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9EO4

Outward-open structure of human dopamine transporter bound to cocaine

Summary for 9EO4
Entry DOI10.2210/pdb9eo4/pdb
EMDB information19845
DescriptorSodium-dependent dopamine transporter, CHOLESTEROL, CHOLESTEROL HEMISUCCINATE, ... (7 entities in total)
Functional Keywordsneurotransmitter/sodium symporters, monoamine transporter, dopamine transporter, slc6, membrane protein
Biological sourceHomo sapiens (human)
Total number of polymer chains1
Total formula weight74217.76
Authors
Nielsen, J.C.,Salomon, K.,Kalenderoglou, I.E.,Bargmeyer, S.,Pape, T.,Shahsavar, A.,Loland, C.J. (deposition date: 2024-03-14, release date: 2024-07-03)
Primary citationNielsen, J.C.,Salomon, K.,Kalenderoglou, I.E.,Bargmeyer, S.,Pape, T.,Shahsavar, A.,Loland, C.J.
The molecular basis for cocaine binding to the human dopamine transporter
To Be Published,
Experimental method
ELECTRON MICROSCOPY (2.66 Å)
Structure validation

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PDB entries from 2024-07-17

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