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1FQ3
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CRYSTAL STRUCTURE OF HUMAN GRANZYME B
分子名称: GRANZYME B, SULFATE ION, beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose
著者Estebanez-Perpina, E, Fuentes-Prior, P, Belorgey, D, Rubin, H, Bode, W.
登録日2000-09-03
公開日2001-01-31
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献Crystal structure of the caspase activator human granzyme B, a proteinase highly specific for an Asp-P1 residue.
Biol.Chem., 381, 2000
1GQF
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Crystal structure of human procaspase-7
分子名称: Caspase-7, SULFATE ION
著者Riedl, S, Bode, W, Fuentes-Prior, P.
登録日2001-11-23
公開日2002-01-04
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Structural basis for the activation of human procaspase-7.
Proc. Natl. Acad. Sci. U.S.A., 98, 2001
1GTL
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The thermostable serine-carboxyl type proteinase, kumamolisin (KSCP) - complex with Ac-Ile-Pro-Phe-cho
分子名称: ALDEHYDE INHIBITOR, CALCIUM ION, KUMAMOLYSIN, ...
著者Comellas-Bigler, M, Fuentes-Prior, P, Maskos, K, Huber, R, Oyama, H, Uchida, K, Dunn, B.M, Oda, K, Bode, W.
登録日2002-01-16
公開日2002-06-13
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献The 1.4 A Crystal Structure of Kumamolysin. A Thermostable Serine-Carboxyl-Type Proteinase
Structure, 10, 2002
1GT9
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High resolution crystal structure of a thermostable serine-carboxyl type proteinase, kumamolisin (kscp)
分子名称: CALCIUM ION, KUMAMOLYSIN, SULFATE ION
著者Comellas-Bigler, M, Fuentes-Prior, P, Maskos, K, Huber, R, Oyama, H, Uchida, K, Dunn, B.M, Oda, K, Bode, W.
登録日2002-01-14
公開日2002-06-13
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.38 Å)
主引用文献The 1.4 A Crystal Structure of Kumamolysin. A Thermostable Serine-Carboxyl-Type Proteinase
Structure, 10, 2002
1GTJ
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Crystal structure of the thermostable serine-carboxyl type proteinase, kumamolisin (KSCP) - complex with Ac-Ile-Ala-Phe-cho
分子名称: ALDEHYDE INHIBITOR, CALCIUM ION, KUMAMOLYSIN, ...
著者Comellas-Bigler, M, Fuentes-Prior, P, Maskos, K, Huber, R, Oyama, H, Uchida, K, Dunn, B.M, Oda, K, Bode, W.
登録日2002-01-15
公開日2002-06-13
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献The 1.4 A Crystal Structure of Kumamolysin. A Thermostable Serine-Carboxyl-Type Proteinase
Structure, 10, 2002
1GTG
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Crystal structure of the thermostable serine-carboxyl type proteinase, kumamolysin (kscp)
分子名称: CALCIUM ION, KUMAMOLYSIN
著者Comellas-Bigler, M, Fuentes-Prior, P, Maskos, K, Huber, R, Oyama, H, Uchida, K, Dunn, B.M, Oda, K, Bode, W.
登録日2002-01-15
公開日2002-06-13
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献The 1.4 A Crystal Structure of Kumamolysin. A Thermostable Serine-Carboxyl-Type Proteinase
Structure, 10, 2002
7Z9B
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Sam68
分子名称: 1,2-ETHANEDIOL, GLYCEROL, IODIDE ION, ...
著者Nadal, M, Fuentes-Prior, P.
登録日2022-03-20
公開日2023-02-01
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (3.333 Å)
主引用文献Structure and function analysis of Sam68 and hnRNP A1 synergy in the exclusion of exon 7 from SMN2 transcripts.
