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1IKV
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K103N Mutant HIV-1 Reverse Transcriptase in Complex with Efivarenz
分子名称: (-)-6-CHLORO-4-CYCLOPROPYLETHYNYL-4-TRIFLUOROMETHYL-1,4-DIHYDRO-2H-3,1-BENZOXAZIN-2-ONE, POL POLYPROTEIN
著者Lindberg, J, Unge, T.
登録日2001-05-07
公開日2001-06-06
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Structural basis for the inhibitory efficacy of efavirenz (DMP-266), MSC194 and PNU142721 towards the HIV-1 RT K103N mutant.
Eur.J.Biochem., 269, 2002
1IKY
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HIV-1 Reverse Transcriptase in Complex with the Inhibitor MSC194
分子名称: 1-[2-(3-ACETYL-2-HYDROXY-6-METHOXY-PHENYL)-CYCLOPROPYL]-3-(5-CYANO-PYRIDIN-2-YL)-THIOUREA, POL POLYPROTEIN
著者Lindberg, J, Unge, T.
登録日2001-05-07
公開日2001-06-06
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Structural basis for the inhibitory efficacy of efavirenz (DMP-266), MSC194 and PNU142721 towards the HIV-1 RT K103N mutant.
Eur.J.Biochem., 269, 2002
1ZDH
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MS2 COAT PROTEIN/RNA COMPLEX
分子名称: PROTEIN (BACTERIOPHAGE MS2 COAT PROTEIN), RNA (5'-R(*AP*CP*AP*UP*GP*AP*GP*GP*AP*UP*CP*AP*CP*CP*CP*AP*U P*GP*U)-3')
著者Valegard, K, Van Den Worm, S, Liljas, L.
登録日1996-09-24
公開日1997-04-21
最終更新日2023-04-19
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献The three-dimensional structures of two complexes between recombinant MS2 capsids and RNA operator fragments reveal sequence-specific protein-RNA interactions.
J.Mol.Biol., 270, 1997
1ZDI
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RNA BACTERIOPHAGE MS2 COAT PROTEIN/RNA COMPLEX
分子名称: PROTEIN (RNA BACTERIOPHAGE MS2 COAT PROTEIN), RNA (5'-R(*AP*CP*AP*UP*GP*AP*GP*GP*AP*UP*UP*AP*CP*CP*CP*AP*U P*GP*U)-3')
著者Valegard, K, Van Den Worm, S, Liljas, L.
登録日1996-09-24
公開日1997-04-21
最終更新日2023-04-19
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献The three-dimensional structures of two complexes between recombinant MS2 capsids and RNA operator fragments reveal sequence-specific protein-RNA interactions.
J.Mol.Biol., 270, 1997
1BMS
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BU of 1bms by Molmil
CRYSTAL STRUCTURE OF MS2 CAPSIDS WITH MUTATIONS IN THE SUBUNIT FG LOOP
分子名称: BACTERIOPHAGE MS2 CAPSID
著者Liljas, L, Stonehouse, N.J.
登録日1995-08-29
公開日1996-03-08
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Crystal structures of MS2 capsids with mutations in the subunit FG loop.
J.Mol.Biol., 256, 1996
1AQ4
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STRUCTURE OF A MS2 COAT PROTEIN MUTANT IN COMPLEX WITH AN RNA OPERATOR
分子名称: PROTEIN(BACTERIOPHAGE MS2 COAT PROTEIN), RNA (5'-R(*AP*CP*AP*UP*GP*AP*GP*GP*AP*UP*UP*AP*CP*CP*CP*AP*U P*GP*U)-3')
著者Van Den Worm, S.H, Stonehouse, N.J, Valegard, K, Liljas, L.
登録日1997-08-06
公開日1997-12-24
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Crystal structures of MS2 coat protein mutants in complex with wild-type RNA operator fragments.
Nucleic Acids Res., 26, 1998
1AQ3
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BACTERIOPHAGE MS2 CAPSID PROTEIN/RNA COMPLEX
分子名称: PROTEIN (BACTERIOPHAGE MS2 COAT PROTEIN), RNA (5'-R(*AP*CP*AP*UP*GP*AP*GP*GP*AP*UP*UP*AP*CP*CP*CP*AP*U P*GP*U)-3')
著者Van Den Worm, S, Stonehouse, N, Valegard, K, Liljas, L.
登録日1997-08-06
公開日1997-12-24
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Crystal structures of MS2 coat protein mutants in complex with wild-type RNA operator fragments.
