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6ZPC
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BU of 6zpc by Molmil
Cyanophage S-2L HD phosphohydrolase (DatZ) bound to dATP
分子名称: 2'-DEOXYADENOSINE 5'-TRIPHOSPHATE, DatZ, LITHIUM ION, ...
著者Czernecki, D, Legrand, P, Delarue, M.
登録日2020-07-08
公開日2021-03-03
最終更新日2024-05-15
実験手法X-RAY DIFFRACTION (1.2683593 Å)
主引用文献How cyanophage S-2L rejects adenine and incorporates 2-aminoadenine to saturate hydrogen bonding in its DNA.
Nat Commun, 12, 2021
6ZP9
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BU of 6zp9 by Molmil
Cyanophage S-2L Primase-Polymerase (PrimPol), AEP domain (PP-N190)
分子名称: CALCIUM ION, PrimPol AEP domain (PP-N190)
著者Czernecki, D, Legrand, P, Delarue, M.
登録日2020-07-08
公開日2021-03-03
最終更新日2024-05-15
実験手法X-RAY DIFFRACTION (1.50002229 Å)
主引用文献How cyanophage S-2L rejects adenine and incorporates 2-aminoadenine to saturate hydrogen bonding in its DNA.
Nat Commun, 12, 2021
6ZPB
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BU of 6zpb by Molmil
Cyanophage S-2L HD phosphohydrolase (DatZ) bound to dA and two catalytic Co2+ ions
分子名称: (2R,3S,5R)-5-(6-amino-9H-purin-9-yl)-tetrahydro-2-(hydroxymethyl)furan-3-ol, COBALT (II) ION, DatZ
著者Czernecki, D, Legrand, P, Delarue, M.
登録日2020-07-08
公開日2021-03-03
最終更新日2024-05-15
実験手法X-RAY DIFFRACTION (1.72097385 Å)
主引用文献How cyanophage S-2L rejects adenine and incorporates 2-aminoadenine to saturate hydrogen bonding in its DNA.
Nat Commun, 12, 2021
4D3E
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BU of 4d3e by Molmil
Tetramer of IpaD, modified from 2J0O, fitted into negative stain electron microscopy reconstruction of the wild type tip complex from the type III secretion system of Shigella flexneri
分子名称: INVASIN IPAD
著者Cheung, M, Shen, D.-K, Makino, F, Kato, T, Roehrich, D, Martinez-Argudo, I, Walker, M.L, Murillo, I, Liu, X, Pain, M, Brown, J, Frazer, G, Mantell, J, Mina, P, Todd, T, Sessions, R.B, Namba, K, Blocker, A.J.
登録日2014-10-21
公開日2014-12-10
最終更新日2024-05-08
実験手法ELECTRON MICROSCOPY (24 Å)
主引用文献Three-Dimensional Electron Microscopy Reconstruction and Cysteine-Mediated Crosslinking Provide a Model of the T3Ss Needle Tip Complex.
Mol.Microbiol., 95, 2015
6I8Z
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BU of 6i8z by Molmil
Crystal structure of PTK2 in complex with BI-4464.
分子名称: 3-methoxy-~{N}-(1-methylpiperidin-1-ium-4-yl)-4-[[4-[(3-oxidanylidene-1,2-dihydroinden-4-yl)oxy]-5-(trifluoromethyl)pyrimidin-2-yl]amino]benzamide, Focal adhesion kinase 1
著者Bader, G, Zoephel, A.
登録日2018-11-21
公開日2019-02-20
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.99 Å)
主引用文献Highly Selective PTK2 Proteolysis Targeting Chimeras to Probe Focal Adhesion Kinase Scaffolding Functions.
J.Med.Chem., 62, 2019
6GO3
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BU of 6go3 by Molmil
TdT chimera (Loop1 of pol mu) - apoenzyme
分子名称: DNA nucleotidylexotransferase,DNA-directed DNA/RNA polymerase mu,DNA nucleotidylexotransferase
著者Loc'h, J, Gerodimos, C.A, Rosario, S, Lieber, M.R, Delarue, M.
登録日2018-06-01
公開日2019-06-05
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Structural evidence for an intransbase selection mechanism involving Loop1 in polymerase mu at an NHEJ double-strand break junction.
J.Biol.Chem., 294, 2019
6GO4
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BU of 6go4 by Molmil
TdT chimera (Loop1 of pol mu) - binary complex with ddCTP
分子名称: 2',3'-DIDEOXYCYTIDINE 5'-TRIPHOSPHATE, DNA nucleotidylexotransferase,DNA-directed DNA/RNA polymerase mu,DNA nucleotidylexotransferase, MAGNESIUM ION, ...
著者Loc'h, J, Gerodimos, C.A, Rosario, S, Lieber, M.R, Delarue, M.
登録日2018-06-01
公開日2019-06-05
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.96 Å)
主引用文献Structural evidence for an intransbase selection mechanism involving Loop1 in polymerase mu at an NHEJ double-strand break junction.
J.Biol.Chem., 294, 2019
6GO5
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BU of 6go5 by Molmil
TdT chimera (Loop1 of pol mu) - Ternary complex with 1-nt gapped DNA substrate
分子名称: 2'-deoxy-5'-O-[(S)-hydroxy{[(S)-hydroxy(phosphonooxy)phosphoryl]methyl}phosphoryl]cytidine, DNA (5'-D(*AP*CP*AP*GP*CP*G)-3'), DNA (5'-D(*CP*GP*CP*TP*GP*GP*CP*AP*AP*AP*CP*A)-3'), ...
