8XI9
Crystal structure of FRB-FKBP fusion protein in complex with rapamycin
Summary for 8XI9
Entry DOI | 10.2210/pdb8xi9/pdb |
Descriptor | FRB-FKBP fusion protein, RAPAMYCIN IMMUNOSUPPRESSANT DRUG (3 entities in total) |
Functional Keywords | rapamycin, signaling protein |
Biological source | Homo sapiens (human) More |
Total number of polymer chains | 1 |
Total formula weight | 24244.86 |
Authors | Inobe, T.,Sakaguchi, R.,Obita, T.,Mukaiyama, A.,Yokoyama, T.,Mizuguchi, M.,Akiyama, S. (deposition date: 2023-12-19, release date: 2024-08-07, Last modification date: 2024-10-09) |
Primary citation | Inobe, T.,Sakaguchi, R.,Obita, T.,Mukaiyama, A.,Koike, S.,Yokoyama, T.,Mizuguchi, M.,Akiyama, S. Structural insights into rapamycin-induced oligomerization of a FRB-FKBP fusion protein. Febs Lett., 598:2292-2305, 2024 Cited by PubMed: 39031920DOI: 10.1002/1873-3468.14986 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.85 Å) |
Structure validation
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