Nucleic Acids Res., 26, 1998
2CAB
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STRUCTURE, REFINEMENT AND FUNCTION OF CARBONIC ANHYDRASE ISOZYMES. REFINEMENT OF HUMAN CARBONIC ANHYDRASE I
分子名称: CARBONIC ANHYDRASE FORM B, ZINC ION
著者Kannan, K.K, Ramanadham, M, Jones, T.A.
登録日1983-10-05
公開日1984-02-02
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structure, refinement, and function of carbonic anhydrase isozymes: refinement of human carbonic anhydrase I
Ann.N.Y.Acad.Sci., 429, 1984
2CA2
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CRYSTALLOGRAPHIC STUDIES OF INHIBITOR BINDING SITES IN HUMAN CARBONIC ANHYDRASE II. A PENTACOORDINATED BINDING OF THE SCN-ION TO THE ZINC AT HIGH P*H
分子名称: CARBONIC ANHYDRASE II, MERCURY (II) ION, THIOCYANATE ION, ...
著者Eriksson, A.E, Kylsten, P.M, Jones, T.A, Liljas, A.
登録日1989-02-06
公開日1990-01-15
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Crystallographic studies of inhibitor binding sites in human carbonic anhydrase II: a pentacoordinated binding of the SCN- ion to the zinc at high pH.
Proteins, 4, 1988
1CA2
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REFINED STRUCTURE OF HUMAN CARBONIC ANHYDRASE II AT 2.0 ANGSTROMS RESOLUTION
分子名称: CARBONIC ANHYDRASE II, ZINC ION
著者Eriksson, A.E, Jones, T.A, Liljas, A.
登録日1989-02-06
公開日1990-01-15
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Refined structure of human carbonic anhydrase II at 2.0 A resolution.
Proteins, 4, 1988
1D4J
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HIV-1 protease in complex with the inhibitor MSL370
分子名称: 2,5-DIBENZYLOXY-3,4-DIHYDROXY-HEXANEDIOIC ACID 2-CHLORO-6-FLUORO-BENZYLAMIDE (2-HYDROXY-INDAN-1- YL)-AMIDE, HIV-1 PROTEASE
著者Unge, T.
登録日1999-10-04
公開日2002-06-26
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.81 Å)
主引用文献Optimization of P1-P3 groups in symmetric and asymmetric HIV-1 protease inhibitors.
Eur.J.Biochem., 270, 2003
1D4H
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HIV-1 Protease in complex with the inhibitor BEA435
分子名称: 2,5-DIBENZYLOXY-3,4-DIHYDROXY-HEXANEDIOIC ACID BENZYLAMIDE (2-HYDROXY-INDAN-1-YL)-AMIDE, HIV-1 PROTEASE
著者Unge, T.
登録日1999-10-04
公開日2002-06-26
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.81 Å)
主引用文献Optimization of P1-P3 groups in symmetric and asymmetric HIV-1 protease inhibitors.
Eur.J.Biochem., 270, 2003
1D4I
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HIV-1 protease in complex with the inhibitor BEA425
分子名称: 2,5-DIBENZYLOXY-3-HYDROXY-HEXANEDIOIC ACID BIS-[(2-HYDROXY-INDAN-1-YL)-AMIDE], HIV-1 PROTEASE
著者Unge, T.
登録日1999-10-04
公開日2002-06-26
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.81 Å)
主引用文献Optimization of P1-P3 groups in symmetric and asymmetric HIV-1 protease inhibitors.
Eur.J.Biochem., 270, 2003
1EC1
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HIV-1 protease in complex with the inhibitor BEA409
分子名称: HIV-1 PROTEASE, N,N-[2,5-O-[DI-4-THIOPHEN-3-YL-BENZYL]-GLUCARYL]-DI-[VALYL-AMIDO-METHANE]
著者Unge, T.
登録日2000-01-25
公開日2002-06-26
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Optimization of P1-P3 groups in symmetric and asymmetric HIV-1 protease inhibitors
Eur.J.Biochem., 270, 2003
1EBY
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HIV-1 protease in complex with the inhibitor BEA369
分子名称: HIV-1 PROTEASE, N,N-[2,5-O-DIBENZYL-GLUCARYL]-DI-[1-AMINO-INDAN-2-OL]
著者Unge, T.
登録日2000-01-25
公開日2002-06-26
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.294 Å)
主引用文献Optimization of P1-P3 groups in symmetric and asymmetric HIV-1 protease inhibitors
Eur.J.Biochem., 270, 2003
1EBZ
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HIV-1 protease in complex with the inhibitor BEA388
分子名称: HIV-1 PROTEASE, [5-(2-HYDROXY-INDAN-1-YLCARBAMOYL)-3,4-DIHYDROXY-2,5-[DIBENZYL-OXY]-PENTANOYL]-VALINYL-AMIDO-METHANE
著者Unge, T.
