6WNA
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![BU of 6wna by Molmil](/molmil-images/mine/6wna) | Next generation monomeric IgG4 Fc | 分子名称: | Beta-2-microglobulin, IgG receptor FcRn large subunit p51, Immunoglobulin heavy constant gamma 4, ... | 著者 | Oganesyan, V.Y, Shan, L, van Dyk, N, Dall'Acqua, W.F. | 登録日 | 2020-04-22 | 公開日 | 2021-09-15 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | In vivo pharmacokinetic enhancement of monomeric Fc and monovalent bispecific designs through structural guidance. Commun Biol, 4, 2021
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6WOL
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![BU of 6wol by Molmil](/molmil-images/mine/6wol) | Next generation monomeric IgG4 Fc bound to neonatal Fc receptor | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-3)-[2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-6)]beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[beta-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, Beta-2-microglobulin, IgG receptor FcRn large subunit p51, ... | 著者 | Oganesyan, V.Y, Shan, L, van Dyk, N, Dall'Acqua, W.F. | 登録日 | 2020-04-24 | 公開日 | 2021-09-15 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.49 Å) | 主引用文献 | In vivo pharmacokinetic enhancement of monomeric Fc and monovalent bispecific designs through structural guidance. Commun Biol, 4, 2021
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5HVW
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![BU of 5hvw by Molmil](/molmil-images/mine/5hvw) | Monomeric IgG4 Fc | 分子名称: | GLYCEROL, Ig gamma-4 chain C region, ZINC ION, ... | 著者 | Oganesyan, V.Y, Shan, L, Dall'Acqua, W.F. | 登録日 | 2016-01-28 | 公開日 | 2016-08-17 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (1.95 Å) | 主引用文献 | Generation and Characterization of an IgG4 Monomeric Fc Platform. Plos One, 11, 2016
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3K6F
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![BU of 3k6f by Molmil](/molmil-images/mine/3k6f) | |
3K5S
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![BU of 3k5s by Molmil](/molmil-images/mine/3k5s) | |
3K6I
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![BU of 3k6i by Molmil](/molmil-images/mine/3k6i) | |
3K5R
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![BU of 3k5r by Molmil](/molmil-images/mine/3k5r) | |
3K6D
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![BU of 3k6d by Molmil](/molmil-images/mine/3k6d) | |
6BTJ
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![BU of 6btj by Molmil](/molmil-images/mine/6btj) | |
4V0G
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![BU of 4v0g by Molmil](/molmil-images/mine/4v0g) | JAK3 in complex with a covalent EGFR inhibitor | 分子名称: | N-[3-(2-{3-amino-6-[1-(1-methylpiperidin-4-yl)-1H-pyrazol-4-yl]pyrazin-2-yl}-1H-benzimidazol-1-yl)phenyl]propanamide, TYROSINE-PROTEIN KINASE JAK3 | 著者 | Debreczeni, J.E, Hennessy, E.J, Chuaquini, C, Ashton, S, Coclough, N, Cross, D.A.E, Eberlein, C, Gingipalli, L, Klinowska, T.C.M, Orme, J.P, Sha, L, Wu, X. | 登録日 | 2014-09-16 | 公開日 | 2016-01-13 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | Utilisation of Structure Based Design to Identify Novel, Irreversible Inhibitors of the Epidermal Growth Factor Receptor (Egfr) Harboring the Gatekeeper T790M Mutation To be Published
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4H58
