Summary for 6YZ3
Entry DOI | 10.2210/pdb6yz3/pdb |
Related | 6Z07 6Z17 6Z5K |
Descriptor | LysR family transcriptional regulator, 1,2-ETHANEDIOL, 6-chloranyl-3-[(2-hexyl-2,3-dihydro-1,3-thiazol-4-yl)methyl]quinazolin-4-one, ... (4 entities in total) |
Functional Keywords | pseudomonas aeruginosa, antagonist, quorum sensing, dna binding protein |
Biological source | Pseudomonas aeruginosa |
Total number of polymer chains | 1 |
Total formula weight | 27173.15 |
Authors | Richardson, W.K.,Emsley, J. (deposition date: 2020-05-06, release date: 2020-09-16, Last modification date: 2024-01-24) |
Primary citation | Grossman, S.,Soukarieh, F.,Richardson, W.,Liu, R.,Mashabi, A.,Emsley, J.,Williams, P.,Camara, M.,Stocks, M.J. Novel quinazolinone inhibitors of the Pseudomonas aeruginosa quorum sensing transcriptional regulator PqsR. Eur.J.Med.Chem., 208:112778-112778, 2020 Cited by PubMed: 32927392DOI: 10.1016/j.ejmech.2020.112778 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (3 Å) |
Structure validation
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