著者Loc'h, J, Gerodimos, C.A, Rosario, S, Lieber, M.R, Delarue, M.
登録日2018-06-01
公開日2019-06-05
最終更新日2024-05-15
実験手法X-RAY DIFFRACTION (2.35 Å)
主引用文献Structural evidence for an intransbase selection mechanism involving Loop1 in polymerase mu at an NHEJ double-strand break junction.
J.Biol.Chem., 294, 2019
6GO6
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BU of 6go6 by Molmil
TdT chimera (Loop1 of pol mu) - ternary complex with downstream dsDNA
分子名称: 2',3'-DIDEOXYCYTIDINE 5'-TRIPHOSPHATE, DNA (5'-D(*AP*AP*AP*AP*AP*C)-3'), DNA (5'-D(*TP*TP*TP*TP*TP*GP*GP*C)-3'), ...
著者Loc'h, J, Gerodimos, C.A, Rosario, S, Lieber, M.R, Delarue, M.
登録日2018-06-01
公開日2019-06-05
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.09 Å)
主引用文献Structural evidence for an intransbase selection mechanism involving Loop1 in polymerase mu at an NHEJ double-strand break junction.
J.Biol.Chem., 294, 2019
6GO7
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BU of 6go7 by Molmil
TdT chimera (Loop1 of pol mu) - full DNA synapsis complex
分子名称: 2',3'-DIDEOXYCYTIDINE 5'-TRIPHOSPHATE, DNA (5'-D(*AP*AP*AP*AP*AP*C)-3'), DNA (5'-D(*TP*TP*TP*TP*TP*GP*C)-3'), ...
著者Loc'h, J, Gerodimos, C.A, Rosario, S, Lieber, M.R, Delarue, M.
登録日2018-06-01
公開日2019-06-05
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.55 Å)
主引用文献Structural evidence for an intransbase selection mechanism involving Loop1 in polymerase mu at an NHEJ double-strand break junction.
J.Biol.Chem., 294, 2019
2J9T
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BU of 2j9t by Molmil
BipD of Burkholderia Pseudomallei
分子名称: BORIC ACID, CITRATE ANION, MEMBRANE ANTIGEN
著者Johnson, S, Roversi, P, Field, T, Deane, J.E, Galyov, E, Lea, S.M.
登録日2006-11-16
公開日2006-11-20
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Self-Chaperoning of the Type III Secretion System Needle Tip Proteins Ipad and Bipd.
J.Biol.Chem., 282, 2007
4K13
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BU of 4k13 by Molmil
Structure of HCAIX mimic (HCAII with 5 mutations in active site) in complex with dorzolamide
分子名称: (4S-TRANS)-4-(ETHYLAMINO)-5,6-DIHYDRO-6-METHYL-4H-THIENO(2,3-B)THIOPYRAN-2-SULFONAMIDE-7,7-DIOXIDE, Carbonic anhydrase 2, DIMETHYL SULFOXIDE, ...
著者Biswas, S, McKenna, R.
登録日2013-04-04
公開日2014-04-09
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Developing isoform specific inhibitors for hCAIX using CAIX mimic
To be Published
4K1Q
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BU of 4k1q by Molmil
Structure of hCAIX mimic (hCAII with 5 mutations in active site)
分子名称: Carbonic anhydrase 2, ZINC ION
著者Biswas, S, McKenna, R.
登録日2013-04-05
公開日2014-04-09
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.699 Å)
主引用文献Developing isoform specific inhibitors for hCAIX using CAIX mimic
To be Published
4K0Z
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BU of 4k0z by Molmil
Structure of HCAIX mimic (HCAII with 5 mutations in active site) in complex with methazolamide
分子名称: Carbonic anhydrase 2, DIMETHYL SULFOXIDE, N-(3-methyl-5-sulfamoyl-1,3,4-thiadiazol-2(3H)-ylidene)acetamide, ...
著者Biswas, S, McKenna, R.
登録日2013-04-04
公開日2014-04-09
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.799 Å)
主引用文献Developing isoform specific inhibitors for hCAIX using CAIX mimic
To be Published
4K0T
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BU of 4k0t by Molmil
Structure of HCAIX mimic (HCAII with 5 mutations in active site) in complex with chlorzolamide
分子名称: 5-(2-chlorophenyl)-1,3,4-thiadiazole-2-sulfonamide, Carbonic anhydrase 2, DIMETHYL SULFOXIDE, ...
著者Biswas, S, McKenna, R.
登録日2013-04-04
公開日2014-04-09
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.78 Å)
主引用文献Designing isoform specific inhibitors against hCAIX using CAIX mimic
To be Published
4K0S
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BU of 4k0s by Molmil
Structure of HCAIX mimic (HCAII with 5 mutations in active site) in complex with acetazolamide
分子名称: 5-ACETAMIDO-1,3,4-THIADIAZOLE-2-SULFONAMIDE, Carbonic anhydrase 2, ZINC ION
著者Biswas, S, McKenna, R.
登録日2013-04-04
公開日2014-04-09
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.802 Å)
主引用文献Developing isoform specific inhibitors against hCAIX using CAIX mimic
To be Published
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件を2024-06-26に公開中

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