7BI2
PI3KC2aDeltaN and DeltaC-C2
Summary for 7BI2
Entry DOI | 10.2210/pdb7bi2/pdb |
Descriptor | Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit alpha,Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit alpha, 1,2-ETHANEDIOL, 9-(6-aminopyridin-3-yl)-1-[3-(trifluoromethyl)phenyl]benzo[h][1,6]naphthyridin-2(1H)-one, ... (5 entities in total) |
Functional Keywords | pi3kc2 alpha, kinase, transferase |
Biological source | Mus musculus (House Mouse) More |
Total number of polymer chains | 1 |
Total formula weight | 132490.89 |
Authors | Lo, W.T.,Roske, Y.,Daumke, O.,Haucke, V. (deposition date: 2021-01-12, release date: 2022-03-09, Last modification date: 2024-01-31) |
Primary citation | Lo, W.T.,Zhang, Y.,Vadas, O.,Roske, Y.,Gulluni, F.,De Santis, M.C.,Zagar, A.V.,Stephanowitz, H.,Hirsch, E.,Liu, F.,Daumke, O.,Kudryashev, M.,Haucke, V. Structural basis of phosphatidylinositol 3-kinase C2 alpha function. Nat.Struct.Mol.Biol., 29:218-228, 2022 Cited by PubMed: 35256802DOI: 10.1038/s41594-022-00730-w PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (3.25 Å) |
Structure validation
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