Å) | 主引用文献 | Architecture and regulation of an enterobacterial cellulose secretion system. Sci Adv, 7, 2021
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6YB5
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![BU of 6yb5 by Molmil](/molmil-images/mine/6yb5) | Orthorhombic crystal structure of a native BcsRQ complex crystallized in the presence of ADP | 分子名称: | ADENOSINE-5'-TRIPHOSPHATE, Bacterial cellulose secretion regulator BcsQ, Bacterial cellulose secretion regulator BcsR, ... | 著者 | Caleechurn, M, Abidi, W, Zouhir, S, Roche, S, Krasteva, P.V. | 登録日 | 2020-03-15 | 公開日 | 2021-02-24 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.59 Å) | 主引用文献 | Architecture and regulation of an enterobacterial cellulose secretion system. Sci Adv, 7, 2021
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5DCK
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5AEQ
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![BU of 5aeq by Molmil](/molmil-images/mine/5aeq) | Neuronal calcium sensor (NCS-1)from Rattus norvegicus | 分子名称: | CALCIUM ION, NEURONAL CALCIUM SENSOR 1, SODIUM ION | 著者 | Saleem, M, Karuppiah, V, Pandalaneni, S, Burgoyne, R, Derrick, J.P, Lian, L.Y. | 登録日 | 2015-01-08 | 公開日 | 2015-02-18 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.95 Å) | 主引用文献 | Neuronal Calcium Sensor-1 Binds the D2 Dopamine Receptor and G-Protein-Coupled Receptor Kinase 1 (Grk1) Peptides Using Different Modes of Interactions. J.Biol.Chem., 290, 2015
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