3L7D
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![BU of 3l7d by Molmil](/molmil-images/mine/3l7d) | Crystal Structure of Glycogen Phosphorylase DK5 complex | 分子名称: | 1-(2,3-dideoxy-3-fluoro-beta-D-arabino-hexopyranosyl)-4-[(phenylcarbonyl)amino]pyrimidin-2(1H)-one, Glycogen phosphorylase, muscle form | 著者 | Tsirkone, V.G, Lamprakis, C, Hayes, J.M, Skamnaki, V, Drakou, C, Zographos, S.E, Leonidas, D.D. | 登録日 | 2009-12-28 | 公開日 | 2010-10-20 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | 1-(3-Deoxy-3-fluoro-beta-d-glucopyranosyl) pyrimidine derivatives as inhibitors of glycogen phosphorylase b: Kinetic, crystallographic and modelling studies. Bioorg.Med.Chem., 18, 2010
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3LX5
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![BU of 3lx5 by Molmil](/molmil-images/mine/3lx5) | Crystal structure of mGMPPNP-bound NFeoB from S. thermophilus | 分子名称: | 2-amino-9-(5-O-[(R)-hydroxy{[(R)-hydroxy(phosphonoamino)phosphoryl]oxy}phosphoryl]-3-O-{[2-(methylamino)phenyl]carbonyl}-beta-D-erythro-pentofuranosyl-2-ulose)-1,9-dihydro-6H-purin-6-one, Ferrous iron uptake transporter protein B, GLYCEROL, ... | 著者 | Ash, M.R, Guilfoyle, A, Maher, M.J, Clarke, R.J, Guss, J.M, Jormakka, M. | 登録日 | 2010-02-24 | 公開日 | 2010-03-09 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Potassium-activated GTPase reaction in the G Protein-coupled ferrous iron transporter B. J.Biol.Chem., 285, 2010
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3L6D
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![BU of 3l6d by Molmil](/molmil-images/mine/3l6d) | Crystal structure of putative oxidoreductase from Pseudomonas putida KT2440 | 分子名称: | Putative oxidoreductase | 著者 | Malashkevich, V.N, Patskovsky, Y, Toro, R, Sauder, J.M, Burley, S.K, Almo, S.C, New York SGX Research Center for Structural Genomics (NYSGXRC) | 登録日 | 2009-12-23 | 公開日 | 2010-01-12 | 最終更新日 | 2021-02-10 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Crystal structure of putative oxidoreductase from Pseudomonas putida KT2440 To be Published
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3I15
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![BU of 3i15 by Molmil](/molmil-images/mine/3i15) | |
3R59
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![BU of 3r59 by Molmil](/molmil-images/mine/3r59) | Human Cyclophilin D Complexed with a Fragment | 分子名称: | 1-(3-aminophenyl)ethanone, Peptidyl-prolyl cis-trans isomerase F, mitochondrial | 著者 | Colliandre, L, Ahmed-Belkacem, H, Bessin, Y, Pawlotsky, J.M, Guichou, J.F. | 登録日 | 2011-03-18 | 公開日 | 2012-03-21 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (1.1 Å) | 主引用文献 | Fragment-based discovery of a new family of non-peptidic small-molecule cyclophilin inhibitors with potent antiviral activities. Nat Commun, 7, 2016
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3I13
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3I45
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![BU of 3i45 by Molmil](/molmil-images/mine/3i45) | CRYSTAL STRUCTURE OF putative twin-arginine translocation pathway signal protein from Rhodospirillum rubrum Atcc 11170 | 分子名称: | NICOTINIC ACID, Twin-arginine translocation pathway signal protein | 著者 | Malashkevich, V.N, Toro, R, Morano, C, Sauder, J.M, Burley, S.K, Almo, S.C, New York SGX Research Center for Structural Genomics (NYSGXRC) | 登録日 | 2009-07-01 | 公開日 | 2009-07-14 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (1.36 Å) | 主引用文献 | CRYSTAL STRUCTURE OF putative twin-arginine translocation pathway signal protein from Rhodospirillum rubrum
Atcc 11170 To be Published
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3R8F