登録日2000-01-25
公開日2002-06-26
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.01 Å)
主引用文献Optimization of P1-P3 groups in symmetric and asymmetric HIV-1 protease inhibitors
Eur.J.Biochem., 270, 2003
1EBW
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HIV-1 protease in complex with the inhibitor BEA322
分子名称: HIV-1 PROTEASE, N,N-[2,5-O-[DIBENZYL]-GLUCARYL]-DI-[ISOLEUCYL-AMIDO-METHANE]
著者Unge, T.
登録日2000-01-25
公開日2002-06-26
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.81 Å)
主引用文献Optimization of P1-P3 groups in symmetric and asymmetric HIV-1 protease inhibitors
Eur.J.Biochem., 270, 2003
1EC2
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HIV-1 protease in complex with the inhibitor BEA428
分子名称: HIV-1 PROTEASE, N,N-[2,5-O-[DI-4-PYRIDIN-3-YL-BENZYL]-GLUCARYL]-DI-[VALYL-AMIDO-METHANE]
著者Unge, T.
登録日2000-01-25
公開日2002-06-26
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Optimization of P1-P3 groups in symmetric and asymmetric HIV-1 protease inhibitors
Eur.J.Biochem., 270, 2003
1EC3
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HIV-1 protease in complex with the inhibitor MSA367
分子名称: HIV-1 PROTEASE, N,N-[2,5-O-DIBENZYL-GLUCARYL]-DI-[VALINYL-AMINOMETHANYL-PYRIDINE]
著者Unge, T.
登録日2000-01-25
公開日2002-06-26
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Optimization of P1-P3 groups in symmetric and asymmetric HIV-1 protease inhibitors
Eur.J.Biochem., 270, 2003
2BUK
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SATELLITE TOBACCO NECROSIS VIRUS
分子名称: CALCIUM ION, COAT PROTEIN
著者Jones, T.A, Liljas, L.
登録日2005-06-14
公開日2005-08-18
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.45 Å)
主引用文献Structure of Satellite Tobacco Necrosis Virus After Crystallographic Refinement at 2.5 A Resolution.
J.Mol.Biol., 177, 1984
1CRM
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STRUCTURE AND FUNCTION OF CARBONIC ANHYDRASES
分子名称: CARBONIC ANHYDRASE I, CHLORIDE ION, HYDROSULFURIC ACID, ...
著者Yadava, V.S, Kannan, K.K.
登録日1994-03-04
公開日1995-02-07
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structure and Function of Carbonic Anhydrases
Biomolecular Structure, Conformation, Function and Evolution, 1, 1981
1CZM
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DRUG-PROTEIN INTERACTIONS: STRUCTURE OF SULFONAMIDE DRUG COMPLEXED WITH HUMAN CARBONIC ANHYDRASE I
分子名称: 3-ACTOXYMERCURI-4-AMINOBENZENESULFONAMIDE, CARBONIC ANHYDRASE I, MERCURY (II) ION, ...
著者Chakravarty, S, Kannan, K.K.
登録日1993-11-28
公開日1994-04-30
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Drug-protein interactions. Refined structures of three sulfonamide drug complexes of human carbonic anhydrase I enzyme.
J.Mol.Biol., 243, 1994
1AZM
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DRUG-PROTEIN INTERACTIONS: STRUCTURE OF SULFONAMIDE DRUG COMPLEXED WITH HUMAN CARBONIC ANHYDRASE I
分子名称: 5-ACETAMIDO-1,3,4-THIADIAZOLE-2-SULFONAMIDE, CARBONIC ANHYDRASE I, ZINC ION
著者Chakravarty, S, Kannan, K.K.
登録日1993-11-28
公開日1994-04-30
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Drug-protein interactions. Refined structures of three sulfonamide drug complexes of human carbonic anhydrase I enzyme.
J.Mol.Biol., 243, 1994
1BZM
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DRUG-PROTEIN INTERACTIONS: STRUCTURE OF SULFONAMIDE DRUG COMPLEXED WITH HUMAN CARBONIC ANHYDRASE I
分子名称: CARBONIC ANHYDRASE I, N-(3-methyl-5-sulfamoyl-1,3,4-thiadiazol-2(3H)-ylidene)acetamide, ZINC ION
著者Chakravarty, S, Kannan, K.K.
登録日1993-11-28
公開日1994-04-30
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Drug-protein interactions. Refined structures of three sulfonamide drug complexes of human carbonic anhydrase I enzyme.
J.Mol.Biol., 243, 1994
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