6TX9
| |
6TX8
| |
6TX6
| |
6TXX
| CRYSTAL STRUCTURE OF HUMAN FKBP51 FK1 DOMAIN A19T MUTANT IN COMPLEX WITH SAFit2 | 分子名称: | (1R)-3-(3,4-dimethoxyphenyl)-1-{3-[2-(morpholin-4-yl)ethoxy]phenyl}propyl (2S)-1-[(2S)-2-[(1S)-cyclohex-2-en-1-yl]-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxylate, Peptidyl-prolyl cis-trans isomerase FKBP5 | 著者 | Fiegen, D, Draxler, S.W. | 登録日 | 2020-01-14 | 公開日 | 2020-05-27 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Hybrid Screening Approach for Very Small Fragments: X-ray and Computational Screening on FKBP51. J.Med.Chem., 63, 2020
|
|
4YHM
| Reversal Agent for Dabigatran | 分子名称: | N-[(2-{[(4-carbamimidoylphenyl)amino]methyl}-1-methyl-1H-benzimidazol-5-yl)carbonyl]-N-pyridin-2-yl-beta-alanine, aDabi-Fab2b heavy chain, aDabi-Fab2b light chain | 著者 | Schiele, F, Nar, H. | 登録日 | 2015-02-27 | 公開日 | 2016-01-13 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.16 Å) | 主引用文献 | Structure-guided residence time optimization of a dabigatran reversal agent. Mabs, 7, 2015
|
|
4YHI
| Reversal Agent for Dabigatran | 分子名称: | N-[(2-{[(4-carbamimidoylphenyl)amino]methyl}-1-methyl-1H-benzimidazol-5-yl)carbonyl]-N-pyridin-2-yl-beta-alanine, aDabi-Fab2a heavy chain, aDabi-Fab2a light chain | 著者 | Schiele, F, Nar, H. | 登録日 | 2015-02-27 | 公開日 | 2016-01-13 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Structure-guided residence time optimization of a dabigatran reversal agent. Mabs, 7, 2015
|
|
4YHN
| Dabigatran Reversal Agent | 分子名称: | aDabi-Fab3 heavy chain, aDabi-Fab3 light chain | 著者 | Schiele, F, Nar, H. | 登録日 | 2015-02-27 | 公開日 | 2016-02-10 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.31 Å) | 主引用文献 | Structure-guided residence time optimization of a dabigatran reversal agent. Mabs, 7, 2015
|
|
4YHL
| Reversal Agent for Dabigatran | 分子名称: | aDabi-Fab2b heavy chain, aDabi-Fab2b light chain | 著者 | Schiele, F, Nar, H. | 登録日 | 2015-02-27 | 公開日 | 2016-01-13 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.09 Å) | 主引用文献 | Structure-guided residence time optimization of a dabigatran reversal agent. Mabs, 7, 2015
|
|
4YGV
| Reversal Agent for Dabigatran | 分子名称: | GLYCEROL, aDabi-Fab2a heavy chain, aDabi-Fab2a light chain | 著者 | Schiele, F, Nar, H. | 登録日 | 2015-02-26 | 公開日 | 2015-06-17 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.76 Å) | 主引用文献 | Structure-guided residence time optimization of a dabigatran reversal agent. Mabs, 7, 2015
|
|
2WFJ
| Atomic resolution crystal structure of the PPIase domain of human cyclophilin G in complex with cyclosporin A. | 分子名称: | 1,2-ETHANEDIOL, CHLORIDE ION, CYCLOSPORIN A, ... | 著者 | Stegmann, C.M, Sheldrick, G.M, Wahl, M.C. | 登録日 | 2009-04-06 | 公開日 | 2009-06-16 | 最終更新日 | 2019-05-22 | 実験手法 | X-RAY DIFFRACTION (0.75 Å) | 主引用文献 | The Thermodynamic Influence of Trapped Water Molecules on a Protein-Ligand Interaction. Angew.Chem.Int.Ed.Engl., 48, 2009
|
|
4YHO
| Reversal Agent for Dabigatran | 分子名称: | N-[(2-{[(4-carbamimidoylphenyl)amino]methyl}-1-methyl-1H-benzimidazol-5-yl)carbonyl]-N-pyridin-2-yl-beta-alanine, aDabi-Fab3 heavy chain, aDabi-Fab3 light chain | 著者 | Schiele, F, Nar, H. | 登録日 | 2015-02-27 | 公開日 | 2016-01-13 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.82 Å) | 主引用文献 | Structure-guided residence time optimization of a dabigatran reversal agent. Mabs, 7, 2015
|
|
4YHK
| Reversal Agent for Dabigatran | 分子名称: | GLYCEROL, N-[(2-{[(4-carbamimidoylphenyl)amino]methyl}-1-methyl-1H-benzimidazol-5-yl)carbonyl]-N-pyridin-2-yl-beta-alanine, aDabi-Fab2a heavy chain, ... | 著者 | Schiele, F, Nar, H. | 登録日 | 2015-02-27 | 公開日 | 2016-01-13 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.21 Å) | 主引用文献 | Structure-guided residence time optimization of a dabigatran reversal agent. Mabs, 7, 2015
|
|
2WFI
| |
4EOW
| |