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![BU of 4h58 by Molmil](/molmil-images/mine/4h58) | BRAF in complex with compound 3 | 分子名称: | CHLORIDE ION, N-(4-{[(2-methoxyethyl)amino]methyl}phenyl)-6-(pyridin-4-yl)quinazolin-2-amine, Serine/threonine-protein kinase B-raf | 著者 | Vasbinder, M, Aquila, B, Augustin, M, Chueng, T, Cook, D, Drew, L, Fauber, B, Glossop, S, Godin, R, Grondine, M, Hennessy, E, Johannes, J, Lee, S, Lyne, P, Moertl, M, Omer, C, Palakurthi, S, Pontz, T, Read, J, Sha, L, Shen, M, Steinbacher, S, Wang, H, Wu, A, Ye, M, Bagal, B. | 登録日 | 2012-09-18 | 公開日 | 2013-02-27 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | Discovery and Optimization of a Novel Series of Potent Mutant B-Raf(V600E) Selective Kinase Inhibitors. J.Med.Chem., 56, 2013
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4OCS
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![BU of 4ocs by Molmil](/molmil-images/mine/4ocs) | Crystal structure of human Fab CAP256-VRC26.10, a potent V1V2-directed HIV-1 neutralizing antibody | 分子名称: | CAP256-VRC26.10 heavy chain, CAP256-VRC26.10 light chain | 著者 | Gorman, J, Doria-Rose, N.A, Schramm, C.A, Moore, P.L, Mascola, J.R, Shapiro, L, Morris, L, Kwong, P.D. | 登録日 | 2014-01-09 | 公開日 | 2014-02-26 | 最終更新日 | 2023-12-06 | 実験手法 | X-RAY DIFFRACTION (1.901 Å) | 主引用文献 | Developmental pathway for potent V1V2-directed HIV-neutralizing antibodies. Nature, 509, 2014
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4OCW
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![BU of 4ocw by Molmil](/molmil-images/mine/4ocw) | Crystal structure of human Fab CAP256-VRC26.06, a potent V1V2-directed HIV-1 neutralizing antibody | 分子名称: | CAP256-VRC26.06 heavy chain, CAP256-VRC26.06 light chain | 著者 | Gorman, J, Doria-Rose, N.A, Schramm, C.A, Moore, P.L, Mascola, J.R, Shapiro, L, Morris, L, Kwong, P.D. | 登録日 | 2014-01-09 | 公開日 | 2014-02-26 | 最終更新日 | 2023-12-06 | 実験手法 | X-RAY DIFFRACTION (3.001 Å) | 主引用文献 | Developmental pathway for potent V1V2-directed HIV-neutralizing antibodies. Nature, 509, 2014
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4O6M
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![BU of 4o6m by Molmil](/molmil-images/mine/4o6m) | Structure of AF2299, a CDP-alcohol phosphotransferase (CMP-bound) | 分子名称: | AF2299, a CDP-alcohol phosphotransferase, CALCIUM ION, ... | 著者 | Clarke, O.B, Sciara, G, Tomasek, D, Banerjee, S, Rajashankar, K.R, Shapiro, L, Mancia, F, New York Consortium on Membrane Protein Structure (NYCOMPS) | 登録日 | 2013-12-22 | 公開日 | 2014-05-14 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.901 Å) | 主引用文献 | Structural basis for catalysis in a CDP-alcohol phosphotransferase. Nat Commun, 5, 2014
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4O6N
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![BU of 4o6n by Molmil](/molmil-images/mine/4o6n) | Structure of AF2299, a CDP-alcohol phosphotransferase (CDP-bound) | 分子名称: | AF2299, a CDP-alcohol phosphotransferase, CALCIUM ION, ... | 著者 | Clarke, O.B, Sciara, G, Tomasek, D, Banerjee, S, Rajashankar, K.R, Shapiro, L, Mancia, F, New York Consortium on Membrane Protein Structure (NYCOMPS) | 登録日 | 2013-12-22 | 公開日 | 2014-05-14 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Structural basis for catalysis in a CDP-alcohol phosphotransferase. Nat Commun, 5, 2014
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7M8K
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![BU of 7m8k by Molmil](/molmil-images/mine/7m8k) | Cryo-EM structure of Brazil (P.1) SARS-CoV-2 spike glycoprotein variant in the prefusion state (1 RBD up) | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Spike glycoprotein | 著者 | Casner, R.G, Cerutti, G, Shapiro, L, Ho, D.D. | 登録日 | 2021-03-29 | 公開日 | 2021-05-05 | 最終更新日 | 2021-05-26 | 実験手法 | ELECTRON MICROSCOPY | 主引用文献 | Increased resistance of SARS-CoV-2 variant P.1 to antibody neutralization. Cell Host Microbe, 29, 2021