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![BU of 3r8f by Molmil](/molmil-images/mine/3r8f) | Replication initiator DnaA bound to AMPPCP and single-stranded DNA | 分子名称: | 5'-D(P*AP*AP*AP*AP*AP*AP*AP*AP*AP*AP*AP*A)-3', Chromosomal replication initiator protein dnaA, MAGNESIUM ION, ... | 著者 | Duderstadt, K.E, Chuang, K, Berger, J.M. | 登録日 | 2011-03-23 | 公開日 | 2011-09-28 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (3.366 Å) | 主引用文献 | DNA stretching by bacterial initiators promotes replication origin opening. Nature, 478, 2011
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3I6E
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![BU of 3i6e by Molmil](/molmil-images/mine/3i6e) | CRYSTAL STRUCTURE OF MUCONATE LACTONIZING ENZYME FROM Ruegeria pomeroyi. | 分子名称: | MAGNESIUM ION, Muconate cycloisomerase I, SODIUM ION | 著者 | Fedorov, A.A, Fedorov, E.V, Sauder, J.M, Burley, S.K, Gerlt, J.A, Almo, S.C, New York SGX Research Center for Structural Genomics (NYSGXRC) | 登録日 | 2009-07-07 | 公開日 | 2009-07-14 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Crystal structure of muconate lactonizing enzyme from Ruegeria pomeroyi. To be Published
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3HZO
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![BU of 3hzo by Molmil](/molmil-images/mine/3hzo) | |
3HN2
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![BU of 3hn2 by Molmil](/molmil-images/mine/3hn2) | Crystal structure of 2-dehydropantoate 2-reductase FROM Geobacter metallireducens GS-15 | 分子名称: | 2-dehydropantoate 2-reductase | 著者 | Patskovsky, Y, Toro, R, Morano, C, Rutter, M, Chang, S, Sauder, J.M, Burley, S.K, Almo, S.C, New York SGX Research Center for Structural Genomics (NYSGXRC) | 登録日 | 2009-05-29 | 公開日 | 2009-06-09 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Crystal structure of 2-dehydropantoate 2-reductase FROM Geobacter metallireducens To be Published
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3HQC
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![BU of 3hqc by Molmil](/molmil-images/mine/3hqc) | Crystal structure of Phosphotyrosine-binding domain from the Human Tensin-like C1 domain-containing phosphatase (TENC1) | 分子名称: | ACETATE ION, GLYCEROL, SULFATE ION, ... | 著者 | Sampathkumar, P, Romero, R, Wasserman, S, Do, J, Dickey, M, Bain, K, Gheyi, T, Klemke, R, Atwell, S, Sauder, J.M, Burley, S.K, New York SGX Research Center for Structural Genomics (NYSGXRC) | 登録日 | 2009-06-05 | 公開日 | 2009-07-21 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Crystal structure of Phosphotyrosine-binding domain from the Human Tensin-like C1 domain-containing phosphatase (TENC1) To be Published
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3TO0
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![BU of 3to0 by Molmil](/molmil-images/mine/3to0) | Crystal structure of Mus musculus iodotyrosine deiodinase (IYD) C217A, C239A bound to FMN | 分子名称: | ACETATE ION, FLAVIN MONONUCLEOTIDE, Iodotyrosine deiodinase 1, ... | 著者 | Buss, J.M, McTamney, P.M, Rokita, S.E. | 登録日 | 2011-09-02 | 公開日 | 2012-02-29 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.655 Å) | 主引用文献 | Expression of a soluble form of iodotyrosine deiodinase for active site characterization by engineering the native membrane protein from Mus musculus. Protein Sci., 21, 2012
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3HV2
