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6Z55

Crystal structure of CLK3 in complex with macrocycle ODS2004070

Summary for 6Z55
Entry DOI10.2210/pdb6z55/pdb
DescriptorDual specificity protein kinase CLK3, PHOSPHATE ION, 1,2-ETHANEDIOL, ... (6 entities in total)
Functional Keywordskinase, kinase inhibitor, clk3, macrocycle, nanocyclic, structural genomics, structural genomics consortium, sgc, transferase
Biological sourceHomo sapiens (Human)
Total number of polymer chains2
Total formula weight87413.02
Authors
Chaikuad, A.,Benderitter, P.,Hoflack, J.,Denis, A.,Knapp, S.,Structural Genomics Consortium (SGC) (deposition date: 2020-05-26, release date: 2020-06-03, Last modification date: 2024-01-24)
Primary citationChaikuad, A.,Benderitter, P.,Hoflack, J.,Denis, A.,Knapp, S.,Structural Genomics Consortium (SGC)
Crystal structure of CLK3 in complex with macrocycle ODS2004070
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.7 Å)
Structure validation

218500

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