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2ROV
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BU of 2rov by Molmil
The split PH domain of ROCK II
分子名称: Rho-associated protein kinase 2
著者Wen, W, Zhang, M.
登録日2008-04-25
公開日2008-06-24
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献The split PH domain of ROCK II
To be Published
4UYI
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BU of 4uyi by Molmil
Crystal structure of the BTB domain of human SLX4 (BTBD12)
分子名称: STRUCTURE-SPECIFIC ENDONUCLEASE SUBUNIT SLX4
著者Pinkas, D.M, Sanvitale, C.E, Strain-Damerell, C, Fairhead, M, Wang, D, Tallant, C, Cooper, C.D.O, Sorrell, F.J, Kopec, J, Chaikuad, A, Fitzpatrick, F, Pike, A.C.W, Hozjan, V, Ying, Z, Roos, A.K, Savitsky, P, Bradley, A, Nowak, R, Filippakopoulos, P, Krojer, T, Burgess-Brown, N.A, Marsden, B.D, von Delft, F, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Bullock, A.
登録日2014-09-01
公開日2014-10-01
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (1.86 Å)
主引用文献Crystal Structure of the Btb Domain of Human Slx4 (Btbd12)
To be Published
4UR3
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BU of 4ur3 by Molmil
Crystal structure of the PCE reductive dehalogenase from S. multivorans P2(1) crystal form
分子名称: IRON/SULFUR CLUSTER, NORPSEUDO-B12, TETRACHLOROETHENE REDUCTIVE DEHALOGENASE CATALYTIC SUBUNIT
著者Bommer, M, Kunze, C, Fesseler, J, Schubert, T, Diekert, G, Dobbek, H.
登録日2014-06-25
公開日2014-10-15
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.235 Å)
主引用文献Structural Basis for Organohalide Respiration.
Science, 346, 2014
4UR2
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BU of 4ur2 by Molmil
Crystal structure of the PCE reductive dehalogenase from S. multivorans in complex with iodide
分子名称: GLYCEROL, IODIDE ION, IRON/SULFUR CLUSTER, ...
著者Bommer, M, Kunze, C, Fesseler, J, Schubert, T, Diekert, G, Dobbek, H.
登録日2014-06-25
公開日2014-10-15
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.096 Å)
主引用文献Structural Basis for Organohalide Respiration.
Science, 346, 2014
2RPV
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BU of 2rpv by Molmil
Solution Structure of GB1 with LBT probe
分子名称: Immunoglobulin G-binding protein G, LANTHANUM (III) ION
著者Saio, T, Ogura, K, Yokochi, M, Kobashigawa, Y, Inagaki, F.
登録日2008-10-28
公開日2009-09-15
最終更新日2021-11-10
実験手法SOLUTION NMR
主引用文献Two-point anchoring of a lanthanide-binding peptide to a target protein enhances the paramagnetic anisotropic effect
J.Biomol.Nmr, 44, 2009
4UVW
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BU of 4uvw by Molmil
Crystal structure of human tankyrase 2 in complex with 4,5-dimethyl-3- phenyl-1,2-dihydroisoquinolin-1-one
分子名称: 4,5-dimethyl-3-phenylisoquinolin-1(2H)-one, SULFATE ION, TANKYRASE-2, ...
著者Haikarainen, T, Narwal, M, Lehtio, L.
登録日2014-08-08
公開日2015-07-29
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Exploration of the Nicotinamide-Binding Site of the Tankyrases, Identifying 3-Arylisoquinolin-1-Ones as Potent and Selective Inhibitors in Vitro.
Bioorg.Med.Chem., 23, 2015
4UZZ
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BU of 4uzz by Molmil
Crystal structure of the TtIFT52-46 complex
分子名称: INTRAFLAGELLAR TRANSPORT COMPLEX B PROTEIN 46 CARBOXY-TERMINAL PROTEIN, INTRAFLAGELLAR TRANSPORTER-LIKE PROTEIN
著者Braeuer, P, Taschner, M, Lorentzen, E.
