Loading
PDBj
メニューPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help
Search by PDB author
4IAN
DownloadVisualize
BU of 4ian by Molmil
Crystal Structure of apo Human PRPF4B kinase domain
分子名称: SULFATE ION, Serine/threonine-protein kinase PRP4 homolog
著者Mechin, I, Haas, K, Chen, X, Zhang, Y, McLean, L.
登録日2012-12-06
公開日2013-08-28
最終更新日2017-11-15
実験手法X-RAY DIFFRACTION (2.44 Å)
主引用文献Evaluation of Cancer Dependence and Druggability of PRP4 Kinase Using Cellular, Biochemical, and Structural Approaches.
J.Biol.Chem., 288, 2013
2F8G
DownloadVisualize
BU of 2f8g by Molmil
HIV-1 protease mutant I50V complexed with inhibitor TMC114
分子名称: (3R,3AS,6AR)-HEXAHYDROFURO[2,3-B]FURAN-3-YL(1S,2R)-3-[[(4-AMINOPHENYL)SULFONYL](ISOBUTYL)AMINO]-1-BENZYL-2-HYDROXYPROPYLCARBAMATE, ACETIC ACID, CHLORIDE ION, ...
著者Kovalevsky, A.Y, Weber, I.T.
登録日2005-12-02
公開日2006-03-07
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.22 Å)
主引用文献Effectiveness of Nonpeptide Clinical Inhibitor TMC-114 on HIV-1 Protease with Highly Drug Resistant Mutations D30N, I50V, and L90M.
J.Med.Chem., 49, 2006
2F80
DownloadVisualize
BU of 2f80 by Molmil
HIV-1 Protease mutant D30N complexed with inhibitor TMC114
分子名称: (3R,3AS,6AR)-HEXAHYDROFURO[2,3-B]FURAN-3-YL(1S,2R)-3-[[(4-AMINOPHENYL)SULFONYL](ISOBUTYL)AMINO]-1-BENZYL-2-HYDROXYPROPYLCARBAMATE, CHLORIDE ION, POL POLYPROTEIN, ...
著者Kovalevsky, A.Y, Weber, I.T.
登録日2005-12-01
公開日2006-03-07
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.45 Å)
主引用文献Effectiveness of Nonpeptide Clinical Inhibitor TMC-114 on HIV-1 Protease with Highly Drug Resistant Mutations D30N, I50V, and L90M.
J.Med.Chem., 49, 2006
3SMQ
DownloadVisualize
BU of 3smq by Molmil
Crystal structure of protein arginine methyltransferase 3
分子名称: 1-(1,2,3-benzothiadiazol-6-yl)-3-[2-(cyclohex-1-en-1-yl)ethyl]urea, CHLORIDE ION, Protein arginine N-methyltransferase 3, ...
著者Dobrovetsky, E, Dong, A, Walker, J.R, Siarheyeva, A, Senisterra, G, Wasney, G.A, Smil, D, Bolshan, Y, Nguyen, K.T, Allali-Hassani, A, Hajian, T, Poda, G, Bountra, C, Weigelt, J, Edwards, A.M, Al-Awar, R, Brown, P.J, Schapira, M, Arrowsmith, C.H, Vedadi, M, Structural Genomics Consortium (SGC)
登録日2011-06-28
公開日2011-08-31
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献An allosteric inhibitor of protein arginine methyltransferase 3.
Structure, 20, 2012
1HTV
DownloadVisualize
BU of 1htv by Molmil
CRYSTAL STRUCTURE OF DESTRIPEPTIDE (B28-B30) INSULIN
分子名称: INSULIN, ZINC ION
著者Ye, J, Chang, W, Liang, D.
登録日2001-01-01
公開日2001-05-23
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Crystal structure of destripeptide (B28-B30) insulin: implications for insulin dissociation.
