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6Y9H

Thrombin in complex with D-Phe-Pro-m-Trifluoromethylbenzylamide derivative (phe2)

Summary for 6Y9H
Entry DOI10.2210/pdb6y9h/pdb
DescriptorProthrombin, Hirudin variant-2, D-Phe-Pro-m-Trifluoromethylbenzylamide derivative (phe2), ... (9 entities in total)
Functional Keywordscoagulation, blood clotting, convertion of fibrinogen to fibrin, blood clotting inhibitor, thrombin inhibitor, preorganization, glycosylation, blood, hydrolase
Biological sourceHomo sapiens (Human)
More
Total number of polymer chains4
Total formula weight36380.04
Authors
Sandner, A.,Heine, A.,Klebe, G.,Abazi, N. (deposition date: 2020-03-09, release date: 2021-03-31, Last modification date: 2024-01-24)
Primary citationSandner, A.,Heine, A.,Klebe, G.
Thrombin in complex with D-Phe-Pro-m-Trifluoromethylbenzylamide derivative (phe2)
To be published,
Experimental method
X-RAY DIFFRACTION (1.48 Å)
Structure validation

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