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7VKE

Crystal structure of human CD38 ECD in complex with UniDab(TM) F11A

Summary for 7VKE
Entry DOI10.2210/pdb7vke/pdb
DescriptorADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1, Unidab F11A, 1,2-ETHANEDIOL, ... (7 entities in total)
Functional Keywordscomplex, transferase, antibody, receptor, hydrolase
Biological sourceHomo sapiens (Human)
More
Total number of polymer chains2
Total formula weight45610.03
Authors
Schooten, W.V.,Schellenberger, U.,Ugamraj, H.S.,Manicka, S.,Bijpuria, S.,Gondu, R.K. (deposition date: 2021-09-29, release date: 2022-08-03, Last modification date: 2023-11-29)
Primary citationUgamraj, H.S.,Dang, K.,Ouisse, L.H.,Buelow, B.,Chini, E.N.,Castello, G.,Allison, J.,Clarke, S.C.,Davison, L.M.,Buelow, R.,Deng, R.,Iyer, S.,Schellenberger, U.,Manika, S.N.,Bijpuria, S.,Musnier, A.,Poupon, A.,Cuturi, M.C.,van Schooten, W.,Dalvi, P.
TNB-738, a biparatopic antibody, boosts intracellular NAD+ by inhibiting CD38 ecto-enzyme activity.
Mabs, 14:2095949-2095949, 2022
Cited by
PubMed: 35867844
DOI: 10.1080/19420862.2022.2095949
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.9 Å)
Structure validation

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