8E2M
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![BU of 8e2m by Molmil](/molmil-images/mine/8e2m) | Bruton's tyrosine kinase (BTK) with compound 13 | 分子名称: | (5P)-5-[4-methyl-6-(2-methylpropyl)pyridin-3-yl]-4-oxo-N-[(1R,2S)-2-propanamidocyclopentyl]-4,5-dihydro-3H-1-thia-3,5,8-triazaacenaphthylene-2-carboxamide, TRIETHYLENE GLYCOL, Tyrosine-protein kinase BTK | 著者 | Alexander, R, Milligan, C.M. | 登録日 | 2022-08-15 | 公開日 | 2022-11-16 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.904 Å) | 主引用文献 | Discovery of JNJ-64264681: A Potent and Selective Covalent Inhibitor of Bruton's Tyrosine Kinase. J.Med.Chem., 65, 2022
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5NC8
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![BU of 5nc8 by Molmil](/molmil-images/mine/5nc8) | |
4LI4
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![BU of 4li4 by Molmil](/molmil-images/mine/4li4) | |
4LM9
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![BU of 4lm9 by Molmil](/molmil-images/mine/4lm9) | |
4LMC
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![BU of 4lmc by Molmil](/molmil-images/mine/4lmc) | |
4NL9
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![BU of 4nl9 by Molmil](/molmil-images/mine/4nl9) | |
6G05
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![BU of 6g05 by Molmil](/molmil-images/mine/6g05) | |
7V90
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![BU of 7v90 by Molmil](/molmil-images/mine/7v90) | Telomeric mononucleosome | 分子名称: | DNA (145-mer), Histone H2A type 1-B/E, Histone H2B type 1-K, ... | 著者 | Soman, A. | 登録日 | 2021-08-24 | 公開日 | 2022-07-27 | 最終更新日 | 2024-06-12 | 実験手法 | ELECTRON MICROSCOPY (3.5 Å) | 主引用文献 | Columnar structure of human telomeric chromatin. Nature, 609, 2022
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7VA4
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![BU of 7va4 by Molmil](/molmil-images/mine/7va4) | Telomeric tetranucleosome in open state | 分子名称: | DNA (539-MER), Histone H2A type 1-B/E, Histone H2B type 1-K, ... | 著者 | Soman, A. | 登録日 | 2021-08-27 | 公開日 | 2022-07-27 | 最終更新日 | 2024-06-19 | 実験手法 | ELECTRON MICROSCOPY (14 Å) | 主引用文献 | Columnar structure of human telomeric chromatin. Nature, 609, 2022
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7V9J
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![BU of 7v9j by Molmil](/molmil-images/mine/7v9j) | Telomeric trinucleosome | 分子名称: | DNA (408-mer), Histone H2A type 1-B/E, Histone H2B type 1-K, ... | 著者 | Soman, A. | 登録日 | 2021-08-25 | 公開日 | 2022-07-27 | 最終更新日 | 2024-06-12 | 実験手法 | ELECTRON MICROSCOPY (8 Å) | 主引用文献 | Columnar structure of human telomeric chromatin. Nature, 609, 2022
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7V9C
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![BU of 7v9c by Molmil](/molmil-images/mine/7v9c) | Telomeric Dinucleosome in open state | 分子名称: | DNA (275-mer), Histone H2A type 1-B/E, Histone H2B type 1-K, ... | 著者 | Soman, A. | 登録日 | 2021-08-24 | 公開日 | 2022-07-27 | 最終更新日 | 2024-06-12 | 実験手法 | ELECTRON MICROSCOPY (4.5 Å) | 主引用文献 | Columnar structure of human telomeric chromatin. Nature, 609, 2022
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7V9S
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![BU of 7v9s by Molmil](/molmil-images/mine/7v9s) | Telomeric trinucleosome in open state | 分子名称: | DNA (408-MER), Histone H2A type 1-B/E, Histone H2B type 1-K, ... | 著者 | Soman, A. | 登録日 | 2021-08-26 | 公開日 | 2022-07-27 | 最終更新日 | 2024-06-19 | 実験手法 | ELECTRON MICROSCOPY (11 Å) | 主引用文献 | Columnar structure of human telomeric chromatin. Nature, 609, 2022
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7V9K
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![BU of 7v9k by Molmil](/molmil-images/mine/7v9k) | Telomeric tetranucleosome | 分子名称: | DNA (539-mer), Histone H2A type 1-B/E, Histone H2B type 1-K, ... | 著者 | Soman, A. | 登録日 | 2021-08-25 | 公開日 | 2022-07-27 | 最終更新日 | 2024-06-12 | 実験手法 | ELECTRON MICROSCOPY (8.1 Å) | 主引用文献 | Columnar structure of human telomeric chromatin. Nature, 609, 2022
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7V96
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![BU of 7v96 by Molmil](/molmil-images/mine/7v96) | Telomeric Dinucleosome | 分子名称: | DNA (275-mer), Histone H2A type 1-B/E, Histone H2B type 1-K, ... | 著者 | Soman, A. | 登録日 | 2021-08-24 | 公開日 | 2022-07-27 | 最終更新日 | 2024-06-12 | 実験手法 | ELECTRON MICROSCOPY (3.92 Å) | 主引用文献 | Columnar structure of human telomeric chromatin. Nature, 609, 2022
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8T85
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![BU of 8t85 by Molmil](/molmil-images/mine/8t85) | Structure of RssB bound to beryllofluoride | 分子名称: | BERYLLIUM TRIFLUORIDE ION, DI(HYDROXYETHYL)ETHER, MAGNESIUM ION, ... | 著者 | Brugger, C, Schwartz, J, Deaconescu, A.M. | 登録日 | 2023-06-21 | 公開日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (2.38 Å) | 主引用文献 | Structure of phosphorylated-like RssB, the adaptor delivering sigma s to the ClpXP proteolytic machinery, reveals an interface switch for activation. J.Biol.Chem., 299, 2023