Protein Sci., 32, 2023
1E0F
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Crystal structure of the human alpha-thrombin-haemadin complex: an exosite II-binding inhibitor
分子名称: HAEMADIN, THROMBIN
著者Richardson, J.L, Kroeger, B, Hoefken, W, Pereira, P, Huber, R, Bode, W, Fuentes-Prior, P.
登録日2000-03-27
公開日2000-11-03
最終更新日2023-12-06
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献Crystal Structure of the Human Alpha-Thrombin-Haemadin Complex: An Exosite II-Binding Inhibitor
Embo J., 19, 2000
7ZU1
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Crystal structure of mutant AR-LBD (V758A) bound to dihydrotestosterone
分子名称: 2,3-DIHYDROXY-1,4-DITHIOBUTANE, 5-ALPHA-DIHYDROTESTOSTERONE, Androgen receptor, ...
著者Alegre-Marti, A, Jimenez-Panizo, A, Estebanez-Perpina, E, Fuentes-Prior, P.
登録日2022-05-11
公開日2023-03-22
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.68 Å)
主引用文献A hotspot for posttranslational modifications on the androgen receptor dimer interface drives pathology and anti-androgen resistance.
Sci Adv, 9, 2023
7ZU2
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Crystal structure of mutant AR-LBD (Q799E) bound to dihydrotestosterone
分子名称: 5-ALPHA-DIHYDROTESTOSTERONE, Androgen receptor, IMIDAZOLE
著者Alegre-Marti, A, Jimenez-Panizo, A, Estebanez-Perpina, E, Fuentes-Prior, P.
登録日2022-05-11
公開日2023-03-22
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.74 Å)
主引用文献A hotspot for posttranslational modifications on the androgen receptor dimer interface drives pathology and anti-androgen resistance.
Sci Adv, 9, 2023
7ZTX
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Crystal structure of mutant AR-LBD (F755V) bound to dihydrotestosterone
分子名称: 5-ALPHA-DIHYDROTESTOSTERONE, Androgen receptor, IMIDAZOLE, ...
著者Alegre-Marti, A, Jimenez-Panizo, A, Estebanez-Perpina, E, Fuentes-Prior, P.
登録日2022-05-11
公開日2023-03-22
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.89 Å)
主引用文献A hotspot for posttranslational modifications on the androgen receptor dimer interface drives pathology and anti-androgen resistance.
Sci Adv, 9, 2023
7ZTV
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BU of 7ztv by Molmil
Crystal structure of mutant AR-LBD (F755L) bound to dihydrotestosterone
分子名称: 1,2-ETHANEDIOL, 5-ALPHA-DIHYDROTESTOSTERONE, Androgen receptor
著者Alegre-Marti, A, Jimenez-Panizo, A, Estebanez-Perpina, E, Fuentes-Prior, P.
登録日2022-05-11
公開日2023-03-22
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.94 Å)
主引用文献A hotspot for posttranslational modifications on the androgen receptor dimer interface drives pathology and anti-androgen resistance.
Sci Adv, 9, 2023
7ZTZ
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Crystal structure of mutant AR-LBD (Y764C) bound to dihydrotestosterone
分子名称: 5-ALPHA-DIHYDROTESTOSTERONE, Androgen receptor, IMIDAZOLE, ...
著者Alegre-Marti, A, Jimenez-Panizo, A, Estebanez-Perpina, E, Fuentes-Prior, P.
登録日2022-05-11
公開日2023-03-22
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献A hotspot for posttranslational modifications on the androgen receptor dimer interface drives pathology and anti-androgen resistance.
Sci Adv, 9, 2023
1CZS
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BU of 1czs by Molmil
CRYSTAL STRUCTURE OF THE C2 DOMAIN OF HUMAN COAGULATION FACTOR V: COMPLEX WITH PHENYLMERCURY
分子名称: PHENYLMERCURY, PROTEIN (COAGULATION FACTOR V)
著者Macedo-Ribeiro, S, Bode, W, Huber, R, Kane, W.H, Fuentes-Prior, P.