Biochim.Biophys.Acta, 1547, 2001
2F81
DownloadVisualize
BU of 2f81 by Molmil
HIV-1 Protease mutant L90M complexed with inhibitor TMC114
分子名称: (3R,3AS,6AR)-HEXAHYDROFURO[2,3-B]FURAN-3-YL(1S,2R)-3-[[(4-AMINOPHENYL)SULFONYL](ISOBUTYL)AMINO]-1-BENZYL-2-HYDROXYPROPYLCARBAMATE, CHLORIDE ION, GLYCEROL, ...
著者Kovalevsky, A.Y, Weber, I.T.
登録日2005-12-01
公開日2006-03-07
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.25 Å)
主引用文献Effectiveness of Nonpeptide Clinical Inhibitor TMC-114 on HIV-1 Protease with Highly Drug Resistant Mutations D30N, I50V, and L90M.
J.Med.Chem., 49, 2006
2HS1
DownloadVisualize
BU of 2hs1 by Molmil
Ultra-high resolution X-ray crystal structure of HIV-1 protease V32I mutant with TMC114 (darunavir) inhibitor
分子名称: (3R,3AS,6AR)-HEXAHYDROFURO[2,3-B]FURAN-3-YL(1S,2R)-3-[[(4-AMINOPHENYL)SULFONYL](ISOBUTYL)AMINO]-1-BENZYL-2-HYDROXYPROPYLCARBAMATE, CHLORIDE ION, DIMETHYL SULFOXIDE, ...
著者Weber, I.T, Kovalevsky, A.Y.
登録日2006-07-20
公開日2006-10-03
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (0.84 Å)
主引用文献Ultra-high Resolution Crystal Structure of HIV-1 Protease Mutant Reveals Two Binding Sites for Clinical Inhibitor TMC114.
J.Mol.Biol., 363, 2006
2KBU
DownloadVisualize
BU of 2kbu by Molmil
NMR solution structure of Pin1 WW domain mutant with beta turn mimic at position 12
分子名称: Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1
著者Fuller, A.A, Bhabha, G, Case, D.A.
登録日2008-12-08
公開日2009-07-07
最終更新日2023-11-15
実験手法SOLUTION NMR
主引用文献Evaluating beta-turn mimics as beta-sheet folding nucleators.
Proc.Natl.Acad.Sci.USA, 106, 2009
6KZ5
DownloadVisualize
BU of 6kz5 by Molmil
Crystal Structure Analysis of the Csn-B-bounded NUR77 Ligand binding Domain
分子名称: Nuclear receptor subfamily 4 group A member 1, ethyl 2-[2-octanoyl-3,5-bis(oxidanyl)phenyl]ethanoate
著者Hong, W, Chen, H, Wu, Q, Lin, T.
登録日2019-09-23
公開日2020-10-14
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (4.45 Å)
主引用文献Blocking PPAR gamma interaction facilitates Nur77 interdiction of fatty acid uptake and suppresses breast cancer progression.
Proc.Natl.Acad.Sci.USA, 117, 2020
6JYJ
DownloadVisualize
BU of 6jyj by Molmil
Crystal structure of FAM46B (TENT5B)
分子名称: CITRATE ANION, Terminal nucleotidyltransferase 5B
著者Zhang, H, Hu, J.L, Gao, S.
登録日2019-04-26
公開日2020-03-04
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.693199 Å)
主引用文献FAM46B is a prokaryotic-like cytoplasmic poly(A) polymerase essential in human embryonic stem cells.
Nucleic Acids Res., 48, 2020
6M8N
DownloadVisualize
BU of 6m8n by Molmil
Endo-fucoidan hydrolase P5AFcnA from glycoside hydrolase family 107
分子名称: CALCIUM ION, MALONATE ION, P5AFcnA
著者Boraston, A.B, Vickers, C.J, Abe, K, Salama-Alber, O.
登録日2018-08-22
公開日2018-10-03
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (1.55 Å)
主引用文献Endo-fucoidan hydrolases from glycoside hydrolase family 107 (GH107) display structural and mechanistic similarities to alpha-l-fucosidases from GH29.