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![BU of 3hv2 by Molmil](/molmil-images/mine/3hv2) | Crystal structure of signal receiver domain OF HD domain-containing protein FROM Pseudomonas fluorescens Pf-5 | 分子名称: | Response regulator/HD domain protein, SULFATE ION | 著者 | Patskovsky, Y, Ramagopal, U, Toro, R, Freeman, J, Miller, S, Sauder, J.M, Burley, S.K, Almo, S.C, New York SGX Research Center for Structural Genomics (NYSGXRC) | 登録日 | 2009-06-15 | 公開日 | 2009-06-23 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Crystal structure of signal receiver domain oF HD domain-containing protein 3 FROM Pseudomonas fluorescens To be Published
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3HWJ
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![BU of 3hwj by Molmil](/molmil-images/mine/3hwj) | Crystal structure of the second PHR domain of Mouse Myc-binding protein 2 (MYCBP-2) | 分子名称: | DIMETHYL SULFOXIDE, E3 ubiquitin-protein ligase MYCBP2 | 著者 | Sampathkumar, P, Ozyurt, S.A, Wasserman, S.R, Miller, S.A, Bain, K.T, Rutter, M.E, Gheyi, T, Klemke, R.L, Atwell, S, Sauder, J.M, Burley, S.K, New York SGX Research Center for Structural Genomics (NYSGXRC) | 登録日 | 2009-06-17 | 公開日 | 2009-07-21 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (2.25 Å) | 主引用文献 | Structures of PHR domains from Mus musculus Phr1 (Mycbp2) explain the loss-of-function mutation (Gly1092-->Glu) of the C. elegans ortholog RPM-1. J.Mol.Biol., 397, 2010
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3L7A
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![BU of 3l7a by Molmil](/molmil-images/mine/3l7a) | Crystal Structure of Glycogen Phosphorylase DK2 complex | 分子名称: | 1-(3-deoxy-3-fluoro-beta-D-glucopyranosyl)-4-[(phenylcarbonyl)amino]pyrimidin-2(1H)-one, Glycogen phosphorylase, muscle form | 著者 | Tsirkone, V.G, Lamprakis, C, Hayes, J.M, Skamnaki, V, Drakou, C, Zographos, S.E, Leonidas, D.D. | 登録日 | 2009-12-28 | 公開日 | 2010-10-20 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | 1-(3-Deoxy-3-fluoro-beta-d-glucopyranosyl) pyrimidine derivatives as inhibitors of glycogen phosphorylase b: Kinetic, crystallographic and modelling studies. Bioorg.Med.Chem., 18, 2010
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3LLW
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![BU of 3llw by Molmil](/molmil-images/mine/3llw) | Crystal structure of geranyltransferase from helicobacter pylori 26695 | 分子名称: | Geranyltranstransferase (IspA), SULFATE ION | 著者 | Patskovsky, Y, Toro, R, Rutter, M, Sauder, J.M, Burley, S.K, Almo, S.C, New York SGX Research Center for Structural Genomics (NYSGXRC) | 登録日 | 2010-01-29 | 公開日 | 2010-03-31 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Crystal Structure of Geranyltransferase from Helicobacter Pylori To be Published
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3RDA
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![BU of 3rda by Molmil](/molmil-images/mine/3rda) | Human Cyclophilin D Complexed with a Fragment | 分子名称: | 3-methyl-1,2-oxazol-5-amine, Peptidyl-prolyl cis-trans isomerase F, mitochondrial | 著者 | Colliandre, L, Ahmed-Belkacem, H, Bessin, Y, Pawlotsky, J.M, Guichou, J.F. | 登録日 | 2011-04-01 | 公開日 | 2012-03-21 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (1.07 Å) | 主引用文献 | Fragment-based discovery of a new family of non-peptidic small-molecule cyclophilin inhibitors with potent antiviral activities. Nat Commun, 7, 2016
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3RDB
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![BU of 3rdb by Molmil](/molmil-images/mine/3rdb) | Human Cyclophilin D Complexed with a Fragment | 分子名称: | 3-[5-(chloromethyl)-1,2,4-oxadiazol-3-yl]aniline, O-ACETALDEHYDYL-HEXAETHYLENE GLYCOL, Peptidyl-prolyl cis-trans isomerase F, ... | 著者 | Colliandre, L, Ahmed-Belkacem, H, Bessin, Y, Pawlotsky, J.M, Guichou, J.F. | 登録日 | 2011-04-01 | 公開日 | 2012-03-21 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | Fragment-based discovery of a new family of non-peptidic small-molecule cyclophilin inhibitors with potent antiviral activities. Nat Commun, 7, 2016