登録日1999-09-07
公開日1999-11-26
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Crystal structures of the membrane-binding C2 domain of human coagulation factor V.
Nature, 402, 1999
1CZT
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BU of 1czt by Molmil
CRYSTAL STRUCTURE OF THE C2 DOMAIN OF HUMAN COAGULATION FACTOR V
分子名称: PROTEIN (COAGULATION FACTOR V)
著者Macedo-Ribeiro, S, Bode, W, Huber, R, Kane, W.H, Fuentes-Prior, P.
登録日1999-09-07
公開日1999-11-26
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (1.87 Å)
主引用文献Crystal structures of the membrane-binding C2 domain of human coagulation factor V.
Nature, 402, 1999
1CZV
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CRYSTAL STRUCTURE OF THE C2 DOMAIN OF HUMAN COAGULATION FACTOR V: DIMERIC CRYSTAL FORM
分子名称: PROTEIN (COAGULATION FACTOR V)
著者Macedo-Ribeiro, S, Bode, W, Huber, R, Kane, W.H, Fuentes-Prior, P.
登録日1999-09-07
公開日1999-11-26
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Crystal structures of the membrane-binding C2 domain of human coagulation factor V.
Nature, 402, 1999
7ZAF
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Sam68
分子名称: 1,2-ETHANEDIOL, CHLORIDE ION, GLYCEROL, ...
著者Nadal, M, Puestes-Prior, P.
登録日2022-03-22
公開日2023-02-01
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.71 Å)
主引用文献Structure and function analysis of Sam68 and hnRNP A1 synergy in the exclusion of exon 7 from SMN2 transcripts.
Protein Sci., 32, 2023
7ZAB
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Sam68
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, 1,2-ETHANEDIOL, CHLORIDE ION, ...
著者Nadal, M, Puestes-Prior, P.
登録日2022-03-22
公開日2023-02-01
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.46 Å)
主引用文献Structure and function analysis of Sam68 and hnRNP A1 synergy in the exclusion of exon 7 from SMN2 transcripts.
Protein Sci., 32, 2023
5TO3
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Crystal structure of thrombin mutant W215A/E217A fused to EGF456 of thrombomodulin via a 31-residue linker and bound to PPACK
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-beta-D-mannopyranose-(1-4)-beta-D-mannopyranose-(1-4)-alpha-D-mannopyranose-(1-4)-[beta-D-mannopyranose-(1-6)]beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, D-phenylalanyl-N-[(2S,3S)-6-{[amino(iminio)methyl]amino}-1-chloro-2-hydroxyhexan-3-yl]-L-prolinamide, ...
著者Barranco-Medina, S, Murphy, M, Pelc, L, Chen, Z, Di Cera, E, Pozzi, N.
登録日2016-10-16
公開日2017-03-29
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.34 Å)
主引用文献Rational Design of Protein C Activators.
Sci Rep, 7, 2017
1EAW
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Crystal structure of the MTSP1 (matriptase)-BPTI (aprotinin) complex
分子名称: PANCREATIC TRYPSIN INHIBITOR, SUPPRESSOR OF TUMORIGENICITY 14
著者Friedrich, R, Bode, W.
登録日2001-07-17
公開日2002-01-28
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.93 Å)
主引用文献Catalytic Domain Structures of Mt-Sp1/Matriptase, a Matrix-Degrading Transmembrane Serine Proteinase.
J.Biol.Chem., 277, 2002
1EAX
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Crystal structure of MTSP1 (matriptase)
分子名称: BENZAMIDINE, SULFATE ION, SUPPRESSOR OF TUMORIGENICITY 14
著者Friedrich, R, Bode, W.
登録日2001-07-17
公開日2002-01-28
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.3 Å)
主引用文献Catalytic Domain Structures of Mt-Sp1/Matriptase, a Matrix-Degrading Transmembrane Serine Proteinase.
J.Biol.Chem., 277, 2002
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