J. Biol. Chem., 293, 2018
7BI9
DownloadVisualize
BU of 7bi9 by Molmil
PI3KC2a core in complex with PIK90
分子名称: 1,2-ETHANEDIOL, N-(2,3-DIHYDRO-7,8-DIMETHOXYIMIDAZO[1,2-C] QUINAZOLIN-5-YL)NICOTINAMIDE, Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit alpha,Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit alpha
著者Lo, W.T, Roske, Y, Daumke, O, Haucke, V.
登録日2021-01-12
公開日2022-03-09
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.65 Å)
主引用文献Structural basis of phosphatidylinositol 3-kinase C2 alpha function.
Nat.Struct.Mol.Biol., 29, 2022
7BI6
DownloadVisualize
BU of 7bi6 by Molmil
PI3KC2a core in complex with ATP
分子名称: 1,2-ETHANEDIOL, ADENOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, ...
著者Lo, W.T, Roske, Y, Daumke, O, Haucke, V.
登録日2021-01-12
公開日2022-03-09
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.75 Å)
主引用文献Structural basis of phosphatidylinositol 3-kinase C2 alpha function.
Nat.Struct.Mol.Biol., 29, 2022
7BI4
DownloadVisualize
BU of 7bi4 by Molmil
PI3KC2a core apo
分子名称: 1,2-ETHANEDIOL, Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit alpha,Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit alpha, SULFATE ION
著者Lo, W.T, Roske, Y, Daumke, O, Haucke, V.
登録日2021-01-12
公開日2022-03-09
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.42 Å)
主引用文献Structural basis of phosphatidylinositol 3-kinase C2 alpha function.
Nat.Struct.Mol.Biol., 29, 2022
7BI2
DownloadVisualize
BU of 7bi2 by Molmil
PI3KC2aDeltaN and DeltaC-C2
分子名称: 1,2-ETHANEDIOL, 9-(6-aminopyridin-3-yl)-1-[3-(trifluoromethyl)phenyl]benzo[h][1,6]naphthyridin-2(1H)-one, IODIDE ION, ...
著者Lo, W.T, Roske, Y, Daumke, O, Haucke, V.
登録日2021-01-12
公開日2022-03-09
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (3.25 Å)
主引用文献Structural basis of phosphatidylinositol 3-kinase C2 alpha function.
Nat.Struct.Mol.Biol., 29, 2022
6A5F
DownloadVisualize
BU of 6a5f by Molmil
The structure of [4+2] and [6+4] cyclase in the biosynthetic pathway of nargenicin
分子名称: NgnD
著者Zhang, B, Ge, H.M.
登録日2018-06-23
公開日2019-02-06
最終更新日2024-03-27
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献Enzyme-catalysed [6+4] cycloadditions in the biosynthesis of natural products.
Nature, 568, 2019
6A6J
DownloadVisualize
BU of 6a6j by Molmil
Crystal structure of Zebra fish Y-box protein1 (YB-1) Cold-shock domain in complex with 6mer m5C RNA
分子名称: RNA (5'-R(P*CP*AP*UP*(5MC)P*U)-3'), ZINC ION, Zebra fish Y-box protein1 (YB-1)
著者Zhang, M.M, Wu, B.X, Huang, Y, Ma, J.B.
登録日2018-06-28
公開日2019-06-19
最終更新日2024-03-27
実験手法X-RAY DIFFRACTION (2.255 Å)
主引用文献RNA 5-Methylcytosine Facilitates the Maternal-to-Zygotic Transition by Preventing Maternal mRNA Decay.
Mol.Cell, 75, 2019
6A5H
DownloadVisualize
BU of 6a5h by Molmil
The structure of [4+2] and [6+4] cyclase in the biosynthetic pathway of unidentified natural product
分子名称: 101015D
著者Zhang, B, Ge, H.M.
登録日2018-06-23
公開日2019-02-06
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (1.618 Å)
主引用文献Enzyme-catalysed [6+4] cycloadditions in the biosynthesis of natural products.
