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6VKA

HIV Integrase Core domain (IN) in complex with dimer-spanning ligand

Summary for 6VKA
Entry DOI10.2210/pdb6vka/pdb
DescriptorIntegrase, IODIDE ION, 2,2'-{ethane-1,2-diylbis[oxyethane-2,1-diylcarbamoyl-4,1-phenyleneethyne-2,1-diyl(5-methyl-1-benzofuran-2,3-diyl)]}diacetic acid, ... (5 entities in total)
Functional Keywordsvirus, inhibitor, complex, hiv integrase, transferase
Biological sourceHuman immunodeficiency virus 1 (HIV-1)
Total number of polymer chains2
Total formula weight38505.71
Authors
Gorman, M.A.,Parker, M.W. (deposition date: 2020-01-19, release date: 2021-01-20)
Primary citationScanlon, M.,Gorman, M.A.
HIV Integrase core domain (IN) in complex with dimeric spanning inhibitor
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.863 Å)
Structure validation

218853

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