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4MI3
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![BU of 4mi3 by Molmil](/molmil-images/mine/4mi3) | Crystal structure of Gpb in complex with SUGAR (N-{(2R)-2-METHYL-3-[4-(PROPAN-2-YL)PHENYL]PROPANOYL}-BETA-D-GLUCOPYRANOSYLAMINE) (S21) | 分子名称: | Glycogen phosphorylase, muscle form, N-{(2R)-2-methyl-3-[4-(propan-2-yl)phenyl]propanoyl}-beta-D-glucopyranosylamine | 著者 | Kantsadi, L.A, Chatzileontiadou, S.M.D, Leonidas, D.D. | 登録日 | 2013-08-30 | 公開日 | 2014-07-23 | 最終更新日 | 2023-12-06 | 実験手法 | X-RAY DIFFRACTION (2.15 Å) | 主引用文献 | Structure based inhibitor design targeting glycogen phosphorylase b. Virtual screening, synthesis, biochemical and biological assessment of novel N-acyl-beta-d-glucopyranosylamines. Bioorg.Med.Chem., 22, 2014
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1KQY
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![BU of 1kqy by Molmil](/molmil-images/mine/1kqy) | Hevamine Mutant D125A/E127A/Y183F in Complex with Penta-NAG | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, GLYCEROL, Hevamine A, ... | 著者 | Rozeboom, H.J, Dijkstra, B.W. | 登録日 | 2002-01-08 | 公開日 | 2002-01-23 | 最終更新日 | 2023-08-16 | 実験手法 | X-RAY DIFFRACTION (1.92 Å) | 主引用文献 | Expression and characterization of active site mutants of hevamine, a chitinase from the rubber tree Hevea brasiliensis. Eur.J.Biochem., 269, 2002
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1KR0
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![BU of 1kr0 by Molmil](/molmil-images/mine/1kr0) | Hevamine Mutant D125A/Y183F in Complex with Tetra-NAG | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Hevamine A, SULFATE ION | 著者 | Rozeboom, H.J, Dijkstra, B.W. | 登録日 | 2002-01-08 | 公開日 | 2002-01-23 | 最終更新日 | 2023-08-16 | 実験手法 | X-RAY DIFFRACTION (1.92 Å) | 主引用文献 | Expression and Characterization of Active Site Mutants of Hevamine, a
Chitinase from the Rubber Tree Hevea brasiliensis. Eur.J.Biochem., 269, 2002
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1KR1
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![BU of 1kr1 by Molmil](/molmil-images/mine/1kr1) | Hevamine Mutant D125A/E127A in Complex with Tetra-NAG | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Hevamine A, SULFATE ION | 著者 | Rozeboom, H.J, Dijkstra, B.W. | 登録日 | 2002-01-08 | 公開日 | 2002-01-23 | 最終更新日 | 2023-08-16 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Expression and Characterization of Active Site Mutants of Hevamine, a
Chitinase from the Rubber Tree Hevea brasiliensis. Eur.J.Biochem., 269, 2002
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6WE5
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![BU of 6we5 by Molmil](/molmil-images/mine/6we5) | |
8SV9
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![BU of 8sv9 by Molmil](/molmil-images/mine/8sv9) | Crystal structure of ULK1 kinase domain with inhibitor MR-2088 | 分子名称: | (4P)-4-[(2P)-2-(1,2,5,6-tetrahydropyridin-3-yl)-1H-pyrrolo[2,3-b]pyridin-5-yl]-N-(2,2,2-trifluoroethyl)thiophene-2-carboxamide, 1,2-ETHANEDIOL, SULFATE ION, ... | 著者 | Schonbrunn, E, Sun, L. | 登録日 | 2023-05-15 | 公開日 | 2024-03-27 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Development of potent and selective ULK1/2 inhibitors based on 7-azaindole scaffold with favorable in vivo properties. Eur.J.Med.Chem., 266, 2024
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6WSA
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6WSB
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![BU of 6wsb by Molmil](/molmil-images/mine/6wsb) | |
6WTS
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![BU of 6wts by Molmil](/molmil-images/mine/6wts) | CryoEM structure of the C. sordellii lethal toxin TcsL in complex with SEMA6A | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, SEMA6A, ... | 著者 | Kucharska, I, Rubinstein, J.L, Julien, J.P. | 登録日 | 2020-05-03 | 公開日 | 2020-07-08 | 最終更新日 | 2020-08-05 | 実験手法 | ELECTRON MICROSCOPY (3.3 Å) | 主引用文献 | Recognition of Semaphorin Proteins by P. sordellii Lethal Toxin Reveals Principles of Receptor Specificity in Clostridial Toxins. Cell, 182, 2020
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8T4D
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![BU of 8t4d by Molmil](/molmil-images/mine/8t4d) | MD65 N332-GT5 SOSIP in complex with RM_N332_08 Fab and RM20A3 Fab | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, MD65 N332-GT5 SOSIP gp120, ... | 著者 | Ozorowski, G, Torres, J.L, Ward, A.B. | 登録日 | 2023-06-09 | 公開日 | 2024-05-08 | 最終更新日 | 2024-05-29 | 実験手法 | ELECTRON MICROSCOPY (3.1 Å) | 主引用文献 | Vaccine priming of rare HIV broadly neutralizing antibody precursors in nonhuman primates. Science, 384, 2024
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