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6TX9

CRYSTAL STRUCTURE OF HUMAN FKBP51 FK1 DOMAIN A19T MUTANT IN COMPLEX WITH HYDANTOIN

Summary for 6TX9
Entry DOI10.2210/pdb6tx9/pdb
DescriptorPeptidyl-prolyl cis-trans isomerase FKBP5, imidazolidine-2,4-dione, SODIUM ION, ... (4 entities in total)
Functional Keywordsppiase, fragment, isomerase
Biological sourceHomo sapiens (Human)
Total number of polymer chains1
Total formula weight14172.13
Authors
Fiegen, D.,Draxler, S.W. (deposition date: 2020-01-13, release date: 2020-05-27, Last modification date: 2024-01-24)
Primary citationDraxler, S.W.,Bauer, M.,Eickmeier, C.,Nadal, S.,Nar, H.,Rangel Rojas, D.,Seeliger, D.,Zeeb, M.,Fiegen, D.
Hybrid Screening Approach for Very Small Fragments: X-ray and Computational Screening on FKBP51.
J.Med.Chem., 63:5856-5864, 2020
Cited by
PubMed: 32420743
DOI: 10.1021/acs.jmedchem.0c00120
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.42 Å)
Structure validation

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