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8R0Q

Pim1 in complex with 6-bromo-1H-benzo[d]imidazol-2-amine and Pimtide

Summary for 8R0Q
Entry DOI10.2210/pdb8r0q/pdb
Related7QB2 7QFM 7Z6U 8AFR 8R0H
DescriptorSerine/threonine-protein kinase pim-1, Pimtide, 1,2-ETHANEDIOL, ... (6 entities in total)
Functional Keywordsserine kinase, kinase, complex, pim1, pim, pim-1, inhibitor, tumorigenisis, cancer, pimtide, proto oncogen, atp, phosphorylation, apoptosis, cell cycle, transferase
Biological sourceHomo sapiens (human)
More
Total number of polymer chains2
Total formula weight37572.89
Authors
Hochban, P.M.M.,Heine, A.,Diederich, W.E. (deposition date: 2023-10-31, release date: 2024-11-13)
Primary citationHochban, P.M.M.,Hubach, D.,Heine, A.,Diederich, W.E.
Pim1 in complex with 6-bromo-1H-benzo[d]imidazol-2-amine and Pimtide
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.7 Å)
Structure validation

248942

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