登録日2014-09-09
公開日2014-11-05
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.318 Å)
主引用文献Crystal Structures of Ift70/52 and Ift52/46 Provide Insight Into Intraflagellar Transport B Core Complex Assembly.
J.Cell Biol., 207, 2014
4UQU
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BU of 4uqu by Molmil
Crystal structure of the tetrachloroethene reductive dehalogenase from Sulfurospirillum multivorans
分子名称: BENZAMIDINE, GLYCEROL, IRON/SULFUR CLUSTER, ...
著者Bommer, M, Kunze, C, Fesseler, J, Schubert, T, Diekert, G, Dobbek, H.
登録日2014-06-25
公開日2014-10-15
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (1.595 Å)
主引用文献Structural Basis for Organohalide Respiration.
Science, 346, 2014
4URV
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BU of 4urv by Molmil
The crystal structure of H-Ras and SOS in complex with ligands
分子名称: 4-(4-BROMOPHENYL)PIPERIDIN-4-OL, FORMIC ACID, GTPASE HRAS, ...
著者Winter, J.J.G, Anderson, M, Blades, K, Brassington, C, Breeze, A.L, Chresta, C, Embrey, K, Fairley, G, Faulder, P, Finlay, M.R.V, Kettle, J.G, Nowak, T, Overman, R, Patel, S.J, Perkins, P, Spadola, L, Tart, J, Tucker, J, Wrigley, G.
登録日2014-07-02
公開日2015-03-04
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.58 Å)
主引用文献Small Molecule Binding Sites on the Ras:SOS Complex Can be Exploited for Inhibition of Ras Activation.
J.Med.Chem., 58, 2015
4UVU
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BU of 4uvu by Molmil
Crystal structure of human tankyrase 2 in complex with 1-((4-(5- methyl-1-oxo-1,2-dihydroisoquinolin-3-yl)phenyl)methyl)pyrrolidin-1- ium
分子名称: 5-methyl-3-[4-(pyrrolidin-1-ylmethyl)phenyl]isoquinolin-1(2H)-one, GLYCEROL, SULFATE ION, ...
著者Haikarainen, T, Narwal, M, Lehtio, L.
登録日2014-08-08
公開日2015-07-29
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Exploration of the Nicotinamide-Binding Site of the Tankyrases, Identifying 3-Arylisoquinolin-1-Ones as Potent and Selective Inhibitors in Vitro.
Bioorg.Med.Chem., 23, 2015
4UR0
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BU of 4ur0 by Molmil
Crystal structure of the PCE reductive dehalogenase from S. multivorans in complex with trichloroethene
分子名称: 1,1,2-trichloroethene, BENZAMIDINE, GLYCEROL, ...
著者Bommer, M, Kunze, C, Fesseler, J, Schubert, T, Diekert, G, Dobbek, H.
登録日2014-06-25
公開日2014-10-15
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (1.798 Å)
主引用文献Structural Basis for Organohalide Respiration.
Science, 346, 2014
4UZ2
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BU of 4uz2 by Molmil
Crystal structure of the N-terminal LysM domains from the putative NlpC/P60 D,L endopeptidase from T. thermophilus
分子名称: CELL WALL-BINDING ENDOPEPTIDASE-RELATED PROTEIN
著者Wong, J.E.M.M, Blaise, M.
登録日2014-09-04
公開日2015-01-14
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献An Intermolecular Binding Mechanism Involving Multiple Lysm Domains Mediates Carbohydrate Recognition by an Endopeptidase.
Acta Crystallogr.,Sect.D, 71, 2015
2RR3
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BU of 2rr3 by Molmil
Solution structure of the complex between human VAP-A MSP domain and human OSBP FFAT motif
分子名称: Oxysterol-binding protein 1, Vesicle-associated membrane protein-associated protein A
著者Furuita, K, Jee, J, Fukada, H, Mishima, M, Kojima, C.