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3RMR
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![BU of 3rmr by Molmil](/molmil-images/mine/3rmr) | |
3RRN
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![BU of 3rrn by Molmil](/molmil-images/mine/3rrn) | S. cerevisiae dbp5 l327v bound to gle1 h337r and ip6 | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, ATP-dependent RNA helicase DBP5, INOSITOL HEXAKISPHOSPHATE, ... | 著者 | Montpetit, B, Thomsen, N.D, Helmke, K.J, Seeliger, M.A, Berger, J.M, Weis, K. | 登録日 | 2011-04-29 | 公開日 | 2011-05-18 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (4.001 Å) | 主引用文献 | A conserved mechanism of DEAD-box ATPase activation by nucleoporins and InsP6 in mRNA export. Nature, 472, 2011
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3L6E
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![BU of 3l6e by Molmil](/molmil-images/mine/3l6e) | Crystal structure of putative short chain dehydrogenase/reductase family oxidoreductase from Aeromonas hydrophila subsp. hydrophila ATCC 7966 | 分子名称: | Oxidoreductase, short-chain dehydrogenase/reductase family, SULFATE ION | 著者 | Malashkevich, V.N, Patskovsky, Y, Toro, R, Sauder, J.M, Burley, S.K, Almo, S.C, New York SGX Research Center for Structural Genomics (NYSGXRC) | 登録日 | 2009-12-23 | 公開日 | 2010-02-09 | 最終更新日 | 2021-02-10 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Crystal structure of putative short chain dehydrogenase/reductase family oxidoreductase from Aeromonas
hydrophila subsp. hydrophila ATCC 7966 To be Published
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3L7B
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![BU of 3l7b by Molmil](/molmil-images/mine/3l7b) | Crystal Structure of Glycogen Phosphorylase DK3 complex | 分子名称: | 4-amino-1-(3-deoxy-3-fluoro-beta-D-glucopyranosyl)pyrimidin-2(1H)-one, Glycogen phosphorylase, muscle form | 著者 | Tsirkone, V.G, Lamprakis, C, Hayes, J.M, Skamnaki, V, Drakou, C, Zographos, S.E, Leonidas, D.D. | 登録日 | 2009-12-28 | 公開日 | 2010-10-20 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | 1-(3-Deoxy-3-fluoro-beta-d-glucopyranosyl) pyrimidine derivatives as inhibitors of glycogen phosphorylase b: Kinetic, crystallographic and modelling studies. Bioorg.Med.Chem., 18, 2010
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3R54
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![BU of 3r54 by Molmil](/molmil-images/mine/3r54) | Human Cyclophilin D Complexed with a Fragment | 分子名称: | Peptidyl-prolyl cis-trans isomerase F, mitochondrial, pyrrolidine-1-carbaldehyde | 著者 | Colliandre, L, Ahmed-Belkacem, H, Bessin, Y, Pawlotsky, J.M, Guichou, J.F. | 登録日 | 2011-03-18 | 公開日 | 2012-03-21 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (1.35 Å) | 主引用文献 | Fragment-based discovery of a new family of non-peptidic small-molecule cyclophilin inhibitors with potent antiviral activities. Nat Commun, 7, 2016
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3LQ7
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![BU of 3lq7 by Molmil](/molmil-images/mine/3lq7) | Crystal structure of glutathione s-transferase from agrobacterium tumefaciens str. c58 | 分子名称: | Glutathione S-transferase | 著者 | Patskovsky, Y, Toro, R, Gilmore, M, Chang, S, Sauder, J.M, Burley, S.K, Almo, S.C, New York SGX Research Center for Structural Genomics (NYSGXRC) | 登録日 | 2010-02-08 | 公開日 | 2010-02-23 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Crystal Structure of Glutathione S-Transferase from Agrobacterium Tumefaciens To be Published
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