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1M0W
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![BU of 1m0w by Molmil](/molmil-images/mine/1m0w) | Yeast Glutathione Synthase Bound to gamma-glutamyl-cysteine, AMP-PNP and 2 Magnesium Ions | 分子名称: | GAMMA-GLUTAMYLCYSTEINE, MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, ... | 著者 | Gogos, A, Shapiro, L, Burley, S.K, New York SGX Research Center for Structural Genomics (NYSGXRC) | 登録日 | 2002-06-14 | 公開日 | 2002-12-11 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Large Conformational Changes in the Catalytic Cycle of Glutathione Synthase Structure, 10, 2002
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8DXS
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![BU of 8dxs by Molmil](/molmil-images/mine/8dxs) | |
8DW9
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![BU of 8dw9 by Molmil](/molmil-images/mine/8dw9) | |
8DWA
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![BU of 8dwa by Molmil](/molmil-images/mine/8dwa) | |
4FMK
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![BU of 4fmk by Molmil](/molmil-images/mine/4fmk) | Crystal structure of mouse nectin-2 extracellular fragment D1-D2 | 分子名称: | CADMIUM ION, Poliovirus receptor-related protein 2, alpha-D-mannopyranose-(1-3)-[alpha-D-mannopyranose-(1-6)]beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Harrison, O.J, Brasch, J, Shapiro, L. | 登録日 | 2012-06-17 | 公開日 | 2012-08-22 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.56 Å) | 主引用文献 | Nectin ectodomain structures reveal a canonical adhesive interface. Nat.Struct.Mol.Biol., 19, 2012
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4FMT
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![BU of 4fmt by Molmil](/molmil-images/mine/4fmt) | |
4FOM
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![BU of 4fom by Molmil](/molmil-images/mine/4fom) | Crystal structure of human nectin-3 full ectodomain (D1-D3) | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, Poliovirus receptor-related protein 3, alpha-D-mannopyranose-(1-3)-[alpha-D-mannopyranose-(1-6)]beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Harrison, O.J, Jin, X, Brasch, J, Shapiro, L. | 登録日 | 2012-06-20 | 公開日 | 2012-08-22 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (3.93 Å) | 主引用文献 | Nectin ectodomain structures reveal a canonical adhesive interface. Nat.Struct.Mol.Biol., 19, 2012
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4FQP
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![BU of 4fqp by Molmil](/molmil-images/mine/4fqp) | Crystal structure of human Nectin-like 5 full ectodomain (D1-D3) | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Poliovirus receptor, ... | 著者 | Harrison, O.J, Jin, X, Brasch, J, Shapiro, L. | 登録日 | 2012-06-25 | 公開日 | 2012-08-22 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (3.6 Å) | 主引用文献 | Nectin ectodomain structures reveal a canonical adhesive interface. Nat.Struct.Mol.Biol., 19, 2012
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4FN0
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![BU of 4fn0 by Molmil](/molmil-images/mine/4fn0) | Crystal structure of mouse nectin-2 extracellular fragment D1-D2, 2nd crystal form | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, Poliovirus receptor-related protein 2, beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose | 著者 | Harrison, O.J, Brasch, J, Shapiro, L. | 登録日 | 2012-06-18 | 公開日 | 2012-08-22 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (3.35 Å) | 主引用文献 | Nectin ectodomain structures reveal a canonical adhesive interface. Nat.Struct.Mol.Biol., 19, 2012
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