登録日2010-03-09
公開日2010-03-23
最終更新日2024-05-01
実験手法SOLUTION NMR
主引用文献Electrostatic interaction between oxysterol-binding protein and VAMP-associated protein A revealed by NMR and mutagenesis studies
J.Biol.Chem., 285, 2010
4UZY
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BU of 4uzy by Molmil
Crystal structure of the Chlamydomonas IFT70 and IFT52 complex
分子名称: CITRATE ANION, FLAGELLAR ASSOCIATED PROTEIN, INTRAFLAGELLAR TRANSPORT PROTEIN IFT52, ...
著者Taschner, M, Lorentzen, E.
登録日2014-09-09
公開日2014-11-05
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.477 Å)
主引用文献Crystal Structures of Ift70/52 and Ift52/46 Provide Insight Into Intraflagellar Transport B Core Complex Assembly.
J.Cell Biol., 207, 2014
2RS2
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BU of 2rs2 by Molmil
1H, 13C, and 15N Chemical Shift Assignments for Musashi1 RBD1:r(GUAGU) complex
分子名称: RNA (5'-R(*GP*UP*AP*GP*U)-3'), RNA-binding protein Musashi homolog 1
著者Ohyama, T, Nagata, T, Tsuda, K, Imai, T, Okano, H, Yamazaki, T, Katahira, M.
登録日2011-06-27
公開日2011-12-28
最終更新日2024-05-01
実験手法SOLUTION NMR
主引用文献Structure of Musashi1 in a complex with target RNA: the role of aromatic stacking interactions
Nucleic Acids Res., 2011
4V23
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BU of 4v23 by Molmil
RSV Matrix protein
分子名称: MATRIX PROTEIN, POTASSIUM ION
著者Forster, A, Maertens, G, Bajorek, M.
登録日2014-10-05
公開日2015-02-25
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Dimerization of Matrix Protein is Required for Budding of Respiratory Syncytial Virus.
J.Virol., 89, 2015
4V3L
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BU of 4v3l by Molmil
RNF38-UB-UbcH5B-Ub complex
分子名称: 1,2-ETHANEDIOL, E3 UBIQUITIN-PROTEIN LIGASE RNF38, POLYUBIQUITIN-C, ...
著者Buetow, L, Gabrielsen, M, Anthony, N.G, Dou, H, Patel, A, Aitkenhead, H, Sibbet, G.J, Smith, B.O, Huang, D.T.
登録日2014-10-20
公開日2015-04-08
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (1.53 Å)
主引用文献Activation of a Primed Ring E3-E2-Ubiquitin Complex by Non-Covalent Ubiquitin.
Mol.Cell, 58, 2015
2SN3
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BU of 2sn3 by Molmil
STRUCTURE OF SCORPION TOXIN VARIANT-3 AT 1.2 ANGSTROMS RESOLUTION
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, SCORPION NEUROTOXIN (VARIANT 3)
著者Zhao, B, Carson, M, Ealick, S.E, Bugg, C.E.
登録日1992-02-20
公開日1994-01-31
最終更新日2017-11-29
実験手法X-RAY DIFFRACTION (1.2 Å)
主引用文献Structure of scorpion toxin variant-3 at 1.2 A resolution.
J.Mol.Biol., 227, 1992
2TIR
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BU of 2tir by Molmil
CRYSTAL STRUCTURE ANALYSIS OF A MUTANT ESCHERICHIA COLI THIOREDOXIN IN WHICH LYSINE 36 IS REPLACED BY GLUTAMIC ACID
分子名称: COPPER (II) ION, THIOREDOXIN
著者Nikkola, M, Gleason, F.K, Fuchs, J.A, Eklund, H.
登録日1993-01-10
公開日1993-10-31
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Crystal structure analysis of a mutant Escherichia coli thioredoxin in which lysine 36 is replaced by glutamic acid.
Biochemistry, 32, 1993
4WFS
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BU of 4wfs by Molmil
Crystal Structure of tRNA-dihydrouridine(20) synthase catalytic domain
分子名称: CHLORIDE ION, FLAVIN MONONUCLEOTIDE, SULFATE ION, ...