Nature, 568, 2019
6B1V
DownloadVisualize
BU of 6b1v by Molmil
Crystal structure of Ps i-CgsB C78S in complex with i-neocarratetraose
分子名称: 1,2-ETHANEDIOL, 3,6-anhydro-2-O-sulfo-alpha-D-galactopyranose-(1-3)-4-O-sulfo-beta-D-galactopyranose-(1-4)-3,6-anhydro-2-O-sulfo-alpha-D-galactopyranose-(1-3)-4-O-sulfo-beta-D-galactopyranose, CALCIUM ION, ...
著者Hettle, A.G, Boraston, A.B.
登録日2017-09-19
公開日2018-03-14
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.84 Å)
主引用文献The Molecular Basis of Polysaccharide Sulfatase Activity and a Nomenclature for Catalytic Subsites in this Class of Enzyme.
Structure, 26, 2018
6B0K
DownloadVisualize
BU of 6b0k by Molmil
Crystal structure of Ps i-CgsB C78S in complex with k-carrapentaose
分子名称: 1,2-ETHANEDIOL, 3,6-anhydro-D-galactose, 4-O-sulfo-beta-D-galactopyranose, ...
著者Hettle, A, Boraston, A.B.
登録日2017-09-14
公開日2018-03-14
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献The Molecular Basis of Polysaccharide Sulfatase Activity and a Nomenclature for Catalytic Subsites in this Class of Enzyme.
Structure, 26, 2018
6B0J
DownloadVisualize
BU of 6b0j by Molmil
Crystal structure of Ps i-CgsB in complex with k-i-k-neocarrahexaose
分子名称: 1,2-ETHANEDIOL, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, 3,6-anhydro-2-O-sulfo-alpha-D-galactopyranose-(1-3)-4-O-sulfo-beta-D-galactopyranose, ...
著者Hettle, A.G, Boraston, A.B.
登録日2017-09-14
公開日2018-03-14
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献The Molecular Basis of Polysaccharide Sulfatase Activity and a Nomenclature for Catalytic Subsites in this Class of Enzyme.
Structure, 26, 2018
6A5G
DownloadVisualize
BU of 6a5g by Molmil
The structure of [4+2] and [6+4] cyclase in the biosynthetic pathway of streptoseomycin
分子名称: [4+2] and [4+6] cyclase StmD
著者Zhang, B, Ge, H.M.
登録日2018-06-23
公開日2019-02-06
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Enzyme-catalysed [6+4] cycloadditions in the biosynthesis of natural products.
Nature, 568, 2019
6BJ8
DownloadVisualize
BU of 6bj8 by Molmil
TCR55 in complex with Pep20/HLA-B35
分子名称: Beta-2-microglobulin, GLYCEROL, HLA class I histocompatibility antigen, ...
著者Jude, K.M, Sibener, L.V, Yang, X, Garcia, K.C.
登録日2017-11-05
公開日2018-07-25
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Isolation of a Structural Mechanism for Uncoupling T Cell Receptor Signaling from Peptide-MHC Binding.
Cell, 174, 2018
6BIA
DownloadVisualize
BU of 6bia by Molmil
Crystal structure of Ps i-CgsB
分子名称: 1,2-ETHANEDIOL, CALCIUM ION, CITRIC ACID, ...
著者Hettle, A.G, Boraston, A.B.
登録日2017-11-01
公開日2018-03-14
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献The Molecular Basis of Polysaccharide Sulfatase Activity and a Nomenclature for Catalytic Subsites in this Class of Enzyme.
Structure, 26, 2018
6BJ3
DownloadVisualize
BU of 6bj3 by Molmil
TCR55 in complex with HIV(Pol448-456)/HLA-B35
分子名称: 1,2-ETHANEDIOL, Beta-2-microglobulin, HIV Pol B35 peptide, ...
著者Jude, K.M, Sibener, L.V, Garcia, K.C.
登録日2017-11-03
公開日2018-07-25
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (1.898 Å)
主引用文献Isolation of a Structural Mechanism for Uncoupling T Cell Receptor Signaling from Peptide-MHC Binding.
Cell, 174, 2018

221716

件を2024-06-26に公開中

PDB statisticsPDBj update infoContact PDBjnumon