著者Bou-Nader, C, Pecqueur, L, Kamah, A, Bregeon, D, Golinelli-Pimpaneau, B, Guimaraes, B.G, Fontecave, M, Hamdane, D.
登録日2014-09-17
公開日2015-10-07
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.68 Å)
主引用文献An extended dsRBD is required for post-transcriptional modification in human tRNAs.
Nucleic Acids Res., 43, 2015
4WG7
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BU of 4wg7 by Molmil
Room-temperature crystal structure of lysozyme determined by serial synchrotron crystallography using a nano focused beam.
分子名称: CHLORIDE ION, Lysozyme C
著者Coquelle, N, Brewster, A.S, Kappe, U, Shilova, A, Weinhausen, B, Burghammer, M, Colletier, J.P.
登録日2014-09-18
公開日2015-05-06
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Raster-scanning serial protein crystallography using micro- and nano-focused synchrotron beams.
Acta Crystallogr.,Sect.D, 71, 2015
2RUH
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BU of 2ruh by Molmil
Chemical Shift Assignments for MIP and MDM2 in bound state
分子名称: E3 ubiquitin-protein ligase Mdm2
著者Nagata, T, Shirakawa, K, Kobayashi, N, Shiheido, H, Horisawa, K, Katahira, M, Doi, N, Yanagawa, H.
登録日2014-06-03
公開日2014-10-15
最終更新日2024-05-15
実験手法SOLUTION NMR
主引用文献Structural Basis for Inhibition of the MDM2:p53 Interaction by an Optimized MDM2-Binding Peptide Selected with mRNA Display
Plos One, 9, 2014
4WGI
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BU of 4wgi by Molmil
A Single Diastereomer of a Macrolactam Core Binds Specifically to Myeloid Cell Leukemia 1 (MCL1)
分子名称: (2S)-2-[(2S,3R)-10-{[(4-fluorophenyl)sulfonyl]amino}-3-methyl-2-[(methyl{[4-(trifluoromethyl)phenyl]carbamoyl}amino)methyl]-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-5(6H)-yl]propanoic acid, FORMIC ACID, MAGNESIUM ION, ...
著者Clifton, M.C, Fairman, J.W, Fang, C, D'Souza, B, Fulroth, B, Leed, A, McCarren, P, Wang, L, Wang, Y, Kaushik, V, Palmer, M, Wei, G, Golub, T.R, Hubbard, B.K, Serrano-Wu, M.H.
登録日2014-09-18
公開日2014-11-19
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Single Diastereomer of a Macrolactam Core Binds Specifically to Myeloid Cell Leukemia 1 (MCL1).
Acs Med.Chem.Lett., 5, 2014
4WJ3
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BU of 4wj3 by Molmil
Crystal structure of the asparagine transamidosome from Pseudomonas aeruginosa
分子名称: 76mer-tRNA, Aspartate--tRNA(Asp/Asn) ligase, Aspartyl/glutamyl-tRNA(Asn/Gln) amidotransferase subunit B, ...
著者Suzuki, T, Nakamura, A, Kato, K, Tanaka, I, Yao, M.
登録日2014-09-29
公開日2014-12-31
最終更新日2020-02-05
実験手法X-RAY DIFFRACTION (3.705 Å)
主引用文献Structure of the Pseudomonas aeruginosa transamidosome reveals unique aspects of bacterial tRNA-dependent asparagine biosynthesis
Proc.Natl.Acad.Sci.USA, 112, 2015
2RHQ
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PheRS from Staphylococcus haemolyticus- rational protein engineering and inhibitor studies
分子名称: 1-{3-[(4-pyridin-2-ylpiperazin-1-yl)sulfonyl]phenyl}-3-(1,3-thiazol-2-yl)urea, Phenylalanyl-tRNA synthetase alpha chain, Phenylalanyl-tRNA synthetase beta chain, ...
著者Evdokimov, A.G, Mekel, M.
登録日2007-10-09
公開日2007-11-06
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Rational protein engineering in action: the first crystal structure of a phenylalanine tRNA synthetase from Staphylococcus haemolyticus.
J.Struct.Biol., 162, 2008

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